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IDPMIDYEARSequenceNameLengthLinear/CyclicChiralityChem-MODC-ter MODN-ter MODNatureOriginCell LineCancer TypeAssayActivityTesting TimeTissue AffectedPatents
5272
None2015
CHYRVKPKIKRFEKYKGRMW
LPSBD-220LinearLNoneFreeFreeAnticancerSyntheticHep3BLiver CancerCell Proliferation assay~40% cell survival at 60 µg/ml24-hLiverNone
5271
None2015
CHYRVKPKIKRFEKYKGRMW
LPSBD-220LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerCell Proliferation assay~20% cell survival at 60 µg/ml24-hLungNone
5270
None2015
CQYSVNPKIKRFELYFKGRMW
LPSBD-021LinearLNoneFreeFreeAnticancerSyntheticHep3BLiver CancerCell Proliferation assay~40% cell survival at 60 µg/ml24-hLiverNone
5268
258543662015
FIGAIARLL
BmKn-249LinearLNoneFreeFreeAntimicrobialDerivative of Bmkn-2HSC-4Tongue Squamous Cell CarcinomaMTT assayIC50 between 29-97 µg/ml24-hTongueNone
5269
None2015
CQYSVNPKIKRFELYFKGRMW
LPSBD-021LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerCell Proliferation assay~20% cell survival at 60 µg/ml24-hLungNone
5266
258543662015
FIGAIARLLSKI
Bmkn-2112LinearLNoneFreeFreeAntimicrobialDerivative of Bmkn-2HSC-4Tongue Squamous Cell CarcinomaMTT assayIC50 between 29-97 µg/ml24-hTongueNone
5267
258543662015
FIGAIARLLS
BmKn-2310LinearLNoneFreeFreeAntimicrobialDerivative of Bmkn-2HSC-4Tongue Squamous Cell CarcinomaMTT assayIC50 between 29-97 µg/ml24-hTongueNone
5264
258543662015
FIGAIARLLSKIF
BmKn213LinearLNoneFreeFreeAntimicrobialMesobuthus martensii KarschHSC-4Tongue Squamous Cell CarcinomaMTT assayIC50 = 29 µg/mL24-hTongueNone
5265
258543662015
FIGAIARLLSK
Bmkn-2211LinearLNoneFreeFreeAntimicrobialDerivative of Bmkn-2HSC-4Tongue Squamous Cell CarcinomaMTT assayIC50 between 29-97 µg/ml24-hTongueNone
5263
258022812015
AQQICKAPSQTFPGLCFMDSSCRKYCIKEKFTGGHCSKLQRKCLCTKPC
TPP349LinearLNoneFreeFreeAntifungalpistils from tomato flowersU-937Leukemia CancerLDH leakage assay35% cytotoxicity at 10 μMNot AvailableBloodNone
5258
265278622015
RRRQRRKKRGGGGlgaswhrpdkcclgyqkrrlpGGGLRRMADDLNAQY
TAT-DV1-BH349LinearMixNoneFreeFreeAnticancerSynthetic polypeptideMDA-MB-231Breast cancerCCK-8 assaySurvival rate = 28.67±8.22% at 80 µM72-hBreastNone
5259
265278622015
RRRQRRKKRGGGGlgaswhrpdkcclgyqkrrlpGGGLRRMADDLNAQY
TAT-DV1-BH349LinearMixNoneFreeFreeAnticancerSynthetic polypeptideMCF-7Breast cancerCCK-8 assaySurvival rate = 36.97±4.22% at 80 µM72-hBreastNone
5262
258022812015
AQQICKAPSQTFPGLCFMDSSCRKYCIKEKFTGGHCSKLQRKCLCTKPC
TPP349LinearLNoneFreeFreeAntifungalpistils from tomato flowersU-937Leukemia CancerPI uptake assay69.6% cell death at 10 μMNot AvailableBloodNone
5257
254622642015
VKRFKKFFRKLKKEV
B1-Glu15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 36.6 µM24-hBloodNone
5256
254622642015
VKRFKKFFRKLKKEV
B1-Glu15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 38.9 µM24-hBreastNone
5254
254622642015
VKRFKKFFRKLKKDV
B1-Asp15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 19.9 µM24-hBreastNone
5255
254622642015
VKRFKKFFRKLKKDV
B1-Asp15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 44.7 µM24-hBloodNone
5253
254622642015
VKRFKKFFRKLKKHV
B1-His15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 10.5 µM24-hBloodNone
5252
254622642015
VKRFKKFFRKLKKHV
B1-His15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 5.0µM24-hBreastNone
5250
254622642015
VKRFKKFFRKLKKRV
B1-Arg15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 5.5 µM24-hBreastNone
5251
254622642015
VKRFKKFFRKLKKRV
B1-Arg15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 8.7 µM24-hBloodNone
5249
254622642015
VKRFKKFFRKLKKKV
B1-Lys15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562/ADMLeukemia cancerMTT assayIC50 = 5.5 µM24-hBloodNone
5247
254622642015
VKRFKKFFRKLKKKV
B1-Lys15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 5.5 µM24-hBloodNone
5248
254622642015
VKRFKKFFRKLKKKV
B1-Lys15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7/ADMBreast CancerMTT assayIC50 = 8.6 µM24-hBreastNone
5246
254622642015
VKRFKKFFRKLKKKV
B1-Lys15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 8.3 µM24-hBreastNone
5245
254622642015
VKRFKKFFRKLKKTV
B1-Thr15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 17.0 µM24-hBloodNone
5243
254622642015
VKRFKKFFRKLKKQV
B1-Gln15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 16.2 µM24-hBloodNone
5244
254622642015
VKRFKKFFRKLKKTV
B1-Thr15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 19.1 µM24-hBreastNone
5242
254622642015
VKRFKKFFRKLKKQV
B1-Gln15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 14.5 µM24-hBreastNone
5241
254622642015
VKRFKKFFRKLKKGV
B1-Gly15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 14.8 µM24-hBloodNone
5239
254622642015
VKRFKKFFRKLKKFV
B1-Phe15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 3.7 µM24-hBloodNone
5240
254622642015
VKRFKKFFRKLKKGV
B1-Gly15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 15.8 µM24-hBreastNone
5238
254622642015
VKRFKKFFRKLKKFV
B1-Phe15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 1.3 µM24-hBreastNone
5237
254622642015
VKRFKKFFRKLKKLV
B1-Leu15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562/ADMLeukemia cancerMTT assayIC50 = 3.3 µM24-hBloodNone
5236
254622642015
VKRFKKFFRKLKKLV
B1-Leu15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7/ADMBreast CancerMTT assayIC50 = 4.4 µM24-hBreastNone
5235
254622642015
VKRFKKFFRKLKKLV
B1-Leu15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 1.1 µM24-hBloodNone
5233
254622642015
VKRFKKFFRKLKKVV
B1-Val15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 5.0 µM24-hBloodNone
5234
254622642015
VKRFKKFFRKLKKLV
B1-Leu15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 3.6 µM24-hBreastNone
5232
254622642015
VKRFKKFFRKLKKVV
B1-Val15LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 4.9 µM24-hBreastNone
5231
254622642015
VKRFKKFFRKLKKAV
B1-Ala1415LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1K-562Leukemia cancerMTT assayIC50 = 8.6 µM24-hBloodNone
5230
254622642015
VKRFKKFFRKLKKAV
B1-Ala1415LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of B1MCF-7Breast CancerMTT assayIC50 = 8.9 µM24-hBreastNone
5228
254622642015
VKRFKKFFRKLKKSV
B115LinearLNoneAmidationFreeAntimicrobial and AnticancerCathelicidin-BF15MCF-7/ADMBreast CancerMTT assayIC50 = 24.1 µM24-hBreastNone
5229
254622642015
VKRFKKFFRKLKKSV
B115LinearLNoneAmidationFreeAntimicrobial and AnticancerCathelicidin-BF15K-562/ADMLeukemia cancerMTT assayIC50 = 31.6 µM24-hBloodNone
5227
254622642015
VKRFKKFFRKLKKSV
B115LinearLNoneAmidationFreeAntimicrobial and AnticancerCathelicidin-BF15K-562Leukemia cancerMTT assayIC50 = 26.9 µM24-hBloodNone
5224
274860682015
PcatPhexPhexPcat
Lipotetrapeptide-C16-PCatPCatPCatPCat-NH24LinearLPcat = L-4R-aminoproline ; Phex = L-4R-hexyloxyprolineAmidationPalmitic acidAnticancerSyntheticDU-145Prostate CancerMTS assayCC50 = 16.5 µM73-76hProstateNone
5225
274860682015
PcatPhexPhexPcat
Lipotetrapeptide-C16-PCatPCatPCatPCat-NH24LinearLPcat = L-4R-aminoproline ; Phex = L-4R-hexyloxyprolineAmidationPalmitic acidAnticancerSyntheticMiaPaCa.2Pancreatic CancerMTS assayCC50 = 23 µM73-76hPancreasNone
5226
254622642015
VKRFKKFFRKLKKSV
B115LinearLNoneAmidationFreeAntimicrobial and AnticancerCathelicidin-BF15MCF-7Breast CancerMTT assayIC50 = 21.9 µM24-hBreastNone
5221
274860682015
KKKK
C16-Lipotetrapeptide4LinearLNoneAmidationPalmitic acidAnticancerSyntheticDU-145Prostate CancerMTS assayCC50 = 18 µM73-76hProstateNone
5222
274860682015
PcatPhexPhexPcat
Lipotetrapeptide-C16-PCatPCatPCatPCat-NH24LinearLPcat = L-4R-aminoproline ; Phex = L-4R-hexyloxyprolineAmidationPalmitic acidAnticancerSyntheticMDA-MB-231Breast CancerMTS assayCC50 = 12.5 µM73-76hBreastNone
5223
274860682015
PcatPhexPhexPcat
Lipotetrapeptide-C16-PCatPCatPCatPCat-NH24LinearLPcat = L-4R-aminoproline ; Phex = L-4R-hexyloxyprolineAmidationPalmitic acidAnticancerSyntheticJIMT-1Breast CancerMTS assayCC50 = 17 µM73-76hBreastNone
5218
274860682015
KKK
C16-Liptotripeptide3LinearLNoneAmidationPalmitic acidAnticancerSyntheticMiaPaCa.2Pancreatic CancerMTS assayCC50 =16 µM73-76hPancreasNone
5219
274860682015
KKKK
C16-Lipotetrapeptide4LinearLNoneAmidationPalmitic acidAnticancerSyntheticMDA-MB-231Breast CancerMTS assayCC50 = 30 µM73-76hBreastNone
5220
274860682015
KKKK
C16-Lipotetrapeptide4LinearLNoneAmidationPalmitic acidAnticancerSyntheticJIMT-1Breast CancerMTS assayCC50 = 30 µM73-76hBreastNone
5215
274860682015
KKK
C14-Liptotripeptide3LinearLNoneAmidationMyristic acidAnticancerSyntheticDU-145Prostate CancerMTS assayCC50 =10 µM73-76hProstateNone
5216
274860682015
KKK
C16-Liptotripeptide3LinearLNoneAmidationPalmitic acidAnticancerSyntheticJIMT-1Breast CancerMTS assayCC50 = 10 µM73-76hBreastNone
5217
274860682015
KKK
C16-Liptotripeptide3LinearLNoneAmidationPalmitic acidAnticancerSyntheticDU-145Prostate CancerMTS assayCC50 = 9 µM73-76hProstateNone
5214
254475432015
ACYCRIPACIAGERRYGTCIYQGRLWAFCC
Human neutrophil peptide-1 (HNP-1)30Cyclic(C2-C30, C4-C19,C9-C29)LNoneFreeFreeAntimicrobialHomo sapiensPC-3Prostate CancerCytotoxicity assay (LIVE/DEAD® Viability/Cytotoxicity Assay Kit (L-3224))IC50 = 2.2 ± 0.3 μM4hProstateNone
5212
256337172015
Str given in figure
KEMTUB104LinearLNonefluorine atom in para-position on the phenyl ringN-tubuvaline fragment replaced with stable benzyl groupAnti-cancerSynthetic analogue of natural tubulysinsMDA-MB-453Breast CancerMTT assayIC50 = 16.3 ± 5.6 pM72-hBreastNone
5213
256337172015
Str given in figure
KEMTUB104LinearLNonefluorine atom in para-position on the phenyl ringN-tubuvaline fragment replaced with stable benzyl groupAnti-cancerSynthetic analogue of natural tubulysinsSK-BR-3Breast CancerMTT assayIC50 = 12.2 ± 6 pM72-hBreastNone
5210
256337172015
Str given in figure
KEMTUB104LinearLNonefluorine atom in para-position on the phenyl ringN-tubuvaline fragment replaced with stable benzyl groupAnti-cancerSynthetic analogue of natural tubulysinsMCF-7/DDBreast CancerMTT assayIC50 = 68.6 ± 30.1 pM72-hBreastNone
5211
256337172015
Str given in figure
KEMTUB104LinearLNonefluorine atom in para-position on the phenyl ringN-tubuvaline fragment replaced with stable benzyl groupAnti-cancerSynthetic analogue of natural tubulysinsMDA-MB-231Breast CancerMTT assayIC50 = 68 ± 18 pM72-hBreastNone
5209
256337172015
Str given in figure
KEMTUB104LinearLNonefluorine atom in para-position on the phenyl ringN-tubuvaline fragment replaced with stable benzyl groupAnti-cancerSynthetic analogue of natural tubulysinsMCF-7Breast CancerMTT assayIC50 = 30.1 ± 13.2 pM72-hBreastUS 8,580,820; US (US 2011/200581).
5204
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHL-60Leukemia CancerLDH leakage assayIC50 = 23.01 μg/mL24-hBloodNone
5203
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomDU-145Prostrate CancerLDH leakage assayIC50 = 15.91 μg/mL24-hProstateNone
5202
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHepG-2Liver CancerLDH leakage assayIC50 = 28.99 μg/mL24-hLiverNone
5201
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomMCF-7Breast CancerLDH leakage assayIC50 = 23.9 μg/mL24-hBreastNone
5200
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHL-60Leukemia CancerMTT assayIC50 < 20 μg/mL24-hBloodNone
5199
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomDU-145Prostrate CancerMTT assayIC50 ~ 15 μg/mL24-hProstateNone
5198
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHepG-2Liver CancerMTT assayIC50 ~ 20 μg/mL24-hLiverNone
5197
264829322015
LKCKKLVPLFSKTCPAGKNLCYKMFMVAAPHVPVKRGCIDVCPKSSLLVKYVCCNTDKCN
Cytotoxin-II60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomMCF-7Breast CancerMTT assayIC50 ~ 10 μg/mL24-hBreastNone
5192
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHL-60Leukemia CancerLDH leakage assayIC50 = 38.3 μg/mL24-hBloodNone
5191
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomDU-145Prostrate CancerLDH leakage assayIC50 = 20.99 μg/mL24-hProstateNone
5190
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHepG-2Liver CancerLDH leakage assayIC50 = 35.84 μg/mL24-hLiverNone
5189
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomMCF-7Breast CancerLDH leakage assayIC50 = 45.71 μg/mL24-hBreastNone
5188
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHL-60Leukemia CancerMTT assayIC50 < 40 μg/mL24-hBloodNone
5187
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomDU-145Prostrate CancerMTT assayIC50 ~ 20 μg/mL24-hProstateNone
5186
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomHepG-2Liver CancerMTT assayIC50 ~ 40 μg/mL24-hLiverNone
5185
264829322015
LKCNKLVPIAYKTCPEGKNLCYKMFMMSDLTIPVKRGCIDVCPKNSLLVKYVCCNTDRCN
Cytotoxin-I60CyclicLNoneFreeFreeAnticancerCaspian cobra (Naja oxiana) venomMCF-7Breast CancerMTT assayIC50 < 20 μg/mL24-hBreastNone
5183
258210842015
CVLIGQRCDNDRGPRCCSGQGNCVPLPFLGGVCAV
Ep-AMP135CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerEchinopsis pachanoiU-937/GTBLymphoma cancerFluorometric microculture cytotoxicity assayIC50 > 100 µMNot AvailableBloodNone
5182
263227452015
GLPTCGETCFKGKCYTPGCSCSYPICKKD
Cyclotide mela-629CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusHeLaCervical CancerResazurin dye assayCC50 = 11.42 ±1.00 µMNot AvailableCervixNone
5181
263227452015
GLPTCGETCFKGKCYTPGCSCSYPICKKD
Cyclotide mela-629CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusMM96LSkin CancerResazurin dye assayCC50 = 1.58 ±0.48 µMNot AvailableSkinNone
5180
263994952015
GIPCGESCVFIPCLTSAIGCSCKSKVCYRN
Mra3030CyclicLNoneCyclizedCyclizedAntimicrobial and AnticancerViola tricolor, Melicytus ramiflorus, Viola philippicaBGC-823Gastric CancerResazurin dye assayIC50 = 1.75 ±0.05 µMNot AvailableStomachNone
5179
263994952015
GIPCGESCVFIPCLTSAIGCSCKSKVCYRN
Mra3030CyclicLNoneCyclizedCyclizedAntimicrobial and AnticancerViola tricolor, Melicytus ramiflorus, Viola philippicaHeLaCervical CancerResazurin dye assayIC50 = 15.5 ±0.06 µMNot AvailableCervixNone
5178
263994952015
GIPCGESCVFIPCLTSAIGCSCKSKVCYRN
Mra3030CyclicLNoneCyclizedCyclizedAntimicrobial and AnticancerViola tricolor, Melicytus ramiflorus, Viola philippicaMM96LSkin CancerResazurin dye assayIC50 = 4.91 ±0.04 µMNot AvailableSkinNone
5177
263227452015
GKPICGETCFKGKCYTPGCTCSYPICKKD
Mela329CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusHeLaCervical CancerResazurin dye assayCC50 = 18.73 ±1.82 µMNot AvailableCervixNone
5175
259743072015
NYNQPNS
IturinA7CyclicLNoneCyclized; C16 Fatty acid moietyCyclizedLipopeptideBacillus megateriumMDA-MB-468Breast CancerMTT assayIC50 = 13.30 ± 0.97 μM48-hBreastNone
5176
263227452015
GKPICGETCFKGKCYTPGCTCSYPICKKD
Mela329CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusMM96LSkin CancerResazurin dye assayCC50 = 2.04 ±0.26 µMNot AvailableSkinNone
5172
259743072015
NYNQPNS
IturinA7CyclicLNoneCyclized; C16 Fatty acid moietyCyclizedLipopeptideBacillus megateriumMDA-MB-231Breast CancerMTT assayIC50 = 7.98 ± 0.19 μM48-hBreastNone
5173
259743072015
NYNQPNS
IturinA7CyclicLNoneCyclized; C16 Fatty acid moietyCyclizedLipopeptideBacillus megateriumMCF-7Breast CancerMTT assayIC50 = 12.16 ± 0.24 μM48-hBreastNone
5174
259743072015
NYNQPNS
IturinA7CyclicLNoneCyclized; C16 Fatty acid moietyCyclizedLipopeptideBacillus megateriumT-47DBreast CancerMTT assayIC50 = 26.29 ± 0.78 μM48-hBreastNone
5169
267036312015
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntimicrobialPardachirus marmoratusOSCC-SCC-4Oral cancerMTT assayCell Viability <20% at 20μg/mL24-hNot AvailableNone
5167
256260772015
FLFKLIPKVIKGLVKAIRK
AaeAP2a19LinearLNoneAmidationFreeAntimicrobialSynthetic analog of AaeAP2MCF-7Breast CancerMTT assayGraph Figure 424-hBreastNone
5168
256260772015
FLFKLIPKVIKGLVKAIRK
AaeAP2a19LinearLNoneAmidationFreeAntimicrobialSynthetic analog of AaeAP2PC-3Prostate CancerMTT assayGraph Figure 424-hProstateNone
5166
256260772015
FLFKLIPKVIKGLVKAIRK
AaeAP2a19LinearLNoneAmidationFreeAntimicrobialSynthetic analog of AaeAP2MDA-MB-435SSkin CancerMTT assayGraph Figure 424-hSkinNone
5164
256260772015
FLFKLIPKAIKGLVKAIRK
AaeAP1a19LinearLNoneAmidationFreeAntimicrobialSynthetic analog of AaeAP1MCF-7Breast CancerMTT assayGraph Figure 424-hBreastNone
5165
256260772015
FLFKLIPKAIKGLVKAIRK
AaeAP1a19LinearLNoneAmidationFreeAntimicrobialSynthetic analog of AaeAP1PC-3Prostate CancerMTT assayGraph Figure 424-hProstateNone
5163
256260772015
FLFKLIPKAIKGLVKAIRK
AaeAP1a19LinearLNoneAmidationFreeAntimicrobialSynthetic analog of AaeAP1MDA-MB-435SSkin CancerMTT assayGraph Figure 424-hSkinNone
5162
267519702015
GLPLCGETCVGGTCNTPGCSCGWPVCVRN
Vigno 529Cyclic(C5-C19,C9-C21,C14-C21)LNoneFreeFreeAnticancerViola ignobilisHeLaCervical CancerMTT assay24% cell viability at 7.5 μM24-hCervixNone
5158
260643102015
GAFLKCGESCVYLPCLTTVVGCSCQNSVCYRD
DC132CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaDU-145Liver CancerCCK-8 assayIC50 = 3.32 μM72-hLiverNone
5157
260643102015
GAFLKCGESCVYLPCLTTVVGCSCQNSVCYRD
DC132CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaPC-3Prostate CancerCCK-8 assayIC50 = 2.24 μM72-hProstateNone
5156
260643102015
GAFLKCGESCVYLPCLTTVVGCSCQNSVCYRD
DC132CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaLNCaPProstate CancerCCK-8 assayIC50 = 5.03 μM72-hProstateNone
5155
260643102015
GAVPCGETCVYLPCITPDIGCSCQNKVCYRD
DC231CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaDU-145Liver CancerCCK-8 assayIC50 = 3.11 μM72-hLiverNone
5154
260643102015
GAVPCGETCVYLPCITPDIGCSCQNKVCYRD
DC231CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaPC-3Prostate CancerCCK-8 assayIC50 = 2.65 μM72-hProstateNone
5153
260643102015
GAVPCGETCVYLPCITPDIGCSCQNKVCYRD
DC231CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaLNCaPProstate CancerCCK-8 assayIC50 = 4.31 μM72-hProstateNone
5152
260643102015
GTSCGETCVLLPCLSSVLGCTCQNKRCYKD
DC330CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaDU-145Liver CancerCCK-8 assayIC50 = 0.55 μM72-hLiverNone
5151
260643102015
GTSCGETCVLLPCLSSVLGCTCQNKRCYKD
DC330CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaPC-3Prostate CancerCCK-8 assayIC50 = 0.76 μM72-hProstateNone
5150
260643102015
GTSCGETCVLLPCLSSVLGCTCQNKRCYKD
DC330CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaLNCaPProstate CancerCCK-8 assayIC50 = 0.21 μM72-hProstateNone
5149
264027312015
GFGSKPLDSFGLNFF
Chaxapeptin15MixLNoneFreeCyclized to form macrolactam ringAntimicrobial and AnticancerStreptomyces leeuwenhoekii Strain C58A-549Lung CancerCyQUANT Direct assayCell invasion < 50% at 50 μM36-hLungNone
5148
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-668Gastric cancerLDH release assayCytotoxicity ~ 60-80% at 50 μM24-hStomachNone
5147
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-638Gastric cancerLDH release assayCytotoxicity ~ 60-80% at 50 μM24-hStomachNone
5146
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-601Gastric cancerLDH release assayCytotoxicity ~ 60-80% at 50 μM24-hStomachNone
5145
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-484Gastric cancerLDH release assayCytotoxicity ~ 60-80% at 50 μM24-hStomachNone
5144
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-668Gastric cancerMTS assayIC50 ~ 20-50 μM24-hStomachNone
5143
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-638Gastric cancerMTS assayIC50 ~ 20-50 μM24-hStomachNone
5142
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-601Gastric cancerMTS assayIC50 ~ 20-50 μM24-hStomachNone
5141
250474442015
LLCIALRKKLLCIALRKK
CopA318LinearLNoneAmidationFreeAntimicrobialanalogue derived from coprisinSNU-484Gastric cancerMTS assayIC50 ~ 20-50 μM24-hStomachNone
5139
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 1.8 ± 0.02 μM24-hCervixNone
5138
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticB-16Skin CancerMTT assayIC50 = 3.9 ± 0.02 μM24-hSkinNone
5137
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 5.8 ± 0.36 μM24-hLiverNone
5136
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticSGC-7901Gastric cancerMTT assayIC50 = 4.8 ± 0.08 μM24-hStomachNone
5135
264058062015
FKKLKKLFSKLWNWK
HPRP-A115LinearLNoneAmidationAcetylationAnticancerHelicobacter pyloriHeLaCervical CancerMTT assayIC50 = 3.5 ± 0.03 μM24-hCervixNone
5134
264058062015
FKKLKKLFSKLWNWK
HPRP-A115LinearLNoneAmidationAcetylationAnticancerHelicobacter pyloriHepG-2Liver CancerMTT assayIC50 = 7.7 ± 0.23 μM24-hLiverNone
5133
264058062015
FKKLKKLFSKLWNWK
HPRP-A115LinearLNoneAmidationAcetylationAnticancerHelicobacter pyloriSGC-7901Gastric cancerMTT assayIC50 = 5.2 ± 0.14 μM24-hStomachNone
5132
264058062015
FKKLKKLFSKLWNWK
HPRP-A115LinearLNoneAmidationAcetylationAnticancerHelicobacter pyloriB-16Skin CancerMTT assayIC50 = 6.1 ± 0.02 μM24-hSkinNone
5131
262395372015
WWRRWWRRWRRWWRRWWR
RW-AH18LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerMTS assayLC50 = 4.6 ± 0.2 μM24-hSkinNone
5130
262395372015
WWRRWWRRWRRWWRRWWR
RW-AH18LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerMTS assayLC50 = 8.4 ± 0.5 μM24-hSkinNone
5129
262395372015
WWRRWWRRWRRWWRRWWR
RW-AH18LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerPI uptake assayLC50 = 4.5 ± 0.02 μM8-hSkinNone
5128
262395372015
FWQRRIRRWRRFWQRRIRRWRR
DIM-LF11-31822LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerMTS assayLC50 = 9.4 ± 0.5 μM24-hSkinNone
5127
262395372015
FWQRRIRRWRRFWQRRIRRWRR
DIM-LF11-31822LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerMTS assayLC50 = 9.3 ± 0.8 μM24-hSkinNone
5126
262395372015
FWQRRIRRWRRFWQRRIRRWRR
DIM-LF11-31822LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerPI uptake assayLC50 = 3.8 ± 0.5 μM8-hSkinNone
5125
262395372015
PFWRRRIRIRRRRIRIRRRWFP
R-DIM-LF11-33722LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerMTS assayLC50 = 5.0 ± 0.4 μM24-hSkinNone
5124
262395372015
PFWRRRIRIRRRRIRIRRRWFP
R-DIM-LF11-33722LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerMTS assayLC50 = 12.3 ± 1.3 μM24-hSkinNone
5123
262395372015
PFWRRRIRIRRRRIRIRRRWFP
R-DIM-LF11-33722LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerPI uptake assayLC50 = 3.5 ± 0.4 μM8-hSkinNone
5122
262395372015
PFWRIRIRRPRRIRIRWFP
R-DIM-P-LF11-32219LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerMTS assayLC50 = 10.4 ± 0.7 μM24-hSkinEP_2943215_B1
5121
262395372015
