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Browse result page of AntiTbPdb

The total number entries retrieved from this search are 434
IDNameSequenceN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicLengthChiralityNatureSourceOriginSpeciesStrainInhibition ConcentrationIn vitro/ In vivoCell LineIntracellular InhibitionCytotoxicityAnimal ModelEffective Dose in model organismImmune ResponceMechanism of ActionTargetCombination TherapyOther ActivitiesYear of PublicationPubmed ID/ Patent No.
antitb_1334Cairomycin Bnot availableNANANACyclic0MixNANaturalStreptomyces fungusMycobacterium tuberculosis Mycobacterium tuberculosis H37RvMIC= 50 μg/mL BothNANANASwiss mice 3 mg/kg of body weightNANANANAAntimicrobial against S.aureus, B.subtilis, P.aureginosa,Pseudomonas. Antifungal also.1976855995
antitb_1335Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium tuberculosis Mycobacterium tuberculosis H37RvIC50 = <0.0125 μg/mL (50%)BothNANANAICR/JCL male mice and male beagle dogs 10 mg/kg for mice and 50mg/kg for dogNANANANANA19883348603
antitb_1336Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium intracellulareMycobacterium intracellulareIC50 = 1.56 μg/mL (50%)BothNANANAICR/JCL male mice and male beagle dogs 11 mg/kg for mice and 50mg/kg for dogNANANANANA19883348603
antitb_1337Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium kansasiiMycobacterium kansasiiIC50= 0.39 μg/mL (50%)BothNANANAICR/JCL male mice and male beagle dogs 12 mg/kg for mice and 50mg/kg for dogNANANANANA19883348603
antitb_1338Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium tuberculosis Mycobacterium tuberculosis H37RvIC90= 0.05 μg/mL(90%)BothNANANAICR/JCL male mice and male beagle dogs 13 mg/kg for mice and 50mg/kg for dogNANANANANA19883348603
antitb_1339Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium intracellulareMycobacterium intracellulareIC90= 0.78 μg/mL(90%)BothNANANAICR/JCL male mice and male beagle dogs 14 mg/kg for mice and 50mg/kg for dogNANANANANA19883348603
antitb_1340Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium kansasiiMycobacterium kansasiiIC90= 0.78 μg/mL(90%)BothNANANAICR/JCL male mice and male beagle dogs 15 mg/kg for mice and 50mg/kg for dogNANANANANA19883348603
antitb_1341Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium bovisMycobacterium tuberculosis H37RvNABothNANANAICR/JCL Mice 15 mg/kg for mice and 50mg/kg for dogNANANA4mg of DHMPA peptide+ 0.1 mg of IsoniazidNA19883348603
antitb_1342Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium tuberculosis Mycobacterium tuberculosis R-KMNABothNANANAICR/JCL Mice 15 mg/kg for mice and 50mg/kg for dogNANANA4mg of DHMPA peptide+ 0.1 mg of IsoniazidNA19883348603
antitb_1343Dihydromycoplanecin AR-N(CH3)-CH(CH-CH3-CH3)-CO-N(CH-C-CH2-CH3-C-CH)-CO-N(CH3)-CH-C)-NH-CH(CH2-CH-CH3-CH3)-CO-N-CH-C-CH3_C-CH)-CONH-CH(CH2-CH2-CH-CH3-CH3)-Co-N-CH3-Ch-CH(CH3-CH3)-Co-N-(CH-C-Ch)-Co-N(CH3)-CH(CH2-CH-CH3-CH3)-CO-NH-CH2-CO-O-CH(CH3)Propanol is attached FreeR =CH3-CH2-CH(OH)-COCyclic21MixNANaturalAspergillus awajinensisMycobacterium smegmatisMycobacterium smegmatis ATCC 607FIC= 0.250 - 0.375 NANANANANA NANANANADHMPA+ IsoniazidNA19883348603
antitb_1344Tenecin 1 fragment 1-15VTCDILSVEAKGVKL FreeAmidationNoneLinear15NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 607MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANANone19989693108
antitb_1345Tenecin 1 fragment 17-27DAACAAHCLFR FreeAmidationInternal disulphide bondCyclic11NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 608MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANANone19989693108
antitb_1346Tenecin 1 fragment 16-32DAACAAHCLFR FreeAmidationNoneLinear11NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 609MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANANA19989693108
antitb_1347Tenecin 1 fragment 29-43NDAACAAHCLFRGRSGG FreeAmidationNoneLinear17NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 610MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANAAntibacterial against MRSA, bacillus subtilis, E.coli, Shigella at 10-30 μg/ml19989693108
antitb_1348Tenecin 1 Fragment 33-42RSGGYCNGKRVCVCR FreeAmidationNoneLinear15NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 611MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANAAntibacterial against MRSA, bacillus subtilis, E.coli, Shigella at 10-30 μg/ml19989693108
