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ACPs in Clinical Trial Studies

This page allows users to browse Anticancer proteins or peptides in clinical trials. The table below displays detailed information about each protein or peptide, including their sequences, associated NCT ID (clinical trial number), and the condition(s) being studied. Detailed experimental information can be viewed in the CancerPPD2 database peptide card or in the corresponding UniProt protein entry. Additionally, cross-references to DrugBank and ThPDB2 are provided for further research.

Name of the Entry Sequence NCT ID CancerPPD2 ID Uniprot ID Cross-References Phase Condition
p28 LSTAADMQGVVTDGMASGLDKDYLKPDD NCT01975116 7479 NA DB17241 Phase 1 Brain Tumor
p28 LSTAADMQGVVTDGMASGLDKDYLKPDD NCT00914914 7479 NA DB17241 Phase 1 Solid Tumor
ALRN-6924 LTFAEYWAQLaAAAAAa NCT03725436 4676 NA DB17285 Phase 1 Advanced Malignant Solid Neoplasm|Anatomic Stage III Breast Cancer
ALRN-6924 LTFAEYWAQLaAAAAAa NCT03654716 4676 NA DB17285 Phase 1 Leukemia|Brain Tumor|Solid Tumor|Lymphoma
ALRN-6924 LTFAEYWAQLaAAAAAa NCT02264613 4676 NA DB17285 Phase 1| Phase 2 Solid Tumor|Lymphoma|Peripheral T-Cell Lymphoma
ALRN-6924 LTFAEYWAQLaAAAAAa NCT05622058 4676 NA DB17285 Phase 1 Prevention of Chemotherapy-induced Myelosuppression
ALRN-6924 LTFAEYWAQLaAAAAAa NCT04022876 4676 NA DB17285 Phase 1 Non Small Cell Lung Cancer
ALRN-6924 LTFAEYWAQLaAAAAAa NCT02909972 4676 NA DB17285 Phase 1 Acute Myeloid Leukemia
LUNA18 Not Available NCT05012618 7842 NA NA Phase 1 Metastatic Solid Tumors
GV1001 EARPALLTSRLRFIPK NCT00444782 7308 NA DB12747 Phase 1| Phase 2 Hepatocellular Carcinoma
GV1001 EARPALLTSRLRFIPK NCT01579188 7308 NA DB12747 Phase 3 Inoperable Stage III Non-small Cell Lung Cancer
GV1001 EARPALLTSRLRFIPK NCT02854072 7308 NA DB12747 Phase 3 Pancreatic Cancer
Tigapotide PGDSTRKCMDLKGNK NCT00695851 4682 NA DB04985; Th1272 Phase 1 Prostate Cancer
Nelipepimut-S KIFGSLAFL NCT01570036 4174 NA DB06226 Phase 2 Breast Cancer
Nelipepimut-S KIFGSLAFL NCT02297698 4174 NA DB06226 Phase 2 Breast Cancer
Ozarelix Not Available NCT01252693 4695 NA DB12581 Phase 2 Prostate Cancer
LTX-315 KKWWKKW-Dip-K NCT01986426 3308 NA DB12748 Phase 1 Transdermally Accessible Tumours
Balixafortide ACSAp(Dab)RYCYQKpPYH NCT01837095 7848 NA DB15370 Phase 1 Breast Cancer
Balixafortide ACSAp(Dab)RYCYQKpPYH NCT01413568 7848 NA DB15370 Phase 1| Phase 2 Acute Myeloid Leukemia
Balixafortide ACSAp(Dab)RYCYQKpPYH NCT04826016 7848 NA DB15370 Phase 1|Phase 2 Advanced Breast Cancer
Balixafortide ACSAp(Dab)RYCYQKpPYH NCT03786094 7848 NA DB15370 Phase 3 Metastatic Breast Cancer|Locally Recurrent Breast Cancer
Balixafortide ACSAp(Dab)RYCYQKpPYH NCT01105403 7848 NA DB15370 Phase 2 Multiple Myeloma
TAK-448 ywNTF(AzGly)R(Me)W NCT01132404 7851 NA DB11975 Phase 1|Phase 2 Prostate Cancer
Dolastatin 10 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide NCT00003626 4644 NA DB12730 Phase 2 Prostate Cancer
Dolastatin 10 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide NCT00003557 4644 NA DB12730 Phase 2 Gall Bladder Cancer
Dolastatin 10 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide NCT00003693 4644 NA DB12730 Phase 1 Leukemia Cancer
Dolastatin 10 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide NCT00003677 4644 NA DB12730 Phase 2 Pancreatic Cancer