PFWRIRIRRPRRIRIRWFP
R-DIM-P-LF11-32219LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerMTS assayLC50 = 23.3 ± 1.7 μM24-hSkinEP_2943215_B1
5120
262395372015
PFWRIRIRRPRRIRIRWFP
R-DIM-P-LF11-32219LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerPI uptake assayLC50 = 5.9 ± 0.3 μM8-hSkinEP_2943215_B1
5119
262395372015
PFWRIRIRRPRRIRIRWFP
R-DIM-P-LF11-32219LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerPI uptake assayLC50 = 9.5 ± 0.3 μM8-hSkinEP_2943215_B1
5115
259702922015
KKKKKK-Nal-Nal-KKWRKWLAKK
K6-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticSASOral CancerMTT assayGraph Figure 224-hTongueNone
5114
259702922015
KKKKKK-Nal-Nal-KKWRKWLAKK
K6-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticOECM-1Oral CancerMTT assayGraph Figure 224-hNot AvailableNone
5113
259702922015
KKKKKK-Nal-Nal-KKWRKWLAKK
K6-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticC9Oral CancerMTT assayGraph Figure 224-hNot AvailableNone
5112
259702922015
KKKKKK-Nal-Nal-KKWRKWLAKK
K6-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayGraph Figure 224-hLungNone
5111
259702922015
KKKKKK-Nal-Nal-KKWRKWLAKK
K6-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticPC-9GLung CancerMTT assayGraph Figure 224-hLungNone
5110
259702922015
KKKKKK-Nal-Nal-KKWRKWLAKK
K6-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticPC-9Lung CancerMTT assayGraph Figure 224-hLungNone
5109
259702922015
KKKKRR-Nal-Nal-KKWRKWLAKK
K4R2-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticSASOral CancerMTT assayGraph Figure 224-hTongueNone
5108
259702922015
KKKKRR-Nal-Nal-KKWRKWLAKK
K4R2-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticOECM-1Oral CancerMTT assayGraph Figure 224-hNot AvailableNone
5107
259702922015
KKKKRR-Nal-Nal-KKWRKWLAKK
K4R2-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticC9Oral CancerMTT assayGraph Figure 224-hNot AvailableNone
5106
259702922015
KKKKRR-Nal-Nal-KKWRKWLAKK
K4R2-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayGraph Figure 224-hLungNone
5105
259702922015
KKKKRR-Nal-Nal-KKWRKWLAKK
K4R2-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticPC-9GLung CancerMTT assayGraph Figure 224-hLungNone
5104
259702922015
KKKKRR-Nal-Nal-KKWRKWLAKK
K4R2-Nal2-S118LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticPC-9Lung CancerMTT assayGraph Figure 224-hLungNone
5103
259702922015
Nal-Nal-KKWRKWLAKK
Nal2-S112LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticSASOral CancerMTT assayGraph Figure 224-hTongueUS_10093699_B2
5102
259702922015
Nal-Nal-KKWRKWLAKK
Nal2-S112LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticOECM-1Oral CancerMTT assayGraph Figure 224-hNot AvailableUS_10093699_B2
5101
259702922015
Nal-Nal-KKWRKWLAKK
Nal2-S112LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticC9Oral CancerMTT assayGraph Figure 224-hNot AvailableUS_10093699_B2
5100
259702922015
Nal-Nal-KKWRKWLAKK
Nal2-S112LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayGraph Figure 224-hLungUS_10093699_B2
5099
259702922015
Nal-Nal-KKWRKWLAKK
Nal2-S112LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticPC-9GLung CancerMTT assayGraph Figure 224-hLungUS_10093699_B2
5098
259702922015
Nal-Nal-KKWRKWLAKK
Nal2-S112LinearLNal = beta-naphthylalanineAmidationAcetylationAntimicrobialSyntheticPC-9Lung CancerMTT assayGraph Figure 224-hLungUS_10093699_B2
5093
253122532014
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSyntheticU-937Leukemia CancerFITC-Annexin V/PI double staining and flow cytometry assay>20% apoptosis rate at 80 μM24-hBloodNone
5092
253122532014
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSyntheticHL-60Leukemia CancerFITC-Annexin V/PI double staining and flow cytometry assay>20% apoptosis rate at 80 μM24-hBloodNone
5091
253122532014
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSyntheticNB-4Leukemia CancerFITC-Annexin V/PI double staining and flow cytometry assay60% apoptosis rate at 80 μM24-hBloodNone
5090
246924462014
RECKTESNTFPGICITKPPCRKACISEKFTDGHCSKILRRCLCTKPC
NaD147Cyclic(C3-C47,C14-34,C20-C41,C24-C43)LNoneNoneNoneHost DefenseNicotiana alataB16-F10Skin CancerMTT assayIC50 = 1.5 ± 0.6 μM48-hSkinNone
5089
246924462014
RECKTESNTFPGICITKPPCRKACISEKFTDGHCSKILRRCLCTKPC
NaD147Cyclic(C3-C47,C14-34,C20-C41,C24-C43)LNoneNoneNoneHost DefenseNicotiana alataHeLaCervical CancerMTT assayIC50 = 1.0 ± 0.1 μM48-hCervixNone
5088
246924462014
RECKTESNTFPGICITKPPCRKACISEKFTDGHCSKILRRCLCTKPC
NaD147Cyclic(C3-C47,C14-34,C20-C41,C24-C43)LNoneNoneNoneHost DefenseNicotiana alataMM170Skin CancerMTT assayIC50 = 2.4 ± 0.8 μM48-hSkinNone
5087
246924462014
RECKTESNTFPGICITKPPCRKACISEKFTDGHCSKILRRCLCTKPC
NaD147Cyclic(C3-C47,C14-34,C20-C41,C24-C43)LNoneNoneNoneHost DefenseNicotiana alataMCF-7Breast CancerMTT assayIC50 = 2.0 ± 1.3 μM48-hBreastNone
5086
246924462014
RECKTESNTFPGICITKPPCRKACISEKFTDGHCSKILRRCLCTKPC
NaD147Cyclic(C3-C47,C14-34,C20-C41,C24-C43)LNoneNoneNoneHost DefenseNicotiana alataHCT-116Colon CancerMTT assayIC50 = 4.9 ± 3.1 μM48-hColonNone
5085
245033752014
RLGDGCTR
Cyclosaplin8CyclicLNoneCyclizedCyclizedAnticancerSantalum album LMDA-MB-231Breast CancerMTT assayIC50 = 2.06 μg/mL24-hBreast638/KOL/2013
5084
246921992014
Wa(D-allo-i)VlL
Baceridin6CyclicMixNoneCyclizedCyclizedAntimicrobial and Anticancerculture medium of a plant-associated Bacillus strainHeLaCervical CancerMTT assayIC50 between (1–2 µg/mL)72-hCervixNone
5083
246921992014
Wa(D-allo-i)VlL
Baceridin6CyclicMixNoneCyclizedCyclizedAntimicrobial and Anticancerculture medium of a plant-associated Bacillus strainRKOColon CancerMTT assayIC50 between (1–2 µg/mL)72-hColonNone
5082
246921992014
Wa(D-allo-i)VlL
Baceridin6CyclicMixNoneCyclizedCyclizedAntimicrobial and Anticancerculture medium of a plant-associated Bacillus strainHCT-116 -/- p53Colon CancerMTT assayIC50 between (1–2 µg/mL)72-hColonNone
5081
247047572014
GLVGTLLGHIGKAILG
Frenatin 2.1S16LinearLNonealpha-amidationFreeAntimicrobialSphaenorhynchus lacteusA-549Lung CancerTrypan blue assayLC50 = 80 ± 6 μM24-hLungNone
5080
247047572014
GLVGTLLGHIGKAILS
Frenatin 2.2S16LinearLNonealpha-amidationFreeAntimicrobialSphaenorhynchus lacteusA-549Lung CancerTrypan blue assayLC50 = 75 ± 5 μM24-hLungNone
5079
244925202014
ELLVDLL
Gageostatin C7LinearLNoneFree(E)-7,9-dimethylundec-2-enoic acidAntimicrobialBacillus subtilisACHNRenal CancerSulforhodamine B assayGI50 = 12.3 µg/mL48-hKidneyNone
5077
244925202014
ELLVDLL
Gageostatin C7LinearLNoneFree(E)-7,9-dimethylundec-2-enoic acidAntimicrobialBacillus subtilisNCI-H23Lung CancerSulforhodamine B assayGI50 = 10.9 µg/mL48-hLungNone
5078
244925202014
ELLVDLL
Gageostatin C7LinearLNoneFree(E)-7,9-dimethylundec-2-enoic acidAntimicrobialBacillus subtilisNUGC-3Stomach CancerSulforhodamine B assayGI50 = 10.5 µg/mL48-hStomachNone
5075
244925202014
ELLVDLL
Gageostatin C7LinearLNoneFree(E)-7,9-dimethylundec-2-enoic acidAntimicrobialBacillus subtilisHCT-15Colon CancerSulforhodamine B assayGI50 = 23.2 µg/mL48-hColonNone
5076
244925202014
ELLVDLL
Gageostatin C7LinearLNoneFree(E)-7,9-dimethylundec-2-enoic acidAntimicrobialBacillus subtilisPC-3Prostate CancerSulforhodamine B assayGI50 = 11.7 µg/mL48-hProstateNone
5073
244925202014
ELLVDLL
Gageostatin B7LinearLNoneFree3-beta-hydroxy-9,11-dimethyltridecanoic acidAntimicrobialBacillus subtilisACHNRenal CancerSulforhodamine B assayGI50 = 18.4 µg/mL48-hKidneyNone
5074
244925202014
ELLVDLL
Gageostatin C7LinearLNoneFree(E)-7,9-dimethylundec-2-enoic acidAntimicrobialBacillus subtilisMDA-MB-231Breast CancerSulforhodamine B assayGI50 = 11.2 µg/mL48-hBreastNone
5072
244925202014
ELLVDLL
Gageostatin B7LinearLNoneFree3-beta-hydroxy-9,11-dimethyltridecanoic acidAntimicrobialBacillus subtilisNUGC-3Stomach CancerSulforhodamine B assayGI50 = 13.9 µg/mL48-hStomachNone
5070
244925202014
ELLVDLL
Gageostatin B7LinearLNoneFree3-beta-hydroxy-9,11-dimethyltridecanoic acidAntimicrobialBacillus subtilisPC-3Prostate CancerSulforhodamine B assayGI50 = 19.4 µg/mL48-hProstateNone
5071
244925202014
ELLVDLL
Gageostatin B7LinearLNoneFree3-beta-hydroxy-9,11-dimethyltridecanoic acidAntimicrobialBacillus subtilisNCI-H23Lung CancerSulforhodamine B assayGI50 = 11.7 µg/mL48-hLungNone
5068
244925202014
ELLVDLL
Gageostatin B7LinearLNoneFree3-beta-hydroxy-9,11-dimethyltridecanoic acidAntimicrobialBacillus subtilisMDA-MB-231Breast CancerSulforhodamine B assayGI50 = 16.1 µg/mL48-hBreastNone
5069
244925202014
ELLVDLL
Gageostatin B7LinearLNoneFree3-beta-hydroxy-9,11-dimethyltridecanoic acidAntimicrobialBacillus subtilisHCT-15Colon CancerSulforhodamine B assayGI50 = 18.3 µg/mL48-hColonNone
5067
244925202014
ELLVDLL
Gageostatin A7LinearLNoneFree3-beta-hydroxy-11-methyltridecanoic acidAntimicrobialBacillus subtilisACHNRenal CancerSulforhodamine B assayGI50 = 11.5 µg/mL48-hKidneyNone
5065
244925202014
ELLVDLL
Gageostatin A7LinearLNoneFree3-beta-hydroxy-11-methyltridecanoic acidAntimicrobialBacillus subtilisNCI-H23Lung CancerSulforhodamine B assayGI50 = 11.2 µg/mL48-hLungNone
5066
244925202014
ELLVDLL
Gageostatin A7LinearLNoneFree3-beta-hydroxy-11-methyltridecanoic acidAntimicrobialBacillus subtilisNUGC-3Stomach CancerSulforhodamine B assayGI50 = 11.8 µg/mL48-hStomachNone
5064
244925202014
ELLVDLL
Gageostatin A7LinearLNoneFree3-beta-hydroxy-11-methyltridecanoic acidAntimicrobialBacillus subtilisPC-3Prostate CancerSulforhodamine B assayGI50 = 10.8 µg/mL48-hProstateNone
5063
244925202014
ELLVDLL
Gageostatin A7LinearLNoneFree3-beta-hydroxy-11-methyltridecanoic acidAntimicrobialBacillus subtilisHCT-15Colon CancerSulforhodamine B assayGI50 = 11.4 µg/mL48-hColonNone
5062
244925202014
ELLVDLL
Gageostatin A7LinearLNoneFree3-beta-hydroxy-11-methyltridecanoic acidAntimicrobialBacillus subtilisMDA-MB-231Breast CancerSulforhodamine B assayGI50 = 14.9 µg/mL48-hBreastNone
5061
248308452014
ETFADWWKLLAE
mt_S20A/L22 W/P27A12LinearLNoneFreeFreeAnticancerMDM5MCF-7Breast CancerMTT/MTS assayIC50= 8.7 µMNot AvailableBreastNone
5060
248308452014
ESFSDWWKLLAE
mt_T18S/L22 W/P27A12LinearLNoneFreeFreeAnticancerMDM4MCF-7Breast CancerMTT/MTS assayIC50=27 µMNot AvailableBreastNone
5059
248308452014
LTFSDWWKLLAE
mt_E17L/L22 W/P27A12LinearLNoneFreeFreeAnticancerMDM3MCF-7Breast CancerMTT/MTS assayIC50=15.1 µMNot AvailableBreastNone
5058
248308452014
ETFSDWWKLLAE
mt_L22 W/P27A12LinearLNoneFreeFreeAnticancerMDM2MCF-7Breast CancerMTT/MTS assayIC50=16.3 µMNot AvailableBreastNone
5057
247140812014
TKPRKTKPRKTKPRKTKPR
T Peptide19LinearLNoneFreeFreeAnticancerTuftsin derivativeBGC-823Gastric CancerMTT/MTS assay67.2% maximum inhibitory rate at 8 mg/kg48-hStomachNone
5056
247140812014
TKPRKTKPRKTKPRKTKPR
T Peptide19LinearLNoneFreeFreeAnticancerTuftsin derivativeHT-29Colon CancerMTT/MTS assay70% maximum inhibitory rate at 8 mg/kg48-hColonNone
5055
247140812014
TKPRKTKPRKTKPRKTKPR
T Peptide19LinearLNoneFreeFreeAnticancerTuftsin derivativeHepG-2Liver CancerMTT/MTS assay69.6% maximum inhibitory rate at 8 mg/kg48-hLiverNone
5054
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC107Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5053
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC107Colorectal CancerCell Viability assayCell viability >65% at 12.5μM approx24-hColonNone
5052
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC107Colorectal CancerCell Viability assayCell viability >50% at 12.5μM approx24-hColonNone
5051
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >85% at 12.5μM approx24-hColonNone
5050
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >80% at 12.5μM approx24-hColonNone
5049
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5048
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC113Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5047
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC113Colorectal CancerCell Viability assayCell viability >65% at 12.5μM approx24-hColonNone
5046
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC113Colorectal CancerCell Viability assayCell viability >80% at 12.5μM approx24-hColonNone
5045
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5044
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >60% at 12.5μM approx24-hColonNone
5043
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5042
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >85% at 12.5μM approx24-hColonNone
5041
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >80% at 12.5μM approx24-hColonNone
5040
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >45% at 12.5μM approx24-hColonNone
5039
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5038
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5037
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5036
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC18Colorectal CancerCell Viability assayCell viability >75% at 12.5μM approx24-hColonNone
5035
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC18Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5034
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC18Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5033
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >50% at 12.5μM approx24-hColonNone
5032
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >40% at 12.5μM approx24-hColonNone
5031
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >40% at 12.5μM approx24-hColonNone
5030
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability =50% at 12.5μM approx.1-hColonNone
5029
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability =50% at 12.5μM approx.1-hColonNone
5028
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5027
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5026
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5025
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5024
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5023
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5022
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5021
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5020
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5019
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5018
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >50% at 12.5μM approx.1-hColonNone
5017
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability =50% at 12.5μM approx.1-hColonNone
5015
246769012014
KAQ-Dip-QKQAW
LTX-3288LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideFem-XSkin CancerMTT/MTS assayIC50= >350 µM5–60 MinSkinNone
5016
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5013
246769012014
KKWWKKW-Dip-K
LTX-3159LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideA375Skin CancerMTT/MTS assayIC50=12.7 µM30-MinSkinNone
5014
246769012014
KKWWKKW-Dip-K
LTX-3159LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideFem-XSkin CancerMTT/MTS assayIC50=15.3 µM30-MinSkinNone
5012
246769012014
KKWWKKW-Dip-K
LTX-3159LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideB16F1Skin CancerMTT/MTS assayIC50=13.3 µM30-MinSkinNone
5011
246610242014
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneFreeFreeAntimicrobialMain component of honey bee venomSCC25Skin CancerCell Viability assay102.9 ± 4.1% cell growth inhibition at 1 µM24-hSkinNone
5010
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC25Skin CancerCell Viability assay107.0 ± 5.0% cell growth inhibition at 1 µM24-hSkinNone
5009
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC25Skin CancerCell Viability assay0.6 ± 0.6% cell growth inhibition at 10 µM48-hSkinNone
5008
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC25Skin CancerMTT/MTS assayIC50=2.2 µM48-hSkinNone
5007
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC12Skin CancerMTT/MTS assayIC50=1 µM48-hSkinNone
5006
245873502014
LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES
LL 3737LinearLNoneFreeFreeAntimicrobialAlso known human cathelicidinOVRCAR-3Ovarian CancerMTT/MTS assayLC50= 24 at 100 µM72-hOvaryNone
5005
245873502014
GIGKFLKKAKKFGKAFVKILKK
Pexiganan22LinearLNoneAmidationFreeAntimicrobialAnalog of magainin 2OVRCAR-3Ovarian CancerMTT/MTS assayLC50= 13 at 100 µM72-hOvaryNone
5004
245873502014
LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES
LL 3737LinearLNoneFreeFreeAntimicrobialAlso known human cathelicidinLNCaPProstate cancerMTT/MTS assayLC50= 27 at 100 µM72-hProstateNone
5003
245873502014
GIGKFLKKAKKFGKAFVKILKK
Pexiganan22LinearLNoneAmidationFreeAntimicrobialAnalog of magainin 2LNCaPProstate cancerMTT/MTS assayLC50= 6 at 100 µM72-hProstateNone
5002
245873502014
LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES
LL 3737LinearLNoneFreeFreeAntimicrobialAlso known human cathelicidinMCF-7Breast CancerMTT/MTS assayLC50= 21 at 100 µM72-hBreastNone
5001
245873502014
GIGKFLKKAKKFGKAFVKILKK
Pexiganan22LinearLNoneAmidationFreeAntimicrobialAnalog of magainin 2MCF-7Breast CancerMTT/MTS assayLC50= 8 at 100 µM72-hBreastNone
4673
228851722012
GLFGKLIKKFARKAISYAVKKARGKH
ltc2aG11A26LinearLNoneFreeFreeAntimicrobialCentral Asian spider, Lachesana tarabaeviProstate tumor celllineProstate CancerLDH leakage assaygraph fig 8 ANot AvailableProstateNone
4671
230857712012
Not Available
12c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=14 µMNot AvailableBloodNone
4672
228851722012
GLFGKLIKKFGRKAISYAVKKARGKH
Latarcin 2a26LinearLNoneFreeFreeAntimicrobialCentral Asian spider, Lachesana tarabaeviBreast tumor celllineBreast CancerLDH leakage assaygraph fig 8 ANot AvailableBreastNone
4669
230857712012
Not Available
12a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=6.1 µMNot AvailableBloodNone
4670
230857712012
Not Available
12b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=27 µMNot AvailableBloodNone
4667
230857712012
Not Available
11b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=19 µMNot AvailableBloodNone
4668
230857712012
Not Available
11c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=7.2 µMNot AvailableBloodNone
4666
230857712012
Not Available
11a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=5.2 µMNot AvailableBloodNone
4664
230857712012
Not Available
10b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=11.4 µMNot AvailableBloodNone
4665
230857712012
Not Available
10c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=6.6 µMNot AvailableBloodNone
4662
230857712012
Not Available
9c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=3.1 µMNot AvailableBloodNone
4663
230857712012
Not Available
10a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=28 µMNot AvailableBloodNone
4660
230857712012
Not Available
9a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=31 µMNot AvailableBloodNone
4661
230857712012
Not Available
9b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=2.3 µMNot AvailableBloodNone
4658
230857712012
Not Available
8b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=>254 µMNot AvailableBloodNone
4659
230857712012
Not Available
8c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=107 µMNot AvailableBloodNone
4657
230857712012
Not Available
8a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=136 µMNot AvailableBloodNone
4655
230857712012
Not Available
7b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=>78 µMNot AvailableBloodNone
4656
230857712012
Not Available
7c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=79 µMNot AvailableBloodNone
4653
230857712012
Not Available
6c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=4.3 µMNot AvailableBloodNone
4654
230857712012
Not Available
7a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=>63 µMNot AvailableBloodNone
4650
230857712012
Not Available
5c3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=4.1 µMNot AvailableBloodNone
4651
230857712012
Not Available
6a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=14.4 µMNot AvailableBloodNone
4652
230857712012
Not Available
6b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=11.0 µMNot AvailableBloodNone
4648
230857712012
Not Available
5a3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=10.6 µMNot AvailableBloodNone
4649
230857712012
Not Available
5b3LinearLNoneFreeFreeAntimicrobialsynthetic b2,2-amino acid derivativesRamosLymphoma CancerMTT/MTS assayIC50=7.1 µMNot AvailableBloodNone
4600
213513232011
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EGFR-lytic32LinearMixNoneFreeFreeAntitumorSynthetic PeptideMDA-MB-231Breast CancerELISAIC50 =0.46 µM15-MinBreastNone
4599
213513232011
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EGFR-lytic32LinearMixNoneFreeFreeAntitumorSynthetic PeptideMDA-MB-231Breast CancerELISAIC50 =0.12 µM60-MinBreastNone
4598
214039172011
FLPLIGRVLSGIL
Temporin A13LinearLNoneAmidationFreeAntimicrobialFrog Rana temporariaU-943Lymphoma CancerMTT/MTS assayIC50 =80-90 µg/mlNot AvailableBloodNone
4597
214039172011
RGGRLCYCRRRFCVCVGR
Protegrin 118LinearLNoneAmidationFreeAntimicrobialalpha helical peptide without cysteinesU-942Lymphoma CancerMTT/MTS assayIC50 =30-40 µg/mlNot AvailableBloodNone
4596
214039172011
GIGKFLKKAKKFGKAFVKILKK
Pexiganan MSI-7818LinearLNoneAmidationFreeAntimicrobialAnalog of MagaininU-941Lymphoma CancerMTT/MTS assayIC50 =20-30 µg/mlNot AvailableBloodNone
4595
214039172011
ILRWPWWPWRRK
Omiganan MBI-22612LinearLNoneAmidationFreeAntimicrobialBovine neutrophilsU-937Lymphoma CancerMTT/MTS assayIC50 =80-85 µg/mlNot AvailableBloodNone
4594
214039172011
AKRHHGYKRKFH
Demegen P-11312LinearLNoneAmidationFreeAntimicrobialCanaida albicansU-939Lymphoma CancerMTT/MTS assayIC50 =85-90 µg/mlNot AvailableBloodNone
4593
214039172011
GLFDVIKKVASVIGGL
Citropin 1.116LinearLNoneAmidationFreeAntimicrobialAustralian blue mountains tree frog, Litoria citropaU-938Lymphoma CancerMTT/MTS assayIC50 =40 µg/mlNot AvailableBloodNone
4592
214039172011
TRSSRAGLQFPVGRVHRLLRK
Buforin 221LinearLNoneFreeFreeAntimicrobialBufo Bufo GargarizansU-937Lymphoma CancerMTT/MTS assayIC50 =90-95 µg/mlNot AvailableBloodNone
4591
214236132011
QETFSDLWKLLP
P5317-2812LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =30 µMNot AvailableColonNone
4590
214236132011
LTAEHYAAQATS
3A12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 >100 µMNot AvailableColonNone
