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IDPMIDYEARSequenceNameLengthLinear/CyclicChiralityChem-MODC-ter MODN-ter MODNatureOriginCell LineCancer TypeAssayActivityTesting TimeTissue AffectedPatents
4618
209643342010
KWKWKW
Dex-(KW)36LinearLDextranAmidationDextranAnticancerSyntheticPC-3Prostate CancerMTT/MTS assayat 10 µM 60% viablityNot AvailableProstateNone
4619
209643342010
KWKWKW
Dex-(KW)36LinearLDextranAmidationDextranAnticancerSyntheticMCF-7Breast CancerMTT/MTS assayat 10 µM 35-40% viablityNot AvailableBreastNone
4616
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideSkmel-25Skin CancerMTT/MTS assayat 100 µM 55-60% viablity48-hSkinNone
4617
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideSkmel-28Skin CancerMTT/MTS assayat 100 µM 35-40% viablity48-hSkinNone
4614
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideB16F10-Nex 2Skin CancerMTT/MTS assayat 100 µM 50% viablity48-hSkinNone
4615
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideA-2058Skin CancerMTT/MTS assayat 100 µM 30% viablity48-hSkinNone
4612
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideMDA-MB-231Breast CancerMTT/MTS assayat 100 µM 55% viablity48-hBreastNone
4613
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assayat 100 µM 50% viablity48-hCervixNone
4611
208029912010
CSSRTMHHC
Peptide-209Cyclic(C1-C9)LNoneFreeFreeAntitumorSynthetic PeptideHL-60Leukemia CancerMTT/MTS assayat 100 µM 90% viablity48-hBloodNone
4454
17067680, 189574412007
GIKCRFCCGCCTPGICGVCCRF
hepcidin TH1-522Not AvailableLNoneFreeFreeAnticancerTilapia, Oreochromis mossambicusNot AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4453
17561225, 189574412007
LLGMIPLAISAISALSKL
Phylloseptin-L132Not AvailableLNoneFreeFreeAnticancerHylomantis lemur (Hylidae: PhyllomedusinaeNot AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4452
17561225, 189574412007
GLWSKIKEAAKAAGKAALNAVTGLVNQGDQPS
Phylloseptin32Not AvailableLNoneFreeFreeAnticancerHylomantis lemur (Hylidae: PhyllomedusinaeNot AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4439
19341344, 189574412009
ILPILSLIGGLLGK
Temporin-1CEb17Not AvailableLNoneFreeFreeAntimicrobialRana chensinensis, China, AsiaNot AvailableBreast CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4423
18191970, 189574412008
GLLPCAESCVYIPCLTTVIGCSCKSKVCYKN
Vibi H31Not AvailableLNoneFreeFreeAnticancerAlpine violetViola bifloraNot AvailableLung CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4422
18191970, 189574412008
GIPCAESCVWIPCTVTALIGCGCSNKVCYN
Vibi E30Not AvailableLNoneFreeFreeAnticancerAlpine violetViola bifloraNot AvailableLeukemia CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4418
18191970, 189574412008
GTFPCGESCVFIPCLTSAIGCSCKSKVCYKN
Vibi G31Not AvailableLNoneFreeFreeAnticancerAlpine violetViola bifloraNot AvailableSkin CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4403
20198492, 189574412010
GKWMSLLKHILK
Halictine 212Not AvailableLNoneFreeFreeAnticancerVenom, the eusocial bee, Halictus sexcinctusNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4402
20198492, 189574412010
GMWSKILGHLIR
Halictine 112Not AvailableLNoneFreeFreeAnticancervenom, the eusocial bee, Halictus sexcinctusNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4397
20575512, 189574412010
GIACGESCVFLGCFIPGCSCKSKVCYFN
Psyle A28Not AvailableLNoneFreeFreeAntibacterialPsychotria leptothyrsaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4396
20575512, 189574412010
GVIPCGESCVFIPCISSVLGCSCKNKVCYRD
Psyle E31Not AvailableLNoneFreeFreeAntibacterialPsychotria leptothyrsaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4395
20575512, 189574412010
KLCGETCFKFKCYTPGCSCSYPFCK
Psyle C25Not AvailableLNoneFreeFreeAntibacterialPsychotria leptothyrsaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4364
16713189, 189574412006
FLPILASLAAKFGPKLFCLVTKKC
Brevinin-1BYa24Not AvailableLNoneFreeFreeAntibacterialRana boylii, North AmericaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4362
19254736, 189574412009
GLMDTIKGVAKTVAASWLDKLKCKITGC
Ranatuerin-2Ya28Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates yavapaiensisNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4361
19254736, 189574412009
FLPVIAGVAANFLPKLFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4360
19254736, 189574412009
FLPIIAGVAAKVLPKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4359
19254736, 189574412009
FLPIIAGIAAKFLPKIFCTISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4358
19254736, 189574412009
FLPIIAGAAAKVVQKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4357
19254736, 189574412009
FLPIIAGAAAKVVEKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4356
19254736, 189574412009
FLPAIVGAAAKFLPKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4355
17698251, 189574412007
FLIGMTQGLICLITRKC
Dybowskin-217Not AvailableLNoneFreeFreeAntibacterialRana dybowskii, Rana chensinensis, AsiaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4354
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 8.0 µM48-hPancreaticWO_2010_064207_A2
4353
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptidePane- 1Breast CancerWST-1 assayIC50= 14.1 µM48-hBreastWO_2010_064207_A2
4352
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptideCFPAC-IPancreatic CancerWST-1 assayIC50= 9.2 µM48-hPancreaticWO_2010_064207_A2
4351
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 14.7 µM48-hPancreaticWO_2010_064207_A2
4350
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 7.9 µM48-hPancreaticWO_2010_064207_A2
4349
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptidePane- 1Breast CancerWST-1 assayIC50= 13.1 µM48-hBreastWO_2010_064207_A2
4348
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideCFPAC-IPancreatic CancerWST-1 assayIC50= 10.6 µM48-hPancreaticWO_2010_064207_A2
4347
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 12.5 µM48-hPancreaticWO_2010_064207_A2
4346
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideLNCaPProstate CancerWST-1 assayIC50= 4.8 µMNot AvailableProstateUS_8436137_B2
4345
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 7.4 µMNot AvailablePancreaticUS_8436137_B2
4344
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 6.6 µMNot AvailablePancreaticUS_8436137_B2
4343
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideU-251Brain TumorWST-1 assayIC50= 8.4 µMNot AvailableBrainUS_8436137_B2
4342
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBT-20Breast CancerWST-1 assayIC50= 1.9 µMNot AvailableBreastUS_8436137_B2
4341
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideH-322Lung CancerWST-1 assayIC50= 3.2 µMNot AvailableLungUS_8436137_B2
4340
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideLNCaPProstate CancerWST-1 assayIC50= 10 µMNot AvailableProstateUS_8436137_B2
4339
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 12 µMNot AvailablePancreaticUS_8436137_B2
4338
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 12 µMNot AvailablePancreaticUS_8436137_B2
4337
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideU-251Brain TumorWST-1 assayIC50= 12 µMNot AvailableBrainUS_8436137_B2
4336
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBT-20Breast CancerWST-1 assayIC50= 6.5 µMNot AvailableBreastUS_8436137_B2
4335
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideH-322Lung CancerWST-1 assayIC50= 6.8 µMNot AvailableLungUS_8436137_B2
4262
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay2% apoptosis at 50 µM8-hNot AvailableNone
4261
