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| ID | PMID | YEAR | Sequence | Name | Length | Linear/Cyclic | Chirality | Chem-MOD | C-ter MOD | N-ter MOD | Nature | Origin | Cell Line | Cancer Type | Assay | Activity | Testing Time | Tissue Affected | Patents |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 37251837 | 2023 | Not Available | CPSA-CPSC-L-ACAN | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Recombinant Fusion Peptide | HeLa | Cervical Cancer | MTT assay | IC50 = 63.15 μg/ml | 24-h | Cervix | None | |
| 34361728 | 2021 | Structure given in figure | GA - 8 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 60.70 ± 0.6 µg/mL | 24-h | Colon | None | |
| 34361728 | 2021 | Structure given in figure | GA - 7 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.30 ± 0.1 µg/mL | 24-h | Liver | None | |
| 34361728 | 2021 | Structure given in figure | GA - 8 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 6.90 ± 1.1 µg/mL | 24-h | Breast | None | |
| 34361728 | 2021 | Structure given in figure | GA - 7 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.70 ± 0.2 µg/mL | 24-h | Breast | None | |
| 34361728 | 2021 | Structure given in figure | GA - 7 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.0 ± 1.1 µg/mL | 24-h | Colon | None | |
| 34361728 | 2021 | Structure given in figure | GA - 5 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.0 ± 0.3 µg/mL | 24-h | Breast | None | |
| 34361728 | 2021 | Structure given in figure | GA - 5 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 5.2 ± 0.8 µg/mL | 24-h | Colon | None | |
| 34361728 | 2021 | Structure given in figure | GA - 4 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 73.0 ± 1.4 µg/mL | 24-h | Colon | None | |
| 34361728 | 2021 | Structure given in figure | GA - 3 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 7.40 ± 0.4 µg/mL | 24-h | Colon | None | |
| 34361728 | 2021 | Structure given in figure | GA - 4 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 6.10 ± 0.4 µg/mL | 24-h | Breast | None | |
| 34361728 | 2021 | Structure given in figure | GA - 2 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 70.30 ± 0.9 µg/mL | 24-h | Colon | None | |
| 34361728 | 2021 | Structure given in figure | GA - 3 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.1 ± 0.7 µg/mL | 24-h | Breast | None | |
| 34361728 | 2021 | Structure given in figure | GA - 2 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.70 ± 1.3 µg/mL | 24-h | Breast | None | |
| 33005727 | 2020 | Not Available | LRH7-G5 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Synthetic | HCC-1937 | Breast Cancer | MTT assay | 60% cell viability at 0.1 μM | 48-h | Breast | None | |
| 33005727 | 2020 | Not Available | LRH7-G5 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | 60% cell viability at 0.01 μM | 48-h | Breast | None | |
| 32121469 | 2020 | Figure given in Scheme 1 | branched tetrapeptide Schiff bases derivative 5e | Not Available | Cyclic | L | chiral N3,N5-bis[(l-phenylalaninyl-l-leucinyl) substituted aryl or heterocyclic Schiff base]pyridine | Not Available | Not Available | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM | NA | Breast | None | |
| 32121469 | 2020 | Figure given in Scheme 1 | branched tetrapeptide Schiff bases derivative 5d | Not Available | Cyclic | L | chiral N3,N5-bis[(l-phenylalaninyl-l-leucinyl) substituted aryl or heterocyclic Schiff base]pyridine | Not Available | Not Available | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM | NA | Breast | None | |
| 32121469 | 2020 | Figure given in Scheme 1 | branched tetrapeptide Schiff bases derivative 5c | Not Available | Cyclic | L | chiral N3,N5-bis[(l-phenylalaninyl-l-leucinyl) substituted aryl or heterocyclic Schiff base]pyridine | Not Available | Not Available | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM | NA | Breast | None | |