4588
214236132011
PRFWEYWLRLME
MIP12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =0.12 µMNot AvailableColonNone
4589
214236132011
LTFEHYWAQLTS
DI12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =1.6 µMNot AvailableColonNone
4587
214236132011
PRFWEYWLRLAE
MIP(M11A)12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =0.4 µMNot AvailableColonNone
4585
214236132011
PRFWEYWLALME
MIP(R9A)12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =0.02 µMNot AvailableColonNone
4586
214236132011
PRFWEYWLRAME
MIP(L10A)12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =1.14 µMNot AvailableColonNone
4584
214236132011
PRFWEYALRLME
MIP(W7A)12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 >100 µMNot AvailableColonNone
4583
214236132011
PRFWEAWLRLME
MIP(Y6A)12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 >100 µMNot AvailableColonNone
4582
214236132011
PRAWEYWLRLME
MIP(F3A)12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =0.57 µMNot AvailableColonNone
4580
214236132011
LTAEHYAAQATS
3A12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 >100 µMNot AvailableColonNone
4581
214236132011
QETFSDLWKLLP
P5317-2812LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =4.7 µMNot AvailableColonNone
4579
214236132011
LTFEHYWAQLTS
DI12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =0.29 µMNot AvailableColonNone
4577
219281252012
GVGSPYVSRLLGICL
p77615LinearLNoneFreeFreeAntitumorSynthetic PeptideNot AvailableTumorELISPOT assayNot AvailableNot AvailableNot AvailableNone
4578
214236132011
PRFWEYWLRLME
MIP12LinearLNoneFreeFreeAntitumorE3 ubiquitin-protein ligaseHCT-116-p53+/+Colon CancerImmunoprecipitation assayIC50 =0.01 µMNot AvailableColonNone
4575
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7-TX400Breast CancerMTT/MTS assay~5% cytotoxic at 50 µM24-hBreastNone
4576
219281252012
LIAHNQVRQV
p8510LinearLNoneFreeFreeAntitumorSynthetic PeptideNot AvailableTumorELISPOT assayNot AvailableNot AvailableNot AvailableNone
4574
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7-TX400Breast CancerMTT/MTS assay60-70% cytotoxic at 50 µM24-hBreastNone
4571
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7Breast CancerMTT/MTS assay70% cytotoxic at 50 µM24-hBreastNone
4572
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7Breast CancerMTT/MTS assay0% cytotoxic at 50 µM24-hBreastNone
4573
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7-TX400Breast CancerMTT/MTS assay60-70% cytotoxic at 50 µM24-hBreastNone
4567
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay~0% cytotoxic at 10 µM24-hBreastNone
4568
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay5-10% cytotoxic at 25 µM24-hBreastNone
4569
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay20% cytotoxic at 50 µM24-hBreastNone
4570
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7Breast CancerMTT/MTS assay70% cytotoxic at 50 µM24-hBreastNone
4564
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay5% cytotoxic at 25 µM24-hBreastNone
4565
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay10-15% cytotoxic at 50 µM24-hBreastNone
4566
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4561
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay15-20% cytotoxic at 50 µM24-hBreastNone
4562
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay~5% cytotoxic at 5 µM24-hBreastNone
4563
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay~5% cytotoxic at 10 µM24-hBreastNone
4559
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay10% cytotoxic at 10 µM24-hBreastNone
4560
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay10-15% cytotoxic at 25 µM24-hBreastNone
4557
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10-15% cytotoxic at 50 µM24-hBreastNone
4558
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay10% cytotoxic at 5 µM24-hBreastNone
4555
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay~0% cytotoxic at 10 µM24-hBreastNone
4556
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10% cytotoxic at 25 µM24-hBreastNone
4552
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay10% cytotoxic at 25 µM24-hBreastNone
4553
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay10-15% cytotoxic at 50 µM24-hBreastNone
4554
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4549
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay80-90% cytotoxic at 25 µM24-hBreastNone
4550
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay85-90% cytotoxic at 50 µM24-hBreastNone
4551
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay~5% cytotoxic at 10 µM24-hBreastNone
4546
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay80-90% cytotoxic at 50 µM24-hBreastNone
4547
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay30-40% cytotoxic at 5 µM24-hBreastNone
4548
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay60-70% cytotoxic at 10 µM24-hBreastNone
4544
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay50% cytotoxic at 10 µM24-hBreastNone
4545
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay80% cytotoxic at 25 µM24-hBreastNone
4543
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay10% cytotoxic at 5 µM24-hBreastNone
4540
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay20% cytotoxic at 10 µM24-hBreastNone
4541
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay70-80% cytotoxic at 25 µM24-hBreastNone
4542
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay80-85% cytotoxic at 50 µM24-hBreastNone
4538
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay40-50% cytotoxic at 50 µM24-hBreastNone
4539
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4537
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay20% cytotoxic at 25 µM24-hBreastNone
4534
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay40-50% cytotoxic at 50 µM24-hBreastNone
4535
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4536
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10% cytotoxic at 10 µM24-hBreastNone
4532
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay5% cytotoxic at 10 µM24-hBreastNone
4533
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay20-30% cytotoxic at 25 µM24-hBreastNone
4530
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay85-90% cytotoxic at 50 µM24-hBreastNone
4531
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4528
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay40-50% cytotoxic at 10 µM24-hBreastNone
4529
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay80% cytotoxic at 25 µM24-hBreastNone
4525
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay60-70% cytotoxic at 25 µM24-hBreastNone
4526
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay80-85% cytotoxic at 50 µM24-hBreastNone
4527
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay15-20% cytotoxic at 5 µM24-hBreastNone
4524
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay40-50% cytotoxic at 10 µM24-hBreastNone
4521
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay70% cytotoxic at 25 µM24-hBreastNone
4522
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay80-85% cytotoxic at 50 µM24-hBreastNone
4523
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay30% cytotoxic at 5 µM24-hBreastNone
4520
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay50% cytotoxic at 10 µM24-hBreastNone
4518
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay60% cytotoxic at 50 µM24-hBreastNone
4519
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay30% cytotoxic at 5 µM24-hBreastNone
4517
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay30-35% cytotoxic at 25 µM24-hBreastNone
4515
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay5-10% cytotoxic at 5 µM24-hBreastNone
4516
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10% cytotoxic at 10 µM24-hBreastNone
4514
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay60% cytotoxic at 50 µM24-hBreastNone
4511
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay5% cytotoxic at 5 µM24-hBreastNone
4512
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay5% cytotoxic at 10 µM24-hBreastNone
4513
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay30-35% cytotoxic at 25 µM24-hBreastNone
4504
220572782011
AAKKWAKAKWAKAKKWAKAA
Z1021LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4503
220572782011
AAWKWAWAKKWAKAKKWAKAA
Z921LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =13 µMNot AvailableColonNone
4501
220572782011
KAAKKAWKAAKKAWKAAKKAA
Z721LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =21 µMNot AvailableColonNone
4502
220572782011
AWKKWAKAWKWAKAKWWAKAA
Z821LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =23 µMNot AvailableColonNone
4500
220572782011
KWWKKAAKAAKKAAKAAKKWA
Z621LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =31 µMNot AvailableColonNone
4499
220572782011
KAAKKAWKWAKKAAKWAKKAA
Z521LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =67 µMNot AvailableColonNone
4498
220572782011
KAAKKAWKAAKKAAKWWKKAA
Z421LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =173 µMNot AvailableColonNone
4497
220572782011
KAAKKAWKAWKKAAKAAWKKAA
Z321LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4496
220572782011
KAAKKWAKAWKKAAKAWKKAA
Z221LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4495
220572782011
KAAKKWAKAAKKWAKAWKKAA
Z121LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4494
220572782011
AAKKWAKAKWAKAKKWAKAA
Z1021LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 >211 µMNot AvailableBreastNone
4493
220572782011
AAWKWAWAKKWAKAKKWAKAA
Z921LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =16 µMNot AvailableBreastNone
4492
220572782011
AWKKWAKAWKWAKAKWWAKAA
Z821LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =14 µMNot AvailableBreastNone
4491
220572782011
KAAKKAWKAAKKAWKAAKKAA
Z721LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =15 µMNot AvailableBreastNone
4490
220572782011
KWWKKAAKAAKKAAKAAKKWA
Z621LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =16 µMNot AvailableBreastNone
4489
220572782011
KAAKKAWKWAKKAAKWAKKAA
Z521LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =28 µMNot AvailableBreastNone
4488
220572782011
KAAKKAWKAAKKAAKWWKKAA
Z421LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =68 µMNot AvailableBreastNone
4487
220572782011
KAAKKAWKAWKKAAKAAWKKAA
Z321LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =128 µMNot AvailableBreastNone
4486
220572782011
KAAKKWAKAWKKAAKAWKKAA
Z221LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =173 µMNot AvailableBreastNone
4485
220572782011
KAAKKWAKAAKKWAKAWKKAA
Z121LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =186 µMNot AvailableBreastNone
4484
220572782011
AAKKWAKAKWAKAKKWAKAA
Z1021LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4483
220572782011
AAWKWAWAKKWAKAKKWAKAA
Z921LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =9 µMNot AvailableSkinNone
4482
220572782011
AWKKWAKAWKWAKAKWWAKAA
Z821LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =19 µMNot AvailableSkinNone
4481
220572782011
KAAKKAWKAAKKAWKAAKKAA
Z721LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =15 µMNot AvailableSkinNone
4480
220572782011
KWWKKAAKAAKKAAKAAKKWA
Z621LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =17 µMNot AvailableSkinNone
4479
220572782011
KAAKKAWKWAKKAAKWAKKAA
Z521LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =42 µMNot AvailableSkinNone
4478
220572782011
KAAKKAWKAAKKAAKWWKKAA
Z421LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =155 µMNot AvailableSkinNone
4477
220572782011
KAAKKAWKAWKKAAKAAWKKAA
Z321LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4476
220572782011
KAAKKWAKAWKKAAKAWKKAA
Z221LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4475
220572782011
KAAKKWAKAAKKAAKAWKKAA
Z121LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4474
220769542011
RRRRRRRRGGC-Pem
Peptide-311LinearLPem= PemetrexedAmidationFreeAnticancerSyntheticNCI-H358Lung CancerMTT/MTS assayIC50 = 8.41 µM3-hLungNone
4473
220769542011
IELLQARGGC-Pem-GGRRRRRRRR
Peptide-220LinearLPem= PemetrexedAmidationFreeAnticancerSyntheticNCI-H358Lung CancerMTT/MTS assayIC50 = 2.19 µM3-hLungNone
4472
220769542011
IELLQARGGC-Pem
Peptide-110LinearLPem= PemetrexedAmidationFreeAnticancerSyntheticNCI-H358Lung CancerMTT/MTS assayIC50 = 4.63 mM3-hLungNone
4471
220769542011
RRRRRRRRGGC-Pem
Peptide-311LinearLPem= PemetrexedAmidationFreeAnticancerSyntheticHL-60Leukemia CancerMTT/MTS assayIC50 = 6.24 µM3-hBloodNone
4470
220769542011
IELLQARGGC-Pem-GGRRRRRRRR
Peptide-210LinearLPem= PemetrexedAmidationFreeAnticancerSyntheticHL-60Leukemia CancerMTT/MTS assayIC50 = 2.64 µM3-hBloodNone
4469
220769542011
IELLQARGGC-Pem
Peptide-110LinearLPem= PemetrexedAmidationFreeAnticancerSyntheticHL-60Leukemia CancerMTT/MTS assayIC50 = 2.17 µM3-hBloodNone
4427
21434649, 189574412011
GLPVCGETCFGGTCNTPGCTCDPWPVCTRN
Vaby D30Not AvailableLNoneFreeFreeAnticancerAfrican, the Ethiopian highlands, Viola abyssinicaNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4426
21434649, 189574412011
GLPVCGETCAGGTCNTPGCSCSWPICTRN
Vaby A29Not AvailableLNoneFreeFreeAnticancerAfrican, the Ethiopian highlands, Viola abyssinicaNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4416
22771617, 189574412012
GLLGLLGSVVSHVVPAIVGHF
Maculatin 1.321Not AvailableLNoneFreeFreeAnticancerBlue-thighed frog,Litoria chloris, AustraliaNot AvailableSkin CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4415
22771617, 189574412012
GLLGLLGSVVSHVLPAITQHL
Maculatin 1.421Not AvailableLNoneFreeFreeAnticancerBlue-thighed frog,Litoria chloris, AustraliaNot AvailableSkin CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4387
22100226, 189574412012
GFGMALKLLKKVL
Macropin 113Not AvailableLNoneFreeFreeAntibacterialVenom, the solitary beeMacropis fulvipesNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4386
22100226, 189574412012
GTGLPMSERRKIMLMMR
Macropin 217Not AvailableLNoneFreeFreeAntibacterialVenom, the solitary beeMacropis fulvipesNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4384
21596752, 189574412011
GEFLKCGESCVQGECYTPGCSCDWPICKKN
Cliotide T230Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4383
21596752, 189574412011
GIPCGESCVFIPCITAAIGCSCKSKVCYRN
Cliotide T430Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4382
21596752, 189574412011
GIPCGESCVFIPCITGAIGCSCKSKVCYRN
Cliotide T130Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4381
21596752, 189574412011
GLPTCGETCTLGTCYVPDCSCSWPICMKN
Cliotide T329Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4379
21723349, 189574412011
GSIPCEGSCVFIPCISAIIGCSCSNKVCYKN
Viphi G31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4378
21723349, 189574412011
GLPVCGETCVGGTCNTPGCGCSWPVCTRN
Viba1729Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4377
21723349, 189574412011
GLPVCGETCVGGTCNTPGCACSWPVCTRN
Viba 1529Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4376
21723349, 189574412011
GIPCGESCVFIPCLTSAIDCSCKSKVCYRN
Mram 830Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4375
21723349, 189574412011
GSIPCGESCVFIPCISAIIGCSCSSKVCYKN
Viphi F31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4374
21723349, 189574412011
GSIPCGESCVFIPCISSVIGCACKSKVCYKN
Viphi F31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4373
21723349, 189574412011
GSIPCGESCVFIPCISAVIGCSCSNKVCYKN
Viphi E31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4372
22467870, 189574412012
GIPCAESCVWIPPCTITALMGCSCKNNVCYNN
Chassatide C232Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4371
22467870, 189574412012
GEYCGESCYLIPCFTPGCYCVSRQCVNKN
Chassatide C1029Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4370
22467870, 189574412012
GDACGETCFTGICFTAGCSCNPWPTCTRN
Chassatide C429Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4369
22467870, 189574412012
GASCGETCFTGICFTAGCSCNPWPTCTRN
Chassatide C429Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4368
22467870, 189574412012
IPCGESCVWIPCISGMFGCSCKDKVCYS
ChaC1129Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4367
22467870, 189574412012
AIPCGESCVWIPCISTVIGCSCSNKVCYR
Chassatide C829Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4366
22467870, 189574412012
IPCGESCVWIPCITAIAGCSCKNKVCYT
ChaC729Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4365
21882228, 189574412012
AWKLFDDGV
Cr-ACP19Not AvailableLNoneFreeFreeAntibacterialSeeds,Cycas revolutaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
3828
230348932012
MDSNKDERAYAQWVIIILHNVGSSPFKIANLGLSWGKLYADGNKDKEVYP
SDYNGKTVGPDEKIQINSCGRENASSGTEGSFDIVDPNDGNKTIRHFYWECPWGS
KRNTWTPSGSNTKWMVEWSGQNLDSGALGTITVDVLRKGN
AAD (or Aa-Pri1)145LinearLNoneFreeFreeAntitumorPurified from Agrocybe aegeritaSH-SY5YBrain TumorMTT/MTS assayAt 2.5 µM concentration,decrease in cell vibility= 70%48-hBrainNone
3827
230348932012
MDSNKDERAYAQWVIIILHNVGSSPFKIANLGLSWGKLYADGNKDKEVYP
SDYNGKTVGPDEKIQINSCGRENASSGTEGSFDIVDPNDGNKTIRHFYW
ECPWGSKRNTWTPSGSNTKWMVEWSGQNLDSGALGTITVDVLRKGN
AAD (or Aa-Pri1)145LinearLNoneFreeFreeAntitumorPurified from Agrocybe aegeritaHeLaCervical CancerMTT/MTS assayAt 2.5 µM concentration,decrease in cell vibility= 70%48-hCervixNone
3826
230348932012
MDSNKDERAYAQWVIIILHNVGSSPFKIANLGLSWGKLYADGNKDKEVY
PSDYNGKTVGPDEKIQINSCGRENASSGTEGSFDIVDPNDGNKTIRHFYW
ECPWGSKRNTWTPSGSNTKWMVEWSGQNLDSGALGTITVDVLRKGN
AAD (or Aa-Pri1)145LinearLNoneFreeFreeAntitumorPurified from Agrocybe aegeritaHepG-2Liver CancerMTT/MTS assayAt 2.5 µM concentration,decrease in cell vibility= 35%48-hLiverNone
3824
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNF
VLIVSQLQPSQENEMFSIRDSAHRRFLLFRRAFKQL
RGD-mda-7207LinearLNoneFreeFreeAnticancerDerived from wtmda-7/IL-24 by insertion og a glycine residue between Arg(164) and Asp(165).Ket-3TumorMTT assayApoptotic rate(%)= >50% at concentration of 8 µg/ml72-hNot AvailableNone
3823
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNF
VLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAFK
QLDVEAALTKALGEVDILLTWMQKFYKL
RGD-mda-7207LinearLNoneFreeFreeAnticancerDerived from wtmda-7/IL-24 by insertion og a glycine residue between Arg(164) and Asp(165).MCF-7Breast CancerMTT assayApoptotic rate(%)= >70% at concentration of 8 µg/ml72-hBreastNone
3821
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANNF
VLIVSQLQPSQENEMFSIRDSAHRRFLLFRRAF
KQL
wtmda-7/IL-24206LinearLNoneFreeFreeAnticancerNAKet-3TumorMTT assayApoptotic rate(%)= >30% at concentration of 8 µg/ml72-hNot AvailableNone
3820
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANN
FVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRAF
KQL
wtmda-7/IL-24206LinearLNoneFreeFreeAnticancerNAMCF-7Breast CancerMTT assayApoptotic rate(%)= >50% at concentration of 8 µg/ml72-hBreastNone
3819
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANN
FVLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAF
KQLDVEAALTKALGEVDILLTWMQKFYKL
RGD-mda-7207LinearLNoneFreeFreeAnticancerDerived from wtmda-7/IL-24 by insertion og a glycine residue between Arg(164) and Asp(165).Ket-3TumorMTT/MTS assayCell viability(% of control)= 0.5 at concentration 8 µg/ml48-hNot AvailableNone
3818
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANN
FVLIVSQLQPSQENEMFSIRGDSAHRRFLLFRRAF
KQLDVEAALTKALGEVDILLTWMQKFYKL
RGD-mda-7207LinearLNoneFreeFreeAnticancerDerived from wtmda-7/IL-24 by insertion og a glycine residue between Arg(164) and Asp(165).MCF-7Breast CancerMTT/MTS assayCell viability(% of control)=0.5 at concentration 4 µg/ml48-hBreastNone
3817
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLANN
FVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRA
FKQL
wtmda-7/IL-24206LinearLNoneFreeFreeAnticancerNAKet-3TumorMTT/MTS assayCell viability(% of control)= 0.5 at concentration 8 µg/ml48-hNot AvailableNone
3816
229634852012
MNFQQRLQSLWTLARPFCPPLLATASQMQMVVLPCLGFTLLLWSQVSG
AQGQEFHFGPCQVKGVVPQKLWEAFWAVKDTMQAQDNITSARLLQQEVLQ
NVSDAESCYLVHTLLEFYLKTVFKNYHNRTVEVRTLKSFSTLAN
NFVLIVSQLQPSQENEMFSIRDSAHRRFLLFRRA
FKQL
wtmda-7/IL-24206LinearLNoneFreeFreeAnticancerNAMCF-7Breast CancerMTT/MTS assayCell viability(% of control)=0.5 at concentration 7 µg/ml48-hBreastNone
3815
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 1.4±0.1 µM24-hSkinNone
3814
238936052013
KISKRILTGKK
NK-1111LinearLNoneAmidationFreeAnticancerNK2 derived inactive control peptideE42/02Skin CancerMTT/MTS assayIC50 >> 100 µM24-hSkinNone
3813
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 13.1±0.9 µM24-hSkinNone
3812
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 12.3±1.0 µM24-hSkinNone
3811
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 3.7± 4.3 µM24-hSkinNone
3810
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 40 µM (approx)24-hSkinNone
3808
238936052013
KISKRILTGKK
NK-1111LinearLNoneAmidationFreeAnticancerNK2 derived inactive control peptideE42/02Skin CancerMTT/MTS assayIC-50 >> 100 µM4-hSkinNone
3809
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 1.8±0.1 µM4-hSkinNone
3807
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 9.3±1.5 µM4-hSkinNone
3806
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 8.3±0.5 µM4-hSkinNone
3805
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 12.1±1.6 µM4-hSkinNone
3804
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 50 µM (approx)4-hSkinNone
3803
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 2.1±0.1 µM2-hSkinNone
3802
238936052013
KISKRILTGKK
NK-1111LinearLNoneAmidationFreeAnticancerNK2 derived inactive control peptideE42/02Skin CancerMTT/MTS assayIC-50 >> 100 µM2-hSkinNone
3801
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 13.8±2.0 µM2-hSkinNone
3800
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 12.3±2.0 µM2-hSkinNone
3799
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 13.0±1.0 µM2-hSkinNone
3798
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 50 µM (approx)2-hSkinNone
3797
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 3.2±0.1 µM30-MinSkinNone
3796
238936052013
KISKRILTGKK
NK-1111LinearLNoneAmidationFreeAnticancerNK2 derived inactive control peptideE42/02Skin CancerMTT/MTS assayIC-50>> 100 µM30-MinSkinNone
3795