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay1% apoptosis at 20 µM8-hNot AvailableNone
4260
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay0% apoptosis at 10 µM8-hNot AvailableNone
4259
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay3% apoptosis at 50 µM8-hNot AvailableNone
4258
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay2% apoptosis at 20 µM8-hNot AvailableNone
4257
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay1% apoptosis at 10 µM8-hNot AvailableNone
4256
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay5% apoptosis at 50 µM8-hBrainNone
4255
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay1% apoptosis at 20 µM8-hBrainNone
4254
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay2% apoptosis at 10 µM8-hBrainNone
4253
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay3% apoptosis at 50 µM8-hBrainNone
4252
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay2% apoptosis at 20 µM8-hBrainNone
4251
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay1% apoptosis at 10 µM8-hBrainNone
4250
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay55% apoptosis at 50 µM8-hNot AvailableNone
4249
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay35% apoptosis at 20 µM8-hNot AvailableNone
4248
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay23% apoptosis at 10 µM8-hNot AvailableNone
4247
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay79% apoptosis at 50 µM8-hNot AvailableNone
4246
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay46% apoptosis at 20 µM8-hNot AvailableNone
4245
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay43% apoptosis at 10 µM8-hNot AvailableNone
4244
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay68% apoptosis at 50 µM8-hBrainNone
4243
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay66% apoptosis at 20 µM8-hBrainNone
4242
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay25% apoptosis at 10 µM8-hBrainNone
4241
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay65% apoptosis at 50 µM8-hBrainNone
4240
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay45% apoptosis at 20 µM8-hBrainNone
4239
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay8% apoptosis at 10 µM8-hBrainNone
4238
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay50% apoptosis at 50 µM8-hNot AvailableNone
4237
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay20% apoptosis at 20 µM8-hNot AvailableNone
4236
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay15% apoptosis at 10 µM8-hNot AvailableNone
4235
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay30% apoptosis at 50 µM8-hNot AvailableNone
4234
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay>50% apoptosis at 20 µM8-hNot AvailableNone
4233
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay20% apoptosis at 10 µM8-hNot AvailableNone
4232
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay80% apoptosis at 50 µM8-hBrainNone
4231
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay80% apoptosis at 20 µM8-hBrainNone
4230
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay30% apoptosis at 10 µM8-hBrainNone
4229
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay30% apoptosis at 50 µM8-hBrainNone
4228
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay10% apoptosis at 20 µM8-hBrainNone
4227
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay0% apoptosis at 10 µM8-hBrainNone
4025
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay47.0% inhibition at 10-3M31.92-MinColonNone
4026
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay2.2% inhibition at 10-6M31.92-MinBreastNone
4027
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay7.1% inhibition at 10-5M31.92-MinBreastNone
4028
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay6.9% inhibition at 10-4M31.92-MinBreastNone
4029
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay25.9% inhibition at 10-3M31.92-MinBreastNone
4021
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay70.7% inhibition at 10-5M31.92-MinSkinNone
4022
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay34.4% inhibition at 10-3M31.92-MinSkinNone
4023
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay9.2% inhibition at 10-3M31.92-MinColonNone
4024
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay11.08% inhibition at 10-5M31.92-MinColonNone
4016
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay29.9% inhibition at 10-3M23.03-MinBreastNone
4017
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay3.9% inhibition at 10-5M31.92-MinLarynxNone
4018
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay45% inhibition at 10-3M31.92-MinLarynxNone
4019
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay9.3% inhibition at 10-3M31.92-MinCervixNone
4020
167226322006
YGGFMA*
236LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay4.1% inhibition at 10-6M31.92-MinSkinNone
4012
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay10.9% inhibition at 10-5M23.03-MinColonNone
4013
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay12.1% inhibition at 10-4M23.03-MinColonNone
4014
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay8.1% inhibition at 10-3M23.03-MinColonNone
4015
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay9.6% inhibition at 10-4M23.03-MinBreastNone
4008
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay13.1% inhibition at 10-5M23.03-MinColonNone
4009
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay14.6% inhibition at 10-4M23.03-MinColonNone
4010
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay38.4% inhibition at 10-3M23.03-MinColonNone
4011
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay17.7% inhibition at 10-6M23.03-MinColonNone
4003
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay16.2% inhibition at 10-6M23.03-MinColonNone
4004
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay6.6% inhibition at 10-5M23.03-MinColonNone
4005
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay5.1% inhibition at 10-4M23.03-MinColonNone
4006
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay14.5% inhibition at 10-3M23.03-MinColonNone
4007
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay26.4% inhibition at 10-6M23.03-MinColonNone
3999
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay2.4% inhibition at 10-6M23.03-MinSkinNone
4000
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay4.5% inhibition at 10-5M23.03-MinSkinNone
4001
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay11.4% inhibition at 10-4M23.03-MinSkinNone
4002
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay23.2% inhibition at 10-3M23.03-MinSkinNone
3994
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay44.5% inhibition at 10-3M23.03-MinLarynxNone
3995
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay8.5% inhibition at 10-6M23.03-MinCervixNone
3996
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay9.5% inhibition at 10-5M23.03-MinCervixNone
3997
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay15.4% inhibition at 10-4M23.03-MinCervixNone
3998
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay24.1% inhibition at 10-3M23.03-MinCervixNone
3991
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay13.7% inhibition at 10-6M23.03-MinLarynxNone
3992
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay25.8% inhibition at 10-5M23.03-MinLarynxNone
3993
167226322006
YA*GFM
185LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay34.7% inhibition at 10-4M23.03-MinLarynxNone
3988
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay18.5% inhibition at 10-4M26.70-MinColonNone
3989
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay10.6% inhibition at 10-3M26.70-MinColonNone
3990
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay22.8% inhibition at 10-3M26.70-MinBreastNone
3986
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay3.0% inhibition at 10-6M26.70-MinColonNone
3987
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay8.4% inhibition at 10-5M26.70-MinColonNone
3984
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay24.7% inhibition at 10-4M26.70-MinColonNone
3985
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay29.0% inhibition at 10-3M26.70-MinColonNone
3981
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay23.7% inhibition at 10-3M26.70-MinColonNone
3982
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay12.2% inhibition at 10-6M26.70-MinColonNone
3983
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay15.5% inhibition at 10-5M26.70-MinColonNone
3978
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay3.3% inhibition at 10-6M26.70-MinColonNone
3979
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay11.0% inhibition at 10-5M26.70-MinColonNone
3980
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay7.9% inhibition at 10-4M26.70-MinColonNone
3976
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay2.4% inhibition at 10-4M26.70-MinSkinNone
3977
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay18.3% inhibition at 10-3M26.70-MinSkinNone
3971
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay10.2% inhibition at 10-5M26.70-MinCervixNone
3972
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay13.3% inhibition at 10-4M26.70-MinCervixNone
3973
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay28.0% inhibition at 10-3M26.70-MinCervixNone
3974
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay0.8% inhibition at 10-6M26.70-MinSkinNone
3975
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay1.4% inhibition at 10-5M26.70-MinSkinNone
3970
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay4.9% inhibition at 10-6M26.70-MinCervixNone
3969
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay36.1% inhibition at 10-3M26.70-MinLarynxNone
3968
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay16.8% inhibition at 10-4M26.70-MinLarynxNone
3967
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay10.1% inhibition at 10-5M26.70-MinLarynxNone
3966
167226322006
YA*GFM
175LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay1.0% inhibition at 10-6M26.70-MinLarynxNone
3964
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay8.6% inhibition at 10-3M10.79-MinColonNone
3965
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay15.6% inhibition at 10-3M10.79-MinBreastNone
3962
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay6.9% inhibition at 10-5M10.79-MinColonNone
3963
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay8.1% inhibition at 10-4M10.79-MinColonNone
3959
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay13.5% inhibition at 10-4M10.79-MinColonNone
3960
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay25.3% inhibition at 10-3M10.79-MinColonNone
3961
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay8.1% inhibition at 10-6M10.79-MinColonNone
3957
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay17.0% inhibition at 10-6M10.79-MinColonNone
3958
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay13.5% inhibition at 10-5M10.79-MinColonNone
3955
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay12.4% inhibition at 10-4M10.79-MinColonNone
3956
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay22.4% inhibition at 10-3M10.79-MinColonNone
3952
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay19.4% inhibition at 10-3M10.79-MinSkinNone
3953
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay7.6% inhibition at 10-6M10.79-MinColonNone
3954
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay3.8% inhibition at 10-5M10.79-MinColonNone
3949
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay28.2% inhibition at 10-3M10.79-MinCervixNone
3950
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay1.2% inhibition at 10-5M10.79-MinSkinNone
3951
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay3.3% inhibition at 10-4M10.79-MinSkinNone
3947
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay11.7% inhibition at 10-5M10.79-MinCervixNone
3948
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay11.6% inhibition at 10-4M10.79-MinCervixNone
3944
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay12.6% inhibition at 10-4M10.79-MinLarynxNone
3945
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay26.4% inhibition at 10-3M10.79-MinLarynxNone
3946
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay11.0% inhibition at 10-6M10.79-MinCervixNone
3942
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay4.6% inhibition at 10-6M10.79-MinLarynxNone
3943
167226322006
YRA*G
164LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay4.9% inhibition at 10-5M10.79-MinLarynxNone
3940
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay6.2% inhibition at 10-3M9.53-MinColonNone
3941
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay21.2% inhibition at 10-3M9.53-MinBreastNone
3937
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay2.2% inhibition at 10-6M9.53-MinColonNone
3938
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay4.2% inhibition at 10-5M9.53-MinColonNone
3939
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay6.4% inhibition at 10-4M9.53-MinColonNone
3935
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay14.4% inhibition at 10-4M9.53-MinColonNone
3936
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay23.4% inhibition at 10-3M9.53-MinColonNone
3932
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay15.7% inhibition at 10-3M9.53-MinColonNone
3933
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay13.6% inhibition at 10-6M9.53-MinColonNone
3934
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay20.4% inhibition at 10-5M9.53-MinColonNone
3930
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay7.4% inhibition at 10-5M9.53-MinColonNone
3931
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay9.5% inhibition at 10-4M9.53-MinColonNone
3927
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay5.9% inhibition at 10-4M9.53-MinSkinNone
3928
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay17.9% inhibition at 10-3M9.53-MinSkinNone
3929
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay5.4% inhibition at 10-6M9.53-MinColonNone
3925
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay1.6% inhibition at 10-6M9.53-MinSkinNone
3926
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay2.9% inhibition at 10-5M9.53-MinSkinNone
3922
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay7.3% inhibition at 10-5M9.53-MinCervixNone
3923
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay9.9% inhibition at 10-4M9.53-MinCervixNone
3924
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay28.2% inhibition at 10-3M9.53-MinCervixNone
3920
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay26.7% inhibition at 10-3M9.53-MinLarynxNone
3921
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay9.8% inhibition at 10-6M9.53-MinCervixNone
3917
