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| ID | PMID | YEAR | Sequence | Name | Length | Linear/Cyclic | Chirality | Chem-MOD | C-ter MOD | N-ter MOD | Nature | Origin | Cell Line | Cancer Type | Assay | Activity | Testing Time | Tissue Affected | Patents |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| None | 2020 | Seq ID No. 17 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | NCI-H460 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 17 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | HOP-062 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 16 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | Calu-1 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 16 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | NCI-H460 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 16 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | HOP-062 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 15 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | Calu-1 | Lung Cancer | Tetrazolium-based assay | Cell viability < 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 15 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | NCI-H460 | Lung Cancer | Tetrazolium-based assay | Cell viability < 25% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 15 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | HOP-062 | Lung Cancer | Tetrazolium-based assay | Cell viability ~ 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2022 | ATRA1-R3W2 - HYD | 21 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | H-358 | Lung Cancer | Cytotoxicity assay | LD50 ~24.5 μM | 6-h | Lung | US011447533B2 | ||
| 37853814 | 2024 | NRC-07 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | 52.5 ± 5.0% cell viability at 150 µM | 24-h | Breast | None | ||
| 37853814 | 2024 | NRC-07 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | 14.0 ± 3.0% cell viability at 150 µM | 24-h | Breast | None | ||
| 37880286 | 2023 | MC–FA | 27 | Linear | L | None | Folic Acid | Free | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 12.63 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | MC–FA | 27 | Linear | L | None | Folic Acid | Free | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 66.43 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | MC–FA | 27 | Linear | L | None | Folic Acid | Free | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 35.22 µg/ mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | CM–FA | 27 | Linear | L | None | Amidation | Folic Acid | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 35.75 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | CM–FA | 27 | Linear | L | None | Amidation | Folic Acid | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 10.38 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | CM–FA | 27 | Linear | L | None | Amidation | Folic Acid | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 67.34 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | Mel-C | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 160.62 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | Mel-C | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 58.63 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | Mel-C | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 50.72 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | C-Mel | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 110.59 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | C-Mel | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 44.76 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | C-Mel | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 64.15 µg/mL | 24-h | Cervix | None | ||
| 36873017 | 2023 | LK-LE3 | 30 | Cyclic | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 10.2 µM at pH 6 | 24-h | Cervix | None | ||
| 36873017 | 2023 | LK-LE2 | 30 | Cyclic | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 12.9 µM at pH 6 | 24-h | Cervix | None | ||
| 36873017 | 2023 | LK-LE1 | 30 | Cyclic(C1-C16) | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 11.3 µM at pH 6 | 24-h | Cervix | None | ||
| 37734650 | 2023 | NKL-MUT | 27 | Linear | L | None | Free | Free | Antimicrobial | Trematomus bernacchii | B16-F10 | Skin Cancer | luciferase-based ATPlite assay | ATP level = 0.023 ± 0.007 at 40 μM | 12-h | Skin | None | ||
| 37734650 | 2023 | NKL-WT | 27 | Linear | L | None | Free | Free | Antimicrobial | Trematomus bernacchii | B16-F10 | Skin Cancer | luciferase-based ATPlite assay | ATP level = 0.753 ± 0.254 at 40 μM | 12-h | Skin | None | ||
| 36840453 | 2023 | AMP-WF3 | 25 | Linear | L | None | Free | Free | Anticancer | Poecilia Mexicana fish | Jurkat | Blood Cancer | MTT assay | IC50 = 50 µM | 24-h | Blood | None | ||
| 36626098 | 2023 | bLF | 25 | Linear | L | None | Free | Free | Antimicrobial | Bos Taurus | Jurkat | Blood Cancer | MTT assay | cell viability ~ 17.5% at 20 µM | 4-h | Blood | None | ||
