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IDPMIDYEARSequenceNameLengthLinear/CyclicChiralityChem-MODC-ter MODN-ter MODNatureOriginCell LineCancer TypeAssayActivityTesting TimeTissue AffectedPatents
7704
384915562024
AAEKEFIKYPYPTPLQYQQLATRLKVEKKLVRRW
HMM-ID34LinearLNoneFreeFreeAnticancerRed Sea BrineU2OSOsteosarcomaMTT assayIC50 = 100.5 µg/ml24-hBoneNone
7607
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisHCT-116Colon CancerLDH leakage assayLDH release above 80%24-hColonNone
7606
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisHCT-116Colon CancerMTT assayIC50 = 2.02 μM24-hColonNone
7605
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisU-251-MGBrain TumorMTT assayIC50 = 2.32 μM24-hBrainNone
7604
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisMDA-MB-435Breast CancerMTT assayIC50 = 18.99 μM24-hBreastNone
7603
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisH-460Lung CancerMTT assayIC50 = 3.47 μM24-hLungNone
7601
366260982023
FKCRRWQWRMKKLG-K-RSKNKGFKEQAKSLLKWILD
LFchimera35LinearLNoneAmidationFreeAntimicrobialSynthetic - Lectoferrin chimeraJurkatBlood CancerMTT assaycell viability ~ 8% at 20 µM6-hBloodNone
7600
366260982023
FKCRRWQWRMKKLG-K-RSKNKGFKEQAKSLLKWILD
LFchimera35LinearLNoneAmidationFreeAntimicrobialSynthetic - Lectoferrin chimeraHepG-2Liver CancerMTT assaycell viability ~ 44% at 10 µM12-hLiverNone
7494
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticZR-75-30Breast CancerCell Viability assayIC50 = 12.92 µM72-hBreastNone
7493
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticU-251BrainTumorCell Viability assayIC50 = 18.17 µM72-hBrainNone
7492
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticA-549Lung CancerCell Viability assayIC50 = 22.00 µM72-hLungNone
7491
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticHCT-116Colon CancerCell Viability assayIC50 = 9.08 µM72-hColonNone
7490
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSynthetic786-0Renal CancerCell Viability assayIC50 = 13.5 µM72-hRenalNone
7489
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticHeLaCervical CancerCell Viability assayIC50 = 31.83 µM72-hCervixNone
7488
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSynthetic5637Bladder cancerCell Viability assayIC50 = 9.33 µM72-hBladderNone
7487
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerCell Viability assayIC50 = 24.25 µM72-hBreastNone
7443
374959882023
TKEQKEQIAKATGLTTKQVRNWYVQLNASIKVCMCSC
37-mer peptide37LinearLNoneFreeFreeAntimicrobialSyntheticSK-OV-3Ovarian cancerMTT assayIC50 = 27.45 ± 1.5085 μM24-hOvaryNone
7442
374959882023
TKEQKEQIAKATGLTTKQVRNWYVQLNASIKVCMCSC
37-mer peptide37LinearLNoneFreeFreeAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 33.65 ± 1.09 μM24-hLiverNone
7441
374959882023
TKEQKEQIAKATGLTTKQVRNWYVQLNASIKVCMCSC
37-mer peptide37LinearLNoneFreeFreeAntimicrobialSyntheticSNU-449Liver CancerMTT assayIC50 = 76.4 ± 0.6015 μM24-hLiverNone
7312
352467582022
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin ZP34CyclicLNoneCyclizedCyclizedAntimicrobialLactococcus lactisH-1299Lung CancerMTT assayIC50 = 137.3 ± 9.1 μM48-hLungNone
7311
352467582022
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin ZP34CyclicLNoneCyclizedCyclizedAntimicrobialLactococcus lactisA-549Lung CancerMTT assayIC50 = 132.4 ± 6.4 μM48-hLungNone
7292
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticT98GBrain TumorAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hBrainNone
7291
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticA-549Lung CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hLungNone
7290
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticDU-145Prostate CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hProstateNone
7289
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticA-375Skin CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hSkinNone
7288
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hBreastNone
7287
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticU-251Brain TumorAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hBrainNone
6862
347897532021
GFLDIIKDTGKEFAVKILNNLKCKLAGGCPP
Palustrin - Ca31LinearLNoneFreeFreeHost Defence PeptideLithobates catesbeianusSGC-7901Gastric CancerNot AvailableIC50 = 0.951 μg/mlNot AvailableStomachNone
6834
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticHT-29Colon CancerMTT assayNot AvailableNot AvailableColonNone
6833
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticRKOColon CancerMTT assay25% cell viability at at 20 μM24-hColonNone
6832
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticHCT-15Colon CancerMTT assayNot AvailableNot AvailableColonNone
6831
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticHCT-116Colon CancerMTT assay20% cell viability at at 20 μM24-hColonNone
6813
343093732021
FPWWWPFLRDVFTKGYGFGLGRKKRRQRRRPQ
Pal-pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinMCF-7Breast CancerMTT assayIC50 = 11.85 μM24-hBreastNone
6812
343093732021
FPWWWPFLRDVFTKGYGFGLGRKKRRQRRRPQ
Pal-pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-549Lung CancerMTT assayIC50 = 31.17 μM24-hLungNone
6811
343093732021
FPWWWPFLRDVFTKGYGFGLGRKKRRQRRRPQ
Pal-pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50 = 5.5 ± 1.1 μM24-hSkinNone
6810
343093732021
FPWWWPFL-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATpFL = hydrophobic peptide fragment (FPWWWPFL)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50 = 11.1 ± 0.1 μM24-hSkinNone
6782
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaLoVoColon CancerMTT assayIC50 = 128 µM24-hColonNone
6781
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaHeLaCervical CancerMTT assayIC50 > 128 µM24-hCervixNone
6780
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaMCF-7Breast CancerMTT assayIC50 > 128 µM24-hBreastNone
6779
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaA-549Lung CancerMTT assayIC50 > 128 µM24-hLungNone
6765
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiLoVoColon CancerMTT assayIC50 = 35.05 µM24-hColonNone
6764
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiHeLaCervical CancerMTT assayIC50 = 23.26 µM24-hCervixNone
6763
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiMCF-7Breast CancerMTT assayIC50 = 37.84 µM24-hBreastNone