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay2.7% inhibition at 10-6M9.53-MinLarynxNone
3918
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay2.0% inhibition at 10-5M9.53-MinLarynxNone
3919
167226322006
YSA*G
154LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay18.8% inhibition at 10-4M9.53-MinLarynxNone
3915
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay7.7% inhibition at 10-4M14.05-MinBreastNone
3916
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay18.7% inhibition at 10-3M14.05-MinBreastNone
3913
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay10.7% inhibition at 10-614.05-MinColonNone
3914
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay10.0% inhibition at 10-514.05-MinColonNone
3910
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay8.3% inhibition at 10-514.05-MinColonNone
3911
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay10.5% inhibition at 10-414.05-MinColonNone
3912
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay21.8% inhibition at 10-314.05-MinColonNone
3908
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay7.3% inhibition at 10-314.05-MinSkinNone
3909
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay0.7% inhibition at 10-614.05-MinColonNone
3905
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay3.0% inhibition at 10-614.05-MinSkinNone
3906
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay4.7% inhibition at 10-514.05-MinSkinNone
3907
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay2.7% inhibition at 10-414.05-MinSkinNone
3903
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay11.0% inhibition at 10-414.05-MinCervixNone
3904
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay20.5% inhibition at 10-314.05-MinCervixNone
3901
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay7.2% inhibition at 10-614.05-MinCervixNone
3902
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay17.1% inhibition at 10-514.05-MinCervixNone
3898
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay4.9% inhibition at 10-514.05-MinLarynxNone
3899
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay1.9% inhibition at 10-414.05-MinLarynxNone
3900
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay16.2% inhibition at 10-314.05-MinLarynxNone
3896
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay17.8% inhibition at 10-312.46-MinBreastNone
3897
167226322006
YSA*
103LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay8.5% inhibition at 10-614.05-MinLarynxNone
3893
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay14.5% inhibition at 10-312.46-MinColonNone
3894
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay1.1% inhibition at 10-512.46-MinBreastNone
3895
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay1.2% inhibition at 10-412.46-MinBreastNone
3892
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay8.4% inhibition at 10-412.46-MinColonNone
3891
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay16.5% inhibition at 10-512.46-MinColonNone
3890
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay3.7% inhibition at 10-612.46-MinColonNone
3889
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay17.9% inhibition at 10-312.46-MinColonNone
3888
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay11.8% inhibition at 10-412.46-MinColonNone
3887
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay21.9% inhibition at 10-512.46-MinColonNone
3886
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay10.5% inhibition at 10-612.46-MinColonNone
3885
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay20.8% inhibition at 10-312.46-MinColonNone
3884
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay3.4% inhibition at 10-412.46-MinColonNone
3883
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay8.9% inhibition at 10-512.46-MinColonNone
3882
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay4.9% inhibition at 10-612.46-MinColonNone
3881
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay7.3% inhibition at 10-312.46-MinSkinNone
3880
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay3.9% inhibition at 10-512.46-MinSkinNone
3879
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay14.8% inhibition at 10-312.46-MinCervixNone
3877
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay6.1% inhibition at 10-512.46-MinCervixNone
3878
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay3.1% inhibition at 10-412.46-MinCervixNone
3876
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay7.5% inhibition at 10-612.46-MinCervixNone
3875
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay21.2% inhibition at 10-312.46-MinLarynxNone
3874
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay8.2% inhibition at 10-412.46-MinLarynxNone
3873
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay6.4% inhibition at 10-512.46-MinLarynxNone
3872
167226322006
YSA*
93LinearLA* = Cα -dialkylated glycine (Aaa2,2 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay6.2% inhibition at 10-612.46-MinLarynxNone
3871
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay7.5% inhibition at 10-412.81-MinBreastNone
3870
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideMCF-7Breast CancerMTT/MTS assay2.4% inhibition at 10-512.81-MinBreastNone
3868
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay18.9% inhibition at 10-412.81-MinColonNone
3869
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay26.4% inhibition at 10-312.81-MinColonNone
3867
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay22.7% inhibition at 10-512.81-MinColonNone
3866
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideCaCo-2Colon CancerMTT/MTS assay3.5% inhibition at 10-612.81-MinColonNone
3864
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay28.1% inhibition at 10-412.81-MinColonNone
3865
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay58.2% inhibition at 10-312.81-MinColonNone
3863
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay16.5% inhibition at 10-512.81-MinColonNone
3862
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideSW-620Colon CancerMTT/MTS assay12.9% inhibition at 10-612.81-MinColonNone
3861
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay26.5% inhibition at 10-312.81-MinColonNone
3859
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay1.6% inhibition at 10-512.81-MinColonNone
3860
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay5.4% inhibition at 10-412.81-MinColonNone
3857
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay14% inhibition at 10-312.81-MinSkinNone
3858
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHT-29Colon CancerMTT/MTS assay9.8% inhibition at 10-612.81-MinColonNone
3856
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay7.5% inhibition at 10-412.81-MinSkinNone
3855
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay14% inhibition at 10-512.81-MinSkinNone
3854
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHBLSkin CancerMTT/MTS assay6.5% inhibition at 10-612.81-MinSkinNone
3853
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay36.1% inhibition at 10-312.81-MinNot AvailableNone
3852
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay8.2% inhibition at 10-412.81-MinNot AvailableNone
3851
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHeLaCervical CancerMTT/MTS assay10% inhibition at 10-512.81-MinNot AvailableNone
3850
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay30.4% inhibition at 10-312.81-MinNot AvailableNone
