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| ID | PMID | YEAR | Sequence | Name | Length | Linear/Cyclic | Chirality | Chem-MOD | C-ter MOD | N-ter MOD | Nature | Origin | Cell Line | Cancer Type | Assay | Activity | Testing Time | Tissue Affected | Patents |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 20964334 | 2010 | Dex-(KW)3 | 6 | Linear | L | Dextran | Amidation | Dextran | Anticancer | Synthetic | PC-3 | Prostate Cancer | MTT/MTS assay | at 10 µM 60% viablity | Not Available | Prostate | None | ||
| 20964334 | 2010 | Dex-(KW)3 | 6 | Linear | L | Dextran | Amidation | Dextran | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT/MTS assay | at 10 µM 35-40% viablity | Not Available | Breast | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | Skmel-25 | Skin Cancer | MTT/MTS assay | at 100 µM 55-60% viablity | 48-h | Skin | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | Skmel-28 | Skin Cancer | MTT/MTS assay | at 100 µM 35-40% viablity | 48-h | Skin | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | B16F10-Nex 2 | Skin Cancer | MTT/MTS assay | at 100 µM 50% viablity | 48-h | Skin | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | A-2058 | Skin Cancer | MTT/MTS assay | at 100 µM 30% viablity | 48-h | Skin | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | MDA-MB-231 | Breast Cancer | MTT/MTS assay | at 100 µM 55% viablity | 48-h | Breast | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | at 100 µM 50% viablity | 48-h | Cervix | None | ||
| 20802991 | 2010 | Peptide-20 | 9 | Cyclic(C1-C9) | L | None | Free | Free | Antitumor | Synthetic Peptide | HL-60 | Leukemia Cancer | MTT/MTS assay | at 100 µM 90% viablity | 48-h | Blood | None | ||
| 17067680, 18957441 | 2007 | hepcidin TH1-5 | 22 | Not Available | L | None | Free | Free | Anticancer | Tilapia, Oreochromis mossambicus | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 17561225, 18957441 | 2007 | Phylloseptin-L1 | 32 | Not Available | L | None | Free | Free | Anticancer | Hylomantis lemur (Hylidae: Phyllomedusinae | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 17561225, 18957441 | 2007 | Phylloseptin | 32 | Not Available | L | None | Free | Free | Anticancer | Hylomantis lemur (Hylidae: Phyllomedusinae | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 19341344, 18957441 | 2009 | Temporin-1CEb | 17 | Not Available | L | None | Free | Free | Antimicrobial | Rana chensinensis, China, Asia | Not Available | Breast Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 18191970, 18957441 | 2008 | Vibi H | 31 | Not Available | L | None | Free | Free | Anticancer | Alpine violetViola biflora | Not Available | Lung Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 18191970, 18957441 | 2008 | Vibi E | 30 | Not Available | L | None | Free | Free | Anticancer | Alpine violetViola biflora | Not Available | Leukemia Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 18191970, 18957441 | 2008 | Vibi G | 31 | Not Available | L | None | Free | Free | Anticancer | Alpine violetViola biflora | Not Available | Skin Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 20198492, 18957441 | 2010 | Halictine 2 | 12 | Not Available | L | None | Free | Free | Anticancer | Venom, the eusocial bee, Halictus sexcinctus | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20198492, 18957441 | 2010 | Halictine 1 | 12 | Not Available | L | None | Free | Free | Anticancer | venom, the eusocial bee, Halictus sexcinctus | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20575512, 18957441 | 2010 | Psyle A | 28 | Not Available | L | None | Free | Free | Antibacterial | Psychotria leptothyrsa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20575512, 18957441 | 2010 | Psyle E | 31 | Not Available | L | None | Free | Free | Antibacterial | Psychotria leptothyrsa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20575512, 18957441 | 2010 | Psyle C | 25 | Not Available | L | None | Free | Free | Antibacterial | Psychotria leptothyrsa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 16713189, 18957441 | 2006 | Brevinin-1BYa | 24 | Not Available | L | None | Free | Free | Antibacterial | Rana boylii, North America | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Ranatuerin-2Ya | 28 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates yavapaiensis | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 17698251, 18957441 | 2007 | Dybowskin-2 | 17 | Not Available | L | None | Free | Free | Antibacterial | Rana dybowskii, Rana chensinensis, Asia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | SU.86.86 | Pancreatic Cancer | WST-1 assay | IC50= 8.0 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | Pane- 1 | Breast Cancer | WST-1 assay | IC50= 14.1 µM | 48-h | Breast | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | CFPAC-I | Pancreatic Cancer | WST-1 assay | IC50= 9.2 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BxPC-3 | Pancreatic Cancer | WST-1 assay | IC50= 14.7 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa363-377) -nLytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | SU.86.86 | Pancreatic Cancer | WST-1 assay | IC50= 7.9 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa363-377) -nLytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | Pane- 1 | Breast Cancer | WST-1 assay | IC50= 13.1 µM | 48-h | Breast | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa363-377) -nLytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | CFPAC-I | Pancreatic Cancer | WST-1 assay | IC50= 10.6 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa363-377) -nLytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BxPC-3 | Pancreatic Cancer | WST-1 assay | IC50= 12.5 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | EB(H2R)-lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | LNCaP | Prostate Cancer | WST-1 assay | IC50= 4.8 µM | Not Available | Prostate | US_8436137_B2 | ||
| None | 2009 | EB(H2R)-lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | SU.86.86 | Pancreatic Cancer | WST-1 assay | IC50= 7.4 µM | Not Available | Pancreatic | US_8436137_B2 | ||
| None | 2009 | EB(H2R)-lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BxPC-3 | Pancreatic Cancer | WST-1 assay | IC50= 6.6 µM | Not Available | Pancreatic | US_8436137_B2 | ||
| None | 2009 | EB(H2R)-lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | U-251 | Brain Tumor | WST-1 assay | IC50= 8.4 µM | Not Available | Brain | US_8436137_B2 | ||
| None | 2009 | EB(H2R)-lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BT-20 | Breast Cancer | WST-1 assay | IC50= 1.9 µM | Not Available | Breast | US_8436137_B2 | ||
| None | 2009 | EB(H2R)-lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | H-322 | Lung Cancer | WST-1 assay | IC50= 3.2 µM | Not Available | Lung | US_8436137_B2 | ||