| 32121469 | 2020 | Figure given in Scheme 1 | branched tetrapeptide Schiff bases derivative 4c | Not Available | Cyclic | L | chiral N3,N5-bis[(l-phenylalaninyl-l-leucinyl) substituted aryl or heterocyclic Schiff base]pyridine | Not Available | Not Available | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM | NA | Breast | None | |
| 32121469 | 2020 | Figure given in Scheme 1 | branched tetrapeptide Schiff bases derivative 4b | Not Available | Cyclic | L | chiral N3,N5-bis[(l-phenylalaninyl-l-leucinyl) substituted aryl or heterocyclic Schiff base]pyridine | Not Available | Not Available | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM | NA | Breast | None | |
| 32121469 | 2020 | Figure given in Scheme 1 | branched tetrapeptide Schiff bases derivative 4a | Not Available | Cyclic | L | chiral N3,N5-bis[(l-phenylalaninyl-l-leucinyl) substituted aryl or heterocyclic Schiff base]pyridine | Not Available | Not Available | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 between 8.12 ± 0.14 to 17.55 ± 0.27 μM | NA | Breast | None | |
| 31089358 | 2019 | Not Available | ICD-85 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Active fractions from Gloydius halys and Hemiscorpius lepturus | MCF-7 | Breast Cancer | Neutral Red Uptake assay | IC50 = 21.97 ± 0.63 μg/mL | 24 h | Breast | None | |
| 31089358 | 2019 | Not Available | ICD-85 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Active fractions from Gloydius halys and Hemiscorpius lepturus | MCF-7 | Breast Cancer | MTT assay | IC50 = 36.45 ± 0.38 μg/mL | 24 h | Breast | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | LN229 | Brain Tumor | MTT assay | IC50 = 13.32 ± 1.15 mg/ml | 72-h | Brain | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | PC-9 | Lung Cancer | MTT assay | IC50 = 7.921 ± 1.19 mg/ml | 72-h | Lung | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | HT-29 | Colon Cancer | MTT assay | IC50 = 11.55 ± 3.33 mg/ml | 72-h | Colon | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | PANC-1 | Pancreatic Cancer | MTT assay | IC50 = 8.224 ± 1.43 mg/ml | 72-h | Pancreas | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | A-549 | Lung Cancer | MTT assay | IC50 = 9.921 ± 0.82 mg/ml | 72-h | Lung | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | H-460 | Lung Cancer | MTT assay | IC50 = 9.083 ± 1.22 mg/ml | 72-h | Lung | None | |
| 29921888 | 2019 | Not Available | Silk Fibroin peptide | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Silkworm Cocoons | SW-1990 | Pancreatic Cancer | MTT assay | IC50 = 8.005 ± 1.34 mg/ml | 72-h | Pancreas | None | |
| 27218227 | 2017 | Not Available | Tr3 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | HT-29 | Colon Cancer | MTT assay | IC50 = 112.89 μg/mL | 48-h | Colon | None | |
| 27218227 | 2017 | Not Available | Tr4 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | MCF-7 | Breast Cancer | MTT assay | IC50 = 238.86 μg/mL | 48-h | Breast | None | |
| 27218227 | 2017 | Not Available | Tr4 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | HepG-2 | Liver Cancer | MTT assay | IC50 = 176.37 μg/mL | 48-h | Liver | None | |
| 27218227 | 2017 | Not Available | Tr2 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | HepG-2 | Liver Cancer | MTT assay | IC50 = 36.42 μg/mL | 48-h | Liver | None | |
| 27218227 | 2017 | Not Available | Tr2 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | SGC-7901 | Gastric Cancer | MTT assay | IC50 = 48.25 μg/mL | 48-h | Stomach | None | |
| 27218227 | 2017 | Not Available | Tr1 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | HepG-2 | Liver Cancer | MTT assay | IC50 = 147.03 μg/mL | 48-h | Liver | None | |
| 27218227 | 2017 | Not Available | Tr2 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | MCF-7 | Breast Cancer | MTT assay | IC50 < 31.25 μg/mL | 48-h | Breast | None | |
| 27218227 | 2017 | Not Available | Tr1 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Protein extraction from Spirulina platensis | MCF-7 | Breast Cancer | MTT assay | IC50 = 60.12 μg/mL | 48-h | Breast | None | |