3849
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay24.9% inhibition at 10-412.81-MinNot AvailableNone
3848
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay19.7% inhibition at 10-512.81-MinNot AvailableNone
3847
167226322006
YA*
82LinearLA* = Cαα -dialkylated glycine (Aaa1,1 )FreeFreeAntitumorSynthetic PeptideHEp-2Larynx CancerMTT/MTS assay14.2% inhibition at 10-612.81-MinNot AvailableNone
3842
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP(O)25Cyclic(C2-C10,CLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay52% inhibition at 10µg/mlNANot AvailableNone
3841
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP(O)25Cyclic(C2-C10,CLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay42% inhibition at 5µg/mlNANot AvailableNone
3840
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP(O)25Cyclic(C2-C10,CLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay40% inhibition at 2.5µg/mlNANot AvailableNone
3839
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP25LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay75% inhibition at 10µg/mlNANot AvailableNone
3838
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP25LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay40% inhibition at 5µg/mlNANot AvailableNone
3837
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP25LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay50% inhibition at 2.5µg/mlNANot AvailableNone
3836
205150452010
IVRRADRAAVP
ES-211LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay60% inhibition at 10µg/mlNANot AvailableNone
3835
205150452010
IVRRADRAAVP
ES-211LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay60% inhibition at 5µg/mlNANot AvailableNone
3834
205150452010
IVRRADRAAVP
ES-211LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay60% inhibition at 2.5µg/mlNANot AvailableNone
3299
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideA-375Skin CancerMTT/MTS assay6.5 ± 1.07% cell viability at 80 µMNASkinNone
3298
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideA-375Skin CancerMTT/MTS assay26.9 ± 0.5% cell viability at 60 µMNASkinNone
3297
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideA-375Skin CancerMTT/MTS assay47.5 ± 1.66% cell viability at 40 µMNASkinNone
3296
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideA-375Skin CancerMTT/MTS assay63.8 ± 0.8% cell viability at 20 µMNASkinNone
3295
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideA-375Skin CancerMTT/MTS assay86 ± 0.57% cell viability at 10 µMNASkinNone
3294
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideM14Skin CancerMTT/MTS assay13.8 ± 1.44% cell viability at 80 µMNASkinNone
3293
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideM14Skin CancerMTT/MTS assay31.5 ± 1.49% cell viability at 60 µMNASkinNone
3292
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideM14Skin CancerMTT/MTS assay50 ± 3.09% cell viability at 40 µMNASkinNone
3291
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialSynthetic peptideM14Skin CancerMTT/MTS assay71.1 ± 2.84% cell viability at 20 µMNASkinNone
3290
199570172010
KWKLFKKIPKFLHLAKKF
P1818LinearLNoneFreeFreeAntibacterialBovine lactoferrin (Lf-B)M14Skin CancerMTT/MTS assay92.2 ± 1.02% cell viability at 10 µMNASkinNone
3289
195274902009
KAAKKAAKAAKKAAKAAKKAA
KW521LinearLNoneFreeFreeAnticancerSynthetic peptideHT-29Colon CancerMTT/MTS assayIC50 =55±14 µMNAColonNone
3288
195274902009
KAAKKAAKAAKKAAKAAKKAA
KW521LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)FEMXSkin CancerMTT/MTS assayIC50 =30±3 µMNASkinNone
3287
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)RamosLymphoma CancerMTT/MTS assayIC50 = 10 µMNABloodNone
3286
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)RajiLymphoma CancerMTT/MTS assayIC50 = 13 µMNABloodNone
3285
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)Sudhl-4Skin CancerMTT/MTS assayIC50 = 16 µMNASkinNone
3284
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)KMM-1Skin CancerMTT/MTS assayIC50 = 57 µMNASkinNone
3283
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)U-266Lymphoma CancerMTT/MTS assayIC50 = 55 µMNABloodNone
3282
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)KMS-5Skin CancerMTT/MTS assayIC50 = 38 µMNASkinNone
3281
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)HT-29Colon CancerMTT/MTS assayIC50 =148±8 µMNAColonNone
3280
19527490, 235337102009
FKCRRWQWRMKK
LfcinB12LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)FEMXSkin CancerMTT/MTS assayIC50 =40±7 µMNASkinNone
3278
188157342008
KKKFPWWWPFKKKKKKFPWWWPFKKKK
di-PST13-RK-K27LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinMDA-MB-361Breast CancerMTT/MTS assayIC50 =10 µg/mlNABreastNone
3277
188157342008
KKKFPWWWPFKKKKKKFPWWWPFKKKK
di-PST13-RK-K27LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinA-549Lung CancerMTT/MTS assayIC50 =15 µg/mlNALungNone
3275
188157342008
KKKFPWWWPFKKKCKKKFPWWWPFKKKC
di-PST13-RK-C28LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinMDA-MB-361Breast CancerMTT/MTS assayIC50 =17 µg/mlNABreastNone
3274
188157342008
KKKFPWWWPFKKKCKKKFPWWWPFKKKC
di-PST13-RK-C28LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinA-549Lung CancerMTT/MTS assayIC50 =17 µg/mlNALungNone
3272
188157342008
KKKFPWWWPFKKK
PST13-RK13LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinMDA-MB-361Breast CancerMTT/MTS assayIC50 =80 µg/mlNABreastNone
3271
188157342008
KKKFPWWWPFKKK
PST13-RK13LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinA-549Lung CancerMTT/MTS assayIC50 =90 µg/mlNALungNone
3269
188157342008
VRRFPWWWPFLRR
Tritrpticin13LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinMDA-MB-361Breast CancerMTT/MTS assayIC50 =142 µg/mlNABreastNone
3268
188157342008
VRRFPWWWPFLRR
Tritrpticin13LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinA-549Lung CancerMTT/MTS assayIC50 >200 µg/mlNALungNone
3197
177870262007
(K-Aib-C(CH2CO-2'-Pac))4
Tetramer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateMCF-7Breast CancerMTT/MTS assayIC50 =0.64nM24-hBreastNone
3195
177870262007
(K-Aib-C(CH2CO-2'-Pac))4
Tetramer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateHeLaCervical CancerMTT/MTS assayIC50 =0.96nM24-hCervixNone
3196
177870262007
(K-Aib-C(CH2CO-2'-Pac))4
Tetramer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateDUProstate CancerMTT/MTS assayIC50 =1.30nM24-hProstateNone
3194
177870262007
(K-Aib-C(CH2CO-2'-Pac))3
Trimer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateMCF-7Breast CancerMTT/MTS assayIC50 =3.00nM24-hBreastNone
3192
177870262007
(K-Aib-C(CH2CO-2'-Pac))3
Trimer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateHeLaCervical CancerMTT/MTS assayIC50 =1.70nM24-hCervixNone
3193
177870262007
(K-Aib-C(CH2CO-2'-Pac))3
Trimer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateDUProstate CancerMTT/MTS assayIC50 =3.88nM24-hProstateNone
3191
177870262007
(K-Aib-C(CH2CO-2'-Pac))4
Dimer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateMCF-7Breast CancerMTT/MTS assayIC50 =0.62nM24-hBreastNone
3190
177870262007
(K-Aib-C(CH2CO-2'-Pac))3
Dimer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateDUProstate CancerMTT/MTS assayIC50 =2.85nM24-hProstateNone
3189
177870262007
(K-Aib-C(CH2CO-2'-Pac))2
Dimer of peptide-paclitaxel conjugate3LinearLAib = 1-amino-isobutyric acid ,Pac = PaclitaxelAmidationAcetylationAnticancerSynthetic peptide paclitaxel conjugateHeLaCervical CancerMTT/MTS assayIC50 =1.31nM24-hCervixNone
3188