| 36626098 | 2023 | bLF | 25 | Linear | L | None | Free | Free | Antimicrobial | Bos Taurus | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 21% at 10 µM | 24-h | Liver | None | ||
| 37098530 | 2023 | Mellitin | 26 | Linear | L | None | Amidation | Free | Anticancer | Main component of honey bee venom | K-562 | Leukemia Cancer | Sulforhodamine B assay | IC50 = 1.84 ± 0.75 μg/ml | 96-h | Blood | None | ||
| 36830725 | 2023 | Pep-1-Phor21 | 30 | Linear | L | None | Free | Free | Anticancer | Hybrid peptide PEP1 and Phor 21 | PC-3 | Prostrate Cancer | AlamarBlue assay | IC50 ≤ 0.6 μM | 24-h | Prostate | None | ||
| 36830725 | 2023 | Pep-1-Phor21 | 30 | Linear | L | None | Free | Free | Anticancer | Hybrid peptide PEP1 and Phor 21 | DU-145 | Prostrate Cancer | AlamarBlue assay | IC50 = 2.57 ± 2.02 µM | 24-h | Prostate | None | ||
| 36830725 | 2023 | Pep-1-Phor21 | 30 | Linear | L | None | Free | Free | Anticancer | Hybrid peptide PEP1 and Phor 21 | LNCaP | Liver Cancer | AlamarBlue assay | IC50 = 55.13 ± 13.56 µM | 24-h | Liver | None | ||
| 37580909 | 2023 | mPNC-NLS | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | Cytotoxicity assay | IC50 = 45 μM | 24-h | Lung | None | ||
| 37580909 | 2023 | mPNC-NLS | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | U-87 | Brain Tumor | MTT assay | IC50 = 56.9 μM | 24-h | Brain | None | ||
| 37580909 | 2023 | mPNC-NLS | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 44.9 μM | 24-h | Lung | None | ||
| 37483971 | 2023 | ATMP1 | 24 | Linear | L | None | Free | Free | Antimicrobial | Anabas testudineus | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 8.25 ± 0.14 μg/ml | 48-h | Breast | None | ||
| 37483971 | 2023 | ATMP5 | 24 | Linear | L | None | Free | Free | Anticancer; Antimicrobial | Synthetic Analog of ATMP1 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 64.04 ± 0.021 μg /ml | 24-h | Breast | None | ||
| None | 2023 | Raniseptin-3 | 28 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Boana raniceps | B16-F10 | Skin Cancer | MTT assay | IC50 = 6.56 uM | 3-h | Skin | None | ||
| None | 2023 | Raniseptin-6 | 29 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Boana raniceps | B16-F10 | Skin Cancer | MTT assay | IC50 = 8.69 uM | 3-h | Skin | None | ||
| 37310533 | 2023 | PMAP-NC | 23 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analgog of PMAP-24 | A-549 | Lung Cancer | MTT assay | IC50 = 7.1 μM | 4-h | Lung | None | ||
| 37310533 | 2023 | PMAP-NC | 23 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analgog of PMAP-23 | MDA-MB-361 | Breast Cancer | MTT assay | IC50 = 6.4 μM | 4-h | Breast | None | ||
| 37764334 | 2023 | 14VL23 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 16.4 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14VL23 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 5.7 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V5K | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 6.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V5K | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 8.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L2V | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 0.6 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L2V | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 2.2 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14G | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 31.7 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14G | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 48.7 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 4.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 7.0 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L14 | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 20.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L14 | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 64.4 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | Dermaseptin-SS1 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Brown-belly leaf frog, Phyllomedusa Tarsius | H-460 | Lung Cancer | MTT assay | IC50 = 1.3 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | Dermaseptin-SS1 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Brown-belly leaf frog, Phyllomedusa Tarsius | H-838 | Lung Cancer | MTT assay | IC50 = 7.7 µM | 24-h | Lung | None | ||
| 37228702 | 2023 | B1AW-K | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | analogue of B1AW | U251-MG | Brain Tumor | MTT assay | IC50 = 3.860 µM | 24-h | Brain | None | ||
| 37228702 | 2023 | B1AW-K | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | analogue of B1AW | H-838 | Lung Cancer | MTT assay | IC50 = 5.15 µM | 24-h | Lung | None | ||
| 37228702 | 2023 | B1AW-K | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | analogue of B1AW | PC-3 | Prostate Cancer | MTT assay | IC50 = 4.283 µM | 24-h | Prostate | None | ||
| 37228702 | 2023 | B1AW | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Wuyi torrent frog, Amolops wuyiensis | U251-MG | Brain Tumor | MTT assay | IC50 = 33.56 µM | 24-h | Brain | None | ||