antitb_1349Tenecin 1 Fragment 33-43YCNGKRVCVC FreeAmidationInternal disulphide bondCyclic10NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 612MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANAAntibacterial against MRSA, bacillus subtilis, E.coli, Shigella at 10-30 μg/ml19989693108
antitb_1350Tenecin 1 Fragment 34-43YCNGKRVCVCR FreeAmidationNoneLinear11NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 613MIC = >100 μg/mlin vitroHuman erythrocyteNACytotoxic at >10 μg/mlNA NANAMembrane disruption as reported by membrane leaky assayNANANone19989693108
antitb_1351Tenecin 1 Fragment 35-43CNGKRVCVCR FreeAmidationNoneLinear10NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 614MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANAMembrane disruption as reported by membrane leaky assayNANANone19989693108
antitb_1352Tenecin 1 Fragment 34-42NGKRVCVCR FreeAmidationNoneLinear9NANANaturalLarvae of tenebrio molitor(beetle)Mycobacterium smegmatisMycobacterium smegmatis ATCC 615MIC = >100 μg/mlin vitroHuman erythrocyteNANoneNA NANANANANANone19989693108
antitb_1354Nk-lysinNEDTVTQAASRVCDKMKILRGVCKKIMRTFLRRISKDFreeFreeInternal disuphide bond 13 -23Cyclic37LNANaturalPig cytolytic lymphocytesMycobacterium tuberculosis Mycobacterium tuberculosis H37Rv ATCC 25618IC90 = 30 μMIn vitroHuman erythroleukaemia cell line K562 NA30 % cytolytic activity in range of 3 -7 μM peptide concentrationNA NANANANANAAntibacterial against bacillus megaterium, E.coli, P.aeuroginosaand S.aureus199910585872
antitb_1355NKLF1VTQAASRVCDKMKILRGVCKKIMRTFLRRFreeFreeInternal disulphide bond at residue between 9-13Cyclic29LNANaturalPig cytolytic lymphocytesMycobacterium tuberculosis Mycobacterium tuberculosis H37Rv ATCC 25619IC90 = 30 μMIn vitroHuman erythroleukaemia cell line K562 NA31 % cytolytic activity in range of 3 -7 μM peptide concentrationNA NANANANANAAntibacterial against bacillus megaterium, E.coli, P.aeuroginosaand S.aureus199910585872
antitb_1356NKLF2VCDKMKILRGVCKKIMRTFLRRFreeFreeNoneCyclic22LNANaturalPig cytolytic lymphocytesMycobacterium tuberculosis Mycobacterium tuberculosis H37Rv ATCC 25620IC90 = 30 μMIn vitroHuman erythroleukaemia cell line K562 NA32 % cytolytic activity in range of 3 -7 μM peptide concentrationNA NANANANANAAntibacterial against bacillus megaterium, E.coli, P.aeuroginosaand S.aureus199910585872
antitb_1357Gran F2VCRTGRSRWRDVCRNFMRRYQSRFreeFreeInternal disulphide bond at residue between 2-13Cyclic23LNANaturalHuman cytolytic lymphocytesMycobacterium tuberculosis Mycobacterium tuberculosis H37Rv ATCC 25621IC90 = 30 μMIn vitroHuman erythroleukaemia cell line K562 NA33 % cytolytic activity in range of 3 -7 μM peptide concentrationNA NANANANANAAntibacterial against bacillus megaterium, E.coli, P.aeuroginosaand S.aureus199910585872
antitb_1358Gran F1VSNAATRVCRTGRSRWRDVCRNFMRRYQSRFreeFreeNoneLinear30LNANaturalHuman cytolytic lymphocytesMycobacterium tuberculosis Mycobacterium tuberculosis H37Rv ATCC 25622IC90 = 30 μMIn vitroHuman erythroleukaemia cell line K562 NA34 % cytolytic activity in range of 3 -7 μM peptide concentrationNA NANANANANAAntibacterial against bacillus megaterium, E.coli, P.aeuroginosaand S.aureus199910585872
antitb_1359GranulysinTQRSVSNAATRVCRTGRSRWRDVCRNFMRRYQSRVTQGFreeFreeNoneLinear38LNANaturalHuman cytolytic lymphocytesMycobacterium tuberculosis Mycobacterium tuberculosis H37Rv ATCC 25623IC90 = 30 μMIn vitroHuman erythroleukaemia cell line K562 NA35 % cytolytic activity in range of 3 -7 μM peptide concentrationNA NANANANANAAntibacterial against bacillus megaterium, E.coli, P.aeuroginosaand S.aureus199910585872
antitb_1360PleurocidinGWGSFFKKAAHVGKHVGKAALTHYL FreeFreeNoneLinear25LNANaturalPleuronectes americanus Mycobacterium smegmatisMycobacterium smegmatisMIC = 80 μg/mlIn vitroNoneNANANA NANANANANAAntibacterial against P.aeruginosa, K.pneumoniae,S.aureus and C.albicans200010898673
antitb_1361PleurocidinGWGSFFKKAAHVGKHVGKAALTHYL FreeFreeNoneLinear25LNANaturalPleuronectes americanus Mycobacterium smegmatisMycobacterium smegmatisMIC = 20 μg/mlIn vitroNoneNANANA NANANANA185 μM OF D-CYCLOSERINE DRUG + 5.2 μM OF Peptide reduces ~ 4 time MIC of drug Antibacterial against P.aeruginosa, K.pneumoniae,S.aureus and C.albicans200010898673