| None | 2009 | EB-Lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | LNCaP | Prostate Cancer | WST-1 assay | IC50= 10 µM | Not Available | Prostate | US_8436137_B2 | ||
| None | 2009 | EB-Lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | SU.86.86 | Pancreatic Cancer | WST-1 assay | IC50= 12 µM | Not Available | Pancreatic | US_8436137_B2 | ||
| None | 2009 | EB-Lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BxPC-3 | Pancreatic Cancer | WST-1 assay | IC50= 12 µM | Not Available | Pancreatic | US_8436137_B2 | ||
| None | 2009 | EB-Lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | U-251 | Brain Tumor | WST-1 assay | IC50= 12 µM | Not Available | Brain | US_8436137_B2 | ||
| None | 2009 | EB-Lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BT-20 | Breast Cancer | WST-1 assay | IC50= 6.5 µM | Not Available | Breast | US_8436137_B2 | ||
| None | 2009 | EB-Lytic | 32 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | H-322 | Lung Cancer | WST-1 assay | IC50= 6.8 µM | Not Available | Lung | US_8436137_B2 | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 2% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 1% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 0% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 3% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 2% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 1% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 5% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 1% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 2% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 3% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 2% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 1% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 55% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 35% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 23% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 79% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 46% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 43% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 68% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 66% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 25% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 65% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 45% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 8% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 50% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 20% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 15% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 30% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | >50% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 20% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 80% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 80% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 30% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 30% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 10% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BadBH3 | 35 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 0% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 47.0% inhibition at 10-3M | 31.92-Min | Colon | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 2.2% inhibition at 10-6M | 31.92-Min | Breast | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 7.1% inhibition at 10-5M | 31.92-Min | Breast | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 6.9% inhibition at 10-4M | 31.92-Min | Breast | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 25.9% inhibition at 10-3M | 31.92-Min | Breast | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 70.7% inhibition at 10-5M | 31.92-Min | Skin | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 34.4% inhibition at 10-3M | 31.92-Min | Skin | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 9.2% inhibition at 10-3M | 31.92-Min | Colon | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 11.08% inhibition at 10-5M | 31.92-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 29.9% inhibition at 10-3M | 23.03-Min | Breast | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 3.9% inhibition at 10-5M | 31.92-Min | Larynx | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 45% inhibition at 10-3M | 31.92-Min | Larynx | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 9.3% inhibition at 10-3M | 31.92-Min | Cervix | None | ||
| 16722632 | 2006 | 23 | 6 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 4.1% inhibition at 10-6M | 31.92-Min | Skin | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 10.9% inhibition at 10-5M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 12.1% inhibition at 10-4M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 8.1% inhibition at 10-3M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 9.6% inhibition at 10-4M | 23.03-Min | Breast | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 13.1% inhibition at 10-5M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 14.6% inhibition at 10-4M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 38.4% inhibition at 10-3M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 17.7% inhibition at 10-6M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 16.2% inhibition at 10-6M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 6.6% inhibition at 10-5M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 5.1% inhibition at 10-4M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 14.5% inhibition at 10-3M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 26.4% inhibition at 10-6M | 23.03-Min | Colon | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 2.4% inhibition at 10-6M | 23.03-Min | Skin | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 4.5% inhibition at 10-5M | 23.03-Min | Skin | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 11.4% inhibition at 10-4M | 23.03-Min | Skin | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 23.2% inhibition at 10-3M | 23.03-Min | Skin | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 44.5% inhibition at 10-3M | 23.03-Min | Larynx | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 8.5% inhibition at 10-6M | 23.03-Min | Cervix | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 9.5% inhibition at 10-5M | 23.03-Min | Cervix | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 15.4% inhibition at 10-4M | 23.03-Min | Cervix | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 24.1% inhibition at 10-3M | 23.03-Min | Cervix | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 13.7% inhibition at 10-6M | 23.03-Min | Larynx | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 25.8% inhibition at 10-5M | 23.03-Min | Larynx | None | ||