| 37228702 | 2023 | B1AW | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Wuyi torrent frog, Amolops wuyiensis | H-838 | Lung Cancer | MTT assay | IC50 = 32.15 µM | 24-h | Lung | None | ||
| 37228702 | 2023 | B1AW | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Wuyi torrent frog, Amolops wuyiensis | PC-3 | Prostate Cancer | MTT assay | IC50 = 33.46 µM | 24-h | Prostate | None | ||
| 37508198 | 2023 | Figanin 2BN | 27 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | HT-29 | Colon Cancer | MTT assay | LC50 = 14.1 uM | 24-h | Colon | None | ||
| 37508198 | 2023 | Figanin 2BN | 27 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | MDA-MB-231 | Breast Cancer | MTT assay | LC50 = 8.1 uM | 24-h | Breast | None | ||
| 37508198 | 2023 | Figanin 2BN | 27 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | A-549 | Lung Cancer | MTT assay | LC50 = 6.7 uM | 24-h | Lung | None | ||
| 37508198 | 2023 | Picturin 1BN | 25 | Linaer | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | HT-29 | Colon Cancer | MTT assay | LC50 = 84.9 uM | 24-h | Colon | None | ||
| 37508198 | 2023 | Picturin 1BN | 25 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | MDA-MB-231 | Breast Cancer | MTT assay | LC50 = 64.2 uM | 24-h | Breast | None | ||
| 37508198 | 2023 | Picturin 1BN | 25 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | A-549 | Lung Cancer | MTT assay | LC50 = 30.7 µM | 24-h | Lung | None | ||
| 37508198 | 2023 | Picturin 2BN | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | HT-29 | Colon Cancer | MTT assay | LC50 52.2 uM | 24-h | Colon | None | ||
| 37508198 | 2023 | Picturin 2BN | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | MDA-MB-231 | Breast Cancer | MTT assay | LC50 26.3 uM | 24-h | Breast | None | ||
| 37508198 | 2023 | Picturin 2BN | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | A-549 | Lung Cancer | MTT assay | LC50 = 23 µM | 24-h | Lung | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 32.47 µM | 36-h | Lung | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | CCK-8 assay | IC50 = 25.65 µM | 36-h | Bone | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | CCK-8 assay | IC50 = 42.95 µM | 36-h | Cervix | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | ZR-75-30 | Breast Cancer | CCK-8 assay | IC50 = 23.57 µM | 36-h | Breast | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 31.05 µM | 36-h | Breast | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | CCK-8 assay | IC50 = 18.15 µM | 36-h | Breast | None | ||
| 37396945 | 2023 | p28 | 28 | Linear | L | None | Free | Free | Antitumor | Pseudomonas aeruginosa | CT-26 | Colorectal Cancer | MTT assay | IC50 ~ 150 μg/ml | 24-h | Colon | None | ||
| 37396945 | 2023 | p28 | 28 | Linear | L | None | Free | Free | Antitumor | Pseudomonas aeruginosa | HT-29 | Colon Cancer | MTT assay | IC50 ~ 200 μg/ml | 24-h | Colon | None | ||
| 36410436 | 2023 | FHV-2D5 | 23 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-G | 48-h | Liver | None | ||
| 36410436 | 2023 | HTLV-II-Rex-2D5 | 21 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-G | 48-h | Liver | None | ||
| 36410436 | 2023 | TAT-2D5 | 21 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-G | 48-h | Liver | None | ||
| 36410436 | 2023 | 6E(V116-M135) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-D | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D(Q44-R55) | 22 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2C(Q44-Q58) | 25 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2A(F39-Q58) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | #6(M108-L127) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | MCF-7 | Breast Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Breast | None | ||
| 36410436 | 2023 | #6(M108-L127) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Liver | None | ||
| 36410436 | 2023 | #5(D93-F112) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Liver | None | ||
| 36410436 | 2023 | #2(D33-N52) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | MCF-7 | Breast Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Breast | None | ||
| 36410436 | 2023 | #2(D33-N52) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Liver | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 24.60 μM | 24-h | Breast | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | U-251-MG | Brain Tumor | MTT assay | IC50 = 25.06 μM | 24-h | Brain | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | H-157 | Non-small cell lung cancer | MTT assay | IC50 = 24 μM | 24-h | Lung | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | PC-3 | Prostate cancer | MTT assay | IC50 = 31.27 μM | 24-h | Prostate | None | ||
| 35606468 | 2022 | Nigrocin-PN | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Pelophylax nigromaculatus | PC-3 | Prostate cancer | MTT assay | IC50 = 53.03 μM | 24-h | Prostate | None | ||
| 35606468 | 2022 | Nigrocin-PN | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Pelophylax nigromaculatus | U-251-MG | Brain Tumor | MTT assay | IC50 = 73.65 μM | 24-h | Brain | None | ||
