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KRWWKWIRW details
Primary information
ID antitb_1219,
Name23231581
N-Terminal modificationCathelicidin HHC-10
C-Terminal ModificationKRWWKWIRW
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature9
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium bovis
In Vitro/ In vivoMycobacterium tuberculosis complex bacteria, Mycobacterium bovis bacille calmette guerin (BCG) (Mycobacterium bovis BCG Pasteur 1173P2)
Cell Line69 % decrease in CFU at 50 μg/ ml
Inhibition ConcentrationBoth
Sequence2013
CytotoxicityNone
In vivo ModelNA
Lethal DoseNA
Immune Responce8–9 weeks old C57BL/6 mice
Mechanism of ActionCFUs in mouse lungs were reduced 77.8% at 1.25 mg
TargetSignificant reduction of IFN-γ transcription
Combination TherapyCell envelope disruption
Other activitiesCell envelope
PMIDNone
Year of PublicationAntibacterial (such as Pseudomonas aeruginosa, Escherichia coli, Klebsiella pneumonia, and S. aureus etc
Tertiary Structure
(Technique)
Not Predicted),
Primary information
ID antitb_1220,
Name23231581
N-Terminal modificationCathelicidin HHC-10
C-Terminal ModificationKRWWKWIRW
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature9
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium bovis
In Vitro/ In vivoMycobacterium tuberculosis complex bacteria, Mycobacterium bovis bacille calmette guerin (BCG) (Mycobacterium bovis BCG Pasteur 1173P2)
Cell Line88 % decrease in CFU at 100 μg/ ml
Inhibition ConcentrationBoth
Sequence2013
CytotoxicityNone
In vivo ModelNA
Lethal DoseNA
Immune Responce8–9 weeks old C57BL/6 mice
Mechanism of ActionCFUs in mouse lungs were reduced 95.8% at 2.5 mg k
TargetSignificant reduction of IFN-γ transcription
Combination TherapyCell envelope disruption
Other activitiesCell envelope
PMIDNone
Year of PublicationAntibacterial (such as Pseudomonas aeruginosa, Escherichia coli, Klebsiella pneumonia, and S. aureus etc
Tertiary Structure
(Technique)
Not Predicted),