6762
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiA-549Lung CancerMTT assayIC50 = 24.01 µM24-hLungNone
6761
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiLoVoColon CancerMTT assayIC50 = 55.22 µM24-hColonNone
6760
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiHeLaCervical CancerMTT assayIC50 = 52.83 µM24-hCervixNone
6759
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiMCF-7Breast CancerMTT assayIC50 = 41.21 µM24-hBreastNone
6758
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiA-549Lung CancerMTT assayIC50 = 27.31 µM24-hLungNone
6757
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisLoVoColon CancerMTT assayIC50 = 59.78 µM24-hColonNone
6755
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisMCF-7Breast CancerMTT assayIC50 = 45.25 µM24-hBreastNone
6756
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisHeLaCervical CancerMTT assayIC50 = 37.23 µM24-hCervixNone
6754
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisA-549Lung CancerMTT assayIC50 = 15.32 µM24-hLungNone
6753
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiLoVoColon CancerMTT assayIC50 = 8.05 µg/ml24-hColonNone
6752
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiHeLaCervical CancerMTT assayIC50 = 19.69 µg/ml24-hCervixNone
6751
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiMCF-7Breast CancerMTT assayIC50 = 25.74 µg/ml24-hBreastNone
6750
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiA-549Lung CancerMTT assayIC50 = 2.975 µg/ml24-hLungNone
6657
330295952020
{[LLKKLLKK]2kC}2
4-arm branched peptide36LinearLthermal oxidation between the thiol group of cysteine residue in the two 2-arm branchedFreeFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayCell Viability (%) ~ 49.0 ± 0.8 at 30 µg/mL48-hProstateNone
6656
330295952020
{[LLKKLLKK]2kC}2
4-arm branched peptide36LinearLthermal oxidation between the thiol group of cysteine residue in the two 2-arm branchedFreeFreeAntimicrobialSyntheticBcap-37Breast CancerMTT assayCell Viability (%) ~ 51.4 ± 4.2 at 30 µg/mL48-hBreastNone
6654
330295952020
{[LLKKLLKK]2kC}2
4-arm branched peptide36LinearLthermal oxidation between the thiol group of cysteine residue in the two 2-arm branchedFreeFreeAntimicrobialSyntheticSK-HEP-1Liver CancerMTT assayCell Viability (%) ~ 31.7 ± 5.1 at 30 µg/mL48-hLiverNone
6655
330295952020
{[LLKKLLKK]2kC}2
4-arm branched peptide36LinearLthermal oxidation between the thiol group of cysteine residue in the two 2-arm branchedFreeFreeAntimicrobialSyntheticHCT-116Colon CancerMTT assayCell Viability (%) ~ 67.6 ± 5.8 at 30 µg/mL48-hColonNone
6579
319409272020
GPKTKAACKMACKLATCGKKPGGWKCKLCELGCDAV
Turgencin A36Cyclic(C8-C33,C12-C29,C17-C26)LNoneAmidationFreeAntimicrobial and AnticancerSynoicum turgensA-2058Skin CancerCell Viability assayIC50 1.4 µM72-hSkinNone
6578
319409272020
GIKEMLCNMACAQTVCKKSGGPLCDTCQAACKALG
Turgencin B35Cyclic(C7-C31,C11-C27,C16-C24)LNoneAmidationFreeAntimicrobial and AnticancerSynoicum turgensA-2058Skin CancerCell Viability assayIC50 4.1 µM72-hSkinNone
6534
332373352020
MSSSNCANVCQTENFPGGECKAEGATRKCFCKNC
MzDef34LinearLNoneFreeFreeAntimicrobial and AnticancerZea mays L.HCT-116Colon CancerMTT assayIC50 = 29.85 µg/mL24-hColonNone
6533
332373352020
MSSSNCANVCQTENFPGGECKAEGATRKCFCKNC
MzDef34LinearLNoneFreeFreeAntimicrobial and AnticancerZea mays L.MCF-7Breast CancerMTT assayIC50 = 14.85 µg/mL24-hBreastNone
6532
332373352020
MSSSNCANVCQTENFPGGECKAEGATRKCFCKNC
MzDef34LinearLNoneFreeFreeAntimicrobial and AnticancerZea mays L.HepG-2Liver CancerMTT assayIC50 ~ 22 µg/mL24-hLiverNone
6216
304611972019
ALWKTMLKKLGTVALHAGKAALGAVADTISQ
Dermaseptin-PS131LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvageiU251-MGBrain TumorLDH leakage assay20% LDH release at 10⁻⁴ M24-hBrainNone
6215
304611972019
ALWKTMLKKLGTVALHAGKAALGAVADTISQ
Dermaseptin-PS131LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvageiU251-MGBrain TumorMTT assay5.419 μmol/L24-hBrainNone
6212
312343332019
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensiHCT-116Colon CancerMTT assayIC50 = 2.02 µM24-hColonNone
6211
312343332019
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensiU251-MGBrain TumorMTT assayIC50 = 2.32 µM24-hBrainNone
6210
312343332019
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensiMDA-MB-435SBreast CancerMTT assayIC50 = 18.99 µM24-hBreastNone
6209
312343332019
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensiH-460Lung CancerMTT assayIC50 = 3.47 µM24-hLungNone
5980
296289172018
NLVSALIEGRKYLKNVLKKLNRLKEKNKAKNSKENN
DLP-PH36LinearLNoneFreeFreeAntimicrobialPhyllomedusa hypochondrialisPC-3Prostate CancerMTT assayIC50 = 32.25 μg/mL24-hProstateNone
5979
296289172018
NLVSALIEGRKYLKNVLKKLNRLKEKNKAKNSKENN
DLP-PH36LinearLNoneFreeFreeAntimicrobialPhyllomedusa hypochondrialisH-157Lung CancerMTT assayIC50 = 15.41 μg/mL24-hLungNone
5978
304815572018
HSDGIFTDSYSRYRKQMAVKKYLAAVLGRRYRQRFRNK
PACAP3838LinearLNoneAmidationFreeAntimicrobial and AnticancerClarias gariepinusH-460Lung CancerCrystal Violet assayIC50=14.97± 1.16 µM48-hLungNone
5975
304831332018
GRWKIFKKIEKVGQNIRDGIVKAGPAVAVVGQAATI
myristoyl-CM436LinearLNoneAmidationN-myristoylationAntimicrobialBombyx moriMCF-7Breast cancerMTT assayIC50 = 6 μM24-hBreastNone
5976
304831332018
GRWKIFKKIEKVGQNIRDGIVKAGPAVAVVGQAATI
myristoyl-CM436LinearLNoneAmidationN-myristoylationAntimicrobialBombyx moriMDA-MB-231Breast cancerMTT assayIC50 = 4 μM24-hBreastNone
5977
304831332018
GRWKIFKKIEKVGQNIRDGIVKAGPAVAVVGQAATI
myristoyl-CM436LinearLNoneAmidationN-myristoylationAntimicrobialBombyx moriMX-1Breast cancerMTT assayIC50 = 3 μM24-hBreastNone
5967
298757732018
RRRRRRRRRRRIKKKRKWEASALVCIRLVTSSKPRTVa
R11-NLS-pep838LinearMixNoneFreeAcetylationAnticancerNKp44 derived synthetic peptideMDA-MD-231Breast CancerPrestoBlue assayED50 = 5.6 μM24-hBreastNone
5966
298757732018
RRRRRRRRRRRIKKKRKWEASALVCIRLVTSSKPRTVa
R11-NLS-pep838LinearMixNoneFreeAcetylationAnticancerNKp44 derived synthetic peptideHepG-2Liver CancerPrestoBlue assayED50 = 5.9 μM24-hLiverNone
5965
298757732018
RRRRRRRRRRRIKKKRKWEASALVCIRLVTSSKPRTVa
R11-NLS-pep838LinearMixNoneFreeAcetylationAnticancerNKp44 derived synthetic peptidePANC-1Pancreatic CancerPrestoBlue assayED50 = 7.8 μM24-hPancreasNone
5964
298757732018