| 16722632 | 2006 | 18 | 5 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 34.7% inhibition at 10-4M | 23.03-Min | Larynx | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 18.5% inhibition at 10-4M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 10.6% inhibition at 10-3M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 22.8% inhibition at 10-3M | 26.70-Min | Breast | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 3.0% inhibition at 10-6M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 8.4% inhibition at 10-5M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 24.7% inhibition at 10-4M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 29.0% inhibition at 10-3M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 23.7% inhibition at 10-3M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 12.2% inhibition at 10-6M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 15.5% inhibition at 10-5M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 3.3% inhibition at 10-6M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 11.0% inhibition at 10-5M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 7.9% inhibition at 10-4M | 26.70-Min | Colon | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 2.4% inhibition at 10-4M | 26.70-Min | Skin | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 18.3% inhibition at 10-3M | 26.70-Min | Skin | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 10.2% inhibition at 10-5M | 26.70-Min | Cervix | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 13.3% inhibition at 10-4M | 26.70-Min | Cervix | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 28.0% inhibition at 10-3M | 26.70-Min | Cervix | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 0.8% inhibition at 10-6M | 26.70-Min | Skin | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 1.4% inhibition at 10-5M | 26.70-Min | Skin | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 4.9% inhibition at 10-6M | 26.70-Min | Cervix | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 36.1% inhibition at 10-3M | 26.70-Min | Larynx | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 16.8% inhibition at 10-4M | 26.70-Min | Larynx | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 10.1% inhibition at 10-5M | 26.70-Min | Larynx | None | ||
| 16722632 | 2006 | 17 | 5 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 1.0% inhibition at 10-6M | 26.70-Min | Larynx | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 8.6% inhibition at 10-3M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 15.6% inhibition at 10-3M | 10.79-Min | Breast | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 6.9% inhibition at 10-5M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 8.1% inhibition at 10-4M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 13.5% inhibition at 10-4M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 25.3% inhibition at 10-3M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 8.1% inhibition at 10-6M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 17.0% inhibition at 10-6M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 13.5% inhibition at 10-5M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 12.4% inhibition at 10-4M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 22.4% inhibition at 10-3M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 19.4% inhibition at 10-3M | 10.79-Min | Skin | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 7.6% inhibition at 10-6M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 3.8% inhibition at 10-5M | 10.79-Min | Colon | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 28.2% inhibition at 10-3M | 10.79-Min | Cervix | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 1.2% inhibition at 10-5M | 10.79-Min | Skin | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 3.3% inhibition at 10-4M | 10.79-Min | Skin | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 11.7% inhibition at 10-5M | 10.79-Min | Cervix | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 11.6% inhibition at 10-4M | 10.79-Min | Cervix | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 12.6% inhibition at 10-4M | 10.79-Min | Larynx | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 26.4% inhibition at 10-3M | 10.79-Min | Larynx | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 11.0% inhibition at 10-6M | 10.79-Min | Cervix | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 4.6% inhibition at 10-6M | 10.79-Min | Larynx | None | ||
| 16722632 | 2006 | 16 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 4.9% inhibition at 10-5M | 10.79-Min | Larynx | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 6.2% inhibition at 10-3M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 21.2% inhibition at 10-3M | 9.53-Min | Breast | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 2.2% inhibition at 10-6M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 4.2% inhibition at 10-5M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 6.4% inhibition at 10-4M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 14.4% inhibition at 10-4M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 23.4% inhibition at 10-3M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 15.7% inhibition at 10-3M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 13.6% inhibition at 10-6M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 20.4% inhibition at 10-5M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 7.4% inhibition at 10-5M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 9.5% inhibition at 10-4M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 5.9% inhibition at 10-4M | 9.53-Min | Skin | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 17.9% inhibition at 10-3M | 9.53-Min | Skin | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 5.4% inhibition at 10-6M | 9.53-Min | Colon | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 1.6% inhibition at 10-6M | 9.53-Min | Skin | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 2.9% inhibition at 10-5M | 9.53-Min | Skin | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 7.3% inhibition at 10-5M | 9.53-Min | Cervix | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 9.9% inhibition at 10-4M | 9.53-Min | Cervix | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 28.2% inhibition at 10-3M | 9.53-Min | Cervix | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 26.7% inhibition at 10-3M | 9.53-Min | Larynx | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 9.8% inhibition at 10-6M | 9.53-Min | Cervix | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 2.7% inhibition at 10-6M | 9.53-Min | Larynx | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 2.0% inhibition at 10-5M | 9.53-Min | Larynx | None | ||