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assayED50 =0.29 µM24-hBloodNone
3187
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assayED50 >10 µM24-hColonNone
3186
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assayED50 =0.210 µM24-hPancreaticNone
3185
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assayED50 =2.1 µM24-hOral mucosaNone
3184
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay94.5 % inhibition of cell proliferation at 10 µM24-hBloodNone
3183
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay54.3 % inhibition of cell proliferation at 1 µM24-hBloodNone
3182
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay34.7 % inhibition of cell proliferation at 100 nM72-hBloodNone
3181
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay18.7 % inhibition of cell proliferation at 10 nM24-hBloodNone
3180
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay10.4 % inhibition of cell proliferation at 1 nM24-hBloodNone
3179
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay27.9 % inhibition of cell proliferation at 10 µM24-hColonNone
3178
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay21.7 % inhibition of cell proliferation at 1 µM24-hColonNone
3177
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay16.8 % inhibition of cell proliferation at 100 nM72-hColonNone
3176
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay14.2 % inhibition of cell proliferation at 10 nM24-hColonNone
3175
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay16.5 % inhibition of cell proliferation at 1 nM24-hColonNone
3174
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay84.5 % inhibition of cell proliferation at 10 µM24-hPancreaticNone
3173
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay59.6 % inhibition of cell proliferation at 1 µM24-hPancreaticNone
3172
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay48.2 % inhibition of cell proliferation at 100 nM72-hPancreaticNone
3171
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay37.8 % inhibition of cell proliferation at 10 nM24-hPancreaticNone
3170
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay24.2 % inhibition of cell proliferation at 1 nM24-hPancreaticNone
3169
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay98.3 % inhibition of cell proliferation at 10 µM24-hOral mucosaNone
3168
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay43.1 % inhibition of cell proliferation at 1 µM24-hOral mucosaNone
3167
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay30.7 % inhibition of cell proliferation at 100 nM72-hOral mucosaNone
3166
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay18.2 % inhibition of cell proliferation at 10 nM24-hOral mucosaNone
3165
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay10.6 % inhibition of cell proliferation at 1 nM24-hOral mucosaNone
2900
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay35.2 % Cell viability at 100 µM72-hLiverNone
2899
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay41.1 % Cell viability at 75 µM72-hLiverNone
2898
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay49.7 % Cell viability at 50 µM72-hLiverNone
2897
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay63.3 % Cell viability at 25 µM72-hLiverNone
2896
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay72.1 % Cell viability at 12.5 µM72-hLiverNone
2895
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay48.6 % Cell viability at 100 µM48-hLiverNone
2894
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay54.3 % Cell viability at 100 µM48-hLiverNone
2893
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay62.8 % Cell viability at 75 µM48-hLiverNone
2892
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay75.6 % Cell viability at 50 µM48-hLiverNone
2891
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay87.3 % Cell viability at 25 µM48-hLiverNone
2890
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay54.2 % Cell viability at 100 µM24-hLiverNone
2889
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay71.5 % Cell viability at 75 µM24-hLiverNone
2888
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay76.3% Cell viability at 50 µM24-hLiverNone
2887
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay84.1% Cell viability at 25 µM24-hLiverNone
2886
203834642010
MNFNKLFVFVALVLAVCIGQSEAGWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLKG
Ceropin63LinearLNoneFreeFreeAntimicrobialMusca domesticaBEL-7402Liver CancerTrypan blue assay91.8% Cell viability at 12.5 µM24-hLiverNone
2881
202124532010
KWKLFKKIGAVLKVL
Camel15LinearLNoneFreeFreeAntimicrobialCeropin-Melittin hybridWM1158Skin CancerMTT/MTS assayLC50 = 4.1 µM24-hSkinNone
2880
202124532010
KWKLFKKIGAVLKVL
Camel15LinearLNoneFreeFreeAntimicrobialCeropin-Melittin hybrid4T1Breast CancerMTT/MTS assayLC50 = 6.2 µM24-hBreastNone
2879
202124532010
KWKLFKKIGAVLKVL
Camel15LinearLNoneFreeFreeAntimicrobialCeropin-Melittin hybridRENCARenal CancerMTT/MTS assayLC50 = 1.3 µM24-hRenalNone
2878
202124532010
KWKLFKKIGAVLKVL
Camel15LinearLNoneFreeFreeAntimicrobialCeropin-Melittin hybridB16-F10Skin CancerMTT/MTS assayLC50 = 1.75 µM24-hSkinNone
2871
167074642006
LKlLKKLlkKLLkLL
D-K6L915LinearMixNoneAmidationFreeAnticancerHost Defense lytic PeptideMB-231Prostate CancerEnzyme Immunoassay (EIA)LC50=3 µMol/L960-hProstateNone
2870
167074642006
LKlLKKLlkKLLkLL
D-K6L915LinearMixNoneAmidationFreeAnticancerHost DefenseÐLike Lytic PeptideCL-1Lung CancerEnzyme Immunoassay (EIA)LC50=3 µMol/LNot AvailableLungNone
2869
167074642006
LKlLKKLlkKLLkLL
D-K6L915LinearMixNoneAmidationFreeAnticancerHost Defense lytic Peptide22RV1Prostate CancerEnzyme Immunoassay (EIA)LC50=6 µMol/LNot AvailableProstateNone
1549
186563522008
KAQIRAMECNILGRKKRRQRRR
Tat-a522LinearLNoneFreeFreeAnticancerHIV-Tat (49-57)HCT-116Colon CancerMTT/MTS assay~80% Cytotoxicity at 100 µM24-hColonNone
1547
186563522008
KAQIRAMECNIL
A512LinearLNoneFreeFreeAnticancerCyclin B (285-296)HCT-116Colon CancerMTT/MTS assayNot Available24-hColonNone
1548
186563522008
RKKRRQRRR
Tat9LinearLNoneFreeFreeAnticancerHIV-Tat (49-57)HCT-116Colon CancerMTT/MTS assay~10% Cytotoxicity at 100 µM24-hColonNone
1542
166376462006
FKRIVQRIKDFLRNLV
dLL-37(17-32)c16LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayNot Available24-hNot AvailableNone
1541
166376462006
LLGDFKRIVQRIKDF
LL-37(1-4,17-27)15LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayNot Available24-hNot AvailableNone
1539
166376462006
FKRIVQRIKDFLRNLV
LL-37(17-32)b16LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayLC50=25 µM24-hNot AvailableNone
1540
166376462006
FKRIVQRIKDFLR
LL-37(17-29)13LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayLC50=55 µM24-hNot AvailableNone
1538
166376462006
IGKEFKRIVQRIKDFLRNLVPRTES
LL-37(13-37)25LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayLC50=38 µM24-hNot AvailableNone
1537
166376462006
LLGDFFRKSKEK
LL-37(1-12)12LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayNot Available24-hNot AvailableNone
1536
166376462006
FKRIVQRIKDFLRNLV
dLL-37(17-32)c16LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayNot Available24-hNot AvailableNone
1534
166376462006
FKRIVQRIKDFLR
LL-37(17-29)13LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayLC50=57 µM24-hNot AvailableNone
1535
166376462006
LLGDFKRIVQRIKDF
LL-37(1-4,17-27)15LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayNot Available24-hNot AvailableNone
1533
166376462006
FKRIVQRIKDFLRNLV
