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Browse result page of AntiTbPdb

The total number entries retrieved from this search are 434
IDNameSequenceN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicLengthChiralityNatureSourceOriginSpeciesStrainInhibition ConcentrationIn vitro/ In vivoCell LineIntracellular InhibitionCytotoxicityAnimal ModelEffective Dose in model organismImmune ResponceMechanism of ActionTargetCombination TherapyOther ActivitiesYear of PublicationPubmed ID/ Patent No.
antitb_1403LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 25μg/ml (24 hours incubation)in vitroNANANANA NANANANANANA201121790937
antitb_1404LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 100 μg/mL (72 hours incubation)in vitroNANANANA NANANANANANA201121790937
antitb_1477Nocathiacinsnot availableNANANABranched cyclic0NACationicNaturalDerived from Nocardia speciesMycobacterium pneumoniaeMycobacterium pneumoniaeMIC = ≤0.008 mg/mlin vitroMcCoy cell linesNA0.25 μg/mlNA NANABind to the 23S rRNA of the 50S ribosomal subunit and inhibit translation23srRNA subunit of bacteriaNANA201525681127
antitb_1478Lariatin AGSQLVYRWVGHSNVIKGPNANAAlpha carbon of glutamine form amide bond with first glycine and gamma carbon of glutamine involved in side chain formationCyclic18DCationicNaturalDerived from Rhodococcusjostii K01‐B0171Mycobacterium tuberculosisMycobacterium tuberculosis RvMIC = 0.39 mg/Lin vitroNANANANA NANAInhibit cell wall biosynthesisNANANA201525681127
antitb_1479Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacterium tuberculosisMycobacterium tuberculosis RvIC50= 0.0125-25mg/ml in vitroNANANANA NANANANANANA201525681127
antitb_1480Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacterium tuberculosisMycobacterium tuberculosis RvIC90= 0.05 μg/mLin vitroNANANANA NANANANANANA201525681127
antitb_1481Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacterium intracellulareMycobacterium intracellulareIC50= 1.56 μg/ml in vitroNANANANA NANANANANANA201525681127
antitb_1482Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacterium intracellulareMycobacterium intracellulareIC90= 25 μg/mLin vitroNANANANA NANANANANANA201525681127
antitb_1483Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacteria kansaiiMycobacteria kansaiiIC50= 0.39 μg/mL in vitroNANANANA NANANANANANA201525681127
antitb_1484Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacteria kansaiiMycobacteria kansaiiIC90= 0.78 μg/mLin vitroNANANANA NANANANANANA201525681127
antitb_1485Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacteria smegmatisMycobacteria smegmatis ATCC 607MIC = 12.5 μg/mLin vitroNANANANA NANANANADHMP A + INHNA201525681127
antitb_1486Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 25177Reduction in zone of growth to 25 mm at 100 μg conc.LoVo cancer cells NAIC50= 2.25 μg/ml for M.Smegmatis ATCC 25177 NA NANANANANANA201525681127
antitb_1487Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 25177Reduction in zone of growth to 10 mm at 25 μgLoVo cancer cells NAIC50= 2.25μg/ml for M.Smegmatis ATCC 25177 NA NANANANANANA201525681127
antitb_1488Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 35818Reduction in zone of growth to 15 mm at 100 μgLoVo cancer cells NAIC50= 1.95 μg/ml for m.Smegmatis ATCC35818NA NANANANANANA201525681127
antitb_1489Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 35818Reduction in zone of growth to 9 mm at 25 μgLoVo cancer cells NAIC50= 1.95 μg/ml for m.Smegmatis ATCC35818NA NANANANANANA201525681127
antitb_1490Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 25177Reduction in zone of growth to 30 mm at 100 μgLoVo cancer cells NAIC50= 2.25 μg/ml for M.Smegmatis ATCC 25177 NA NANANANANANA201525681127
antitb_1491Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 25177Reduction in zone of growth to 15 mm at 25 μgLoVo cancer cells NAIC50= 2.25μg/ml for M.Smegmatis ATCC 25177 NA NANANANANANA201525681127
antitb_1492Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 35818Reduction in zone of growth to 15 mm at 100 μgLoVo cancer cells NAIC50= 1.95 μg/ml for m.Smegmatis ATCC35818NA NANANANANANA201525681127
antitb_1493Pitipeptolides Anot availableNANANABranched cyclic0DCationicNaturalDerived from Cyanobacterium Lyngbya majusculaMycobacterium tuberculosisMycobacteria smegmatis ATCC 35818Reduction in zone of growth to 10 mm at 25 μgLoVo cancer cells NA IC50= 1.95 μg/ml for m.Smegmatis ATCC35818 NA NANANANANANA201525681127
antitb_1494Lacticin 3147not availableNANANABranched cyclic0DCationicNaturalDerived from Lactococcuslactis Mycobacterium tuberculosisMycobacterium tuberculosis H37 RaIC90= 7.5 mg/ml (±0.36)in vitroNANANANA NANAInhibit biosynthesis of peptidoglycan and form pores in bacterial membraneNANANA201525681127
antitb_1495Lacticin 3148not availableNANANABranched cyclic0DCationicNaturalDerived from Lactococcuslactis Mycobacterium tuberculosisMycobacteria kansasii CIT11/06 IC90= 60 mg/ml (±0.75)in vitroNANANANA NANAInhibit biosynthesis of peptidoglycan and form pores in bacterial membraneNANANA201525681127
antitb_1496Lacticin 3149not availableNANANABranched cyclic0DCationicNaturalDerived from Lactococcuslactis Mycobacterium avium Mycobacterium avium subspecies paratuberculosis ATCC 19698 IC90= 15mg/ml (±0.30) in vitroNANANANA NANAInhibit biosynthesis of peptidoglycan and form pores in bacterial membraneNANANA201525681127
antitb_1497Nisin Anot availableNANANABranched cyclic0DCationicNaturalDerived from Lactococcus lactis Mycobacterium tuberculosisMycobacterium tuberculosis H37 RaIC90= >60mg/ml (±0.18)in vitroNANANANA NANAInhibit biosynthesis of peptidoglycan and form pores in bacterial membraneNANANA201525681127
antitb_1498Nisin Anot availableNANANABranched cyclic0DCationicNaturalDerived from Lactococcuslactis Mycobacterium tuberculosisMycobacteria kansasii CIT11/06 IC90= 60 mg/ml (±0.13)in vitroNANANANA NANAInhibit biosynthesis of peptidoglycan and form pores in bacterial membraneNANANA201525681127