| 16722632 | 2006 | 15 | 4 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 18.8% inhibition at 10-4M | 9.53-Min | Larynx | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 7.7% inhibition at 10-4M | 14.05-Min | Breast | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 18.7% inhibition at 10-3M | 14.05-Min | Breast | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 10.7% inhibition at 10-6 | 14.05-Min | Colon | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 10.0% inhibition at 10-5 | 14.05-Min | Colon | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 8.3% inhibition at 10-5 | 14.05-Min | Colon | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 10.5% inhibition at 10-4 | 14.05-Min | Colon | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 21.8% inhibition at 10-3 | 14.05-Min | Colon | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 7.3% inhibition at 10-3 | 14.05-Min | Skin | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 0.7% inhibition at 10-6 | 14.05-Min | Colon | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 3.0% inhibition at 10-6 | 14.05-Min | Skin | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 4.7% inhibition at 10-5 | 14.05-Min | Skin | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 2.7% inhibition at 10-4 | 14.05-Min | Skin | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 11.0% inhibition at 10-4 | 14.05-Min | Cervix | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 20.5% inhibition at 10-3 | 14.05-Min | Cervix | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 7.2% inhibition at 10-6 | 14.05-Min | Cervix | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 17.1% inhibition at 10-5 | 14.05-Min | Cervix | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 4.9% inhibition at 10-5 | 14.05-Min | Larynx | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 1.9% inhibition at 10-4 | 14.05-Min | Larynx | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 16.2% inhibition at 10-3 | 14.05-Min | Larynx | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 17.8% inhibition at 10-3 | 12.46-Min | Breast | None | ||
| 16722632 | 2006 | 10 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 8.5% inhibition at 10-6 | 14.05-Min | Larynx | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 14.5% inhibition at 10-3 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 1.1% inhibition at 10-5 | 12.46-Min | Breast | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 1.2% inhibition at 10-4 | 12.46-Min | Breast | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 8.4% inhibition at 10-4 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 16.5% inhibition at 10-5 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 3.7% inhibition at 10-6 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 17.9% inhibition at 10-3 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 11.8% inhibition at 10-4 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 21.9% inhibition at 10-5 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 10.5% inhibition at 10-6 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 20.8% inhibition at 10-3 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 3.4% inhibition at 10-4 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 8.9% inhibition at 10-5 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 4.9% inhibition at 10-6 | 12.46-Min | Colon | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 7.3% inhibition at 10-3 | 12.46-Min | Skin | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 3.9% inhibition at 10-5 | 12.46-Min | Skin | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 14.8% inhibition at 10-3 | 12.46-Min | Cervix | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 6.1% inhibition at 10-5 | 12.46-Min | Cervix | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 3.1% inhibition at 10-4 | 12.46-Min | Cervix | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 7.5% inhibition at 10-6 | 12.46-Min | Cervix | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 21.2% inhibition at 10-3 | 12.46-Min | Larynx | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 8.2% inhibition at 10-4 | 12.46-Min | Larynx | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 6.4% inhibition at 10-5 | 12.46-Min | Larynx | None | ||
| 16722632 | 2006 | 9 | 3 | Linear | L | A* = Cα -dialkylated glycine (Aaa2,2 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 6.2% inhibition at 10-6 | 12.46-Min | Larynx | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 7.5% inhibition at 10-4 | 12.81-Min | Breast | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | MCF-7 | Breast Cancer | MTT/MTS assay | 2.4% inhibition at 10-5 | 12.81-Min | Breast | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 18.9% inhibition at 10-4 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 26.4% inhibition at 10-3 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 22.7% inhibition at 10-5 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | CaCo-2 | Colon Cancer | MTT/MTS assay | 3.5% inhibition at 10-6 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 28.1% inhibition at 10-4 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 58.2% inhibition at 10-3 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 16.5% inhibition at 10-5 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | SW-620 | Colon Cancer | MTT/MTS assay | 12.9% inhibition at 10-6 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 26.5% inhibition at 10-3 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 1.6% inhibition at 10-5 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 5.4% inhibition at 10-4 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 14% inhibition at 10-3 | 12.81-Min | Skin | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HT-29 | Colon Cancer | MTT/MTS assay | 9.8% inhibition at 10-6 | 12.81-Min | Colon | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 7.5% inhibition at 10-4 | 12.81-Min | Skin | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 14% inhibition at 10-5 | 12.81-Min | Skin | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HBL | Skin Cancer | MTT/MTS assay | 6.5% inhibition at 10-6 | 12.81-Min | Skin | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 36.1% inhibition at 10-3 | 12.81-Min | Not Available | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 8.2% inhibition at 10-4 | 12.81-Min | Not Available | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HeLa | Cervical Cancer | MTT/MTS assay | 10% inhibition at 10-5 | 12.81-Min | Not Available | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 30.4% inhibition at 10-3 | 12.81-Min | Not Available | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 24.9% inhibition at 10-4 | 12.81-Min | Not Available | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 19.7% inhibition at 10-5 | 12.81-Min | Not Available | None | ||