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 7.5±0.4 µM30-MinSkinNone
3794
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 8.4±0.2 µM30-MinSkinNone
3793
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 10.6±0.4 µM30-MinSkinNone
3792
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 70 µM (approx)30-MinSkinNone
3791
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 1.4±0.1 µM4-hSkinNone
3790
238936052013
KISKRILTGKK
NK-1111LinearLNoneAmidationFreeAnticancerNK2 derived inactive control peptideE42/02Skin CancerMTT/MTS assayIC-50 >> 100 µM4-hSkinNone
3789
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 4.3±0.3 µM4-hSkinNone
3788
229334122012
KW β2,2KK
c85LinearL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 226±21 µMol/LNABloodNone
3787
229334122012
KK β2,2WKK
c76LinearL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 157±30 µMol/LNABloodNone
3786
229334122012
KW β2,2WKK
c66LinearL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 26±2 µMol/LNABloodNone
3785
229334122012
KKW β2,2WKK
c57LinearL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 23±3 µMol/LNABloodNone
3784
229334122012
KW β2,2KK
c45LinearL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 99±15 µMol/LNABloodNone
3783
229334122012
KK β2,2WKK
c36LinearL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 92±2 µMol/LNABloodNone
3782
229334122012
KW β2,2WKK
c26LinearL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 1.71±0.6 µMol/LNABloodNone
3781
229334122012
KKWβ2,2WKK
c17LinearL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)AmidationFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 22±5 µMol/LNABloodNone
3780
229334122012
KW β2,2KK
c85CyclicL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 20±2 µMol/LNABloodNone
3779
229334122012
KK β2,2WKK
c76CyclicL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 16±5 µMol/LNABloodNone
3778
229334122012
KW β2,2WKK
c66CyclicL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 8±1 µMol/LNABloodNone
3775
229334122012
KK β2,2WKK
c36CyclicL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 15±2 µMol/LNABloodNone
3776
229334122012
KW β2,2KK
c45CyclicL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 12.6±0.6 µMol/LNABloodNone
3777
229334122012
KKW β2,2WKK
c57CyclicL(2,2-di(4-[trifluoromethyl]benzyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 11±2 µMol/LNABloodNone
3773
229334122012
KKWβ2,2WKK
c17CyclicL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 10±2 µMol/LNABloodNone
3774
229334122012
KW β2,2WKK
c26CyclicL(2,2-di(naphthalen-2-ylmethyl)-3-amino-propionic acid)FreeFreeAnticancerKKWβ2,2WKKRamosLymphoma CancerMTT/MTS assayIC50= 7.9±0.3 µMol/LNABloodNone
3772
228376672012
KWKSFlKTFKSlKKTVlHTllKAISS
Peptide L6D/L12D/L17D/L20D/L21D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 12.88±0.15 µMol/L1-hCervixNone
3771
228376672012
KWKSFlKTFKSlKKTVlHTlLKAISS
Peptide L6D/L12D/L17D/L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 9.69±0.38 µMol/L1-hCervixNone
3769
228376672012
KWKSFLKTFKSlKKTVLHTlLKAISS
Peptide L12D/L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 3.14±0.06 µMol/L1-hCervixNone
3770
228376672012
KWKSFlKTFKSlKKTVLHTlLKAISS
Peptide L6D/L12D/L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 7.80±0.26 µMol/L1-hCervixNone
3767
228376672012
KWKSFLKTFKSLKKTVLHTlLKAISS
Peptide L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.33±0.06 µMol/L1-hCervixNone
3768
228376672012
KWKSFlKTFKSlKKTVLHTLLKAISS
Peptide L6D/L12D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 3.01±0.08 µMol/L1-hCervixNone
3766
228376672012
KWKSFLKTFKSlKKTVLHTLLKAISS
Peptide L12D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.63±0.07 µMol/L1-hCervixNone
3765
228376672012
KWKSFlKTFKSLKKTVLHTLLKAISS
Peptide L6D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.23±0.10 µMol/L1-hCervixNone
3764
228376672012
kWkSFLkTFkSLKkTVLHTLLkAISS
Peptide K1D/K3D/K7D /K10D/K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 18.07±0.48 µMol/L1-hCervixNone
3762
228376672012
KWKSFLkTFkSLKkTVLHTLLkAISS
Peptide K7D /K10D/K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 4.79±0.23 µMol/L1-hCervixNone
3763
228376672012
KWkSFLkTFkSLKkTVLHTLLkAISS
Peptide K3D/K7D /K10D/K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 20.41±0.64 µMol/L1-hCervixNone
3761
228376672012
KWKSFLkTFKSLKkTVLHTLLKAISS
Peptide K7D /K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 4.45±0.19 µMol/L1-hCervixNone
3760
228376672012
KWKSFLKTFKSLKkTVLHTLLkAISS
Peptide K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.40±0.09 µMol/L1-hCervixNone
3759
228376672012
KWKSFLkTFKSLKkTVLHTLLKAISS
Peptide K7D /K14D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.06±0.01 µMol/L1-hCervixNone
3758
228376672012
KWKSFLKTFKSLKKTVLHTLLkAISS
Peptide K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.39±0.02 µMol/L1-hCervixNone
3757
228376672012
KWKSFLKTFKSLKkTVLHTLLKAISS
Peptide K14D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.52±0.05 µMol/L1-hCervixNone
3756
228376672012
KWKSFLkTFKSLKKTVLHTLLKAISS
Peptide K7D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.29±0.03 µMol/L1-hCervixNone
3755
228376672012
KWKSFLKTFKSLKKTVLHTLLKAISS
Peptide P26LinearLNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.71±0.07 µMol/L1-hCervixNone
3753
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50= 22.25 µM72-hSkinNone
3754
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50= 12.55 µM72-hOvaryNone
3751
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50= 22.51 µM72-hStomachNone
3752
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50= 29.10 µM72-hProstateNone
3750
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50= 14.8 µM72-hColonNone
3748
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-498Renal CancerMTT/MTS assayIC50= 21.48 µM72-hRenalNone
3749
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-549Lung CancerMTT/MTS assayIC50= 14.53 µM72-hLungNone
3746
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50= 27.39 µM72-hSkinNone
3747
226448472012
FLKWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50= 24.76 µM72-hOvaryNone
3745
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50= 47.69 µM72-hProstateNone
3743
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50= 27.00 µM72-hColonNone
3744
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50= 26.70 µM72-hStomachNone
3741
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-498Renal CancerMTT/MTS assayIC50= 41.21 µM72-hRenalNone
3742
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-549Lung CancerMTT/MTS assayIC50= 25.20 µM72-hLungNone
3740
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50= 14.58 µM72-hOvaryNone
3738
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50= 24.32 µM72-hProstateNone
3739
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50= 13.16 µM72-hSkinNone
3736
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50= 14.80 µM72-hColonNone
3737
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50= 13.77 µM72-hStomachNone
3735
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-549Lung CancerMTT/MTS assayIC50= 15.88 µM72-hLungNone
3733
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50= 22.06 µM72-hOvaryNone
3734
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-498Renal CancerMTT/MTS assayIC50= 22.59 µM72-hRenalNone
3732
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50= 13.97 µM72-hSkinNone
3730
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50= 24.31 µM72-hStomachNone
3731
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50= 46.51 µM72-hProstateNone
3728
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-549Lung CancerMTT/MTS assayIC50= 20.36 µM72-hLungNone
3729
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50= 24.63 µM72-hColonNone
3726
224812512012
PLLQATLGGGS
P711LinearLNoneFreeFreeAntiproliferative and AntiangiogenicNAB16-F10Skin CancerWST-1 assayIC50= 1 µM48-hSkinNone
3727
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneFreeFreeAnticancer and AntimicrobialBrevinin-1EMaA-498Renal CancerMTT/MTS assayIC50= 22.88 µM72-hRenalNone
3717
221002262012
GKWLSLLKHILK
HAL-2/1112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3718
241768522013
YGRKKRRQRRRREADFFWSLCTADMS
KilerFLIP26linearLNoneFreeFreeNANAJurkatBlood CancerNot AvailableNANABloodNone
3716
221002262012
GKWMTLLKHILK
HAL-2/1312LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3714
221002262012
GKFMSLLKHILK
HAL-2/2412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3715
221002262012
GKWMSFLKHILK
HAL-2/612LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3713
221002262012
GKWMSLWKHILK
HAL-2/2012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3711
221002262012
GKWMSLLKHIWK
HAL-2/1812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3712
221002262012
GKWMSLLKHWLK
HAL-2/1912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3709
221002262012
GKWKSLLKHILK
HAL-2/112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 > 40 µM48-hBloodNone
3710
221002262012
GKWMSLLKHILK
HAL-2/812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3708
221002262012
GKWMKLLKHILK
HAL-2/212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 > 40 µM48-hBloodNone
3706
221002262012
gkwmsllkhilk
HAL-2/2212LinearDNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3707
221002262012
GKWMSLLKKILK
HAL-2/412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3704
221002262012
GMWSKLLGHLLR
HAL-1/1512LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 > 40 µM48-hBloodNone
3705
221002262012
GKWMSLLKHILK
HAL-212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 34 µM48-hBloodNone
3703
221002262012
GMWSKILGHLIR
HAL-1/2912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3701
221002262012
GKWKKILGHLIR
HAL-1/1912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3702
221002262012
GKWKKILGKLIR
HAL-1/2112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3700
221002262012
GKWSKILGKLIR
HAL-1/2012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 > 40 µM48-hBloodNone
3698
221002262012
KMWSKILGHLIR
HAL-1/1712LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3699
221002262012
GMWKKILGKLIR
HAL-1/1012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3696
221002262012
GMWKKILGHLIR
HAL-1/512LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 > 40 µM48-hBloodNone
3697
221002262012
GKWSKILGHLIR
HAL-1/1212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 > 40 µM48-hBloodNone
3695
221002262012
GMWSKILKHLIR
HAL-1/1812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3693
221002262012
GMWSKILGHLKR
HAL-1/412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3694
221002262012
GMWSKILGKLIR
HAL-1/912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 30±10 µM48-hBloodNone
3692
221002262012
GMWSKILGHLIK
HAL-1/612LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3691
221002262012
gmwskilghlir
HAL-1/2212LinearDNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3689
221002262012
GKWLSLLKHILK
HAL-2/1112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 40 µM48-hColonNone
3690
221002262012
GMWSKILGHLIR
HAL-112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 49±9 µM48-hBloodNone
3688
221002262012
GKWMTLLKHILK
HAL-2/1312LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 60 µM48-hColonNone
3687
221002262012
GKWMSFLKHILK
HAL-2/612LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3686
221002262012
GKFMSLLKHILK
HAL-2/2412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3685
221002262012
GKWMSLWKHILK
HAL-2/2012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3684
221002262012
GKWMSLLKHWLK
HAL-2/1912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3683
221002262012
GKWMSLLKHIWK
HAL-2/1812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3682
221002262012
GKWMSLLKHILK
HAL-2/812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3681
221002262012
GKWKSLLKHILK
HAL-2/112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3680
221002262012
GKWMKLLKHILK
HAL-2/212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 35±5 µM48-hColonNone
3679
221002262012
GKWMSLLKKILK
HAL-2/412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 38±6 µM48-hColonNone
3678
221002262012
gkwmsllkhilk
HAL-2/2212LinearDNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3677
221002262012
GKWMSLLKHILK
HAL-212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 35±3 µM48-hColonNone
3676
221002262012
GMWSKLLGHLLR
HAL-1/1512LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3675
221002262012
GMWSKILGHLIR
HAL-1/2912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3674
221002262012
GKWKKILGKLIR
HAL-1/2112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3673
221002262012
GKWKKILGHLIR
HAL-1/1912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3672
221002262012
GKWSKILGKLIR
HAL-1/2012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3671
221002262012
GMWKKILGKLIR
HAL-1/1012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 60 µM48-hColonNone
3666
221002262012
GMWSKILGKLIR
HAL-1/912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 50 µM48-hColonNone
3667
221002262012
GMWSKILKHLIR
HAL-1/1812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 18±2 µM48-hColonNone
3668
221002262012
GMWKKILGHLIR
HAL-1/512LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 44±5 µM48-hColonNone
3669
221002262012
GKWSKILGHLIR
HAL-1/1212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3670
221002262012
KMWSKILGHLIR
HAL-1/1712LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3661
221002262012
GKWLSLLKHILK
HAL-2/1112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 14±3 µM48-hCervixNone
3662
221002262012
GMWSKILGHLIR
HAL-112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 = 44±8 µM48-hColonNone
3663
221002262012
gmwskilghlir
HAL-1/2212LinearDNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3664
221002262012
GMWSKILGHLIK
HAL-1/612LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3665
221002262012
GMWSKILGHLKR
HAL-1/412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3656
221002262012
GKWMSLLKHWLK
HAL-2/1912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 16±4 µM48-hCervixNone
3657
221002262012
GKWMSLWKHILK
HAL-2/2012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 30±5 µM48-hCervixNone
3658
221002262012
GKFMSLLKHILK
HAL-2/2412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 34 µM48-hCervixNone
3659
221002262012
GKWMSFLKHILK
HAL-2/612LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 23±3 µM48-hCervixNone
3660
221002262012
GKWMTLLKHILK
HAL-2/1312LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 13±3 µM48-hCervixNone
3652
221002262012
GKWMKLLKHILK
HAL-2/212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 6±1 µM48-hCervixNone
3653
221002262012
GKWKSLLKHILK
HAL-2/112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 14±2 µM48-hCervixNone
3654
221002262012
GKWMSLLKHILK
HAL-2/812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 15±3 µM48-hCervixNone
3655
221002262012
GKWMSLLKHIWK
HAL-2/1812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 14±2 µM48-hCervixNone
3647
221002262012
GMWSKILGHLIR
HAL-1/2912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 > 100 µM48-hCervixNone
3648
221002262012
GMWSKLLGHLLR
HAL-1/1512LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 14±2 µM48-hCervixNone
3649
221002262012
GKWMSLLKHILK
HAL-212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 12±1 µM48-hCervixNone
3650
221002262012
gkwmsllkhilk
HAL-2/2212LinearDNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 12 µM48-hCervixNone
3651
221002262012
GKWMSLLKKILK
HAL-2/412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 > 40 µM48-hCervixNone
3645
221002262012
GKWKKILGHLIR
HAL-1/1912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 > 100 µM48-hCervixNone
3646
221002262012
GKWKKILGKLIR
HAL-1/2112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 30±3 µM48-hCervixNone
3644
221002262012
GKWSKILGKLIR
HAL-1/2012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 22±3 µM48-hCervixNone
3643
221002262012
GMWKKILGKLIR
HAL-1/1012LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 13±2 µM48-hCervixNone
3642
221002262012
KMWSKILGHLIR
HAL-1/1712LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 35±3 µM48-hCervixNone
3640
221002262012
GMWKKILGHLIR
HAL-1/512LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 9±1 µM48-hCervixNone
3641
221002262012
GKWSKILGHLIR
HAL-1/1212LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 43±14 µM48-hCervixNone
3639
221002262012
GMWSKILKHLIR
HAL-1/1812LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 4±2 µM48-hCervixNone
3638
221002262012
GMWSKILGKLIR
HAL-1/912LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 9±1 µM48-hCervixNone
3637
221002262012
GMWSKILGHLKR
HAL-1/412LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 > 100 µM48-hCervixNone
3636
221002262012
GMWSKILGHLIK
HAL-1/612LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 15±1 µM48-hCervixNone
3634
221002262012
GMWSKILGHLIR
HAL-112LinearLNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 11±2 µM48-hCervixNone
3635
221002262012
gmwskilghlir
HAL-1/2212LinearDNoneAmidationFreeAntimicrobial and AntifungalHalictines and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 15±3 µM48-hCervixNone
3633
221002262012
GFGMA-(AC6C)-KLLKKVL
MAC1/2613LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 9±2 µM48-hBloodNone
3631
221002262012
GFGMALKL-(AC6C)-KKVL
MAC1/2413LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 11 µM48-hBloodNone
3632
221002262012
GFGMALK-(AC6C)-LKKVL
MAC1/2513LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 12±2 µM48-hBloodNone
3630
221002262012
GFGMALRLLRRVL
MAC1/2113LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 22±4 µM48-hBloodNone
3629
221002262012
GFGMALOLLOOVL
MAC1/2013LinearLO = OrnithineAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 25±3 µM48-hBloodNone
3628
221002262012
GFGMALKLLKKVL
MAC1/1913LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 43±11 µM48-hBloodNone
3626
221002262012
GFKMALKLLKKVL
MAC1/1013LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 16 µM48-hBloodNone
3627
221002262012
GFGMALKLLKKVL
MAC1/1613LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 70 µM48-hBloodNone
3625
221002262012
GFKMALKLLKKVL
MAC1/913LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 14±4 µM48-hBloodNone
3624
221002262012
GFGMALKLLKKVL
MAC1/613LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 15 µM48-hBloodNone
3622
221002262012
LFGMALKLLKKVL
MAC1/313LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 22 µM48-hBloodNone
3623
221002262012
GFGMALKLLKKVL
MAC1/413LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 29 µM48-hBloodNone
3621
221002262012
AFGMALKLLKKVL
MAC1/213LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 17 µM48-hBloodNone
3620
221002262012
gfgmalkllkkvl
MAC1/113LinearDNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 11 µM48-hBloodNone
3619
221002262012
GTGLPMSERRKIMLMMR
MAC217LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 32 µM48-hBloodNone
3616
221002262012
GFGMALK-(AC6C)-LKKVL
MAC1/2513LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 14±1 µM48-hColonNone
3617
221002262012
GFGMA-(AC6C)-KLLKKVL
MAC1/2613LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 18±1 µM48-hColonNone
3618
221002262012
GFGMALKLLKKVL
MAC113LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 12±6 µM48-hBloodNone
3615
221002262012
GFGMALKL-(AC6C)-KKVL
MAC1/2413LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 16±1 µM48-hColonNone
3613
221002262012
GFGMALOLLOOVL
MAC1/2013LinearLO = OrnithineAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 35±4 µM48-hColonNone
3614
221002262012
GFGMALRLLRRVL
MAC1/2113LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 17±2 µM48-hColonNone
3612
221002262012
GFGMALKLLKKVL
MAC1/1913LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 68±2 µM48-hColonNone
3611
221002262012
GFGMALKLLKKVL
MAC1/1613LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3610
221002262012
GFKMALKLLKKVL
MAC1/1013LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3609
221002262012
GFKMALKLLKKVL
MAC1/913LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 13±3 µM48-hColonNone
3607
221002262012
GFGMALKLLKKVL
MAC1/413LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 49±9 µM48-hColonNone
3608
221002262012
GFGMALKLLKKVL
MAC1/613LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 29±3 µM48-hColonNone
3606
221002262012
LFGMALKLLKKVL
MAC1/313LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 11±1 µM48-hColonNone
3604
221002262012
gfgmalkllkkvl
MAC1/113LinearDNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 19±2 µM48-hColonNone
3605
221002262012
AFGMALKLLKKVL
MAC1/213LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 16 µM48-hColonNone
3603
221002262012
GTGLPMSERRKIMLMMR
MAC217LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3601
221002262012
GFGMA-(AC6C)-KLLKKVL
MAC1/2613LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 8±2 µM48-hCervixNone
3602
221002262012
GFGMALKLLKKVL
MAC113LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsSWColon CancerMTT/MTS assayIC50 = 23±4 µM48-hColonNone
3599
221002262012
GFGMALKL-(AC6C)-KKVL
MAC1/2413LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 8±2 µM48-hCervixNone
3600
221002262012
GFGMALK-(AC6C)-LKKVL
MAC1/2513LinearLAC6C = cyclohexyl-1-carboxylic acidAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 7±1 µM48-hCervixNone
3597
221002262012
GFGMALOLLOOVL
MAC1/2013LinearLO = OrnithineAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 10±1 µM48-hCervixNone
3598
221002262012
GFGMALRLLRRVL
MAC1/2113LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 9±3 µM48-hCervixNone
3595
221002262012
GFGMALKLLKKVL
MAC1/1613LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 32±2 µM48-hCervixNone
3596
221002262012
GFGMALKLLKKVL
MAC1/1913LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 21±4 µM48-hCervixNone
3594
221002262012
GFKMALKLLKKVL