antitb_1499Nisin Anot availableNANANABranched cyclic0DCationicNaturalDerived from Lactococcuslactis Mycobacterium avium Mycobacterium avium subspecies paratuberculosis ATCC 19698IC90= >60 mg/ml (± 2.02)in vitroNANANANA NANAInhibit biosynthesis of peptidoglycan and form pores in bacterial membraneNANANA201525681127
antitb_1500Sansanmycins A (Ssa)not availableNANANABranched cyclic0DCationicNaturalDerived from Streptomyces speciesMycobacterium tuberculosisMycobacterium tuberculosis H37RvIC50= 16 μg/mlin vitroNANANANA NANAInhibit the MraY translocase present in the bacterial cell membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1501Sansanmycins A (Ssa)not availableNANANABranched cyclic0DCationicNaturalDerived from Streptomyces speciesMycobacterium tuberculosisMycobacterium tuberculosis 2199IC50= 32 μg/mlIn vitroNANANANA NANAInhibit the MraY translocase present in the bacterial cell membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1502Cyclomarin Anot availableNANANABranched cyclic0DCationicNaturalDerived from Streptomyces speciesMycobacterium tuberculosisMycobacterium tuberculosis H37RvIC50= 0.3mg/mlin vitroNANANANA NAChange the clp1subunit of casinolytic protease by allosteric bindingNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1503Massetolide Anot availableNANANABranched cyclic0DCationicNaturalDerived from Pseudomonas fluorescens SS101Mycobacterium tuberculosisMycobacterium tuberculosis h37RVMIC = 5 mg/mlin vitroNANANANA NAinterfere with bacterial cell wall biosynthesisNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1504Visconsinnot availableNANANABranched cyclic0DCationicNaturalDerived from Pseudomonas speciesMycobacterium tuberculosisMycobacterium avium intercellularaeMIC = 10 mg/mlin vitroNANANANA NAinterfere with bacterial cell wall biosynthesisNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1505Bacitracinnot availableNANANABranched cyclic0DCationicNaturalDerived from Bacillus subtilisMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 130mg/mlin vitroNANANANA NANAinhibit bacterial cell wall synthesisNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1506SP508AR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 31.25 μg/mlin vitroNANANANA NANASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1507SP508BR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue Cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1508SP22AR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 7.8 μg/mlin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1509SP22BR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 31.25 μg/mlin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1510SP508AR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to15 mm at 31.25 mg/Lin vitroNANANANA NANASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1511SP508BR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue Cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to 18 mm at 62.5 mg/Lin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1512SP22AR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to 12 mm 7.8 mg/Lin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1513SP22BR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to 14 mm at 31.25 mg/Lin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1514Hirsutatins Anot availableFreeFreeNoneBranched cyclic0DCationicNaturalDerived from HirsutellaniveaMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC =50 mg/mlin vitroNANANANA NANANANANANA201525681127
antitb_1515Hirsutatins Bnot availableFreeFreeNoneBranched cyclic0DCationicNaturalDerived from HirsutellaniveaMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 50 mg/mlin vitroNANANANA NANANANANANA201525681127
antitb_1516PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium tuberculosisMycobacterium tuberculosis H37RvReduction in growth is inhibited to to 30 % at conc. 6.25 mg/Lin vitroNANANANA NANANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1517PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium tuberculosisMycobacterium tuberculosis H37RvReduction in growth is inhibited to to80% at conc. 50 mg/Lin vitroNANANANA NANANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1518PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium tuberculosisMycobacterium tuberculosis H37RvIC50 = 17± 9 mg/Lin vitroNANANANA NANANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1519PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium tuberculosisMycobacterium tuberculosis E1380/94 (MDR resistant stain)IC50= 93± 12 mg/Lin vitroNANANANA NANANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1520PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium smegmatis Mycobacterium smegmatis susceptible strain50 mg/Lin vitroNANANANA NANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1521PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium tuberculosisMycobacterium tuberculosis H37RvIC50= 50 mg/Lin vitroNANANANA NANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1522PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium tuberculosisMycobacterium tuberculosis E1380/94 (MDR resistant stain)IC50= 50 mg/Lin vitroNANANANA NANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1523PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium avium Mycobacterium avium susceptible strainMIC= 50 mg/Lin vitroNANANANA NANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1535Human neutrohil peptide (HNP-1)DCYCRIPACIAGERRYGTCIYQGRLWAFCCFreeFreeDisulphide linkage between cys2-cys30, cys4-cys19,cys9-cys29Cyclic30LCationicNaturalHuman neutrophil Mycobacterium tuberculosisMycobacterium tuberculosis H37Rv2.5 μg/mlin vitroNANANo cytotoxicityNA NAMediate macrophage to induce TNF-α expression Inhibit lipid biosynthesiNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525613372