RRRRRRRRRRRIKKKRKWEASALVCIRLVTSSKPRTVa
R11-NLS-pep838LinearMixNoneFreeAcetylationAnticancerNKp44 derived synthetic peptideB-16Skin CancerPrestoBlue assayED50 = 7.1 μM24-hSkinNone
5951
290547982018
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin Z34LinearLNoneFreeFreeAntimicrobial and AnticancerLactococcus lactisA-375Skin CancerLDH leakage assay60% LDH release at 60 µM24-hSkinNone
5950
290547982018
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin Z34LinearLNoneFreeFreeAntimicrobial and AnticancerLactococcus lactisA-375Skin CancerMTT assayIC50 = 188.5 ± 8.7 µM24-hSkinNone
5731
288676312017
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin Z34CyclicLNoneCyclizedCyclizedAntimicrobialLactococcus lactisSW-480Colon CancerMTT assay79.22% cytotoxicity at 1000 μg/mL24-hColonNone
5719
283477402017
RWKIFKKIERVGQNVRDGIIKAGKAIQVLGTAKALGK
ABP-dHC-Cecropin A-K(24)37LinearLNoneFreeFreeHost Defence PeptideSyntheticTHP-1Leukemia CancerMTT assayIC50 = 196.1 μM24-hBloodNone
5718
283477402017
RWKIFKKIERVGQNVRDGIIKAGKAIQVLGTAKALGK
ABP-dHC-Cecropin A-K(24)37LinearLNoneFreeFreeHost Defence PeptideSyntheticU-937Leukemia CancerMTT assayIC50 = 223.9 μM24-hBloodNone
5717
283477402017
RWKIFKKIERVGQNVRDGIIKAGKAIQVLGTAKALGK
ABP-dHC-Cecropin A-K(24)37LinearLNoneFreeFreeHost Defence PeptideSyntheticK-562Leukemia CancerMTT assayIC50 = 184.9 μM24-hBloodNone
5716
283477402017
RWKIFKKIERVGQNVRDGIIKAGPAIQVLGTAKALGK
ABP-dHC-Cecropin A37LinearLNoneFreeFreeHost Defence PeptideSyntheticTHP-1Leukemia CancerMTT assayIC50 = 228.5 μM24-hBloodNone
5715
283477402017
RWKIFKKIERVGQNVRDGIIKAGPAIQVLGTAKALGK
ABP-dHC-Cecropin A37LinearLNoneFreeFreeHost Defence PeptideSyntheticU-937Leukemia CancerMTT assayIC50 = 303.2 μM24-hBloodNone
5714
283477402017
RWKIFKKIERVGQNVRDGIIKAGPAIQVLGTAKALGK
ABP-dHC-Cecropin A37LinearLNoneFreeFreeHost Defence PeptideSyntheticK-562Leukemia CancerMTT assayIC50 = 349.5 μM24-hBloodNone
5710
281573212017
GGAGHVPEYFVGIGTPISFYG-WxEAAYQrFL
MccJ25-18-431LinearMixx = NorleucineFreeFreeAntimicrobialSyntheticMDA-MB-435-MDRBreast CancerMTT assayIC50 = 25.0 ± 0.5 μM48-hBreastNone
5709
281573212017
GGAGHVPEYFVGIGTPISFYG-WxEAAYQrFL
MccJ25-18-431LinearMixx = NorleucineFreeFreeAntimicrobialSyntheticMDA-MB-435Breast CancerMTT assayIC50 = 20.0 ± 0.5 μM48-hBreastNone
5708
281573212017
GGAGHVPEYFVGIGTPISFYG-WxEAAYQrFL
MccJ25-18-431LinearMixx = NorleucineFreeFreeAntimicrobialSyntheticMCF-7Breast CancerMTT assayIC50 = 14.2 ± 1.5 μM48-hBreastNone
5550
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorPC-3Prostate CancerLDH leakage assay100% cytotoxicity at 2.5 μM3-hProstateNone
5549
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorLNCaPProstate CancerCrystal Violet assayGI50 = 2.65 ± 1.09 μM24-hProstateNone
5548
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorPC-3Prostate CancerCrystal Violet assayGI50 = 2.17 ± 0.48 μM24-hProstateNone
5547
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorDU-145Prostate CancerCrystal Violet assayGI50 = 0.71 ± 0.55 μM24-hProstateNone
5546
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorA-375Skin CancerCrystal Violet assayGI50 > 10 μM24-hSkinNone
5545
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorSK-Mel-28Skin CancerCrystal Violet assayGI50 > 10 μM24-hSkinNone
5544
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorHT-144Skin CancerCrystal Violet assayGI50 = 5.08 ± 0.72 μM24-hSkinNone
5543
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorMIA PaCa-2Pancreatic CancerCrystal Violet assayGI50 = 7.91 ± 1.40 μM24-hPancreasNone
5542
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorBxPC-3Pancreatic CancerCrystal Violet assayGI50 = 2.31 ± 0.41 μM24-hPancreasNone
5541
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorPANC-1Pancreatic CancerCrystal Violet assayGI50 > 10 μM24-hPancreasNone
5540
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorMDA-MB-453Breast CancerCrystal Violet assayGI50 > 10 μM24-hBreastNone
5539
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorBT-474Breast CancerCrystal Violet assayGI50 > 10 μM24-hBreastNone
5538
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorMDA-MB-231Breast CancerCrystal Violet assayGI50 > 10 μM24-hBreastNone
5537
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorU-373-MGBrain TumorCrystal Violet assayGI50 > 10 μM24-hBrainNone
5536
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorU-138-MGBrain TumorCrystal Violet assayGI50 > 10 μM24-hBrainNone
5535
287970922017
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Dermaseptin - B233LinearLNoneAmidationFreeAntimicrobialPhyllomedusa bicolorU-87-MGBrain TumorCrystal Violet assayGI50 > 10 μM24-hBrainNone
5321
268310102016
VCMPCFTTDQQMARKCSDCCGGKGRGKCYGPQCLCR
CTX-2336LinearLNoneFreeFreeAnticancerSyntheticU-251Brain TumorMTT assayGraph Figure 248-hBrainNone
5320
268310102016
CGPCFTTDHNMARKCDECCGGKGRGKCFGPQCLCR
CA435LinearLNoneFreeFreeAnticancerSyntheticU-251Brain TumorMTT assayGraph Figure 248-hBrainNone
5290
271874672016
GMWSKIKNAGKAAAKAAAKAAGKAALDAVSEAI
dermaseptin-PD-233LinearLNoneFreeFreeAntimicrobialphyllomedusine leaf frogs,Pachymedusa dacnicolorU251-MGBrain TumorMTT assayIC50 = 13.43 μM24-hBrainNone
5289
271874672016
GMWSKIKNAGKAAAKAAAKAAGKAALDAVSEAI
dermaseptin-PD-233LinearLNoneFreeFreeAntimicrobialphyllomedusine leaf frogs,Pachymedusa dacnicolorPC-3Prostate CancerMTT assayIC50 = 3.17 μM24-hProstateNone
5288
271874672016
GMWSKIKNAGKAAAKAAAKAAGKAALDAVSEAI
dermaseptin-PD-233LinearLNoneFreeFreeAntimicrobialphyllomedusine leaf frogs,Pachymedusa dacnicolorH-157Lung CancerMTT assayIC50 = 6.43 μM24-hLungNone
5287
271874672016
GMWSKIKETAMAAAKEAAKAAGKTISDMIKQ
dermaseptin-PD-131LinearLNoneFreeFreeAntimicrobialphyllomedusine leaf frogs,Pachymedusa dacnicolorU251-MGBrain TumorMTT assayIC50 = 15.08 μM24-hBrainNone
5183
258210842015
CVLIGQRCDNDRGPRCCSGQGNCVPLPFLGGVCAV
Ep-AMP135CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerEchinopsis pachanoiU-937/GTBLymphoma cancerFluorometric microculture cytotoxicity assayIC50 > 100 µMNot AvailableBloodNone
5169
267036312015
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntimicrobialPardachirus marmoratusOSCC-SCC-4Oral cancerMTT assayCell Viability <20% at 20μg/mL24-hNot AvailableNone
5158
260643102015
