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Browse result page of AntiTbPdb

The total number entries retrieved from this search are 619
IDNameSequenceN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicLengthChiralityNatureSourceOriginSpeciesStrainInhibition ConcentrationIn vitro/ In vivoCell LineIntracellular InhibitionCytotoxicityAnimal ModelEffective Dose in model organismImmune ResponceMechanism of ActionTargetCombination TherapyOther ActivitiesYear of PublicationPubmed ID/ Patent No.
antitb_1876Dhvar4KRLFKKLLFSLRKYFreeFreeNoneLinear14LCationicProtein DerivedHuman salivary Histatin derivativeMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1877Crot(1–9,38–42)YKQCHKKGGKKGSGFreeFreeNoneLinear14LCationicNaturalCrotamine, a toxin of Crotalus durissus terrificusMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1878CM15KWKLFKKIGAVLKVLFreeFreeNoneLinear15LCationicSyntheticFrom Cecropin A and Melittin sequencesMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at 18.9 ± 1.71 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1879MelittinGIGAVLKVLTTGLPALISWIKRKRQQFreeFreeNoneLinear26LCationicNaturalVenom of Apis melliferaMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at 0.339 ± 0.0854 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1880OT20TKPKGTKPKGTKPKGTKPKGFreeFreeNoneLinear20LCationicSyntheticTetramer derivative of tuftsin sequenceMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1893Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC50 = 15.8 ± 4.5 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1894Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC90 = 34.6 ± 22.4 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1895Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC50 = 11.0 ± 4.1 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1896Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC90 = 65.8 ± 19.13 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1897Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC50 = 15.2± 2.9 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1898Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC90 = 37.9 ± 15.9 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1899Human lactoferricin 1-11GKKKKSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1900Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC50 = 14.2 ± 1.5 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1901Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC90 = 18.9 ± 4.0 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1902Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC50 = 8.0 ± 1.5 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1903Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC90 = 22.8 ± 9.1 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1904Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC50 = 12.4± 0.3 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1905Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC90 = 21.5± 4.0 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1906Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14DCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1907Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14DCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1908Bovine lactoferricin 17-30 all KFKCKKWQWKMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1909Bovine lactoferricin 17-30 all KFKCKKWQWKMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1910Bovine lactoferricin 17-30 all RFRCRRWQWRMRRLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1911Bovine lactoferricin 17-30 all RFRCRRWQWRMRRLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1912NoneILSLRWRWKWWKKFreeFreeNoneLinear13LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatisMIC = 8 μMIn vitroJ774.16 mouse macrophages and A549 human lung epithelial cellsNANo cytotoxicity against J774.16 mouse macrophages and A549 human lung epithelial cellsNA NANANALipid bilayerNAAntibacterial against Streptococcus pyogenes, Streptococcus agalactiae, Streptococcus pneumoniae ATCC 49619, Klebsiella pneumoniae, Pseudomonas aeruginosa ATCC27853, Bacillus subtilis BGSC 1A1. 201626902758
antitb_1913NoneILSLRWRWKWWKKFreeFreeNoneLinear13LCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis mc2 6020MIC = 32 μMIn vitroJ774.16 mouse macrophages and A549 human lung epithelial cellsNANo cytotoxicity against J774.16 mouse macrophages and A549 human lung epithelial cellsNA NANANALipid bilayerNAAntibacterial against Streptococcus pyogenes, Streptococcus agalactiae, Streptococcus pneumoniae ATCC 49619, Klebsiella pneumoniae, Pseudomonas aeruginosa ATCC 27853, Bacillus subtilis BGSC 1A1. 201626902758
antitb_1914NoneILSLRWRWKWWKKFreeFreeNoneLinear13LCationicSyntheticNAMycobacterium bovis Mycobacterium bovis BCG pasteur strainMIC = 32 μMIn vitroJ774.16 mouse macrophages and A549 human lung epithelial cellsNANo cytotoxicity against J774.16 mouse macrophages and A549 human lung epithelial cellsNA NANANALipid bilayerNAAntibacterial against Streptococcus pyogenes, Streptococcus agalactiae, Streptococcus pneumoniae ATCC 49619, Klebsiella pneumoniae, Pseudomonas aeruginosa ATCC 27853, Bacillus subtilis BGSC 1A1. 201626902758
antitb_1915Laterosporulin 10ACVNQCPDAIDRFIVKDKGCHGVEKKYYKQVYVACMNGQHLYCRTEWGGPCQLFreeFreeDisulphide bond between residues 2-43, 6-35 and 20-51 Cyclic53DCationicNaturalDerived from Brevibacillus species SKDU10Mycobacterium smegmatisMycobacterium smegmatis MC2 155MIC = 45 μMIn vitro and ex vivoRAW 264.7 murine macrophageNANo cytotoxicity upto 40 μM/ml concentrationNA NANANACell wall pore formation0.00625 μM of rifampicin with 0.25 μM of peptide, a fourfold reduction in MIC of rifampicin against H37 RVAntibacterial against Staphylococcus aureus MTCC 1430, Bacillus subtilis MTCC 121, Pseudomonas aeruginosa MTCC 1934, Vibrio cholerae MTCC 3904, Escherichia coli MTCC 1610201627267959