| 16722632 | 2006 | 8 | 2 | Linear | L | A* = Cαα -dialkylated glycine (Aaa1,1 ) | Free | Free | Antitumor | Synthetic Peptide | HEp-2 | Larynx Cancer | MTT/MTS assay | 14.2% inhibition at 10-6 | 12.81-Min | Not Available | None | ||
| 20515045 | 2010 | AP(O) | 25 | Cyclic(C2-C10,C | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 52% inhibition at 10µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP(O) | 25 | Cyclic(C2-C10,C | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 42% inhibition at 5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP(O) | 25 | Cyclic(C2-C10,C | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 40% inhibition at 2.5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP | 25 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 75% inhibition at 10µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP | 25 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 40% inhibition at 5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP | 25 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 50% inhibition at 2.5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | ES-2 | 11 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 60% inhibition at 10µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | ES-2 | 11 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 60% inhibition at 5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | ES-2 | 11 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 60% inhibition at 2.5µg/ml | NA | Not Available | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 6.5 ± 1.07% cell viability at 80 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 26.9 ± 0.5% cell viability at 60 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 47.5 ± 1.66% cell viability at 40 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 63.8 ± 0.8% cell viability at 20 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 86 ± 0.57% cell viability at 10 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 13.8 ± 1.44% cell viability at 80 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 31.5 ± 1.49% cell viability at 60 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 50 ± 3.09% cell viability at 40 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 71.1 ± 2.84% cell viability at 20 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Bovine lactoferrin (Lf-B) | M14 | Skin Cancer | MTT/MTS assay | 92.2 ± 1.02% cell viability at 10 µM | NA | Skin | None | ||
| 19527490 | 2009 | KW5 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic peptide | HT-29 | Colon Cancer | MTT/MTS assay | IC50 =55±14 µM | NA | Colon | None | ||
| 19527490 | 2009 | KW5 | 21 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | FEMX | Skin Cancer | MTT/MTS assay | IC50 =30±3 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | Ramos | Lymphoma Cancer | MTT/MTS assay | IC50 = 10 µM | NA | Blood | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | Raji | Lymphoma Cancer | MTT/MTS assay | IC50 = 13 µM | NA | Blood | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | Sudhl-4 | Skin Cancer | MTT/MTS assay | IC50 = 16 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | KMM-1 | Skin Cancer | MTT/MTS assay | IC50 = 57 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | U-266 | Lymphoma Cancer | MTT/MTS assay | IC50 = 55 µM | NA | Blood | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | KMS-5 | Skin Cancer | MTT/MTS assay | IC50 = 38 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | HT-29 | Colon Cancer | MTT/MTS assay | IC50 =148±8 µM | NA | Colon | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | FEMX | Skin Cancer | MTT/MTS assay | IC50 =40±7 µM | NA | Skin | None | ||
| 18815734 | 2008 | di-PST13-RK-K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =10 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | di-PST13-RK-K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 =15 µg/ml | NA | Lung | None | ||
| 18815734 | 2008 | di-PST13-RK-C | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =17 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | di-PST13-RK-C | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 =17 µg/ml | NA | Lung | None | ||
| 18815734 | 2008 | PST13-RK | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =80 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | PST13-RK | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 =90 µg/ml | NA | Lung | None | ||
| 18815734 | 2008 | Tritrpticin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =142 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | Tritrpticin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 >200 µg/ml | NA | Lung | None | ||
| 17787026 | 2007 | Tetramer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 =0.64nM | 24-h | Breast | None | ||
| 17787026 | 2007 | Tetramer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | HeLa | Cervical Cancer | MTT/MTS assay | IC50 =0.96nM | 24-h | Cervix | None | ||
| 17787026 | 2007 | Tetramer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | DU | Prostate Cancer | MTT/MTS assay | IC50 =1.30nM | 24-h | Prostate | None | ||
| 17787026 | 2007 | Trimer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 =3.00nM | 24-h | Breast | None | ||
| 17787026 | 2007 | Trimer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | HeLa | Cervical Cancer | MTT/MTS assay | IC50 =1.70nM | 24-h | Cervix | None | ||
| 17787026 | 2007 | Trimer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | DU | Prostate Cancer | MTT/MTS assay | IC50 =3.88nM | 24-h | Prostate | None | ||
| 17787026 | 2007 | Dimer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 =0.62nM | 24-h | Breast | None | ||
| 17787026 | 2007 | Dimer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | DU | Prostate Cancer | MTT/MTS assay | IC50 =2.85nM | 24-h | Prostate | None | ||