GAFLKCGESCVYLPCLTTVVGCSCQNSVCYRD
DC132CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaDU-145Liver CancerCCK-8 assayIC50 = 3.32 μM72-hLiverNone
5157
260643102015
GAFLKCGESCVYLPCLTTVVGCSCQNSVCYRD
DC132CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaPC-3Prostate CancerCCK-8 assayIC50 = 2.24 μM72-hProstateNone
5156
260643102015
GAFLKCGESCVYLPCLTTVVGCSCQNSVCYRD
DC132CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaLNCaPProstate CancerCCK-8 assayIC50 = 5.03 μM72-hProstateNone
5155
260643102015
GAVPCGETCVYLPCITPDIGCSCQNKVCYRD
DC231CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaDU-145Liver CancerCCK-8 assayIC50 = 3.11 μM72-hLiverNone
5154
260643102015
GAVPCGETCVYLPCITPDIGCSCQNKVCYRD
DC231CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaPC-3Prostate CancerCCK-8 assayIC50 = 2.65 μM72-hProstateNone
5153
260643102015
GAVPCGETCVYLPCITPDIGCSCQNKVCYRD
DC231CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaLNCaPProstate CancerCCK-8 assayIC50 = 4.31 μM72-hProstateNone
5010
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC25Skin CancerCell Viability assay107.0 ± 5.0% cell growth inhibition at 1 µM24-hSkinNone
5009
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC25Skin CancerCell Viability assay0.6 ± 0.6% cell growth inhibition at 10 µM48-hSkinNone
5008
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC25Skin CancerMTT/MTS assayIC50=2.2 µM48-hSkinNone
5007
246610242014
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneFreeFreeAntimicrobialIsolated from the giant silk moth Hyalophora cecropiaSCC12Skin CancerMTT/MTS assayIC50=1 µM48-hSkinNone
5006
245873502014
LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES
LL 3737LinearLNoneFreeFreeAntimicrobialAlso known human cathelicidinOVRCAR-3Ovarian CancerMTT/MTS assayLC50= 24 at 100 µM72-hOvaryNone
5004
245873502014
LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES
LL 3737LinearLNoneFreeFreeAntimicrobialAlso known human cathelicidinLNCaPProstate cancerMTT/MTS assayLC50= 27 at 100 µM72-hProstateNone
5002
245873502014
LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES
LL 3737LinearLNoneFreeFreeAntimicrobialAlso known human cathelicidinMCF-7Breast CancerMTT/MTS assayLC50= 21 at 100 µM72-hBreastNone
4601
154965972004
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
CB36LinearLNoneFreeFreeAntibacterialSyntheticAgsGastric CancerNot AvailableNot AvailableNot AvailableStomachNone
4600
213513232011
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EGFR-lytic32LinearMixNoneFreeFreeAntitumorSynthetic PeptideMDA-MB-231Breast CancerELISAIC50 =0.46 µM15-MinBreastNone
4599
213513232011
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EGFR-lytic32LinearMixNoneFreeFreeAntitumorSynthetic PeptideMDA-MB-231Breast CancerELISAIC50 =0.12 µM60-MinBreastNone
4453
17561225, 189574412007
LLGMIPLAISAISALSKL
Phylloseptin-L132Not AvailableLNoneFreeFreeAnticancerHylomantis lemur (Hylidae: PhyllomedusinaeNot AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4452
17561225, 189574412007
GLWSKIKEAAKAAGKAALNAVTGLVNQGDQPS
Phylloseptin32Not AvailableLNoneFreeFreeAnticancerHylomantis lemur (Hylidae: PhyllomedusinaeNot AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4434
7628632, 189574411995
DHYNCVSSGGQCLYSACPIFTKIQGTCYRGKAKCCK
hBD-136Not AvailableLNoneFreeFreeAntibacterialkeratinocytes; skin; platelets;Homo sapiensNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4423
18191970, 189574412008
GLLPCAESCVYIPCLTTVIGCSCKSKVCYKN
Vibi H31Not AvailableLNoneFreeFreeAnticancerAlpine violetViola bifloraNot AvailableLung CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4420
7916722, 189574411993
GWLKKIGKKIERVGQHTRDATIQTIGVAQQAANVAATLK
Cecropin 239Not AvailableLNoneFreeFreeAntibacterialThe Medfly, Ceratitis capitata; also housefly, Musca domesticaNot AvailableLeukemia CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4418
18191970, 189574412008
GTFPCGESCVFIPCLTSAIGCSCKSKVCYKN
Vibi G31Not AvailableLNoneFreeFreeAnticancerAlpine violetViola bifloraNot AvailableSkin CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4396
20575512, 189574412010
GVIPCGESCVFIPCISSVLGCSCKNKVCYRD
Psyle E31Not AvailableLNoneFreeFreeAntibacterialPsychotria leptothyrsaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4379
21723349, 189574412011
GSIPCEGSCVFIPCISAIIGCSCSNKVCYKN
Viphi G31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4375
21723349, 189574412011
GSIPCGESCVFIPCISAIIGCSCSSKVCYKN
Viphi F31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4374
21723349, 189574412011
GSIPCGESCVFIPCISSVIGCACKSKVCYKN
Viphi F31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4373
21723349, 189574412011
GSIPCGESCVFIPCISAVIGCSCSNKVCYKN
Viphi E31Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4372
22467870, 189574412012
GIPCAESCVWIPPCTITALMGCSCKNNVCYNN
Chassatide C232Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4350
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 7.9 µM48-hPancreaticWO_2010_064207_A2
4349
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptidePane- 1Breast CancerWST-1 assayIC50= 13.1 µM48-hBreastWO_2010_064207_A2
4348
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideCFPAC-IPancreatic CancerWST-1 assayIC50= 10.6 µM48-hPancreaticWO_2010_064207_A2
4347
None2009
NYQWVPYQGRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa363-377) -nLytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 12.5 µM48-hPancreaticWO_2010_064207_A2
4346
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideLNCaPProstate CancerWST-1 assayIC50= 4.8 µMNot AvailableProstateUS_8436137_B2
4345
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 7.4 µMNot AvailablePancreaticUS_8436137_B2
4344
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 6.6 µMNot AvailablePancreaticUS_8436137_B2
4343
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideU-251Brain TumorWST-1 assayIC50= 8.4 µMNot AvailableBrainUS_8436137_B2
4342
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBT-20Breast CancerWST-1 assayIC50= 1.9 µMNot AvailableBreastUS_8436137_B2
4341
None2009
YRWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB(H2R)-lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideH-322Lung CancerWST-1 assayIC50= 3.2 µMNot AvailableLungUS_8436137_B2