MAC1/1013LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 15±6 µM48-hCervixNone
3592
221002262012
GFGMALKLLKKVL
MAC1/613LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 8±2 µM48-hCervixNone
3593
221002262012
GFKMALKLLKKVL
MAC1/913LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 8±1 µM48-hCervixNone
3591
221002262012
GFGMALKLLKKVL
MAC1/413LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 15±5 µM48-hCervixNone
3589
221002262012
AFGMALKLLKKVL
MAC1/213LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 16±3 µM48-hCervixNone
3590
221002262012
LFGMALKLLKKVL
MAC1/313LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 9±2 µM48-hCervixNone
3588
221002262012
gfgmalkllkkvl
MAC1/113LinearDNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 12±4 µM48-hCervixNone
3587
221002262012
GTGLPMSERRKIMLMMR
MAC217LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 > 100 µM48-hCervixNone
3586
221002262012
GFGMALKLLKKVL
MAC113LinearLNoneAmidationFreeAntimicrobial and AntifungalMacropins and their analogsHeLaCervical CancerMTT/MTS assayIC50 = 10±4 µM48-hCervixNone
3569
221002262012
VNWKKILGKIIKVVK
LL-III/3715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50= 4±1 µM48-hBloodNone
3567
221002262012
NKWKKILGKIIKVVK
LL-III/3415LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 5±3 µM48-hBloodNone
3568
221002262012
VNWKKILAKIIKVVK
LL-III/3615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3566
221002262012
VNWKKVLGKVVKVVK
LL-III/2715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 18 µM48-hBloodNone
3565
221002262012
VYWKKILGKIIKVVK
LL-III/2615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 6 µM48-hBloodNone
3563
221002262012
VNWOOILGOIIOVVO
LL-III/2415LinearLO = OrnithineAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 5±2 µM48-hBloodNone
3564
221002262012
vnwkkllgkllkvvk
LL-III/2515LinearDNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 4 µM48-hBloodNone
3562
221002262012
VNWKKLLGKLLKVVK
LL-III/2315LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 6 µM48-hBloodNone
3561
221002262012
KNWKK-Aib-LKK-Aib-IK-Aib-VK
LL-III/2215LinearLAib = 1-amino-isobutyric acidAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 25±4 µM48-hBloodNone
3560
221002262012
VNWKK-Aib-LGK-Aib-IK-Aib-VK
LL-III/1915LinearLAib = 1-amino-isobutyric acidAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 8±2 µM48-hBloodNone
3559
221002262012
KNWKKILKKIIKVVK
LL-III/1815LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 7±2 µM48-hBloodNone
3558
221002262012
VNWRRILGRIIRVVR
LL-III/1715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3557
221002262012
VN-Nal-KKLLGKLLKVVK
LL-III/1615LinearLNal = 3-(1-naphthyl)alanineAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3556
221002262012
VNFKKLLGKLLKVVK
LL-III/1515LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 9±3 µM48-hBloodNone
3555
221002262012
vnwkkilgkiikvvk
LL-III/1215LinearDNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 5±2 µM48-hBloodNone
3554
221002262012
VNWKKIILGKIIKVVK
LL-III/1115LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 4±1 µM48-hBloodNone
3552
221002262012
VNWKKILGKIIKVVK
LL-III/915LinearLNoneMethoxylationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3553
221002262012
KNWKKILGKIIKVVK
LL-III/1015LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 9 µM48-hBloodNone
3551
221002262012
VNWKKILGKIIKVVK
LL-III/815LinearLNoneFreeFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 9 µM48-hBloodNone
3549
221002262012
VNWKKILGKIKKVVK
LL-III/415LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 18 µM48-hBloodNone
3550
221002262012
VNWKKILPKIIKVVK
LL-III/615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 6±3 µM48-hBloodNone
3548
221002262012
VNWKKILKKIIKVVK
LL-III/315LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayNot tested48-hBloodNone
3547
221002262012
NVWKKILGKIIKVVK
LL-III/215LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 7±2 µM48-hBloodNone
3545
221002262012
VNWKKILGKIIKVVK
LL-III15LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 5±3 µM48-hBloodNone
3546
221002262012
VNWKKILAKIIKVVK
LL-III/115LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsCCRF-CEMLeukemia CancerMTT/MTS assayIC50 = 3±1 µM48-hBloodNone
3544
221002262012
VNWKKILGKIIKVVK
LL-III/3715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 13 µM48-hColonNone
3542
221002262012
NKWKKILGKIIKVVK
LL-III/3415LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 37 µM48-hColonNone
3543
221002262012
VNWKKILAKIIKVVK
LL-III/3615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3541
221002262012
VNWKKVLGKVVKVVK
LL-III/2715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3539
221002262012
vnwkkllgkllkvvk
LL-III/2515LinearDNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 20 µM48-hColonNone
3540
221002262012
VYWKKILGKIIKVVK
LL-III/2615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 30 µM48-hColonNone
3538
221002262012
VNWOOILGOIIOVVO
LL-III/2415LinearLO = OrnithineAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 20 µM48-hColonNone
3537
221002262012
VNWKKLLGKLLKVVK
LL-III/2315LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 15 µM48-hColonNone
3535
221002262012
VNWKK-Aib-LGK-Aib-IK-Aib-VK
LL-III/1915LinearLAib = 1-amino-isobutyric acidAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 28 µM48-hColonNone
3536
221002262012
KNWKK-Aib-LKK-Aib-IK-Aib-VK
LL-III/2215LinearLAib = 1-amino-isobutyric acidAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 > 100 µM48-hColonNone
3534
221002262012
KNWKKILKKIIKVVK
LL-III/1815LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3533
221002262012
VNWRRILGRIIRVVR
LL-III/1715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3532
221002262012
VN-Nal-KKLLGKLLKVVK
LL-III/1615LinearLNal = 3-(1-naphthyl)alanineAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3531
221002262012
VNFKKLLGKLLKVVK
LL-III/1515LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 42 µM48-hColonNone
3530
221002262012
vnwkkilgkiikvvk
LL-III/1215LinearDNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 20 µM48-hColonNone
3528
221002262012
KNWKKILGKIIKVVK
LL-III/1015LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3529
221002262012
VNWKKIILGKIIKVVK
LL-III/1115LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 48 µM48-hColonNone
3527
221002262012
VNWKKILGKIIKVVK
LL-III/915LinearLNoneMethoxylationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 25± 5 µM48-hColonNone
3525
221002262012
VNWKKILPKIIKVVK
LL-III/615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3526
221002262012
VNWKKILGKIIKVVK
LL-III/815LinearLNoneFreeFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayNot tested48-hColonNone
3524
221002262012
VNWKKILGKIKKVVK
LL-III/415LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3522
221002262012
NVWKKILGKIIKVVK
LL-III/215LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 11 µM48-hColonNone
3523
221002262012
VNWKKILKKIIKVVK
LL-III/315LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 > 40 µM48-hColonNone
3521
221002262012
VNWKKILAKIIKVVK
LL-III/115LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 12± 3 µM48-hColonNone
3519
221002262012
VNWKKILGKIIKVVK
LL-III/3715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 5±1 µM48-hColonNone
3520
221002262012
VNWKKILGKIIKVVK
LL-III15LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsSWColon CancerMTT/MTS assayIC50 = 18±4 µM48-hColonNone
3518
221002262012
VNWKKILAKIIKVVK
LL-III/3615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 8 µM48-hCervixNone
3516
221002262012
VNWKKVLGKVVKVVK
LL-III/2715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 13±2 µM48-hCervixNone
3517
221002262012
NKWKKILGKIIKVVK
LL-III/3415LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 5±2 µM48-hCervixNone
3515
221002262012
VYWKKILGKIIKVVK
LL-III/2615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 5±1 µM48-hCervixNone
3513
221002262012
VNWOOILGOIIOVVO
LL-III/2415LinearLO = OrnithineAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 3±1 µM48-hCervixNone
3514
221002262012
vnwkkllgkllkvvk
LL-III/2515LinearDNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 4±2 µM48-hCervixNone
3512
221002262012
VNWKKLLGKLLKVVK
LL-III/2315LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 4 µM48-hCervixNone
3511
221002262012
KNWKK-Aib-LKK-Aib-IK-Aib-VK
LL-III/2215LinearLAib = 1-amino-isobutyric acidAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 11±7 µM48-hCervixNone
3509
221002262012
KNWKKILKKIIKVVK
LL-III/1815LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 3 µM48-hCervixNone
3510
221002262012
VNWKK-Aib-LGK-Aib-IK-Aib-VK
LL-III/1915LinearLAib = 1-amino-isobutyric acidAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 3±1 µM48-hCervixNone
3508
221002262012
VNWRRILGRIIRVVR
LL-III/1715LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50= 9 µM48-hCervixNone
3505
221002262012
vnwkkilgkiikvvk
LL-III/1215LinearDNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 6±2 µM48-hCervixNone
3506
221002262012
VNFKKLLGKLLKVVK
LL-III/1515LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 7±1 µM48-hCervixNone
3507
221002262012
VN-Nal-KKLLGKLLKVVK
LL-III/1615LinearLNal = 3-(1-naphthyl)alanineAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 6±1 µM48-hCervixNone
3502
221002262012
VNWKKILGKIIKVVK
LL-III/915LinearLNoneMethoxylationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 3±1 µM48-hCervixNone
3503
221002262012
KNWKKILGKIIKVVK
LL-III/1015LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 9±4 µM48-hCervixNone
3504
221002262012
VNWKKIILGKIIKVVK
LL-III/1115LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 8±1 µM48-hCervixNone
3499
221002262012
VNWKKILGKIKKVVK
LL-III/415LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 7±1 µM48-hCervixNone
3500
221002262012
VNWKKILPKIIKVVK
LL-III/615LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 > 40 µM48-hCervixNone
3501
221002262012
VNWKKILGKIIKVVK
LL-III/815LinearLNoneFreeFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 12±1 µM48-hCervixNone
3497
221002262012
NVWKKILGKIIKVVK
LL-III/215LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayNot tested48-hCervixNone
3498
221002262012
VNWKKILKKIIKVVK
LL-III/315LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayNot tested48-hCervixNone
3495
221002262012
VNWKKILGKIIKVVK
LL-III15LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 4±1 µM48-hCervixNone
3496
221002262012
VNWKKILAKIIKVVK
LL-III/115LinearLNoneAmidationFreeAntimicrobial and AntifungalLasioglossin III and its analogsHeLaCervical CancerMTT/MTS assayIC50 = 3±1 µM48-hCervixNone
3468
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay~30% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3469
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay>40% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3466
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay<20% cytotoxicity at 1 µM48-hBladderWO_2012042540_A2
3467
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay20% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3464
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay40% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3465
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay~50% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3462
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3463
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3460
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 1 µM48-hBladderWO2012042540A2
3461
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<3% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3458
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<15% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3459
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay~15% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3456
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<20% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3457
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay~15% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3454
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 1 µM48-hBladderWO_2012042540_A2
3455
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<3% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3452
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay20% cytotoxicity at 1 µM24-hBladderWO2012042540A2
3453
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay~10% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3450
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3451
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~45% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3449
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~55% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3447
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~40% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3448
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3445
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay>20% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3446
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3443
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3444
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~15% cytotoxicity at 1 µM72-hCervixWO2012042540A2
3441
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~15% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3442
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay<3% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3439
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay20% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3440
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~5% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3437
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay<10% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3438
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay<20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3435
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~5% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3436
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~10% cytotoxicity at 1 µM48-hCervixWO2012042540A2
3433
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay~45% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3434
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~15% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3432
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3431
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay~50% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3430
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay<20% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3429
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay>40% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3428
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay>20% cytotoxicity at 1 µM24-hCervixWO2012042540A2
3427
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay~40% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3426
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3425
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3424
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay<3% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3423
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay>10% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3422
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay5% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3421
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay20% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3420
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay<20% cytotoxicity at 1 µM72-hCervixWO2012042540A2
3419
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay<10% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3418
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay10% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3417
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay5% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3416
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay~15% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3415
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay~40% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3414
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay>30% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3413
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3412
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay<20% cytotoxicity at 1 µM48-hColonWO2012042540A2
3411
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay50% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3410
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay>40% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3409
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3408
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3407
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3406
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay~5% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3405
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay15% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3404
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<15% cytotoxicity at 1 µM24-hColonWO2012042540A2
3403
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay15% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3402
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<20% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3399
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay10% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3400
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3401
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<3% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3396
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay>40% cytotoxicity at 1 µM72-hBladderWO2012042540A2
3397
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay~50% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3398
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay20% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3395
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay~50% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3394
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay<30% cytotoxicity at 1 µM48-hBladderWO_2012042540_A2
3393
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay<30% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3392
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay~30% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3391
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay<45% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3390
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~45% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3389
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay>25% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3388
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 1 µM48-hBladderWO2012042540A2
3387
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3386
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3385
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay<45% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3384
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~45% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3383
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay<25% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3382
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 1 µM48-hBladderWO_2012042540_A2
3381
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay<10% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3380
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay10% cytotoxicity at 1 µM24-hBladderWO2012042540A2
3379
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay~20% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3378
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3377
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay~35% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3376
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay>20% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3375
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3374
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3373
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3372
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay>10% cytotoxicity at 1 µM72-hColonWO2012042540A2
3371
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay>10% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3370
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay10% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3369
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay~10% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3368
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3367
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3366
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3365
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3362
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3363
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<20% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3364
None2012
NHFTLKCPKTALTEPPTLAY
TG2020LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay~15% cytotoxicity at 1 µM48-hColonWO2012042540A2
3338
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =2.1 ± 0.1 µM2-hSkinNone
3339
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =1.8 ± 0.1 µM4-hSkinNone
3340
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =1.4 ± 0.1 µM24-hSkinNone
3341
235337102013
FKCRRWQWRMKK
LfcinB12LinearLNoneAmidationFreeAntihypertensive and Antimicrobial and Antiviral and AntioxidantBovine milkAZ-97Colon CancerMTT/MTS assayInhibition at 0.1g/lNAColonNone
3342
235337102013
YPFPG