| 17787026 | 2007 | Dimer of peptide-paclitaxel conjugate | 3 | Linear | L | Aib = 1-amino-isobutyric acid ,Pac = Paclitaxel | Amidation | Acetylation | Anticancer | Synthetic peptide paclitaxel conjugate | HeLa | Cervical Cancer | MTT/MTS assay | IC50 =1.31nM | 24-h | Cervix | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MOLT-4 | Leukemia Cancer | MTT/MTS assay | ED50 =0.29 µM | 24-h | Blood | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | PTC | Colon Cancer | MTT/MTS assay | ED50 >10 µM | 24-h | Colon | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | ED50 =0.210 µM | 24-h | Pancreatic | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | KB | Oral Cancer | MTT/MTS assay | ED50 =2.1 µM | 24-h | Oral mucosa | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MOLT-4 | Leukemia Cancer | MTT/MTS assay | 94.5 % inhibition of cell proliferation at 10 µM | 24-h | Blood | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MOLT-4 | Leukemia Cancer | MTT/MTS assay | 54.3 % inhibition of cell proliferation at 1 µM | 24-h | Blood | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MOLT-4 | Leukemia Cancer | MTT/MTS assay | 34.7 % inhibition of cell proliferation at 100 nM | 72-h | Blood | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MOLT-4 | Leukemia Cancer | MTT/MTS assay | 18.7 % inhibition of cell proliferation at 10 nM | 24-h | Blood | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MOLT-4 | Leukemia Cancer | MTT/MTS assay | 10.4 % inhibition of cell proliferation at 1 nM | 24-h | Blood | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | PTC | Colon Cancer | MTT/MTS assay | 27.9 % inhibition of cell proliferation at 10 µM | 24-h | Colon | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | PTC | Colon Cancer | MTT/MTS assay | 21.7 % inhibition of cell proliferation at 1 µM | 24-h | Colon | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | PTC | Colon Cancer | MTT/MTS assay | 16.8 % inhibition of cell proliferation at 100 nM | 72-h | Colon | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | PTC | Colon Cancer | MTT/MTS assay | 14.2 % inhibition of cell proliferation at 10 nM | 24-h | Colon | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | PTC | Colon Cancer | MTT/MTS assay | 16.5 % inhibition of cell proliferation at 1 nM | 24-h | Colon | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | 84.5 % inhibition of cell proliferation at 10 µM | 24-h | Pancreatic | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | 59.6 % inhibition of cell proliferation at 1 µM | 24-h | Pancreatic | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | 48.2 % inhibition of cell proliferation at 100 nM | 72-h | Pancreatic | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | 37.8 % inhibition of cell proliferation at 10 nM | 24-h | Pancreatic | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | 24.2 % inhibition of cell proliferation at 1 nM | 24-h | Pancreatic | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | KB | Oral Cancer | MTT/MTS assay | 98.3 % inhibition of cell proliferation at 10 µM | 24-h | Oral mucosa | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | KB | Oral Cancer | MTT/MTS assay | 43.1 % inhibition of cell proliferation at 1 µM | 24-h | Oral mucosa | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | KB | Oral Cancer | MTT/MTS assay | 30.7 % inhibition of cell proliferation at 100 nM | 72-h | Oral mucosa | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | KB | Oral Cancer | MTT/MTS assay | 18.2 % inhibition of cell proliferation at 10 nM | 24-h | Oral mucosa | None | ||
| 17559067 | 2007 | Peptide 5 | 40 | Linear | Mix | Aib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and Pen | Amidation | Free | Anticancer | Synthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P a | KB | Oral Cancer | MTT/MTS assay | 10.6 % inhibition of cell proliferation at 1 nM | 24-h | Oral mucosa | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 35.2 % Cell viability at 100 µM | 72-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 41.1 % Cell viability at 75 µM | 72-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 49.7 % Cell viability at 50 µM | 72-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 63.3 % Cell viability at 25 µM | 72-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 72.1 % Cell viability at 12.5 µM | 72-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 48.6 % Cell viability at 100 µM | 48-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 54.3 % Cell viability at 100 µM | 48-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 62.8 % Cell viability at 75 µM | 48-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 75.6 % Cell viability at 50 µM | 48-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 87.3 % Cell viability at 25 µM | 48-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 54.2 % Cell viability at 100 µM | 24-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 71.5 % Cell viability at 75 µM | 24-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 76.3% Cell viability at 50 µM | 24-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 84.1% Cell viability at 25 µM | 24-h | Liver | None | ||
| 20383464 | 2010 | Ceropin | 63 | Linear | L | None | Free | Free | Antimicrobial | Musca domestica | BEL-7402 | Liver Cancer | Trypan blue assay | 91.8% Cell viability at 12.5 µM | 24-h | Liver | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | WM1158 | Skin Cancer | MTT/MTS assay | LC50 = 4.1 µM | 24-h | Skin | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | 4T1 | Breast Cancer | MTT/MTS assay | LC50 = 6.2 µM | 24-h | Breast | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | RENCA | Renal Cancer | MTT/MTS assay | LC50 = 1.3 µM | 24-h | Renal | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | B16-F10 | Skin Cancer | MTT/MTS assay | LC50 = 1.75 µM | 24-h | Skin | None | ||
| 16707464 | 2006 | D-K6L9 | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Host Defense lytic Peptide | MB-231 | Prostate Cancer | Enzyme Immunoassay (EIA) | LC50=3 µMol/L | 960-h | Prostate | None | ||
| 16707464 | 2006 | D-K6L9 | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Host DefenseÐLike Lytic Peptide | CL-1 | Lung Cancer | Enzyme Immunoassay (EIA) | LC50=3 µMol/L | Not Available | Lung | None | ||
| 16707464 | 2006 | D-K6L9 | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Host Defense lytic Peptide | 22RV1 | Prostate Cancer | Enzyme Immunoassay (EIA) | LC50=6 µMol/L | Not Available | Prostate | None | ||
| 18656352 | 2008 | Tat-a5 | 22 | Linear | L | None | Free | Free | Anticancer | HIV-Tat (49-57) | HCT-116 | Colon Cancer | MTT/MTS assay | ~80% Cytotoxicity at 100 µM | 24-h | Colon | None | ||
| 18656352 | 2008 | A5 | 12 | Linear | L | None | Free | Free | Anticancer | Cyclin B (285-296) | HCT-116 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | None | ||
| 18656352 | 2008 | Tat | 9 | Linear | L | None | Free | Free | Anticancer | HIV-Tat (49-57) | HCT-116 | Colon Cancer | MTT/MTS assay | ~10% Cytotoxicity at 100 µM | 24-h | Colon | None | ||