4340
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideLNCaPProstate CancerWST-1 assayIC50= 10 µMNot AvailableProstateUS_8436137_B2
4339
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 12 µMNot AvailablePancreaticUS_8436137_B2
4338
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 12 µMNot AvailablePancreaticUS_8436137_B2
4337
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideU-251Brain TumorWST-1 assayIC50= 12 µMNot AvailableBrainUS_8436137_B2
4336
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideBT-20Breast CancerWST-1 assayIC50= 6.5 µMNot AvailableBreastUS_8436137_B2
4335
None2009
YHWYGYTPQNVIGGGKLlLKlLkkLLKlLKKK
EB-Lytic32LinearMixNoneFreeFreeAnticancerSynthetic PeptideH-322Lung CancerWST-1 assayIC50= 6.8 µMNot AvailableLungUS_8436137_B2
4238
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay50% apoptosis at 50 µM8-hNot AvailableNone
4237
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay20% apoptosis at 20 µM8-hNot AvailableNone
4236
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay15% apoptosis at 10 µM8-hNot AvailableNone
4235
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay30% apoptosis at 50 µM8-hNot AvailableNone
4234
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay>50% apoptosis at 20 µM8-hNot AvailableNone
4233
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay20% apoptosis at 10 µM8-hNot AvailableNone
4232
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay80% apoptosis at 50 µM8-hBrainNone
4231
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay80% apoptosis at 20 µM8-hBrainNone
4230
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay30% apoptosis at 10 µM8-hBrainNone
4229
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay30% apoptosis at 50 µM8-hBrainNone
4228
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay10% apoptosis at 20 µM8-hBrainNone
4227
165680932006
rrrrrrrrGNLWAAQRYGRELRRMSDEFVDSFKK
r8-BadBH335LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay0% apoptosis at 10 µM8-hBrainNone
3188
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assayED50 =0.29 µM24-hBloodNone
3187
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assayED50 >10 µM24-hColonNone
3186
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assayED50 =0.210 µM24-hPancreaticNone
3185
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assayED50 =2.1 µM24-hOral mucosaNone
3184
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay94.5 % inhibition of cell proliferation at 10 µM24-hBloodNone
3183
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay54.3 % inhibition of cell proliferation at 1 µM24-hBloodNone
3182
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay34.7 % inhibition of cell proliferation at 100 nM72-hBloodNone
3181
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay18.7 % inhibition of cell proliferation at 10 nM24-hBloodNone
3180
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMOLT-4Leukemia CancerMTT/MTS assay10.4 % inhibition of cell proliferation at 1 nM24-hBloodNone
3179
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay27.9 % inhibition of cell proliferation at 10 µM24-hColonNone
3178
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay21.7 % inhibition of cell proliferation at 1 µM24-hColonNone
3177
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay16.8 % inhibition of cell proliferation at 100 nM72-hColonNone
3176
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay14.2 % inhibition of cell proliferation at 10 nM24-hColonNone
3175
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aPTCColon CancerMTT/MTS assay16.5 % inhibition of cell proliferation at 1 nM24-hColonNone
3174
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay84.5 % inhibition of cell proliferation at 10 µM24-hPancreaticNone
3173
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay59.6 % inhibition of cell proliferation at 1 µM24-hPancreaticNone
3172
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay48.2 % inhibition of cell proliferation at 100 nM72-hPancreaticNone
3171
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay37.8 % inhibition of cell proliferation at 10 nM24-hPancreaticNone
3170
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aMiaPaCa.2Pancreatic CancerMTT/MTS assay24.2 % inhibition of cell proliferation at 1 nM24-hPancreaticNone
3169
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay98.3 % inhibition of cell proliferation at 10 µM24-hOral mucosaNone
3168
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay43.1 % inhibition of cell proliferation at 1 µM24-hOral mucosaNone
3167
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay30.7 % inhibition of cell proliferation at 100 nM72-hOral mucosaNone
3166
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay18.2 % inhibition of cell proliferation at 10 nM24-hOral mucosaNone
3165
175590672007
fCYwO-CyLeu-Pen-TKKrPKPfQwFwL-CyLeu-KKLMYPTYLKKfQWAV-Aib-HL
Peptide 540LinearMixAib = = 1-amino-isobutyric acid, O= Ornithine, Pen=penicillamine, CyLeu=cycloleucine or 1-aminocyclopentane-1-carboxylic acid and disulfide bond between Cys and PenAmidationFreeAnticancerSynthetic peptide of four designed analogs of vasoactive intestinal peptide, bombesin, substance P aKBOral CancerMTT/MTS assay10.6 % inhibition of cell proliferation at 1 nM24-hOral mucosaNone
3031
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
3030
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay5 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
3028
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
3029
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay15 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
3027
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
3026
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay38 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
3024
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay39 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
3025
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay28 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
3023
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay95 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
3021
