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Browse result page of AntiTbPdb

The total number entries retrieved from this search are 668
IDNameSequenceN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicLengthChiralityNatureSourceOriginSpeciesStrainInhibition ConcentrationIn vitro/ In vivoCell LineIntracellular InhibitionCytotoxicityAnimal ModelEffective Dose in model organismImmune ResponceMechanism of ActionTargetCombination TherapyOther ActivitiesYear of PublicationPubmed ID/ Patent No.
antitb_1550Lacticin 3147AA-(Dhb)-N-(Dhb)-FALADYWGNNGAWA-(Abu)-L-(Abu)-HEAMAWAKFreeFreeDhb= Didehydroaminobutyric acid, Abu= 2-aminobutyric acidLinear30LCationicNaturalDerived from Lactococcus lactisMycobacterium tuberculosisMycobacterium tuberculosis H37RaIC90= 7.5 μg/mlin vitroNANANANA NANANANANANA201525613372
antitb_1551Lacticin 3147AA-(Dhb)-N-(Dhb)-FALADYWGNNGAWA-(Abu)-L-(Abu)-HEAMAWAKFreeFreeDhb= Didehydroaminobutyric acid, Abu= 2-aminobutyric acidLinear30LCationicNaturalDerived from Lactococcus lactisMycobacterium aviumMycobacterium aviumIC90= 60 μg/mlin vitroNANANANA NANANANANANA201525613372
antitb_1552Lacticin 3147AA-(Dhb)-N-(Dhb)-FALADYWGNNGAWA-(Abu)-L-(Abu)-HEAMAWAKFreeFreeDhb= Didehydroaminobutyric acid, Abu= 2-aminobutyric acidLinear30LCationicNaturalDerived from Lactococcus lactisMycobacterium KansaiiMycobacterium KansaiiIC90= 15 μg/mlin vitroNANANANA NANANANANANA201525613372
antitb_1553E50-52TTKNYGNGVCNSVNWCQCGNVWASCNLATGCAAWLCKLAFreeFreeNoneLinear39LCationicNaturalDerived from Enterococcus faecalisMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC= 0.1mg/L (within macrophage)in vitro NANANANA NANANANANANA201525613372
antitb_1554E50-52TTKNYGNGVCNSVNWCQCGNVWASCNLATGCAAWLCKLAFreeFreeNoneLinear39LCationicNaturalDerived from Enterococcus faecalisMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 1μg/mlin vitroNANANANA NANANANANANA201525613372
antitb_1555Pk34PRVIETKVHGREVTGLARNVSEENVDRLAKRWIKFreeFreeNoneLinear34LCationicMycobacteriophage derivedDerived from mycobacteriophage Mycobacterium tuberculosisMycobacterium tuberculosis H37RvIC50= 50 μg/mlin vitroNANAMacrophage like J774A.1 cell lineBALB/C mice 20mg/KgIncrease production of cytokine like IFN-γ,TNF-α,IL-12,MCp-1, IL-10, IL-6 NANANABactericidal against E.coli, pseudomonas, S.aureus, Bacillus subtilis201525613372
antitb_1557Vgf-1ECYRKSDIVTCEPWQKFCYREVTFFPNHPVYLSGCASECTETNSKWCCTTDKCNRARGGFreeFreeNoneLinear59LNANaturalDerived from snake venom N.atraMycobacterium tuberculosisMycobacterium tuberculosis H37Rv ATCC25618 (resistant to INH) DR-iMIC = 8.5 ± 0.1 mg/Lin vitroNANANANA NANANANANANA200312927960
antitb_1558Vgf-1ECYRKSDIVTCEPWQKFCYREVTFFPNHPVYLSGCASECTETNSKWCCTTDKCNRARGGFreeFreeNoneLinear59LNANaturalDerived from snake venom N.atraMycobacterium tuberculosisMycobacterium tuberculosis H37Rv ATCC25618 (resistant to INH+Rif) DR-irMIC = 8.5 ± 0.1 mg/Lin vitroNANANANA NANANANANANA200412927960
antitb_1559Vgf-1ECYRKSDIVTCEPWQKFCYREVTFFPNHPVYLSGCASECTETNSKWCCTTDKCNRARGGFreeFreeNoneLinear59LNANaturalDerived from snake venom N.atraMycobacterium tuberculosisMycobacterium tuberculosis H37Rv ATCC25618 (resistant to INH+Streptomycin) DR-isMIC = 8.5 ± 0.1 mg/Lin vitroNANANANA NANANANANANA200512927960
antitb_1560Vgf-1ECYRKSDIVTCEPWQKFCYREVTFFPNHPVYLSGCASECTETNSKWCCTTDKCNRARGGFreeFreeNoneLinear59LNANaturalDerived from snake venom N.atraMycobacterium tuberculosisMycobacterium tuberculosis H37Rv ATCC25618 (resistant to INH+Streptomycin) DR-isMIC = 8.5 ± 0.1 mg/Lin vitroNANANANA NANANANANANA200612927960
antitb_1561Vgf-1ECYRKSDIVTCEPWQKFCYREVTFFPNHPVYLSGCASECTETNSKWCCTTDKCNRARGGFreeFreeNoneLinear59LNANaturalDerived from snake venom N.atraMycobacterium tuberculosisMycobacterium tuberculosis H37Rv ATCC25618 (resistant to INH+Rif+Streptomycin) DR-irsMIC = 8.5 ± 0.1 mg/Lin vitroNANANANA NANANANANANA200712927960