antitb_1916Peptide-1GF(A6c)G(A6c)KK(A6c)G(A6c)F(A6c)G(A6c)GKK(A6c)KKKKAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Linear22DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC =4.92 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1917Peptide-2GF(A6c)G(A6c)R(A6c)G(A6c)F(A6c)G(A6c)GR(A6c)RRRRAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Linear19DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 40.75 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1918Peptide-3GF(A6c)G(A6c)Orn(A6c)G(A6c)F(A6c)G(A6c)GOrn(A6c)Orn-Orn- Orn- OrnAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, orn = ornithineLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 11.37 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1919Peptide-4GF(A6c)G(A6c)Dab(A6c)G(A6c)F(A6c)G(A6c)GDab(A6c)Dab-Dab-Dab-DabAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Dab = 2,4-diaminobutyric acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC =11.83 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1920Peptide-5GF(A6c)G(A6c)Dpr(A6c)G(A6c)F(A6c)G(A6c)GDpr(A6c) Dpr-Dpr-Dpr- DprAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Dpr = 2,4-diaminopropanoic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 24.63 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1921Peptide-6GF(A5c)G(A5c)K(A5c)G(A5c)F(A5c)G(A5c)GK(A5c)KKKKAcetylationAmidationA5c = 1-aminocyclopentane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 11.42 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1922Peptide-7GF(A5c)G(A5c)R(A5c)G(A5c)F(A5c)G(A5c)GR(A5c)RRRRAcetylationAmidationA5c = 1-aminocyclopentane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC =21.22 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1923Peptide-8GF(A6c)G(Tic)K(A6c)G(Tic)F(A6c)G(Tic)GK(Tic)KKKKAcetylationAmidation Tic = Tetrahydroisoquinolinecarboxylic acid, A6c 1-aminocyclohexane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 10.33 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1924Peptide-9GF(A6c)G(Oic)K(A6c)G(Oic)F(A6c)G(Oic)GK(Oic)KKKKAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Oic = Octahydroindolecarboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 20.92 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1925Peptide-10GF(A5c)G(A6c)K(A5c)G(A6c)F(A5c)G(A6c)GK(A5c)KKKKAcetylationAmidationA5c = 1-aminocyclopentane carboxylic acid, A6c 1-aminocyclohexane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 22.42 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1926Peptide-11KKKKGF(A6c)G(A6c)K(A6c)G(A6c)F(A6c)G(A6c)GK(A6c)AcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Linear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 21.87 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1927Peptide-1GF(A6c)G(A6c)KK(A6c)G(A6c)F(A6c)G(A6c)GKK(A6c)KKKKAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Linear22DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC =4.92 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1928Peptide-2GF(A6c)G(A6c)R(A6c)G(A6c)F(A6c)G(A6c)GR(A6c)RRRRAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Linear19DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 40.75 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1929Peptide-3GF(A6c)G(A6c)Orn(A6c)G(A6c)F(A6c)G(A6c)GOrn(A6c)Orn-Orn- Orn- OrnAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, orn = ornithineLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 11.37 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1930Peptide-4GF(A6c)G(A6c)Dab(A6c)G(A6c)F(A6c)G(A6c)GDab(A6c)Dab-Dab-Dab-DabAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Dab = 2,4-diaminobutyric acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC =25.65 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1931Peptide-5GF(A6c)G(A6c)Dpr(A6c)G(A6c)F(A6c)G(A6c)GDpr(A6c) Dpr-Dpr-Dpr- DprAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Dpr = 2,4-diaminopropanoic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 49.26 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1932Peptide-6GF(A5c)G(A5c)K(A5c)G(A5c)F(A5c)G(A5c)GK(A5c)KKKKAcetylationAmidationA5c = 1-aminocyclopentane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 22.85 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1933Peptide-7GF(A5c)G(A5c)R(A5c)G(A5c)F(A5c)G(A5c)GR(A5c)RRRRAcetylationAmidationA5c = 1-aminocyclopentane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC >43 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1934Peptide-8GF(A6c)G(Tic)K(A6c)G(Tic)F(A6c)G(Tic)GK(Tic)KKKKAcetylationAmidation Tic = Tetrahydroisoquinolinecarboxylic acid, A6c 1-aminocyclohexane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 20.6μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1935Peptide-9GF(A6c)G(Oic)K(A6c)G(Oic)F(A6c)G(Oic)GK(Oic)KKKKAcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Oic = Octahydroindolecarboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 20.92 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1936Peptide-10GF(A5c)G(A6c)K(A5c)G(A6c)F(A5c)G(A6c)GK(A5c)KKKKAcetylationAmidationA5c = 1-aminocyclopentane carboxylic acid, A6c 1-aminocyclohexane carboxylic acidLinear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 11.21 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357
antitb_1937Peptide-11KKKKGF(A6c)G(A6c)K(A6c)G(A6c)F(A6c)G(A6c)GK(A6c)AcetylationAmidationA6c = 1-aminocyclohexane carboxylic acid, Linear20DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis MDRMIC = 5.47 μMIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against Enterobacter aerogenes, Acinetobacter baumannii, Psuedomonas aeruginosa, Klebsiella pneumoniae, Eenterococcus faecalis, Staphylococcus aureus201627387357