Dolastatin 10 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide NCT00003914 4644 NA DB12730 Phase 2 Kidney Cancer
Dolastatin 10 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N-[3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide NCT00003778 4644 NA DB12730 Phase 2 Ovarian Cancer
Bleomycin A6 MAKLTSAVPVLTARDVAGAVEFWTDRLGFSRDFVEDDFAGVVRDDVTLFISAVQDQVVPDNTLAWVWVRGLDELYAEWSEVVSTNFRDASGPAMTEIGEQPWGREFALRDPAGNCVHFVAEEQD NCT01660399 Available in Uniprot Proteins section P17493 DB12992 Phase 2 Lung Squamous Cell Cancer
Pegfilgrastim MTPLGPASSLPQSFLLKCLEQVRKIQGDGAALQEKLCATYKLCHPEELVLLGHSLGIPWAPLSSCPSQALQLAGCLSQLHSGLFLYQGLLQALEGISPELGPTLDTLQLDVADFATTIWQQMEELGMAPALQPTQGAMPAFASAFQRRAGGVLVASHLQSFLEVSYRVLRHLAQP NCT01516736 Available in Uniprot Proteins section P09919 DB00019; Th1016 Phase 3 Breast Cancer
Endostatin QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF NCT02104323 4690 NA DB06423; Th1356 Phase 2 NF2-Related Tumors
Endostatin QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF NCT03208335 4690 NA DB06423; Th1356 Phase 2 Hepatocellular Carcinoma
Endostatin QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF NCT04356118 4690 NA DB06423; Th1356 Phase 4 Non-Small Cell Lung Cancer
Endostatin QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF NCT02745561 4690 NA DB06423; Th1356 Phase 2 Esophageal Cancer
Endostatin QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF NCT00604435 4690 NA DB06423; Th1356 Phase 2 Breast Cancer
Endostatin QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF NCT05551247 4690 NA DB06423; Th1356 Phase 2 Colorectal Cancer
Stem Bromelain AVPQSIDWRDYGAVTSVKNQNPCGACWAFAAIATVESIYKIKKGILEPLSEQQVLDCAKGYGCKGGWEFRAFEFIISNKGVASGAIYPYKAAKGTCKTDGVPNSAYITGYARVPRNNESSMMYAVSKQPITVAVDANANFQYYKSGVFNGPCGTSLNHAVTAIGYGQDSIIYPKKWGAKWGEAGYIRMARDVSSSSGICGIAIDPLYPTLEE NCT02340845 Available in Uniprot Proteins section P14518 DB12249; Th1476 Phase 2 Breast Cancer, Lung Cancer, Colon Cancer, Cervical Cancer, Ovarian Cancer, Uterine Cancer
ADH-1 GLKAADNDPTAPPYDSLLVFDYEGSGSTAGSLSSLNSSSSGGDQDYDYLNDWGPRFKKLADMYGGGDD NCT00264433 Available in Uniprot Proteins section Q80XX1 DB05485; Th1722 Phase 2 Neoplasm
ADH-1 GLKAADNDPTAPPYDSLLVFDYEGSGSTAGSLSSLNSSSSGGDQDYDYLNDWGPRFKKLADMYGGGDD NCT00421811 Available in Uniprot Proteins section Q80XX1 DB05485; Th1722 Phase 1|Phase 2 Neoplasm
ADH-1 GLKAADNDPTAPPYDSLLVFDYEGSGSTAGSLSSLNSSSSGGDQDYDYLNDWGPRFKKLADMYGGGDD NCT01825603 Available in Uniprot Proteins section Q80XX1 DB05485; Th1722 Phase 1 Neoplasm
ADH-1 GLKAADNDPTAPPYDSLLVFDYEGSGSTAGSLSSLNSSSSGGDQDYDYLNDWGPRFKKLADMYGGGDD NCT00265057 Available in Uniprot Proteins section Q80XX1 DB05485; Th1722 Phase 1| Phase 2 Neoplasm
ADH-1 GLKAADNDPTAPPYDSLLVFDYEGSGSTAGSLSSLNSSSSGGDQDYDYLNDWGPRFKKLADMYGGGDD NCT00225550 Available in Uniprot Proteins section Q80XX1 DB05485; Th1722 Phase 1| Phase 2 Neoplasm
ADH-1 GLKAADNDPTAPPYDSLLVFDYEGSGSTAGSLSSLNSSSSGGDQDYDYLNDWGPRFKKLADMYGGGDD NCT00421811 Available in Uniprot Proteins section Q80XX1 DB05485; Th1722 Phase 1 Neoplasm
LL-37 SKWQHQQDSCRKQLQGVNLTPCEKHIMEKIQGRGDDDDDDDDD NCT02225366 1527 NA DB16532 Phase 1| Phase 2 Melanoma
SOR-C13 KEFLHPSKVDLPR NCT01578564 7847 NA DB15366 Phase 1 Advanced Solid tumors
CIGB-300 GRKKRRQRRRPPQ-X-CWMSPRHLGTC NCT01639625 7250 NA DB16464 Phase 2 Cervical Cancer