antitb_1362Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusMycobacterium tuberculosis Mycobacterium tuberculosis H37RvMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1363Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusMycobacterium vallée Mycobacterium vallée bovineMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1364Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusMycobacterium R1Rv attenuated Mycobacterium R1Rv attenuated humanMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1365Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusBCG-phipps attenuated BCG-phipps attenuated bovineMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1366Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusMycobacterium H37Ra Mycobacterium H37Ra avirlant RaMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1367Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusMycobacterium sigerson Mycobacterium sigerson aviumMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1368Thymus peptidenot availableNANANoneNA0NANANaturalcalf thymusMycobacterium smegmatis Mycobacterium smegmatis SaprophyteMIC = 300 μg/mlIn vitroNoneNANANA NANANANANANA195313118063
antitb_1369Thymus peptidenot availableNANANoneNA0NANANaturalCalf thymusMycobacterium tuberculiiMycobacterium tuberculii BCG-PhippsMIC = 100 μg/mLIn vitroNoneNANANA NANANANANANA195313118063
antitb_1388HepcidinDTHFPICIFCCGCCHRSKCGMCCKTFreeFreeDisulphide linkage between cys7-23, cys10-13, cys11-19,cys14-22Cyclic25LCationicNaturalHuman alveolar type 2 epithiliumMycobacterium tuberculosisMycobacterium H37RvNAin vivoA549 cell lineNANo cytotoxicityBALB/C NAIncreased production of TNF-α, IL-1αNAMycobacterium tuberculosis + IFN-Υantimicrobial201121482189
antitb_1389LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /mlin vitroJ774.A1 macrophage cell lines14% bacteria is cleared NANA NANANANANANA201121790937
antitb_1390LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /ml (after 6 hours)in vitroJ774.A1 macrophage cell lines34% bacteria is cleared NANA NANANANANANA201121790937
antitb_1391LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg/mlin vitroJ774.A1 macrophage cell lines41% bacteria is clearedNANA NANANANANANA201121790937
antitb_1392LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg /ml (after 6 hours incubation)in vitroJ774.A1 macrophage cell lines67% bacteria is cleared NANA NANANANANANA201121790937
antitb_1393GEK-31RKSKEKIGKEFKRIVQR IKDFLRNLVPRTES FreeFreeNoneLinear33LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155NAin vitroJ774.A1 macrophage cell linesNANANA NANANANANANA201121790937
antitb_1394LL-18KEFKRIVQRIKDFLRNLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155NAin vitroJ774.A1 macrophage cell linesNANANA NANANANANANA201121790937
antitb_1395LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /mlin vitroJ774.A1 macrophage cell lines67% bacteria is cleared NANA NANANANANANA201121790937
antitb_1396LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /ml (after 6 hours)in vitroJ774.A1 macrophage cell lines89% bacteria is cleared NANA NANANANANANA201121790937
antitb_1397LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg/mlin vitroJ774.A1 macrophage cell lines81% bacteria is cleared NANA NANANANANANA201121790937
antitb_1398LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg /ml (after 6 hours incubation)in vitroJ774.A1 macrophage cell lines98% bacteria is cleared NANA NANANANANANA201121790937
antitb_1399LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria bovisMycobacteria bovis BCGMIC = 25μg/mlin vitroTHP-1 cells NANANA NANANANANANA201121790937
antitb_1400LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria bovisMycobacteria bovis BCGMIC = 25μg /ml (after 624hours incubation)in vitroTHP-1 cells > 60% bacteria is cleared NANA NANANANANANA201121790937
antitb_1401LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /mlin vitroJ774.A1 macrophage cell lines51% bacteria is cleared NANA NANANANANANA201121790937
antitb_1402LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg/mlin vitroJ774.A1 macrophage cell lines80% bacteria is clearedNANA NANANANANANA201121790937