β-Casomorphins 5 f(60_64)4LinearLNoneAmidationFreeImmunomodulant, Antihypertensive, Antimicrobial,Antiviral, and AntioxidantBovine milkAZ-97Colon CancerMTT/MTS assayInhibition at 9-11g/lNAColonNone
3343
235337102013
RYLGYL
αs1-casein f(90_95)6LinearLNoneAmidationFreeImmunomodulant, Antihypertensive, Antimicrobial,Antiviral, and AntioxidantBovine milkAZ-97Colon CancerMTT/MTS assayInhibition at 12-15g/lNAColonNone
3344
235337102013
PPPEE
Caseinphosphopeptides5LinearLNoneAmidationFreeImmunomodulant, Antihypertensive, Antimicrobial,Antiviral, and AntioxidantBovine milkAZ-97Colon CancerMTT/MTS assayInhibition at 24-28g/lNAColonNone
3345
228201492012
Structure Given
BAA-1Not AvailableLinearLNoneAmidationFreeAntimicrobialBovine lactoferrin (Lf-B)RamosLymphoma CancerMTT/MTS assayIC50 = 8.1 µg/ml1-hBloodNone
3346
228201492012
Structure Given
BAA-2Not AvailableLinearLNoneAmidationFreeAntimicrobialBovine lactoferrin (Lf-B)RamosLymphoma CancerMTT/MTS assayIC50 = 3.8 µg/ml8-hBloodNone
3329
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =7.5 ± 0.4 µM30-MinSkinNone
3330
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =13.8 ± 2.0 µM2-hSkinNone
3331
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =9.3 ± 1.5 µM4-hSkinNone
3332
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =13.1 ± 0.9 µM24-hSkinNone
3333
238936052013
KISKRILTGKK
NK1111LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 >>100 µM30-MinSkinNone
3334
238936052013
KISKRILTGKK
NK1111LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 >>100 µM2-hSkinNone
3335
238936052013
KISKRILTGKK
NK1111LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 >>100 µM4-hSkinNone
3336
238936052013
KISKRILTGKK
NK1111LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 >>100 µM24-hSkinNone
3337
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =3.2 ± 0.1 µM30-MinSkinNone
3328
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =12.3 ± 1.0 µM24-hSkinNone
3327
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =8.3 ± 0.5 µM4-hSkinNone
3326
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =12.3 ± 2.0 µM2-hSkinNone
3325
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =8.4 ± 0.2 µM30-MinSkinNone
3324
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =37 ± 4.3 µM24-hSkinNone
3323
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =12.1 ± 1.6 µM4-hSkinNone
3322
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =13.0 ± 1.0 µM2-hSkinNone
3321
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =10.6 ± 0.4 µM30-MinSkinNone
3320
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~40 µM24-hSkinNone
3319
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~50 µM4-hSkinNone
3318
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~50 µM2-hSkinNone
3317
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~70 µM30-MinSkinNone
3316
21453492, 235337102011
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAntimicrobial and AnticancerBovine lactoferrin (Lf-B)KellyBrain TumorMTT/MTS assayIC50 =141 ± 3 µM30-MinBrainNone
3315
21453492, 235337102011
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAntimicrobial and AnticancerBovine lactoferrin (Lf-B)MT-1Breast CancerMTT/MTS assayIC50 > 160 µM30-MinBreastNone
3313
214534922011
OOW-Dip-OOWWO
LTX-3189LinearLDip = diphenylalanine, O=ornithineAmidationFreeAntimicrobialSynthetic peptideKellyBrain TumorMTT/MTS assayIC50 =78 ± 7 µM30-MinBrainNone
3314
21453492, 235337102011
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAntimicrobial and AnticancerBovine lactoferrin (Lf-B)HT-29Colon CancerMTT/MTS assayIC50 > 160 µM30-MinColonNone
3312
214534922011
OOW-Dip-OOWWO
LTX-3189LinearLDip = diphenylalanine, O=ornithineAmidationFreeAntimicrobialSynthetic peptideMT-1Breast CancerMTT/MTS assayIC50 =216 ± 36 µM30-MinBreastNone
3311
214534922011
OOW-Dip-OOWWO
LTX-3189LinearLDip = diphenylalanine, O=ornithineAmidationFreeAntimicrobialSynthetic peptideHT-29Colon CancerMTT/MTS assayIC50 =248 ± 5 µM30-MinColonNone
3309
214534922011
KKWWKKW-Dip-K
LTX-3159LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideMT-1Breast CancerMTT/MTS assayIC50 =31 ± 3 µM30-MinBreastNone
3310
214534922011
KKWWKKW-Dip-K
LTX-3159LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideKellyBrain TumorMTT/MTS assayIC50 =14 ± 1 µM30-MinBrainNone
3308
214534922011
KKWWKKW-Dip-K
LTX-3159LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideHT-29Colon CancerMTT/MTS assayIC50 =38 ± 3 µM30-MinColonNone
3307
214534922011
WKKW-Dip-KKWK
LTX-3029LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideKellyBrain TumorMTT/MTS assayIC50 =28 ± 0 µM30-MinBrainNone
3306
214534922011
WKKW-Dip-KKWK
LTX-3029LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideMT-1Breast CancerMTT/MTS assayIC50 =73 ± 2 µM30-MinBreastNone
3305
214534922011
WKKW-Dip-KKWK
LTX-3029LinearLDip = diphenylalanineAmidationFreeAntimicrobialSynthetic peptideHT-29Colon CancerMTT/MTS assayIC50 =75 ± 5 µM30-MinColonNone
3267
229346012012
FLGALFKALSHLL
PTP-7b13LinearLNoneFreeFreeAnticancerSynthetic peptideA-549Lung CancerMTT/MTS assayIC50 =32 µMNALungNone
3266
229346012012
FLGALFHALSKLL
PTP-7a13LinearLNoneFreeFreeAnticancerSynthetic peptideA-549Lung CancerMTT/MTS assayIC50 =28 µMNALungNone
3265
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<40% cell viability at 50 µMNAStomachNone
3264
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay100% cell viability at 5 µMNAStomachNone
3263
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<60% cell viability at 50 µMNABloodNone
3262
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µMNABloodNone
3261
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay60% cell viability at 50 µMNAColonNone
3260
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay>100% cell viability at 5 µMNAColonNone
3259
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<20% cell viability at 50 µMNAStomachNone
3258
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<100% cell viability at 5 µMNAStomachNone
3257
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<40% cell viability at 50 µMNABloodNone
3256
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µMNABloodNone
3255
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay40% cell viability at 50 µMNAColonNone
3254
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay100% cell viability at 5 µMNAColonNone
3253
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50 =12.55 µM72-hOvaryNone
3252
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50 =22.25 µM72-hSkinNone
3251
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50 =29.10 µM72-hProstateNone
3250
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50 =22.51 µM72-hStomachNone
3249
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50 =14.80 µM72-hColonNone
3248
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-549Lung CancerMTT/MTS assayIC50 =14.53 µM72-hLungNone
3247
226448472012
FLKWLFKWAKK
GA-K411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-498Renal CancerMTT/MTS assayIC50 =21.48 µM72-hRenalNone
3246
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC5072-hOvaryNone
3245
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50 =27.39 µM72-hSkinNone
3244
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50 =47.69 µM72-hProstateNone
3242
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50 =27.00 µM72-hColonNone
3243
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50 =26.70 µM72-hStomachNone
3240
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-498Renal CancerMTT/MTS assayIC50 =41.21 µM72-hRenalNone
3241
226448472012
FLGWLFKWAKK
GA-K311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-549Lung CancerMTT/MTS assayIC50 =25.20 µM72-hLungNone
3238
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50 =13.16 µM72-hSkinNone
3239
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50 =14.58 µM72-hOvaryNone
3235
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50 =14.80 µM72-hColonNone
3236
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50 =13.77 µM72-hStomachNone
3237
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50 =24.32 µM72-hProstateNone
3233
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-498Renal CancerMTT/MTS assayIC50 =22.59 µM72-hRenalNone
3234
226448472012
FLWWLFKWAWK
GA-W411LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-549Lung CancerMTT/MTS assayIC50 =15.88 µM72-hLungNone
3232
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-OV-3Ovarian CancerMTT/MTS assayIC50 =22.06 µM72-hOvaryNone
3230
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaPC-3Prostate CancerMTT/MTS assayIC50 =46.51 µM72-hProstateNone
3231
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaSK-MEL-2Skin CancerMTT/MTS assayIC50 =13.97 µM72-hSkinNone
3229
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaMKN-45Gastric CancerMTT/MTS assayIC50 =24.31 µM72-hStomachNone
3228
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaHCT-116Colon CancerMTT/MTS assayIC50 =24.63 µM72-hColonNone
3227
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-549Lung CancerMTT/MTS assayIC50 =20.36 µM72-hLungNone
3226
226448472012
FLGWLFKWAWK
GA-W311LinearLNoneAmidationFreeAntimicrobialUndecapeptide analogues derived from Brevinin-1EMaA-498Renal CancerMTT/MTS assayIC50 =22.88 µM72-hRenalNone
3225
224138592012
KVKVKVKVPPTKVKVKVK
SVS-218LinearLNoneAmidationFreeAntimicrobialSynthetic peptideMDA-MB-436Breast CancerMTT/MTS assayIC50 >100 µM24-hBreastNone
3224
224138592012
KVKVKVKVPPTKVKVKVK
SVS-218LinearLNoneAmidationFreeAntimicrobialSynthetic peptideMCF-7Breast CancerMTT/MTS assayIC50 >100 µM24-hBreastNone
3223
224138592012
KVKVKVKVPPTKVKVKVK
SVS-218LinearLNoneAmidationFreeAntimicrobialSynthetic peptideKBOral CancerMTT/MTS assayIC50 >100 µM24-hOral mucosaNone
3222
224138592012
KVKVKVKVPPTKVKVKVK
SVS-218LinearLNoneAmidationFreeAntimicrobialSynthetic peptideA-549Lung CancerMTT/MTS assayIC50 >100 µM24-hLungNone
3221
224138592012
kvkvkvkvPptkvkvkvk
D-SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideMDA-MB-436Breast CancerMTT/MTS assayIC50 =3.2±0.4 µM24-hBreastNone
3220
224138592012
kvkvkvkvPptkvkvkvk
D-SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideMCF-7Breast CancerMTT/MTS assayIC50 =4.7±0.4 µM24-hBreastNone
3219
224138592012
kvkvkvkvPptkvkvkvk
D-SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideKBOral CancerMTT/MTS assayIC50 =4.5±0.5 µM24-hOral mucosaNone
3218
224138592012
kvkvkvkvPptkvkvkvk
D-SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideA-549Lung CancerMTT/MTS assayIC50 =3.2±0.6 µM24-hLungNone
3217
224138592012
KVKVKVKVpPTKVKVKVK
SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideMDA-MB-436Breast CancerMTT/MTS assayIC50 =5.6±0.5 µM24-hBreastNone
3216
224138592012
KVKVKVKVpPTKVKVKVK
SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideMCF-7Breast CancerMTT/MTS assayIC50 =8.1±0.8 µM24-hBreastNone
3215
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3213
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3214
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3211
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3212
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3210
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIVeroRenal CancerMTT/MTS assayNA48-hRenalNone
3208
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IICEFTumorMTT/MTS assayNA48-hNot AvailableNone
3207
224138592012
KVKVKVKVpPTKVKVKVK
SVS-118LinearMixNoneAmidationFreeAntimicrobialBovine lactoferrin (Lf-B)KBOral CancerMTT/MTS assayNA24-hOral mucosaNone
3206
224138592012
KVKVKVKVpPTKVKVKVK
SVS-118LinearMixNoneAmidationFreeAntimicrobialSynthetic peptideA-549Lung CancerMTT/MTS assayNA24-hLungNone
3204
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3205
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3203
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3201
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3202
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIMDBKRenal CancerMTT/MTS assayNA48-hRenalNone
3198
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IICEFTumorMTT/MTS assayNA48-hNot AvailableNone
3200
221841212011
MTLTG
BPP-II5LinearLNoneFreeFreeAntitumorImmunomodulatory bursal-derived Pentapeptide-IIVeroRenal CancerMTT/MTS assayNA48-hRenalNone
3164
233015192013
RWRWRWRW
linear (RW)4-Dox8LinearLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPMDA-MB-468Breast CancerMTT/MTS assay60-74% antiproliferative activity at 1 µM72 to 120-hBreastNone
3163
233015192013
RWRWRWRW
linear (RW)4-Dox8LinearLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPHCT-116Colon CancerMTT/MTS assay21-61% antiproliferative activity at 1 µM72 to 120-hColonNone
3161
233015192013
RWRWRWRW
linear (RW)4-Dox8LinearLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPCCRF-CEMLeukemia CancerMTT/MTS assay46-69% antiproliferative activity at 1 µM72 to 120-hBloodNone
3162
233015192013
RWRWRWRW
linear (RW)4-Dox8LinearLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPSK-OV-3Ovarian CancerMTT/MTS assay28-34% antiproliferative activity at 1 µM72 to 120-hOvaryNone
3160
233015192013
WRWRWRWRW
Cyclic [W(RW)4 ]-Dox9CyclicLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPMDA-MB-468Breast CancerMTT/MTS assay60-79% inhibition of cell proliferation at 1 µM72 to 120-hBreastNone
3156
236274742013
CHHNLTAAC
PTPRJ-pep19.79Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay20 ± 1.4% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3157
233015192013
WRWRWRWRW
Cyclic [W(RW)4 ]-Dox9CyclicLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPCCRF-CEMLeukemia CancerMTT/MTS assay62-73% inhibition of cell proliferation at 1 µM72 to 120-hBloodNone
3158
233015192013
WRWRWRWRW
Cyclic [W(RW)4 ]-Dox9CyclicLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPSK-OV-3Ovarian CancerMTT/MTS assay51-74% inhibition of cell proliferation at 1 µM72 to 120-hOvaryNone
3159
233015192013
WRWRWRWRW
Cyclic [W(RW)4 ]-Dox9CyclicLDoxorubicin (Dox) which is anthracycline attached with linker to CPP [W(RW)4 ]FreeFreeAnticancerDoxorubicin (Dox) is a well-known anthracycline which has been conjugated to a CPPHCT-116Colon CancerMTT/MTS assay50-67% inhibition of cell proliferation at 1 µM72 to 120-hColonNone
3152
236274742013
CHHNATHAC
PTPRJ-pep19.59Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay2 ± 1.5% cell growth inhibition at 160 µM in 48 hours48-hCervixNone
3153
236274742013
CHHNATHAC
PTPRJ-pep19.59Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay19 ± 4.2% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3154
236274742013
CHHNLAHAC
PTPRJ-pep19.69Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay19 ± 4.2% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3155
236274742013
CHHNLTAAC
PTPRJ-pep19.79Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay4.5 ± 2.13% cell growth inhibition at 160 µM in 48 hours48-hCervixNone
3148
236274742013
CHANLTHAC
PTPRJ-pep19.39Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay51 ± 1.4% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3149
236274742013
CHHALTHAC
PTPRJ-pep19.49Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay48.0 ± 2.82% cell growth inhibition at 160 µM in 24 hours24-hCervixNone
3150
236274742013
CHHALTHAC
PTPRJ-pep19.49Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay62.5 ± 4.9% cell growth inhibition at 160 µM in 48 hours48-hCervixNone
3151
236274742013
CHHALTHAC
PTPRJ-pep19.49Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay66.5 ± 2.12% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3144
236274742013
CAHNLTHAC
PTPRJ-pep19.29Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay30 ± 2.82% cell growth inhibition at 160 µM in 48 hours48-hCervixNone
3145
236274742013
CAHNLTHAC
PTPRJ-pep19.29Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay32.0 ± 4.2% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3146
236274742013
CHANLTHAC
PTPRJ-pep19.39Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay28 ± 5.5% cell growth inhibition at 160 µM in 24 hours24-hCervixNone
3147
236274742013
CHANLTHAC
PTPRJ-pep19.39Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay46 ± 4.2% cell growth inhibition at 160 µM in 48 hours48-hCervixNone
3140
236274742013
CHHNLTHAC
PTPRJ-pep199Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay4.5 ± 0.1.4% cell growth inhibition at 160 µM in 48 hours48-hCervixNone
3141
236274742013
CHHNLTHAC
PTPRJ-pep199Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay19 ± 2.82% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3142
236274742013
CHHNLTHAC
PTPRJ-pep19.09LinearLNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay4 ± 1.4% cell growth inhibition at 160 µM in 72 hours72-hCervixNone
3143
236274742013
CAHNLTHAC
PTPRJ-pep19.29Cyclic(C1-C9)LNoneFreeFreeAnticancerPTPRJ agonist peptidesHeLaCervical CancerTrypan blue assay16.5 ± 2.12% cell growth inhibition at 160 µM in 24 hours24-hCervixNone
3137
237704402013
FLGMIPKLIKKLIKAFK
TsAP-S217LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideMCF-7Breast CancerMTT/MTS assayIC50 = 1.8 µM24-hBreastNone
3138
237704402013
FLGMIPKLIKKLIKAFK
TsAP-S217LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptidePC-3Prostate CancerMTT/MTS assayIC50 = 1.6 µM24-hProstateNone
3139
237704402013
FLGMIPKLIKKLIKAFK
TsAP-S217LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideU251-MGBrain TumorMTT/MTS assayIC50 = 2.0 µM24-hBrainNone
3135
237704402013
FLGMIPKLIKKLIKAFK
TsAP-S217LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideHI-57Lung CancerMTT/MTS assayIC50 = 0.83 µM24-hLungNone
3136
237704402013
FLGMIPKLIKKLIKAFK
TsAP-S217LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideH-838Lung CancerMTT/MTS assayIC50 = 1.6 µM24-hLungNone
3132
237704402013
FLSLIPKLVKKIIKAFK
TsAP-S117LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideMCF-7Breast CancerMTT/MTS assayIC50 = 1.8 µM24-hBreastNone
3133
237704402013
FLSLIPKLVKKIIKAFK
TsAP-S117LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptidePC-3Prostate CancerMTT/MTS assayIC50 = 2.1 µM24-hProstateNone
3134
237704402013
FLSLIPKLVKKIIKAFK
TsAP-S117LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideU251-MGBrain TumorMTT/MTS assayIC50 = 2.9 µM24-hBrainNone
3129
237704402013
FLGMIPGLIGGLISAFK
TsAP-217LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusU251-MGBrain TumorMTT/MTS assayIC50 = 15.4 µM24-hBrainNone
3130
237704402013
FLSLIPKLVKKIIKAFK
TsAP-S117LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideHI-57Lung CancerMTT/MTS assayIC50 = 1.5 µM24-hLungNone
3131
237704402013
FLSLIPKLVKKIIKAFK
TsAP-S117LinearLNoneAmidationFreeAntimicrobialDerivative of TsAP-1, Brazilian yellow scorpion venom peptideH-838Lung CancerMTT/MTS assayIC50 = 1.6 µM24-hLungNone
3126
237704402013
FLGMIPGLIGGLISAFK
TsAP-217LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusH-838Lung CancerMTT/MTS assayIC50 = 11.0 µM24-hLungNone
3127
237704402013
FLGMIPGLIGGLISAFK
TsAP-217LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusMCF-7Breast CancerMTT/MTS assayIC50 = 6.4 µM24-hBreastNone
3128
237704402013
FLGMIPGLIGGLISAFK
TsAP-217LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusPC-3Prostate CancerMTT/MTS assayIC50 = 13.3 µM24-hProstateNone
3123
237704402013
FLSLIPSLVGGSISAFK
TsAP-117LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusHI-57Lung CancerMTT/MTS assayIC50 =55.9 µM24-hLungNone
3124
237704402013
FLSLIPSLVGGSISAFK
TsAP-117LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusH-838Lung CancerMTT/MTS assayIC50 =52.5 µM24-hLungNone
3125
237704402013
FLGMIPGLIGGLISAFK
TsAP-217LinearLNoneAmidationFreeAntimicrobialVenom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatusHI-57Lung CancerMTT/MTS assayIC50 = 4.1 µM24-hLungNone
3120
239933312013
KRLRRVWRRWR
MAP-04-0411LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability >80% at 75 µM48-hBreastNone
3121
239933312013
KRLRRVWRRWR
MAP-04-0411LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability >80% at 100 µM48-hBreastNone
3122
239933312013
KWLRRVWRWWR
MAP-04-0311LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayIC50=61.5 µM48-hBreastNone
3116
239933312013
KWLRRVWRWWR
MAP-04-0311LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability <40% at 75 µM48-hBreastNone
3117
239933312013
KWLRRVWRWWR
MAP-04-0311LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability >20% at 100 µM48-hBreastNone
3118
239933312013
KWLRRVWRWWR
MAP-04-0311LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability ~100% at 25 µM48-hBreastNone
3119
239933312013
KRLRRVWRRWR
MAP-04-0411LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability >80% at 50 µM48-hBreastNone
3114
239933312013
KWLRRVWRWWR
MAP-04-0311LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability >80% at 25 µM48-hBreastNone
3115
239933312013
KWLRRVWRWWR
MAP-04-0311LinearLNoneAmidationFreeAntimicrobialAnalogs of Ixosin-B amideMCF-7Breast CancerMTT/MTS assayCell viability ~50% at 50 µM48-hBreastNone
3112
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<100% cell viability at 5 µM24-hStomachNone
3113
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<40% cell viability at 50 µM24-hStomachNone
3109
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay60% cell viability at 50 µM24-hColonNone
3110
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µM24-hBloodNone
3111
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<60% cell viability at 50 µM24-hBloodNone
3108
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay>100% cell viability at 5 µM24-hColonNone
3107
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<20% cell viability at 50 µM24-hStomachNone
3106
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<100% cell viability at 5 µM24-hStomachNone
3105
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<40% cell viability at 50 µM24-hBloodNone
3104
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µM24-hBloodNone
3103
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay40% cell viability at 50 µM24-hColonNone
3102