LL-37(17-32)b16LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayLC50=30 µM24-hNot AvailableNone
1532
166376462006
IGKEFKRIVQRIKDFLRNLVPRTES
LL-37(13-37)25LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayLC50=40 µM24-hNot AvailableNone
1531
166376462006
LLGDFFRKSKEK
LL-37(1-12)12LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayNot Available24-hNot AvailableNone
1530
166376462006
FKRiVQRiKDFlRNLV
dLL-37(17-32)c16LinearMixNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayNot Available24-hNot AvailableNone
1529
166376462006
LLGDFKRIVQRIKDF
LL-37(1-4,17-27)15LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayNot Available24-hNot AvailableNone
1528
166376462006
FKRIVQRIKDFLR
LL-37(17-29)13LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayLC50=60 µM24-hNot AvailableNone
1527
166376462006
FKRIVQRIKDFLRNLV
LL-37(17-32)b16LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayLC50=30 µM24-hNot AvailableNone
1526
166376462006
IGKEFKRIVQRIKDFLRNLVPRTES
LL-37(13-37)25LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayLC50=39 µM24-hNot AvailableNone
1525
166376462006
LLGDFFRKSKEK
LL-37(1-12)12LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayNot Available24-hNot AvailableNone
1423
16512752, 214039172006
AKRHHGYKRKFH
Demegen P-11312LinearLNoneAmidationFreeAntimicrobialAmphibian skin peptideU-937Lymphoma CancerMTT/MTS assay15% Cytotoxicity at 0.5 µg/ml6-hBloodNone
1422
10504394, 214039172009
GLFDVIKKVASVIGGL
Citropin1.116LinearLNoneAmidationFreeAntibacterialAustralian blue mountains tree frog, Litoria citropaU-937Lymphoma CancerMTT/MTS assay60% Cytotoxicity at 0.5 µg/ml6-hBloodNone
1421
10455241, 214039172009
GLFDVIKKVASVIGGL
Citropin1.116LinearLNoneAmidationFreeAntibacterialAustralian blue mountains tree frog, Litoria citropaU-937Lymphoma CancerMTT/MTS assay60% Cytotoxicity at 0.5 µg/ml6-hBloodNone
1353
184259922008
RKAFRWAWRMLKKAAPSITCVR
mPep122LinearLNoneFreeFreeAntimicrobialBovine lactoferrin (Lf-B)HL-60Skin CancerMTT/MTS assayIC50=8 µM24-hBloodNone
1352
184259922008
FKCRRWQWRMKKLGAPSITCVR
pep122LinearLNoneFreeFreeAntimicrobialBovine lactoferrin (Lf-B)HL-60Prostate CancerMTT/MTS assayIC50=77 µM24-hBloodNone
1350
189318812008
ETFSDLWKLL
PNC-2810LinearLNoneFreeFreeAnticancerAntennapediaMiaPaCa.2Pancreatic CancerMTT/MTS assayCytotoxicity=80% µMo/ml48-hPancreaticNone
1351
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothJ82Bladder CancerLDH leakage assayCytotoxicity=196.3 µg/ml48-hBladderNone
1349
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth647VBladder CancerLDH leakage assayIC50=181.1 µg/ml48-hBladderNone
1348
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothRT4Bladder CancerLDH leakage assayIC50=240.4 µg/ml48-hBladderNone
1347
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth486PBladder CancerLDH leakage assayIC50=232.4 µg/ml48-hBladderNone
1344
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)J82Bladder CancerLDH leakage assayIC50=319.2 µg/ml48-hBladderNone
1343
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)647VBladder CancerLDH leakage assayIC50=200.7 µg/ml48-hBladderNone
1342
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)RT4Bladder CancerLDH leakage assayIC50=289.3 µg/ml48-hBladderNone
1341
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)486PBladder CancerLDH leakage assayIC50=373.3/ µg/ml48-hBladderNone
1338
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothJ82Bladder CancerCell Viability assayIC50=77.51 µg/ml48-hBladderNone
1337
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth647VBladder CancerCell Viability assayIC50=61.86 µg/ml48-hBladderNone
1336
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothRT4Bladder CancerCell Viability assayIC50=92.9 µg/ml48-hBladderNone
1335
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth486PBladder CancerCell Viability assayIC50=87.47 µg/ml48-hBladderNone
1332
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)J82Bladder CancerCell Viability assayIC50=99.01 µg/ml48-hBladderNone
1331
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)647VBladder CancerCell Viability assayIC50=28.74 µg/ml48-hBladderNone
1330
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)RT4Bladder CancerCell Viability assayIC50=96.22 µg/ml48-hBladderNone
1329
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)486PBladder CancerCell Viability assayIC50=69.2 µg/ml48-hBladderNone
1326
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothJ82Bladder CancerWST-1 assayIC50=97.93 µg/ml48-hBladderNone
1325
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth647VBladder CancerWST-1 assayIC50=115.12 µg/ml48-hBladderNone
1324
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothRT4Bladder CancerWST-1 assayIC50=184.81 µg/ml48-hBladderNone
1323
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth486PBladder CancerWST-1 assayIC50=161.76 µg/ml48-hBladderNone
1320
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)J82Bladder CancerWST-1 assayIC50=212.07 µg/ml48-hBladderNone
1319
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)647VBladder CancerWST-1 assayIC50=185.39 µg/ml48-hBladderNone
1318
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)RT4Bladder CancerWST-1 assayIC50=231.26 µg/ml48-hBladderNone
1317
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)486PBladder CancerWST-1 assayIC50=251.47 µg/ml48-hBladderNone
1314
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin486P(G4)Bladder CancerCell Viability assayIC50=59.4 µM48-hBladderNone
1313
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin647V(G2)Bladder CancerCell Viability assayIC50=31 µM48-hBladderNone
1312
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skinRT4(G1)Bladder CancerCell Viability assayIC50=135.3 µM48-hBladderNone
1311
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin486P(G4)Bladder CancerWST-1 assayIC50=57.8 µM48-hBladderNone
1310
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin647V(G2)Bladder CancerWST-1 assayIC50=52.4 µM48-hBladderNone
1308
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin486P(G4)Bladder CancerLDH leakage assayIC50=28.6 µM48-hBladderNone
1309
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skinRT4(G1)Bladder CancerWST-1 assayIC50=484 µM48-hBladderNone
1307
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin647V(G2)Bladder CancerLDH leakage assayIC50=54.1 µM48-hBladderNone
1306
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skinRT4(G1)Bladder CancerLDH leakage assayIC50=32.3 µM48-hBladderNone
1115
165724232008
FKCRRWQWRMKKLGA
Lactoferricin B15LinearLNoneAmidationFreeAntimicrobialTemporins familySH-SY-5Y2Brain TumorMTT/MTS assayIC50=60 µM48-hBrainNone
1113
165724232008
FKCRRWQWRMKKLGA
Lactoferricin B15LinearLNoneAmidationFreeAntimicrobialTemporins familySK-N-DZBrain TumorMTT/MTS assayIC50=37 µM48-hBrainNone
1114
165724232008
FKCRRWQWRMKKLGA
Lactoferricin B15LinearLNoneAmidationFreeAntimicrobialTemporins familySHEP-12Brain TumorMTT/MTS assayIC50=45 µM48-hBrainNone
1112
165724232008
FKCRRWQWRMKKLGA
Lactoferricin B15LinearLNoneAmidationFreeAntimicrobialTemporins familyIMR-32Brain TumorMTT/MTS assayIC50=29 µM48-hBrainNone
1111
165724232008
FKCRRWQWRMKKLGA
Lactoferricin B15LinearLNoneAmidationFreeAntibacterialTemporins familyKellyBrain TumorMTT/MTS assayIC50=15.5 µM48-hBrainNone
1110
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ADU-145Prostate CancerMTT/MTS assayIC50=15.3 µg/ml48-hProstateNone
1108