| 28093334 | 2017 | Not Available | Bothropoidin | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antitumor and Antiangiogenic | Bothrops pauloensis snake venom | MDA-MB-231 | Breast Cancer | Cell migration assay | Inhibited cell migration by 45% at 10 μg/mL | 24 h | Breast | None | |
| 28093334 | 2017 | Not Available | Bothropoidin | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antitumor and Antiangiogenic | Bothrops pauloensis snake venom | MDA-MB-231 | Breast Cancer | MTT assay | 30% cytotoxicity at 100 μg/mL | 24 h | Breast | None | |
| 28093334 | 2017 | Not Available | Bothropoidin | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antitumor and Antiangiogenic | Bothrops pauloensis snake venom | MDA-MB-231 | Breast Cancer | Apoptosis assay | Early apoptosis at 10 μg/mL and Late apoptosis at 40 μg/mL | 24 h | Breast | None | |
| 27503270 | 2016 | Not Available | Bmattacin2 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antimicrobial | silkworm Bombyx mori | HCT-116 | Colorectal Cancer | MTS assay | IC50 = 1.70 μM | 24-h | Colon | None | |
| 27503270 | 2016 | Not Available | Bmattacin2 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antimicrobial | silkworm Bombyx mori | A-375 | Skin Cancer | MTS assay | IC50 = 5.23 μM | 24-h | Skin | None | |
| 9492845 | 1998 | 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N- [3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl- 1-(1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin-1- yl]-5-methyl-1-oxoheptan-4-yl]-N,3-dimethylbutanamide | Dolastatin 10 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | DU-145 | Prostate cancer | TUNEL assay | IC50=0.5 nM | 96-h | Prostate | None | |
| 8445676 | 1993 | 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N- [3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1- (1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin- 1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3- dimethylbutanamide | Dolastatin 10 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | RL | Lymphoma Cancer | Cell Viability assay | IC50=.00013-.0013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N- [3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1- (1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin- 1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3- dimethylbutanamide | Dolastatin 10 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | SR | Leukemia Cancer | Cell Viability assay | IC50=.0013-.013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N- [3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1- (1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin- 1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3- dimethylbutanamide | Dolastatin 10 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | HT | Lymphoma Cancer | Cell Viability assay | IC50=.0013-.013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | VV-Nme-VPP-2-hydroxyisovaleryl-2- oxo-4-methoxy-5-benzyl-3-pyrroline | Dolastatin 15 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | SR | Leukemia Cancer | Cell Viability assay | IC50=.00013-.0013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | 2-[[2-(dimethylamino)-3-methylbutanoyl]amino]-N- [3-methoxy-1-[2-[1-methoxy-2-methyl-3-oxo-3-[[2-phenyl-1- (1,3-thiazol-2-yl)ethyl]amino]propyl]pyrrolidin- 1-yl]-5-methyl-1-oxoheptan-4-yl]-N,3- dimethylbutanamide | Dolastatin 10 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | DB | Lymphoma Cancer | Cell Viability assay | IC50=.0013-.013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | VV-Nme-VPP-2-hydroxyisovaleryl-2- oxo-4-methoxy-5-benzyl-3-pyrroline | Dolastatin 15 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | DB | Lymphoma Cancer | Cell Viability assay | IC50=.00013-.0013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | VV-Nme-VPP-2-hydroxyisovaleryl-2- oxo-4-methoxy-5-benzyl-3-pyrroline | Dolastatin 15 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | HT | Lymphoma Cancer | Cell Viability assay | IC50=.00013-.0013 nM | Not Available | Blood | None | |