antitb_1562Vgf-1ECYRKSDIVTCEPWQKFCYREVTFFPNHPVYLSGCASECTETNSKWCCTTDKCNRARGGFreeFreeNoneLinear59LNANaturalDerived from snake venom N.atraMycobacterium tuberculosisMycobacterium tuberculosis H37Rv ATCC25618 (resistant to INH+Rif+Streptomycin+ehambutol) DR-irseMIC = 8.5 ± 0.1 mg/Lin vitroNANANANA NANANANANANA200812927960
antitb_1607TP-5RKDVYFreeAmidationNoneLinear4LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = > 1000mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1608RR-6RRRRRRFreeAmidationNoneLinear5LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = 125 mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1609RR-11RKDVYRRRRRRFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = 125 mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1610RY-11RRRRRRRKDVYFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = 125 mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1611TP-5RKDVYFreeAmidationNoneLinear4LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceNAin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1612RR-6RRRRRRFreeAmidationNoneLinear5LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1613RR-11RKDVYRRRRRRFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1614RY-11RRRRRRRKDVYFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1615RY-11RRRRRRRKDVYFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNARR-11 Peptide(31.25 mg/L) + Rifampicin (1.95mg/L)NA201424411680
antitb_1616LKLLKKLLKKFreeAmidationNoneLinear8LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 125 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1617PPPLLKKLLKKPFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 250 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1618CCCLLKKLLKKCFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 250 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1619IIILLKKLLKKIFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1620MMMLLKKLLKKMFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1621WWWLLKKLLKKWFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1622LKLLKKLLKKFreeAmidationNoneLinear8LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1623PPPLLKKLLKKPFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 125 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1624CCCLLKKLLKKCFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 250 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1625IIILLKKLLKKIFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 15.6 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1626MMMLLKKLLKKMFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 15.6 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1627WWWLLKKLLKKWFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 0.98 μg/mlin vitroRAW 264.7 mouse macrophageNA>500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1628LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTESFreeFreeNoneLinear37LCationicSyntheticNAMycobacterium smegmatisMycobacteria smegmatis mc2 155MIC = 2400 μg/mlin vitro J774 macrophage cell linesNAIC50= 11226 μg/mlNA NAStimulation of TNF-α productioninhibit bacterial Atpase activityNANANA201526218806
antitb_1629LLAPRKSAKKIGKRAKRFreeFreeNoneLinear13LCationicNaturalNAMycobacterium smegmatisMycobacteria smegmatis mc2 155MIC = 600 μg/mlin vitro J774 macrophage cell linesNAIC50= 11226 μg/mlNA NAStimulation of TNF-α productioninhibit bacterial Atpase activityNANANA201526218806
antitb_1653NAWKWLKKWIK FreeFreeNoneLinear9LCationicSyntheticNAMycobacterium Tuberculosis Mycobacterium tuberculosis H37RvIC90 = 1.5 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201626645944