| 16637646 | 2006 | dLL-37(17-32)c | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-4,17-27) | 15 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-32)b | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | LC50=25 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-29) | 13 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | LC50=55 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(13-37) | 25 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | LC50=38 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-12) | 12 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | dLL-37(17-32)c | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-29) | 13 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | LC50=57 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-4,17-27) | 15 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-32)b | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | LC50=30 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(13-37) | 25 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | LC50=40 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-12) | 12 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | dLL-37(17-32)c | 16 | Linear | Mix | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-4,17-27) | 15 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-29) | 13 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | LC50=60 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-32)b | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | LC50=30 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(13-37) | 25 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | LC50=39 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-12) | 12 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16512752, 21403917 | 2006 | Demegen P-113 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Amphibian skin peptide | U-937 | Lymphoma Cancer | MTT/MTS assay | 15% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 10504394, 21403917 | 2009 | Citropin1.1 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Australian blue mountains tree frog, Litoria citropa | U-937 | Lymphoma Cancer | MTT/MTS assay | 60% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 10455241, 21403917 | 2009 | Citropin1.1 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Australian blue mountains tree frog, Litoria citropa | U-937 | Lymphoma Cancer | MTT/MTS assay | 60% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 18425992 | 2008 | mPep1 | 22 | Linear | L | None | Free | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | HL-60 | Skin Cancer | MTT/MTS assay | IC50=8 µM | 24-h | Blood | None | ||
| 18425992 | 2008 | pep1 | 22 | Linear | L | None | Free | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | HL-60 | Prostate Cancer | MTT/MTS assay | IC50=77 µM | 24-h | Blood | None | ||
| 18931881 | 2008 | PNC-28 | 10 | Linear | L | None | Free | Free | Anticancer | Antennapedia | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | Cytotoxicity=80% µMo/ml | 48-h | Pancreatic | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | J82 | Bladder Cancer | LDH leakage assay | Cytotoxicity=196.3 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | 647V | Bladder Cancer | LDH leakage assay | IC50=181.1 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | RT4 | Bladder Cancer | LDH leakage assay | IC50=240.4 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | 486P | Bladder Cancer | LDH leakage assay | IC50=232.4 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | J82 | Bladder Cancer | LDH leakage assay | IC50=319.2 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | 647V | Bladder Cancer | LDH leakage assay | IC50=200.7 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | RT4 | Bladder Cancer | LDH leakage assay | IC50=289.3 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | 486P | Bladder Cancer | LDH leakage assay | IC50=373.3/ µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | J82 | Bladder Cancer | Cell Viability assay | IC50=77.51 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | 647V | Bladder Cancer | Cell Viability assay | IC50=61.86 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | RT4 | Bladder Cancer | Cell Viability assay | IC50=92.9 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | 486P | Bladder Cancer | Cell Viability assay | IC50=87.47 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | J82 | Bladder Cancer | Cell Viability assay | IC50=99.01 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | 647V | Bladder Cancer | Cell Viability assay | IC50=28.74 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | RT4 | Bladder Cancer | Cell Viability assay | IC50=96.22 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | 486P | Bladder Cancer | Cell Viability assay | IC50=69.2 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | J82 | Bladder Cancer | WST-1 assay | IC50=97.93 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | 647V | Bladder Cancer | WST-1 assay | IC50=115.12 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | RT4 | Bladder Cancer | WST-1 assay | IC50=184.81 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin B | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese oak silk moth | 486P | Bladder Cancer | WST-1 assay | IC50=161.76 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | J82 | Bladder Cancer | WST-1 assay | IC50=212.07 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | 647V | Bladder Cancer | WST-1 assay | IC50=185.39 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | RT4 | Bladder Cancer | WST-1 assay | IC50=231.26 µg/ml | 48-h | Bladder | None | ||
| 18315881 | 2008 | Cecropin A | 37 | Linear | L | None | Amidation | Free | Antimicrobial | Hyalophora Cecropia(silkmoth) | 486P | Bladder Cancer | WST-1 assay | IC50=251.47 µg/ml | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 486P(G4) | Bladder Cancer | Cell Viability assay | IC50=59.4 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 647V(G2) | Bladder Cancer | Cell Viability assay | IC50=31 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | RT4(G1) | Bladder Cancer | Cell Viability assay | IC50=135.3 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 486P(G4) | Bladder Cancer | WST-1 assay | IC50=57.8 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 647V(G2) | Bladder Cancer | WST-1 assay | IC50=52.4 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 486P(G4) | Bladder Cancer | LDH leakage assay | IC50=28.6 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | RT4(G1) | Bladder Cancer | WST-1 assay | IC50=484 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 647V(G2) | Bladder Cancer | LDH leakage assay | IC50=54.1 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | RT4(G1) | Bladder Cancer | LDH leakage assay | IC50=32.3 µM | 48-h | Bladder | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | SH-SY-5Y2 | Brain Tumor | MTT/MTS assay | IC50=60 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | SK-N-DZ | Brain Tumor | MTT/MTS assay | IC50=37 