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay100% cell viability at 5 µM24-hColonNone
3071
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
3070
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay1 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
3069
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay20 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
3068
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
3067
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
3066
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay15 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
3065
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
3064
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
3063
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
3062
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
3061
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
3060
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
3059
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay48 % Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
3058
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay84% Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
3057
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay84 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
3056
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay25 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
3055
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
3054
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay45 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
3053
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
3052
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay80 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
3051
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 3.125 mg/L24-hCervixNone
3050
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 6.25 mg/L24-hCervixNone
3049
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 12.5 mg/L24-hCervixNone
3048
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay82 % Cytotoxicity at 25 mg/L24-hCervixNone
3047
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hCervixNone
3046
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L12-hCervixNone
3045
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 6.25 mg/L12-hCervixNone
3044
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 12.5 mg/L12-hCervixNone
3043
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L12-hCervixNone
3042
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay82 % Cytotoxicity at 50 mg/L12-hCervixNone
3041
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 3.125 mg/L6-hCervixNone
3040
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 6.25 mg/L6-hCervixNone
3039
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 12.5 mg/L6-hCervixNone
3038
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L6-hCervixNone
3037
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay78 % Cytotoxicity at 50 mg/L6-hCervixNone
3036
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay1 % Cytotoxicity at 3.125 mg/L3-hCervixNone
3035
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 6.25 mg/L3-hCervixNone
3034
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 12.5 mg/L3-hCervixNone
3033
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay60 % Cytotoxicity at 25 mg/L3-hCervixNone
3032
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 50 mg/L3-hCervixNone
3031
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
3030
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay5 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
3028
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
3029
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay15 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
3027
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
3026
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay38 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
3024
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay39 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
3025
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay28 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
3023
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay95 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
3021
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
3022
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay97 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
3020
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
3019
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
3018
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
3017
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
3016
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
3015
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
3014
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay40 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
3013
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay82 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
3012
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay88 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
3011
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 3.125 mg/L24-hCervixNone
3010
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay12 % Cytotoxicity at 6.25 mg/L24-hCervixNone
3009
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay15 % Cytotoxicity at 12.5 mg/L24-hCervixNone
3008
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay80 % Cytotoxicity at 25 mg/L24-hCervixNone
3007
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hCervixNone
3006
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L12-hCervixNone
3005
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 6.25 mg/L12-hCervixNone
3004
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 12.5 mg/L12-hCervixNone
3003
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay68 % Cytotoxicity at 25 mg/L12-hCervixNone
3002
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay78 % Cytotoxicity at 50 mg/L12-hCervixNone
3001
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 3.125 mg/L6-hCervixNone
3000
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L6-hCervixNone
2999
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75 % Cytotoxicity at 50 mg/L6-hCervixNone
2998
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 12.5 mg/L3-hCervixNone
2997
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay44 % Cytotoxicity at 25 mg/L3-hCervixNone
2996
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay62 % Cytotoxicity at 50 mg/L3-hCervixNone
2994
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay3 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
2995
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay3 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
2993
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay8 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
2992
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay75 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
2990
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay4 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
2991
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
2989
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay4 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
2988
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay12 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
2986
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay76 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
2987
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay70 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
2985
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
2983
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay5 %Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
2984
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay7 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
2982
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay70 % Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
2980
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay5 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
2981
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay75 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
2979
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay10 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2978
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay8 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
2976
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay60 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
2977
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay50 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
2973
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay8 % Cytotoxicity at 12.5 mg/L24-hCervixNone
2974
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay3 % Cytotoxicity at 6.25 mg/L24-hCervixNone
2975
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay3 % Cytotoxicity at 3.125 mg/L24-hCervixNone
2972
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75 % Cytotoxicity at 25 mg/L24-hCervixNone
2970
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 3.125 mg/L12-hCervixNone
2971
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hCervixNone
2969
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 6.25 mg/L12-hCervixNone
2967
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L12-hCervixNone
2968
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay12 % Cytotoxicity at 12.5 mg/L12-hCervixNone
2965
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L6-hCervixNone
2966
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay76 % Cytotoxicity at 50 mg/L12-hCervixNone
2963
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 12.5 mg/L6-hCervixNone
2964
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay7 % Cytotoxicity at 6.25 mg/L6-hCervixNone
2962
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L6-hCervixNone
2961
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75 % Cytotoxicity at 50 mg/L6-hCervixNone
2959
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 6.25 mg/L3-hCervixNone
2960
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 3.125 mg/L3-hCervixNone
2958
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay8 % Cytotoxicity at 12.5 mg/L3-hCervixNone
2957
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay50 % Cytotoxicity at 25 mg/L3-hCervixNone
2956
235980792013
FIFHIIKGLFHAGKMI
Epinecidin-816LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay60 % Cytotoxicity at 50 mg/L3-hCervixNone
2955
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay28 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
2954
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
2952
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
2953
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay38 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
2951
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay84 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
2950
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay28 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
2949
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
2948
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay46 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
2947
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay96 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
2946
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay95 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
2945
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay25 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
2944
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay25 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
2943
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay45 % Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
2942
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay95 % Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
2941
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
2940
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2939
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2938
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2937
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay39 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
2936
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2935
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay42 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
2934
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
2933
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay82 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
2932
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay77 % Cytotoxicity at 25 mg/L24-hCervixNone
2931
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay83% Cytotoxicity at 50 mg/L24-hCervixNone
2930
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay65% Cytotoxicity at 25 mg/L12-hCervixNone
2929
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75 % Cytotoxicity at 50 mg/L12-hCervixNone
2928
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay65% Cytotoxicity at 25 mg/L6-hCervixNone
2927
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75% Cytotoxicity at 50 mg/L6-hCervixNone
2926
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay38% Cytotoxicity at 25 mg/L3-hCervixNone
2925
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay45% Cytotoxicity at 50 mg/L3-hCervixNone
2924
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)COLO-587Human epithelial CancerWST-1 assayIC50=6.4 µM72-hPancreaticNone
2923
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)LNCaPProstate CancerWST-1 assayIC50= 6.2 µM72-hProstateNone
2922
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)HuCCT-1Human epithelial CancerWST-1 assayIC50= 8.3 µM72-hBileductNone
2921
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)U-251Brain TumorWST-1 assayIC50=7.0 µM72-hBrainNone
2920
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SN-19Brain TumorWST-1 assayIC50= 7.8 µM72-hBrainNone
2919
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SF-295Brain TumorWST-1 assayIC50= 6.3 µM72-hBrainNone
2918
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)ZR75-1Breast CancerWST-1 assayIC50= 9.3 µM72-hBreastNone
2917
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)BT-20Breast CancerWST-1 assayIC50= 4.8 µM72-hBreastNone
2916
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)MDA-MB-231Breast CancerWST-1 assayIC50= 7.8 µM72-hBreastNone
2915
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SK-BR-3Breast CancerWST-1 assayIC50= 6.5 µM72-hBreastNone
2914
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)T-47DBreast CancerWST-1 assayIC50= 4.0 µM72-hBreastNone
2913
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)BT-474Breast CancerWST-1 assayIC50= 8.8 µM72-hBreastNone
2911
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)LNCaPProstate CancerWST-1 assayIC50= 15.8 µM72-hProstateNone
2912
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)COLO-587Human epithelial CancerWST-1 assayIC50= 13.5 µM72-hPancreaticNone
2910
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)HuCCT-1Human epithelial CancerWST-1 assayIC50= 17.1 µM72-hBileductNone
2909
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)U-251Brain TumorWST-1 assayIC50= 17.0 µM72-hBrainNone
2907
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SF-295Brain TumorWST-1 assayIC50= 19.1 µM72-hBrainNone
2908
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SN-19Brain TumorWST-1 assayIC50= 21.9 µM72-hBrainNone
2906
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)ZR75-1Breast CancerWST-1 assayIC50= 19.4 µM72-hBreastNone
2905
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)BT-20Breast CancerWST-1 assayIC50= 20.0 µM72-hBreastNone
2904
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)MDA-MB-231Breast CancerWST-1 assayIC50= 27.0 µM72-hBreastNone
2903
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SK-BR-3Breast CancerWST-1 assayIC50= 25.7 µM72-hBreastNone
2902
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)T-47DBreast CancerWST-1 assayIC50= 14.1 µM72-hBreastNone
2901
218490922011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)BT-474Breast CancerWST-1 assayIC50= 34.5 µM72-hBreastNone
2877
235835732013
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.Bcap-37Breast CancerMTT/MTS assay30 % Cell viability at 40 µM1-hBreastNone
2876
235835732013
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.Bcap-37Breast CancerMTT/MTS assay45% Cell viability at 30 µM1-hBreastNone
2874
235835732013
DEVD
caspase 3 inhibitor4LinearLNoneFluoromethyl ketone(fmk)FreeAnticancercaspase 3 inhibitorBcap-37Breast CancerMTT/MTS assay35 % Cell viability at 40 µM1-hBreastNone
2875
235835732013
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.Bcap-37Breast CancerMTT/MTS assay70% Cell viability at 20 µM1-hBreastNone
2872
235835732013
DEVD
caspase 3 inhibitor4LinearLNoneFluoromethyl ketone(fmk)FreeAnticancercaspase 3 inhibitorBcap-37Breast CancerMTT/MTS assay65% Cell viability at 20 µM1-hBreastNone
2873
235835732013
DEVD
caspase 3 inhibitor4LinearLNoneFluoromethyl ketone(fmk)FreeAnticancercaspase 3 inhibitorBcap-37Breast CancerMTT/MTS assay40% Cell viability at 30 µM1-hBreastNone
2868
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainMDA-MB-231Breast CancerWST-1 assayIC50=5.7 µMol/L24-hBreastNone
2867
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainH-322Lung CancerWST-1 assayIC50=3.6 µMol/L24-hLungNone
2866
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainA-172Brain TumorWST-1 assayIC50=6.8 µMol/L24-hBrainNone
2865
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainT98GBrain TumorWST-1 assayIC50=18.5 µMol/L24-hBrainNone
2864
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)KBOral CancerWST-1 assayIC50=13.2 µMol/L24-hOral mucosaNone
2863
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainSU.86.86Pancreatic CancerWST-1 assayIC50=7.5 µMol/L24-hPancreaticNone
2862
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainBXPC-3Pancreatic CancerWST-1 assayIC50=6.8 µMol/L24-hPancreaticNone
2861
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainMDA-MB-231Breast CancerWST-1 assayIC50=18.5 µMol/L24-hBreastNone
2860
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainH-322Lung CancerWST-1 assayIC50=27.1 µMol/L24-hLungNone
2859
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainA-172Brain TumorWST-1 assayIC50=30.5 µMol/L24-hBrainNone
2858
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainT98GBrain TumorWST-1 assayIC50=77.3 µMol/L24-hBrainNone
2857
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)KBOral CancerWST-1 assayIC50=37.4 µMol/L24-hOral mucosaNone
2856
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainSU.86.86Pancreatic CancerWST-1 assayIC50=28.0 µMol/L24-hPancreaticNone
2855
220841652011
KLlLKlLkkLLKlLKKK
Lytik17LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainBXPC-3Pancreatic CancerWST-1 assayIC50=37.1 µMol/L24-hPancreaticNone
2854
23577112, 218719462012
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.MCF-7Breast CancerLDH leakage assay32% Cytotoxicity at 40 µM1-hBreastNone
2853
23577112, 218719462012
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.MCF-7Breast CancerMTT/MTS assay61% Cell viability at 40 µM1-hBreastNone
2851
23577112, 218719462012
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.MDA-MB-231Breast CancerMTT/MTS assay22% Cell viability at 40 µM1-hBreastNone
2852
23577112, 218719462012
FVDLKKIANIINSIF
Tempoprin-1CEa15LinearLNoneAmidationFreeAntimicrobialChinese brown frog Rana chensinensis.MDA-MB-231Breast CancerLDH leakage assay61% Cytotoxicity at 40 µM1-hBreastNone
2850
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorRajiLymphoma CancerLDH leakage assayGI50 =2.57±0.75 µM24-hBloodNone
2849
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorMDA-MB-231Breast CancerLDH leakage assayGI50 =8.06±0.50 µM24-hBreastNone
2848
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorDU-145Liver CancerLDH leakage assayGI50 =0.91±0.04 µM24-hProstateNone
2847
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorLNCaPProstate CancerLDH leakage assayGI50 =0.31±0.15 µM24-hProstateNone
2846
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorPC-3Prostate CancerLDH leakage assayGI50 =1.24±0.23 µM24-hProstateNone
2844
242466472014
GIIKKIIKKIIKKIIKKI
Short α-helical peptides18LinearLNoneAmidationFreeAntimicrobialAlpha-helical proteinsHL-60Leukemia CancerMTT/MTS assay70% Cytotoxicity at 5 µM Approx24-hBloodNone
2843
242466472014
GIIKKIIKKIIKKI
Short α-helical peptides14LinearLNoneAmidationFreeAntimicrobialAlpha-helical proteinsHL-60Leukemia CancerMTT/MTS assay90% Cytotoxicity at 5 µM Approx24-hBloodNone
2842
242466472014
GIIKKIIKKI
Short α-helical peptides10LinearLNoneAmidationFreeAntimicrobialAlpha-helical proteinsHL-60Leukemia CancerMTT/MTS assay100% Cytotoxicity at 5 µM Approx24-hBloodNone
2840
242466472014
GIIKKIIKKIIKKI
Short α-helical peptides14LinearLNoneAmidationFreeAntimicrobialAlpha-helical proteinsHeLaCervical CancerMTT/MTS assay95% Cytotoxicity at 4 µM Approx24-hCervixNone
2841
242466472014
GIIKKIIKKIIKKIIKKI
Short α-helical peptides18LinearLNoneAmidationFreeAntimicrobialAlpha-helical proteinsHeLaCervical CancerMTT/MTS assay80% Cytotoxicity at 4 µM Approx24-hCervixNone
2839
242466472014
GIIKKIIKKI
Short α-helical peptides10LinearLNoneAmidationFreeAntimicrobialAlpha-helical proteinsHeLaCervical CancerMTT/MTS assay99% Cytotoxicity at 4 µM Approx24-hCervixNone
2834
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):J774A.1TumorMTT/MTS assayIC50=12 µM96-hBloodNone
2835