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
3022
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay97 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
3020
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
3019
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
3018
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
3017
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
3016
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
3015
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
3014
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay40 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
3013
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay82 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
3012
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay88 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
3011
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 3.125 mg/L24-hCervixNone
3010
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay12 % Cytotoxicity at 6.25 mg/L24-hCervixNone
3009
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay15 % Cytotoxicity at 12.5 mg/L24-hCervixNone
3008
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay80 % Cytotoxicity at 25 mg/L24-hCervixNone
3007
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hCervixNone
3006
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L12-hCervixNone
3005
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 6.25 mg/L12-hCervixNone
3004
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 12.5 mg/L12-hCervixNone
3003
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay68 % Cytotoxicity at 25 mg/L12-hCervixNone
3002
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay78 % Cytotoxicity at 50 mg/L12-hCervixNone
3001
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 3.125 mg/L6-hCervixNone
3000
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L6-hCervixNone
2999
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75 % Cytotoxicity at 50 mg/L6-hCervixNone
2998
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 12.5 mg/L3-hCervixNone
2997
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay44 % Cytotoxicity at 25 mg/L3-hCervixNone
2996
235980792013
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin-133LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay62 % Cytotoxicity at 50 mg/L3-hCervixNone
2924
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)COLO-587Human epithelial CancerWST-1 assayIC50=6.4 µM72-hPancreaticNone
2923
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)LNCaPProstate CancerWST-1 assayIC50= 6.2 µM72-hProstateNone
2922
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)HuCCT-1Human epithelial CancerWST-1 assayIC50= 8.3 µM72-hBileductNone
2921
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)U-251Brain TumorWST-1 assayIC50=7.0 µM72-hBrainNone
2920
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SN-19Brain TumorWST-1 assayIC50= 7.8 µM72-hBrainNone
2919
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SF-295Brain TumorWST-1 assayIC50= 6.3 µM72-hBrainNone
2918
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)ZR75-1Breast CancerWST-1 assayIC50= 9.3 µM72-hBreastNone
2917
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)BT-20Breast CancerWST-1 assayIC50= 4.8 µM72-hBreastNone
2916
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)MDA-MB-231Breast CancerWST-1 assayIC50= 7.8 µM72-hBreastNone
2915
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)SK-BR-3Breast CancerWST-1 assayIC50= 6.5 µM72-hBreastNone
2914
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)T-47DBreast CancerWST-1 assayIC50= 4.0 µM72-hBreastNone
2913
218490922011
THRPPMWSPVWPGGGKLlLKlLkkLLKlLKKK
Transferrin receptor (TfR)-lytic hybrid peptide32LinearMixNoneFreeFreeAnticancerTransferrin receptor (TfR)BT-474Breast CancerWST-1 assayIC50= 8.8 µM72-hBreastNone
2868
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainMDA-MB-231Breast CancerWST-1 assayIC50=5.7 µMol/L24-hBreastNone
2867
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainH-322Lung CancerWST-1 assayIC50=3.6 µMol/L24-hLungNone
2866
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainA-172Brain TumorWST-1 assayIC50=6.8 µMol/L24-hBrainNone
2865
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainT98GBrain TumorWST-1 assayIC50=18.5 µMol/L24-hBrainNone
2864
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)KBOral CancerWST-1 assayIC50=13.2 µMol/L24-hOral mucosaNone
2863
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainSU.86.86Pancreatic CancerWST-1 assayIC50=7.5 µMol/L24-hPancreaticNone
2862
220841652011
KQLIRFLKRLDRNGGGKLlLKlLkkLLKlLKKK
IL-4RaÐlytic hybrid peptide33LinearMixNoneFreeFreeAnticancerInterleukin-4 receptor a (IL-4Ra) chainBXPC-3Pancreatic CancerWST-1 assayIC50=6.8 µMol/L24-hPancreaticNone
2850
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorRajiLymphoma CancerLDH leakage assayGI50 =2.57±0.75 µM24-hBloodNone
2849
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorMDA-MB-231Breast CancerLDH leakage assayGI50 =8.06±0.50 µM24-hBreastNone
2848
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorDU-145Liver CancerLDH leakage assayGI50 =0.91±0.04 µM24-hProstateNone
2847
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorLNCaPProstate CancerLDH leakage assayGI50 =0.31±0.15 µM24-hProstateNone
2846
230285272012
GLWSKIKEVGKEAAKAAAKAAGKAALGAVSEAV
Adenoregulin33LinearLNoneFreeFreeAntimicrobialSouth American frog Phyllomedusa bicolorPC-3Prostate CancerLDH leakage assayGI50 =1.24±0.23 µM24-hProstateNone
2808
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =250 µg/ml24-hCervixUS_06875744_B2
2727
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =175 µg/ml24-hCervixUS_06875744_B2
2670
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =>1000 µg/ml24-hCervixUS_06875744_B2
2669
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =150 µg/ml24-hCervixUS_06875744_B2
2665
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =370 µg/ml24-hProstateUS_06875744_B2
2584
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =52 µg/ml24-hProstateUS_06875744_B2
2526
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayNot Available24-hProstateUS_06875744_B2
2527