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASW-620Colon CancerMTT/MTS assayIC50=12.7 µg/ml48-hColonNone
1109
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2APC-3Prostate CancerMTT/MTS assayIC50=12 µg/ml48-hProstateNone
1107
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AKM12Colon CancerMTT/MTS assayIC50=12 µg/ml48-hColonNone
1106
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHT-29Colon CancerMTT/MTS assayIC50=17.6 µg/ml48-hColonNone
1105
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHCT-15Colon CancerMTT/MTS assayIC50=13.2 µg/ml48-hColonNone
1103
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ACOLO-205Colon CancerMTT/MTS assayIC50=11.2 µg/ml48-hColonNone
1104
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHCT-116Colon CancerMTT/MTS assayIC50=14.6 µg/ml48-hColonNone
1102
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialHistone H2ASK-OV-3Ovarian CancerMTT/MTS assayIC50=12.6 µg/ml48-hOvaryNone
1101
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-8Ovarian CancerMTT/MTS assayIC50=13 µg/ml48-hOvaryNone
1100
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-5Ovarian CancerMTT/MTS assayIC50=13.8 µg/ml48-hOvaryNone
1099
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-4Ovarian CancerMTT/MTS assayIC50=17.6 µg/ml48-hOvaryNone
1098
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-3Ovarian CancerMTT/MTS assayIC50=15.2 µg/ml48-hOvaryNone
1097
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AIGROV1Ovarian CancerMTT/MTS assayIC50=9 µg/ml48-hOvaryNone
1096
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AUO-31Renal CancerMTT/MTS assayIC50=10.6 µg/ml48-hRenalNone
1094
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASN-12CRenal CancerMTT/MTS assayIC50=11.4 µg/ml48-hRenalNone
1095
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ATK-10Renal CancerMTT/MTS assayIC50=13.1 µg/ml48-hRenalNone
1093
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ARFX393Renal CancerMTT/MTS assayIC50=11 µg/ml48-hRenalNone
1092
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ACAKI-1Renal CancerMTT/MTS assayIC50=14.1 µg/ml48-hRenalNone
1091
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AACHNRenal CancerMTT/MTS assayIC50=12 µg/ml48-hRenalNone
1090
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AA-498Renal CancerMTT/MTS assayIC50=10 µg/ml48-hRenalNone
1089
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2A786-0Renal CancerMTT/MTS assayIC50=12.2 µg/ml48-hRenalNone
1088
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AUACC-62Skin CancerMTT/MTS assayIC50=10.6 µg/ml48-hSkinNone
1087
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AUACC-257Skin CancerMTT/MTS assayIC50=12.5 µg/ml48-hSkinNone
1086
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASK-MEL-5Skin CancerMTT/MTS assayIC50=8.9 µg/ml48-hSkinNone
1085
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASK-MEL-2Skin CancerMTT/MTS assayIC50=11.1 µg/ml48-hSkinNone
1083
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMALME-3MSkin CancerMTT/MTS assayIC50=10.9 µg/ml48-hSkinNone
1084
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AM14Skin CancerMTT/MTS assayIC50=15.1 µg/ml48-hSkinNone
1082
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ALOXIMVISkin CancerMTT/MTS assayIC50=9.5 µg/ml48-hSkinNone
1080
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASNB-75Brain TumorMTT/MTS assayIC50=15.5 µg/ml48-hBrainNone
1081
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AU-251Brain TumorMTT/MTS assayIC50=10.6 µg/ml48-hBrainNone
1079
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASNB-19Brain TumorMTT/MTS assayIC50=13.8 µg/ml48-hBrainNone
1078
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASF-539Brain TumorMTT/MTS assayIC50=9.5 µg/ml48-hBrainNone
1077
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASF-295Brain TumorMTT/MTS assayIC50=12.9 µg/ml48-hBrainNone
1076
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASF-268Brain TumorMTT/MTS assayIC50=12.4 µg/ml48-hBrainNone
1075
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H522Lung CancerMTT/MTS assayIC50=11.2 µg/ml48-hLungNone
1074
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H460Lung CancerMTT/MTS assayIC50=12.1 µg/ml48-hLungNone
1073
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H322MLung CancerMTT/MTS assayIC50=10.7 µg/ml48-hLungNone
1072
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H23Lung CancerMTT/MTS assayIC50=10.8 µg/ml48-hLungNone
1071
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H226Lung CancerMTT/MTS assayIC50=13.3 µg/ml48-hLungNone
1070
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHOP-92Lung CancerMTT/MTS assayIC50=7.2 µg/ml48-hLungNone
1069
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHOP-62Lung CancerMTT/MTS assayIC50=12.6 µg/ml48-hLungNone
1068
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AEKVXLung CancerMTT/MTS assayIC50=12.1 µg/ml48-hLungNone
1067
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AA-549Lung CancerMTT/MTS assayIC50=11.7 µg/ml48-hLungNone
1066
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AT-47DBreast CancerMTT/MTS assayIC50=23.9 µg/ml48-hBreastNone
1065
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ABT-549Breast CancerMTT/MTS assayIC50=12.9 µg/ml48-hBreastNone
1064
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMDA-NBreast CancerMTT/MTS assayIC50=10.6 µg/ml48-hBreastNone
1063
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMDA-MB-435Breast CancerMTT/MTS assayIC50=11.3 µg/ml48-hBreastNone
1062
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHS578TBreast CancerMTT/MTS assayIC50=11.7 µg/ml48-hBreastNone
1061
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMDA-MB-231Breast CancerMTT/MTS assayIC50=11.3 µg/ml48-hBreastNone
1060
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI/ADR-RESBreast CancerMTT/MTS assayIC50=11.5 µg/ml48-hBreastNone
1059
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMCF-7Breast CancerMTT/MTS assayIC50=15.1 µg/ml48-hBreastNone
1058
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASRLeukemia CancerMTT/MTS assayIC50=20.2 µg/ml48-hBloodNone
1057
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ARPMI-8226Leukemia CancerMTT/MTS assayIC50=10.5 µg/ml48-hBloodNone
1056
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMOLT-4Leukemia CancerMTT/MTS assayIC50=17 µg/ml48-hBloodNone
1055
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AK-562Leukemia CancerMTT/MTS assayIC50=8.2 µg/ml48-hBloodNone
1054
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHL-60Leukemia CancerMTT/MTS assayIC50=11.3 µg/ml48-hBloodNone
1053
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ACCRF-CEMLeukemia CancerMTT/MTS assayIC50=14.7 µg/ml48-hBloodNone
4695
206236342010
Not Available
OzarelixNot AvailableLinearLNoneFreeFreeAnticancerLHRH antagonistPC-3Prostate CancerCell Proliferation assayInhibited cell proliferation in a dose and time-dependent manner0-96 hProstateNone
4696
206236342010
Not Available
OzarelixNot AvailableLinearLNoneFreeFreeAnticancerLHRH antagonistDU-145Prostate CancerCell Proliferation assayInhibited cell proliferation in a dose and time-dependent manner0-96 hProstateNone
4690
261257202007
QPVLHLVALNTPLSGGMRGIRGADFQCFQQARAVGLSGTFRAFLSSRLQDLYSIVRRADRGSVPIVNLKDEVLSPSWDSLFSGSQGQLQPGARIFSFDGRDVLRHPAWPQKSVWHGSDPSGRRLMESYCETWRTETTGATGQASSLLSGRLLEQKAASCHNSYIVLCIENSF
Endostatin172LinearLNoneFreeFreeAntiangiogenicP. pastorisMFCStomach CancerIP injectionsTumor inhibition rate = 72.89%14 daysStomachNone