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):J774A.1TumorMTT/MTS assayIC50=17 µM96-hBloodNone
2833
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):J774A.1TumorMTT/MTS assayIC50=26 µM24-hBloodNone
2832
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):J774A.1TumorMTT/MTS assayIC50=47 µM24-hBloodNone
2831
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=36 µM96-hBloodNone
2830
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=25 µM96-hBloodNone
2829
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=45 µM72-hBloodNone
2828
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=36 µM72-hBloodNone
2827
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=43 µM48-hBloodNone
2826
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=37 µM48-hBloodNone
2825
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=43 µM24-hBloodNone
2824
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=39 µM24-hBloodNone
2823
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=38 µM2-hBloodNone
2822
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):HUT-102Lymphoma CancerMTT/MTS assayIC50=93 µM2-hBloodNone
2821
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):MDA-MB-231Breast CancerMTT/MTS assayIC50=10 µM48-hBreastNone
2820
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):MDA-MB-231Breast CancerMTT/MTS assayIC50=16 µM48-hBreastNone
2819
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):MDA-MB-231Breast CancerMTT/MTS assayIC50=12 µM24-hBreastNone
2818
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):MDA-MB-231Breast CancerMTT/MTS assayIC50=29 µM24-hBreastNone
2817
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):MDA-MB-231Breast CancerMTT/MTS assayIC50=18 µM2-hBreastNone
2816
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):MDA-MB-231Breast CancerMTT/MTS assayIC50=39 µM2-hBreastNone
2815
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):LNCaPProstate CancerMTT/MTS assayIC50=8 µM48-hProstateNone
2814
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):LNCaPProstate CancerMTT/MTS assayIC50=28 µM48-hProstateNone
2812
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):LNCaPProstate CancerMTT/MTS assayIC50=23 µM24-hProstateNone
2813
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):LNCaPProstate CancerMTT/MTS assayIC50=9 µM24-hProstateNone
2810
230004742012
RRRRRNWMWC
9R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):LNCaPProstate CancerMTT/MTS assayIC50=44 µM2-hProstateNone
2811
230004742012
RRRRRWCMNW
9S1R10LinearLNoneFreeFreeAnticancerNullomer derived anticancer peptides (NulloPs):LNCaPProstate CancerMTT/MTS assayIC50=26 µM2-hProstateNone
1772
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 14.58 mM24-hOvaryWO_2007133033_A1
1771
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 13.16 mM24-hSkinWO_2007133033_A1
1770
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 24.32 mM24-hProstateWO_2007133033_A1
1769
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayIC50 = 57 mM24-hColonWO_2007133033_A1
1768
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 13.77 mM24-hStomachWO_2007133033_A1
1767
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 14.8 mM24-hColonWO_2007133033_A1
1766
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 15.88 mM24-hLungWO_2007133033_A1
1765
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayNot Available24-hRenalWO_2007133033_A1
1764
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 22.06 mM24-hOvaryWO_2007133033_A1
1763
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 13.97 mM24-hSkinWO_2007133033_A1
1762
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 46.51 mM24-hProstateWO_2007133033_A1
1761
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayIC50 = 48 mM24-hColonWO_2007133033_A1
1760
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 22.31 mM24-hStomachWO_2007133033_A1
1759
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 24.63 mM24-hColonWO_2007133033_A1
1758
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 20.36 mM24-hLungWO_2007133033_A1
1757
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayNot Available24-hRenalWO_2007133033_A1
1756
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 12.55 mM24-hOvaryWO_2007133033_A1
1755
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 22.25 mM24-hSkinWO_2007133033_A1
1754
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 29.1 mM24-hProstateWO_2007133033_A1
1753
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayNot Available24-hColonWO_2007133033_A1
1752
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 22.51 mM24-hStomachWO_2007133033_A1
1751
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 14.8 mM24-hColonWO_2007133033_A1
1750
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 14.53 mM24-hLungWO_2007133033_A1
1749
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayIC50 = 21.48 mM24-hRenalWO_2007133033_A1
1748
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 24.76 mM24-hOvaryWO_2007133033_A1
1747
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 27.39 mM24-hSkinWO_2007133033_A1
1746
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 47.69 mM24-hProstateWO_2007133033_A1
1745
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayNot Available24-hColonWO_2007133033_A1
1744
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 26.7 mM24-hStomachWO_2007133033_A1
1743
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 25.2 mM24-hLungWO_2007133033_A1
1742
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayIC50 = 41.21 mM24-hRenalWO_2007133033_A1
1741
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayIC50 = 57 mM24-hColonUS_008076284_B2
1740
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayIC50 = 48 mM24-hColonUS_008076284_B2
1739
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayNot Available24-hColonUS_008076284_B2
1738
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaNCI-H630Colon CancerMTT/MTS assayNot Available24-hColonUS_008076284_B2
1737
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 14.8 mM24-hColonUS_008076284_B2
1736
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 24.63 mM24-hColonUS_008076284_B2
1735
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 14.8 mM24-hColonUS_008076284_B2
1734
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaHCTl-16Colon CancerMTT/MTS assayIC50 = 27 mM24-hColonUS_008076284_B2
1733
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayNot Available24-hRenalUS_008076284_B2
1732
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 24.32 mM24-hProstateUS_008076284_B2
1731
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 13.77 mM24-hStomachUS_008076284_B2
1730
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 14.58 mM24-hOvaryUS_008076284_B2
1729
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 14.8 mM24-hLungUS_008076284_B2
1728
None2011
FLWWLFKWAWK
Gaegurin peptides SEQID NO: 411LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 13.16 mM24-hSkinUS_008076284_B2
1727
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayNot Available24-hRenalUS_008076284_B2
1726
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 46.51 mM24-hProstateUS_008076284_B2
1725
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 24.31 mM24-hStomachUS_008076284_B2
1724
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 22.06 mM24-hOvaryUS_008076284_B2
1723
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 20.36 mM24-hLungUS_008076284_B2
1722
None2011
FLGWLFKWAWK
Gaegurin peptides SEQID NO: 311LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 13.97 mM24-hSkinUS_008076284_B2
1721
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayIC50 = 21.48 mM24-hRenalUS_008076284_B2
1720
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 29.1 mM24-hProstateUS_008076284_B2
1719
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 22.51 mM24-hStomachUS_008076284_B2
1718
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 12.55 mM24-hOvaryUS_008076284_B2
1717
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 14.53 mM24-hLungUS_008076284_B2
1716
None2011
FLKWLFKWAKK
Gaegurin peptides SEQID NO: 211LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 22.25 mM24-hSkinUS_008076284_B2
1715
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-498Renal CancerMTT/MTS assayIC50 = 41.21 mM24-hRenalUS_008076284_B2
1714
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaPC-3Prostate CancerMTT/MTS assayIC50 = 47.69 mM24-hProstateUS_008076284_B2
1713
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaMKN-45Gastric CancerMTT/MTS assayIC50 = 26.7 mM24-hStomachUS_008076284_B2
1712
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-OV-3Ovarian CancerMTT/MTS assayIC50 = 24.76 mM24-hOvaryUS_008076284_B2
1710
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaSK-MEL-2Skin CancerMTT/MTS assayIC50 = 27.39 mM24-hSkinUS_008076284_B2
1711
None2011
FLGWLFKWAKK
Gaegurin peptides SEQID NO: 111LinearLNoneFreeFreeAntimicrobialKorean frog Rana rugosaA-549Lung CancerMTT/MTS assayIC50 = 25.2 mM24-hLungUS_008076284_B2
1705
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsMECBreast CancerMTT/MTS assay29.33 Inhibition ratio at 50 µg/ml24-hBreastNone
1704
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsMECBreast CancerMTT/MTS assay19.76 Inhibition ratio at 50 µg/ml24-hBreastNone
1703
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyMECBreast CancerMTT/MTS assay27.99 Inhibition ratio at 50 µg/ml24-hBreastNone
1702
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyMECBreast CancerMTT/MTS assay24.15Inhibition ratio at 50 µg/ml24-hBreastNone
1701
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsHEK-293TRenal CancerMTT/MTS assay32.52 Inhibition ratio at 50 µg/ml24-hRenalNone
1700
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsHEK-293TRenal CancerMTT/MTS assay27.86 Inhibition ratio at 50 µg/ml24-hRenalNone
1699
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyHEK-293TRenal CancerMTT/MTS assay30.90 Inhibition ratio at 50 µg/ml24-hRenalNone
1698
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyHEK-293TRenal CancerMTT/MTS assay30.82 Inhibition ratio at 50 µg/ml24-hRenalNone
1697
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsHL7702Liver CancerMTT/MTS assay38.13 Inhibition ratio at 50 µg/ml24-hLiverNone
1696
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsHL7702Liver CancerMTT/MTS assay36.25 Inhibition ratio at 50 µg/ml24-hLiverNone
1695
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyHL7702Liver CancerMTT/MTS assay37.00 Inhibition ratio at 50 µg/ml24-hLiverNone
1694
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyHL7702Liver CancerMTT/MTS assay37.22 Inhibition ratio at 50 µg/ml24-hLiverNone
1693
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsA-549Lung CancerMTT/MTS assay52.50 Inhibition ratio at 50 µg/ml24-hLungNone
1692
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsA-549Lung CancerMTT/MTS assay47.26Inhibition ratio at 50 µg/ml24-hLungNone
1691
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyA-549Lung CancerMTT/MTS assay50.64 Inhibition ratio at 50 µg/ml24-hLungNone
1690
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyA-549Lung CancerMTT/MTS assay45.62 Inhibition ratio at 50 µg/ml24-hLungNone
1689
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsBGC-823Gastric CancerMTT/MTS assay73.705 Inhibition ratio at 50 µg/ml24-hStomachNone
1688
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsBGC-823Gastric CancerMTT/MTS assay62.49 Inhibition ratio at 50 µg/ml24-hStomachNone
1687
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyBGC-823Gastric CancerMTT/MTS assay50.85 Inhibition ratio at 50 µg/ml24-hStomachNone
1686
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyBGC-823Gastric CancerMTT/MTS assay48.19 Inhibition ratio at 50 µg/ml24-hStomachNone
1685
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide aNot Available temporinsHepG-2Liver CancerMTT/MTS assay73.07 Inhibition ratio at 50 µg/ml24-hLiverNone
1684
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide aNot Available temporinsHepG-2Liver CancerMTT/MTS assay60.22 Inhibition ratio at 50 µg/ml24-hLiverNone
1683
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyHepG-2Liver CancerMTT/MTS assay55.98 Inhibition ratio at 50 µg/ml24-hLiverNone
1682
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyHepG-2Liver CancerMTT/MTS assay50.90 Inhibition ratio at 50 µg/ml24-hLiverNone
1681
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsHeLaCervical CancerMTT/MTS assay78.045 Inhibition ratio at 50 µg/ml24-hCervixNone
1680
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsHeLaCervical CancerMTT/MTS assay73.09 Inhibition ratio at 50 µg/ml24-hCervixNone
1679
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familyHeLaCervical CancerMTT/MTS assay56.81 Inhibition ratio at 50 µg/ml24-hCervixNone
1678
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familyHeLaCervical CancerMTT/MTS assay52.32 Inhibition ratio at 50 µg/ml24-hCervixNone
1677
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsSMMC-7721Liver CancerMTT/MTS assay86.175 Inhibition ratio at 50 µg/ml24-hLiverNone
1676
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsSMMC-7721Liver CancerMTT/MTS assay70.39 Inhibition ratio at 50 µg/ml24-hLiverNone
1675
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familySMMC-7721Liver CancerMTT/MTS assay59.37 Inhibition ratio at 50 µg/ml24-hLiverNone
1674
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familySMMC-7721Liver CancerMTT/MTS assay52.77 Inhibition ratio at 50 µg/ml24-hLiverNone
1673
226413522012
RGDLLRHVVKILSKYL
RGD-Las16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsSW-1116Colorectal CancerMTT/MTS assay81.465 Inhibition ratio at 50 µg/ml24-hColonNone
1672
226413522012
RGDLLRHVVKILEKYL
RGD-La16LinearLNoneFreeFreeAnticancerArg-Gly-Asp(RGD) tripeptide ana temporinsSW-1116Colorectal CancerMTT/MTS assay72.69 Inhibition ratio at 50 µg/ml24-hColonNone
1671
226413522012
LLRHVVKILSKYL
Temporin-Las13LinearLNoneFreeFreeAnticancerTemporins familySW-1116Colorectal CancerMTT/MTS assay62.73 Inhibition ratio at 50 µg/ml24-hColonNone
1670
226413522012
LLRHVVKILEKYL
Temporin-La13LinearLNoneFreeFreeAnticancerTemporins familySW-1116Colorectal CancerMTT/MTS assay57.62 Inhibition ratio at 50 µg/ml24-hColonNone
1546
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=14.52 µg/ml24-hFibrous connective tissue None
1545
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=14.51 µg/ml12-hFibrous connective tissue None
1544
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=15.40 µg/ml6-hNot AvailableNone
1543
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=15.74 µg/ml3-hNot AvailableNone
1524
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=2.2 µMo/L36-hCervixNone
1523
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=2 µMo/L36-hCervixNone
1522
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=4.3 µMo/L36-hCervixNone
1521
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=3.8 µMo/L36-hCervixNone
1520
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=10.4 µMo/L36-hCervixNone
1519
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=58.6 µMo/L36-hCervixNone
1518
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=64.7 µMo/L36-hCervixNone
1517
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=>83.6 µMo/L36-hCervixNone
1516
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=>83.6 µMo/L36-hCervixNone
1515
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=>83.6 µMo/L36-hCervixNone
1514
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=4.6 µMo/L36-hSkinNone
1513
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=4.4 µMo/L36-hSkinNone
1512
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=7.8 µMo/L36-hSkinNone
1511
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=5.2 µMo/L36-hSkinNone
1510
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=11.5 µMo/L36-hSkinNone
1509
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=62.5 µMo/L36-hSkinNone
1508
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=63.5 µMo/L36-hSkinNone
1507
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1506
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1505
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1504
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=2.7 µMo/L36-hLungNone
1503
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=4.1 µMo/L36-hLungNone
1502
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=2.9 µMo/L36-hLungNone
1501
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=4.4 µMo/L36-hLungNone
1500
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=4.7 µMo/L36-hLungNone
1499
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=14 µMo/L36-hLungNone
1498
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=15.6 µMo/L36-hLungNone
1497
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=16.4 µMo/L36-hLungNone
1496
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=37.7 µMo/L36-hLungNone
1495
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1494
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=5.5 µMo/L36-hMuscleNone
1493
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=6.4 µMo/L36-hMuscleNone
1492
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=9.8 µMo/L36-hMuscleNone
1491
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=7.5 µMo/L36-hMuscleNone
1490
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=25.2 µMo/L36-hMuscleNone
1488
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1489
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1487
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1486
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1484
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=3.5 µMo/L36-hColonNone
1485
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1483
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=4.3 µMo/L36-hColonNone
1482
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=5 µMo/L36-hColonNone
1481
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=6.4 µMo/L36-hColonNone
1480
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=11.1 µMo/L36-hColonNone
1479
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1478
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1477
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1476
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1475
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1474
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=5.7 µMo/L36-hBreastNone
1473
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=6.2 µMo/L36-hBreastNone
1472
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=5.1 µMo/L36-hBreastNone
1471
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=5 µMo/L36-hBreastNone
1470
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=15.8 µMo/L36-hBreastNone
1469
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=62.3 µMo/L36-hBreastNone
1468
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=70.8 µMo/L36-hBreastNone
1467
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=>83.6 µMo/L36-hBreastNone
1466
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=>83.6 µMo/L36-hBreastNone
1465
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=>83.6 µMo/L36-hBreastNone
1464
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=7.2 µMo/L36-hSkinNone
1463
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=8.7 µMo/L36-hSkinNone
1462
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=6.5 µMo/L36-hSkinNone
1461
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=4.3 µMo/L36-hSkinNone
1460
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=17.8 µMo/L36-hSkinNone
1458
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=59.8 µMo/L36-hSkinNone
1459
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=58.7 µMo/L36-hSkinNone
1455
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1456
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1457
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1452
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=8.7 µMo/L36-hLungNone
1453
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=9.7 µMo/L36-hLungNone
1454
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=9.2 µMo/L36-hLungNone
1449
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=53 µMo/L36-hLungNone
1450
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=33 µMo/L36-hLungNone
1451
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=11.1 µMo/L36-hLungNone
1446
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1447
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1448
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=71 µMo/L36-hLungNone
1445
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1438
219552512011
GIIKKIIIKKIIIKKIIIKKI
Cationic Amphiphilic21CyclicLNoneFreeFreeAntimicrobialAMPHL-60Pancreatic CancerWST-1 assayIC50 = 10 µMNot AvailablePancreaticNone
1437
219552512011
GIIKKIIIKKIIIKKI
Cationic Amphiphilic16CyclicLNoneFreeFreeAntimicrobialAMPHL-60Pancreatic CancerWST-1 assayIC50 = 25 µMNot AvailablePancreaticNone
1436
219552512011
GIIKKIIIKKI
Cationic Amphiphilic11CyclicLNoneFreeFreeAntimicrobialAMPHL-60Pancreatic CancerWST-1 assayIC50 = >500 µMNot AvailablePancreaticNone
1435
219552512011
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneFreeFreeAntimicrobialXenopus laevisHeLaPancreatic CancerWST-1 assayIC50 = >60 µMNot AvailablePancreaticNone
1434
219552512011
GIIKKIIIKKIIIKKIIIKKI
Cationic Amphiphilic21CyclicLNoneFreeFreeAntimicrobialAMPHeLaPancreatic CancerWST-1 assayIC50 = 4 µMNot AvailablePancreaticNone
1433
219552512011
GIIKKIIIKKIIIKKI
Cationic Amphiphilic16CyclicLNoneFreeFreeAntimicrobialAMPHeLaCervical CancerWST-1 assayIC50 = 15 µMNot AvailableCervixNone
1432
219552512011
GIIKKIIIKKI
Cationic Amphiphilic11CyclicLNoneFreeFreeAntimicrobialAMPHeLaCervical CancerWST-1 assayIC50 = 160 µMNot AvailableCervixNone