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =630 µg/ml24-hProstateUS_06875744_B2
2522
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =120 µg/ml24-hLungUS_06875744_B2
2441
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =53 µg/ml24-hLungUS_06875744_B2
2384
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =720 µg/ml24-hLungUS_06875744_B2
2383
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =220 µg/ml24-hLungUS_06875744_B2
2369
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =170 µg/ml24-hSkinUS_06875744_B2
2288
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2231
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =120 µg/ml24-hSkinUS_06875744_B2
2232
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =>1000 µg/ml24-hSkinUS_06875744_B2
2217
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =170 µg/ml24-hSkinUS_06875744_B2
2136
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2080
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =>1000 µg/ml24-hSkinUS_06875744_B2
2079
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =120 µg/ml24-hSkinUS_06875744_B2
2065
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =240 µg/ml24-hColonUS_06875744_B2
1984
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =125 µg/ml24-hColonUS_06875744_B2
1928
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =>1000 µg/ml24-hColonUS_06875744_B2
1927
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =82 µg/ml24-hColonUS_06875744_B2
1913
None2005
LPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
LSB-3738LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =50 µg/ml24-hBreastUS_06875744_B2
1832
None2005
FAKKLAKKLKKLAKKLAKLALALKALALKAL
Shiva-1131LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =96 µg/ml24-hBreastUS_06875744_B2
1776
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AM38LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =540 µg/ml24-hBreastUS_06875744_B2
1775
None2005
MPKWKVFKKIEKVGRNIRNGIVKAGPAIAVLGEAKALG
SB-37 AC38LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =175 µg/ml24-hBreastUS_06875744_B2
1708
96140661998
ALWKTMLKKLGTMALHAGKAALGAAADTISQGTQ
DRS S135LinearLNoneFreeFreeAntimicrobialDermaseptins BMCF-7Breast CancerThymidine Incorporation assayNot Available6-hBreastNone
1546
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=14.52 µg/ml24-hFibrous connective tissue None
1545
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=14.51 µg/ml12-hFibrous connective tissue None
1544
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=15.40 µg/ml6-hNot AvailableNone
1543
220730062011
GFFALIPKIISSPLFKTLLSAVGSALSSSGGQE
Pardaxin33LinearLNoneFreeFreeAntibacterialRed Sea MosessoleHT-1080FibrosarcomaMTT/MTS assayIC50=15.74 µg/ml3-hNot AvailableNone
1351
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothJ82Bladder CancerLDH leakage assayCytotoxicity=196.3 µg/ml48-hBladderNone
1349
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth647VBladder CancerLDH leakage assayIC50=181.1 µg/ml48-hBladderNone
1348
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothRT4Bladder CancerLDH leakage assayIC50=240.4 µg/ml48-hBladderNone
1347
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth486PBladder CancerLDH leakage assayIC50=232.4 µg/ml48-hBladderNone
1344
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)J82Bladder CancerLDH leakage assayIC50=319.2 µg/ml48-hBladderNone
1343
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)647VBladder CancerLDH leakage assayIC50=200.7 µg/ml48-hBladderNone
1342
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)RT4Bladder CancerLDH leakage assayIC50=289.3 µg/ml48-hBladderNone
1341
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)486PBladder CancerLDH leakage assayIC50=373.3/ µg/ml48-hBladderNone
1338
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothJ82Bladder CancerCell Viability assayIC50=77.51 µg/ml48-hBladderNone
1337
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth647VBladder CancerCell Viability assayIC50=61.86 µg/ml48-hBladderNone
1336
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothRT4Bladder CancerCell Viability assayIC50=92.9 µg/ml48-hBladderNone
1335
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth486PBladder CancerCell Viability assayIC50=87.47 µg/ml48-hBladderNone
1332
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)J82Bladder CancerCell Viability assayIC50=99.01 µg/ml48-hBladderNone
1331
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)647VBladder CancerCell Viability assayIC50=28.74 µg/ml48-hBladderNone
1330
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)RT4Bladder CancerCell Viability assayIC50=96.22 µg/ml48-hBladderNone
1329
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)486PBladder CancerCell Viability assayIC50=69.2 µg/ml48-hBladderNone
1326
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothJ82Bladder CancerWST-1 assayIC50=97.93 µg/ml48-hBladderNone
1325
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth647VBladder CancerWST-1 assayIC50=115.12 µg/ml48-hBladderNone
1324
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk mothRT4Bladder CancerWST-1 assayIC50=184.81 µg/ml48-hBladderNone
1323
183158812008
KWKIFKKIEKVGRNIRNGIIKAGPAVAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntimicrobialChinese oak silk moth486PBladder CancerWST-1 assayIC50=161.76 µg/ml48-hBladderNone
1320
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)J82Bladder CancerWST-1 assayIC50=212.07 µg/ml48-hBladderNone
1319
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)647VBladder CancerWST-1 assayIC50=185.39 µg/ml48-hBladderNone
1318
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)RT4Bladder CancerWST-1 assayIC50=231.26 µg/ml48-hBladderNone
1317
183158812008
KWKLFKKIEKVGQNIRDGIIKAGPAVAVVGQATQIAK
Cecropin A37LinearLNoneAmidationFreeAntimicrobialHyalophora Cecropia(silkmoth)486PBladder CancerWST-1 assayIC50=251.47 µg/ml48-hBladderNone
1251
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)MCF-7RBreast CancerMTT assayIC50=24.596-hBreastNone
1250
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)A-2780ROvarian CancerMTT assayIC50=34.596-hOvaryNone
1249
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)HT-29Colon CancerMTT assayIC50=>100 µM96-hColonNone