antitb_1723SEQ ID NO 3NVTSIHSLLFreeFreeNoneLinear9LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1724SEQ ID NO 4ELNNALQNLARTFreeFreeNoneLinear12LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1725SEQ ID NO 7SGSEAYQGVQQKWDAFreeFreeNoneLinear15LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1726SEQ ID NO 8TATELNNALFreeFreeNoneLinear9LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1727SEQ ID NO 9RTISEAGQAMFreeFreeNoneLinear10LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1728SEQ ID NO 10AYQGVQQKWFreeFreeNoneLinear9LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1729SEQ ID NO 11SEAYQGVQQFreeFreeNoneLinear9LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1730SEQ ID NO 12SEAYQGVQQKFreeFreeNoneLinear10LNAProtein DerivedFrom the proetins containing mycobacterial CD8 T cell epitopesMycobacterium tuberculosisMycobacterium tuberculosisNAIn vitroPBMcsNANAβ2-microglobulin gene knowckout mice, TAP-1 null mutant mice and HSP-65 immunized mice NAIFN-γ release increasesBy CD8 T cell responseNANoneNone2002US 2002/013197
antitb_1731Seq ID No 10KMHATNHGGGSFreeFreeNoneLinear11LNASyntheticFrom random peptide libraries diplayed on bacteriophage M13Mycobacterium tuberculosisMycobacterium tuberculosis100 μM completely inhibits the cahpaeron activity of Hsp 16.3In vitroMouse bone marrow derive dmacrophages and THP-1NANANone NANAInhibit chaperon activity of heat shock protein 16.3 (Hsp 16.3)Heat shock protein (Hsp 16.3)NoneNone2007US 2007/003721
antitb_1732Seq ID No 22YPHHFKHRHIPIGGGSFreeFreeNoneLinear16LNASyntheticFrom random peptide libraries diplayed on bacteriophage M14Mycobacterium tuberculosisMycobacterium tuberculosis100 μM completely inhibits the cahpaeron activity of Hsp 16.3In vitroMouse bone marrow derive dmacrophages and THP-1NANANone NANAInhibit chaperon activity of heat shock protein 16.3 (Hsp 16.3)Heat shock protein (Hsp 16.3)NoneNone2007US 2007/003721
antitb_1733Seq ID No 1GVENVSWFreeFreeNoneLinear7LNASyntheticFrom random peptide libraries diplayed on bacteriophage M15Mycobacterium tuberculosisMycobacterium tuberculosis100 μM completely inhibits the cahpaeron activity of Hsp 16.3In vitroMouse bone marrow derive dmacrophages and THP-1NANANone NANAInhibit chaperon activity of heat shock protein 16.3 (Hsp 16.3)Heat shock protein (Hsp 16.3)NoneNone2007US 2007/003721
antitb_1734Seq ID No 2KMHATNHFreeFreeNoneLinear7LNASyntheticFrom random peptide libraries diplayed on bacteriophage M16Mycobacterium tuberculosisMycobacterium tuberculosis100 μM completely inhibits the cahpaeron activity of Hsp 16.3In vitroMouse bone marrow derive dmacrophages and THP-1NANANone NANAInhibit chaperon activity of heat shock protein 16.3 (Hsp 16.3)Heat shock protein (Hsp 16.3)NoneNone2007US 2007/003721
antitb_1735Seq ID No 9KMHATNHGGGSFreeFreeNoneLinear11LNASyntheticFrom random peptide libraries diplayed on bacteriophage M17Mycobacterium tuberculosisMycobacterium tuberculosis100 μM completely inhibits the cahpaeron activity of Hsp 16.3In vitroMouse bone marrow derive dmacrophages and THP-1NANANone NANAInhibit chaperon activity of heat shock protein 16.3 (Hsp 16.3)Heat shock protein (Hsp 16.3)NoneNone2007US 2007/003721
antitb_1736Seq ID No 21YPHHFKHRHIPIFreeFreeNoneLinear12LNASyntheticFrom random peptide libraries diplayed on bacteriophage M18Mycobacterium tuberculosisMycobacterium tuberculosis100 μM completely inhibits the cahpaeron activity of Hsp 16.3In vitroMouse bone marrow derive dmacrophages and THP-1NANANone NANAInhibit chaperon activity of heat shock protein 16.3 (Hsp 16.3)Heat shock protein (Hsp 16.3)NoneNone2007US 2007/003721