| 8445676 | 1993 | VV-Nme-VPP-2-hydroxyisovaleryl-2- oxo-4-methoxy-5-benzyl-3-pyrroline | Dolastatin 15 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Antineoplastic | Dolabella auricularia | RL | Lymphoma Cancer | Cell Viability assay | IC50=.00013-.0013 nM | Not Available | Blood | None | |
| 15887970 | 2005 | Not Available | Sansalv amide A | Not Available | Cyclic | L | None | Free | Free | Antitumor | Synthetic Peptide | S2-13 | Pancreatic Cancer | Cell Viability assay | EC50=7.5 µM | 72-h | Pancreatic | None | |
| 15835725 | 2004 | lw | Psychrophilin D (1) | Not Available | Cyclic | D | Anthranilic acid | Free | Free | Anticancer and Antiplasmodial | Penicillium algidum | P-388 | Leukemia Cancer | Cell Viability assay | ID50=10.1 µg/ml | Not Available | Blood | None | |
| 2387772 | 1989 | I-C28H46N4O6, II-C27H44N4O6, III-C26H42N4O6 | Cepafungin complex | Not Available | Cyclic | Not Available | None | Free | Free | Antitumor | Culture broth of strain Pseudomonas sp. | P-388 | Leukemia Cancer | Not Available | NA | NA | Blood | None | |
| 11943716 | 2002 | Not Available | Hα-Defensin HNPs-2 | Not Available | Not Available | Not Available | Not Available | Amidation | Not Available | Antimicrobial | Not Available | RCCs, HLA-DRB1*10301 | Tumor | Cell Viability assay | Inhibition at 12.5 µg/ml | Not Available | Not Available | None | |
| 11943716 | 2002 | Not Available | Hα-Defensin HNPs-3 | Not Available | Not Available | Not Available | Not Available | Amidation | Not Available | Antimicrobial | Not Available | RCCs, HLA-DRB1*10301 | Tumor | Cell Viability assay | Inhibition at 12.5 µg/ml | Not Available | Not Available | None | |
| 22820149 | 2012 | Structure Given | BAA-1 | Not Available | Linear | L | None | Amidation | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | Ramos | Lymphoma Cancer | MTT/MTS assay | IC50 = 8.1 µg/ml | 1-h | Blood | None | |
| 22820149 | 2012 | Structure Given | BAA-2 | Not Available | Linear | L | None | Amidation | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | Ramos | Lymphoma Cancer | MTT/MTS assay | IC50 = 3.8 µg/ml | 8-h | Blood | None | |
| 11943716 | 2002 | Not Available | Hα-Defensin HNPs-1 | Not Available | Not Available | Not Available | Not Available | Amidation | Not Available | Antimicrobial | Not Available | RCCs, HLA-DRB1*10301 | Tumor | Cell Viability assay | Inhibition at 12.5 µg/ml | Not Available | Not Available | None | |
| 37874670 | 2023 | Not Available | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | NCI-H2122 | NSCLC | CellTiter-Glo Cell Viability assay | IC50 = 1.4 ± 0.3 nmol/L | Not available | Lung | None | |
| 37874670 | 2023 | Not Available | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo Cell Viability assay | IC50 = 1.4 ± 0.2 nmol/L | Not available | Pancreas | None | |
| 37874670 | 2023 | Not Available | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | NCI-H441 | NSCLC | CellTiter-Glo Cell Viability assay | IC50 = 2.9 ± 0.7 nmol/L | Not available | Lung | None | |
| 37874670 | 2023 | Not Available | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | LS 180 | Colon Cancer | CellTiter-Glo Cell Viability assay | IC50 = 2.7 ± 0.4 nmol/L | Not available | Colon | None | |
| 37874670 | 2023 | Not Available | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | GSU | Stomach Cancer | CellTiter-Glo Cell Viability assay | IC50 = 0.17 ± 0.02 nmol/L | Not available | Stomach | None | |
| 20623634 | 2010 | Not Available | Ozarelix | Not Available | Linear | L | None | Free | Free | Anticancer | LHRH antagonist | PC-3 | Prostate Cancer | Cell Proliferation assay | Inhibited cell proliferation in a dose and time-dependent manner | 0-96 h | Prostate | None | |
| 20623634 | 2010 | Not Available | Ozarelix | Not Available | Linear | L | None | Free | Free | Anticancer | LHRH antagonist | DU-145 | Prostate Cancer | Cell Proliferation assay | Inhibited cell proliferation in a dose and time-dependent manner | 0-96 h | Prostate | None |