1248
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)MCF-7Breast CancerMTT assayIC50=42.5 µM96-hBreastNone
1247
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)MAC15AColon CancerMTT assayIC50=37 µM96-hColonNone
1246
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)CHO-KIOvarian CancerMTT assayIC50=32 µM96-hOvaryNone
1245
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)HCLOColon CancerMTT assayIC50=33.5 µM96-hColonNone
1244
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)A-2780Ovarian CancerMTT assayIC50=30.6 µM96-hOvaryNone
1243
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)WEHI-3BLeukemia CancerMTT assayIC50=4.4 µM96-hBloodNone
1242
78494201994
MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVG
Shiva-138LinearLNoneFreeFreeAntibacterialMagaininDLD-1Colon CancerMTT assayIC50=>100 µM96-hColonNone
1241
78494201994
MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVG
Shiva-138LinearLNoneFreeFreeAntibacterialMagaininHRT-18Colon CancerMTT assayIC50=49.3 µM96-hColonNone
1240
78494201994
MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVG
Shiva-138LinearLNoneFreeFreeAntibacterialMagaininBTS-30Breast CancerMTT assayIC50=56 µM96-hBreastNone
1239
78494201994
MPRWRLFRRIDRVGKQIKQGILRAGPAIALVGDARAVG
Shiva-138LinearLNoneFreeFreeAntibacterialMagaininK-562Leukemia CancerMTT assayIC50=28.7 µM96-hBloodNone
1238
78494201994
SWLSKTAKKLENSAKKRISEGIAIAIQGGPR
Cecropin P131LinearLNoneFreeFreeAntibacterialSmall Intestine of PigDLD-1Colon CancerMTT assayIC50=>100 µM96-hColonNone
1237
78494201994
SWLSKTAKKLENSAKKRISEGIAIAIQGGPR
Cecropin P131LinearLNoneFreeFreeAntibacterialSmall Intestine of PigHRT-18Colon CancerMTT assayIC50=>100 µM96-hColonNone
1236
78494201994
SWLSKTAKKLENSAKKRISEGIAIAIQGGPR
Cecropin P131LinearLNoneFreeFreeAntibacterialSmall Intestine of PigBTS-30Breast CancerMTT assayIC50=>100 µM96-hBreastNone
1235
78494201994
SWLSKTAKKLENSAKKRISEGIAIAIQGGPR
Cecropin P131LinearLNoneFreeFreeAntibacterialSmall Intestine of PigK-562Leukemia CancerMTT assayIC50=93 µM96-hBloodNone
1234
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)DLD-1Colon CancerMTT assayIC50=>100 µM96-hColonNone
1233
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)HRT-18Colon CancerMTT assayIC50=25.5 µM96-hColonNone
1232
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)BTS-30Breast CancerMTT assayIC50=24.8 µM96-hBreastNone
1231
78494201994
KWKVFKKIEKMGRNIRNGIVKAGPAIAVLGEAKAL
Cecropin B35LinearLNoneAmidationFreeAntibacterialHyalophora Cecropia(silkmoth)K-562Leukemia CancerMTT assayIC50=15.5 µM96-hBloodNone
7740
None2019
RQIKIWFQNRRMKWKKRQRRNDLRSSFLTLRDHVP
IDP-NLCa0235LinearLNoneFreeFreeAnticancerSyntheticRG1GlioblastomaAlamarBlue assayEC50 ~ 5 μM72-96 hBrainWO 2019/025432 Al
7757
None2020
RQIKWFQNRRMKWKKSKAPKVVILSKALEYLQA
IDP-LLCb0233LinearLNoneFreeFreeAnticancerSyntheticNCl-H187Lung CancerMTT/Alamamar-Blue/Hexosaminidase activity testEC50 ~ 7.5 μM48-72 hLungUS20200239547A1
7758
None2020
RQIKWFQNRRMKWKKSKAPKVVILSKALEYLQA
IDP-LLCb0233LinearLNoneFreeFreeAnticancerSyntheticNCl-H82Lung CancerMTT/Alamamar-Blue/Hexosaminidase activity testEC50 ~ 10 μM48-72 hLungUS20200239547A1
7759
None2020
RQIKWFQNRRMKWKKSKAPKVVILSKALEYLQA
IDP-LLCb0233LinearLNoneFreeFreeAnticancerSyntheticNCl-H510ALung CancerMTT/Alamamar-Blue/Hexosaminidase activity testEC50 ~ 15 μM48-72 hLungUS20200239547A1
7816
None2022
LTSVVFILICCFHLENIFVLLKKRTLRKNDRKKR
Sample Peptide 1 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 48% at 25 μM48-hKidneyUS011339203B2
7817
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 0.4% at 25 μM48-hKidneyUS011339203B2
7818
None2022
WFLREGSMFVALSASVFSLLAIKKRTLRKNDRKKR
Sample Peptide 3 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 45.8% at 25 μM48-hKidneyUS011339203B2
7819
None2022
FLLISACWVISLILGGLPIMGWKKRTLRKNDRKKR
Sample Peptide 4 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 85.6% at 25 μM48-hKidneyUS011339203B2
7821
None2022
VIIVLSVFIACWAPLFILLLLKKRTLRKNDRKKR
Sample Peptide 6 from US011339203B234LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 59.7% at 25 μM48-hKidneyUS011339203B2
7822
None2022
LFRAEYFLVLAVLNSGTNPIIKKRTLRKNDRKKR
Sample Peptide 7 from US011339203B234LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 66.3% at 25 μM48-hKidneyUS011339203B2
7823
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticPC-3Prostate CancerCCK-8 assayCell Viability = 2.5% at 25 μM48-hKidneyUS011339203B2
7824
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticA-2058Skin CancerCCK-8 assayCell Viability = 0.2% at 25 μM48-hSkinUS011339203B2
7825
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 assayCell Viability = 0.6% at 25 μM48-hLungUS011339203B2
7826
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticA-549Lung CancerCCK-8 assayCell Viability = 1.4% at 25 μM48-hLungUS011339203B2
7827
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 / WST-8Cell Viability = 6.8% at 25 μM48-hLungEP3604345B1;US11352408B2
7829
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 / WST-8Cell Viability = 87.7% at 25 μM48-hLungEP3604345B1
7830
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 11.8% at 25 μM48-hLungEP3604345B1
7832
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 120.6% at 25 μM48-hLungEP3604345B1
7833
None2023
PWWWPPVVVQQQMILLIGAARKKRTLRKNDRKKR
Sample Peptide 4 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 102.6% at 25 μM48-hLungEP3604345B1
7836
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticNCI-H446Lung CancerCCK-8 / WST-8Cell Viability = 0.5% at 25 μM48-hLungEP3604345B1
7837
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticNCI-H446Lung CancerCCK-8 / WST-8Cell Viability = 56.7% at 25 μM48-hLungEP3604345B1
7838
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticA-2058Skin CancerCCK-8 / WST-8Cell Viability = 6.7% at 25 μM48-hSkinEP3604345B1
7839
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticA-2058Skin CancerCCK-8 / WST-8Cell Viability = 87.5% at 25 μM48-hSkinEP3604345B1
7840
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerCCK-8 / WST-8Cell Viability = 62.3% at 25 μM48-hBreastEP3604345B1
7841
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerCCK-8 / WST-8Cell Viability = 81.7% at 25 μM48-hBreastEP3604345B1