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | SHEP-12 | Brain Tumor | MTT/MTS assay | IC50=45 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | IMR-32 | Brain Tumor | MTT/MTS assay | IC50=29 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antibacterial | Temporins family | Kelly | Brain Tumor | MTT/MTS assay | IC50=15.5 µM | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | DU-145 | Prostate Cancer | MTT/MTS assay | IC50=15.3 µg/ml | 48-h | Prostate | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SW-620 | Colon Cancer | MTT/MTS assay | IC50=12.7 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | PC-3 | Prostate Cancer | MTT/MTS assay | IC50=12 µg/ml | 48-h | Prostate | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | KM12 | Colon Cancer | MTT/MTS assay | IC50=12 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HT-29 | Colon Cancer | MTT/MTS assay | IC50=17.6 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HCT-15 | Colon Cancer | MTT/MTS assay | IC50=13.2 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | COLO-205 | Colon Cancer | MTT/MTS assay | IC50=11.2 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HCT-116 | Colon Cancer | MTT/MTS assay | IC50=14.6 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | Histone H2A | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50=12.6 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-8 | Ovarian Cancer | MTT/MTS assay | IC50=13 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-5 | Ovarian Cancer | MTT/MTS assay | IC50=13.8 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-4 | Ovarian Cancer | MTT/MTS assay | IC50=17.6 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-3 | Ovarian Cancer | MTT/MTS assay | IC50=15.2 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | IGROV1 | Ovarian Cancer | MTT/MTS assay | IC50=9 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | UO-31 | Renal Cancer | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SN-12C | Renal Cancer | MTT/MTS assay | IC50=11.4 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | TK-10 | Renal Cancer | MTT/MTS assay | IC50=13.1 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | RFX393 | Renal Cancer | MTT/MTS assay | IC50=11 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | CAKI-1 | Renal Cancer | MTT/MTS assay | IC50=14.1 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | ACHN | Renal Cancer | MTT/MTS assay | IC50=12 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | A-498 | Renal Cancer | MTT/MTS assay | IC50=10 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | 786-0 | Renal Cancer | MTT/MTS assay | IC50=12.2 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | UACC-62 | Skin Cancer | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | UACC-257 | Skin Cancer | MTT/MTS assay | IC50=12.5 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SK-MEL-5 | Skin Cancer | MTT/MTS assay | IC50=8.9 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50=11.1 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MALME-3M | Skin Cancer | MTT/MTS assay | IC50=10.9 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | M14 | Skin Cancer | MTT/MTS assay | IC50=15.1 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | LOXIMVI | Skin Cancer | MTT/MTS assay | IC50=9.5 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SNB-75 | Brain Tumor | MTT/MTS assay | IC50=15.5 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | U-251 | Brain Tumor | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SNB-19 | Brain Tumor | MTT/MTS assay | IC50=13.8 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SF-539 | Brain Tumor | MTT/MTS assay | IC50=9.5 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SF-295 | Brain Tumor | MTT/MTS assay | IC50=12.9 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SF-268 | Brain Tumor | MTT/MTS assay | IC50=12.4 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H522 | Lung Cancer | MTT/MTS assay | IC50=11.2 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H460 | Lung Cancer | MTT/MTS assay | IC50=12.1 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H322M | Lung Cancer | MTT/MTS assay | IC50=10.7 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H23 | Lung Cancer | MTT/MTS assay | IC50=10.8 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H226 | Lung Cancer | MTT/MTS assay | IC50=13.3 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HOP-92 | Lung Cancer | MTT/MTS assay | IC50=7.2 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HOP-62 | Lung Cancer | MTT/MTS assay | IC50=12.6 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | EKVX | Lung Cancer | MTT/MTS assay | IC50=12.1 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | A-549 | Lung Cancer | MTT/MTS assay | IC50=11.7 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | T-47D | Breast Cancer | MTT/MTS assay | IC50=23.9 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | BT-549 | Breast Cancer | MTT/MTS assay | IC50=12.9 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MDA-N | Breast Cancer | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MDA-MB-435 | Breast Cancer | MTT/MTS assay | IC50=11.3 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HS578T | Breast Cancer | MTT/MTS assay | IC50=11.7 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=11.3 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI/ADR-RES | Breast Cancer | MTT/MTS assay | IC50=11.5 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=15.1 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SR | Leukemia Cancer | MTT/MTS assay | IC50=20.2 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | RPMI-8226 | Leukemia Cancer | MTT/MTS assay | IC50=10.5 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MOLT-4 | Leukemia Cancer | MTT/MTS assay | IC50=17 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=8.2 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50=11.3 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50=14.7 µg/ml | 48-h | Blood | None | ||
| 20623634 | 2010 | Ozarelix | Not Available | Linear | L | None | Free | Free | Anticancer | LHRH antagonist | PC-3 | Prostate Cancer | Cell Proliferation assay | Inhibited cell proliferation in a dose and time-dependent manner | 0-96 h | Prostate | None | ||
| 20623634 | 2010 | Ozarelix | Not Available | Linear | L | None | Free | Free | Anticancer | LHRH antagonist | DU-145 | Prostate Cancer | Cell Proliferation assay | Inhibited cell proliferation in a dose and time-dependent manner | 0-96 h | Prostate | None | ||
| 26125720 | 2007 | Endostatin | 172 | Linear | L | None | Free | Free | Antiangiogenic | P. pastoris | MFC | Stomach Cancer | IP injections | Tumor inhibition rate = 72.89% | 14 days | Stomach | None |