| 35606468 | 2022 | Nigrocin-PN | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Pelophylax nigromaculatus | H-157 | Non-small cell lung cancer | MTT assay | IC50 = 18.04 μM | 24-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | HCC-827 | Lung Adenocarcinoma | MTT assay | IC50 between 4.0 and 5.5 μM | 72-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | H-1975 | Non Small Cell Lung Cancer (NSCLC) | MTT assay | IC50 between 4.0 and 5.5 μM | 72-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | H-358 | Non Small Cell Lung Cancer (NSCLC) | MTT assay | IC50 = 4.00 ± 0.20 μM | 72-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 5.55 ± 0.13 μM | 72-h | Lung | None | ||
| 36287985 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | HepG-2 | Liver Cancer | MTT assay | IC50 = 5.524 µM | 24-h | Liver | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | H-460 | Lung Cancer | MTT assay | IC50 = 7.07 ± 0.81 µM | 24-h | Lung | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | PC-9 | Lung Cancer | MTT assay | IC50 = 6.34 ± 0.53 µM | 24-h | Lung | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | H-3122 | Lung Cancer | MTT assay | IC50 = 4.64 ± 0.18 µM | 24-h | Lung | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | A-549 | Lung Cancer | MTT assay | IC50 = 4.06 ± 0.60 µM | 24-h | Lung | None | ||
| 35601827 | 2022 | LyeTx-I-b | 24 | Linear | L | None | Amidated | Acetylation | Antimicrobial | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 2.47 µM | 48-h | Breast | None | ||
| 35013881 | 2022 | Brevinin-2R | 25 | Linear | L | None | Free | Free | Antimicrobial | Rana ridibunda | HeLa | Cervical Cancer | MTT assay | IC50 = 131.5 μg/ml | 24-h | Cervix | None | ||
| 36465844 | 2022 | HAZ | 21 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 5.44 μM | 4-h | Lung | None | ||
| 35774163 | 2022 | D-NAF-1 | 24 | Linear | D | None | Free | Free | Anticancer | NAF-1/CISD2 | MDA-MB-231 | Breast Cancer | Not Available | IC50 = 12.8 ± 0.2 μM | NA | Breast | None | ||
| 35774163 | 2022 | NAF-1 | 24 | Linear | L | None | Free | Free | Anticancer | NAF-1/CISD2 | MDA-MB-231 | Breast Cancer | Not Available | IC50 = 18.3 ± 0.4 μM | NA | Breast | None | ||
| 36672551 | 2022 | CIGB-300 | 25 | Cyclic | L | X = Beta- Alanine | Free | Biotinylated | Anticancer | Synthetic | NCI-H-460 | Lung Cancer | Crystal Violet assay | IC50 = 30 ± 5.3 µM | 48-h | Lung | None | ||
| 35745643 | 2022 | BmPLA2 | 24 | Linear | L | None | Free | Free | Anticancer | phospholipase A2 isoform from B. moojeni venom | RD | Rhabdomyosarcoma | MTT assay | 60% reduction in cell viability | 24-h | Muscle | None | ||
| 35745643 | 2022 | BmPLA2 | 24 | Linear | L | None | Free | Free | Anticancer | phospholipase A2 isoform from B. moojeni venom | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 0.6 µM | 24-h | Colon | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | MCF-7 | Breast Cancer | MTT assay | EC50 = 0.724 ± 0.340 mol/L × 10-3 | 24-h | Breast | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | A-2058 | Skin Cancer | MTT assay | EC50 = 0.744 ± 0.208 mol/L × 10-3 | 24-h | Skin | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | U-87 | Brain Tumor | MTT assay | EC50 = 0.427 ± 0.053 mol/L × 10-3 | 24-h | Brain | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | HeLa | Cervical Cancer | MTT assay | EC50 = 0.525 ± 0.160 mol/L × 10-3 | 24-h | Cervix | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | B16-F10-Nex 2 | Skin Cancer | MTT assay | EC50 = 0.263 ± 0.585 mol/L × 10-3 | 24-h | Skin | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | WiDr | Colon Cancer | MTT assay | IC50 = 197.3 μM | 24-h | Colon | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | AGS | Stomach Cancer | MTT assay | IC50 = 29.8 μM | 24-h | Stomach | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | A-549 | Lung Cancer | MTT assay | IC50 = 42.1 μM | 24-h | Lung | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | Hep3B | Liver Cancer | MTT assay | IC50 = 77.5 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | Huh-7 | Liver Cancer | MTT assay | IC50 = 60 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | J5 | Liver Cancer | MTT assay | IC50 = 11 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | AGS | Stomach Cancer | MTT assay | IC50 = 186.5 μM | 24-h | Stomach | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | A-549 | Lung Cancer | MTT assay | IC50 = 300.8 μM | 24-h | Lung | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | Hep3B | Liver Cancer | MTT assay | IC50 = 340.9 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | J5 | Liver Cancer | MTT assay | IC50 = 54.9 μM | 24-h | Liver | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | SNB-19 | Brain Tumor | CCK-8 assay | IC50 = 12.0 ± 0.6 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | SF-268 | Brain Tumor | CCK-8 assay | IC50 = 4.8 ± 0.1 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-138 | Brain Tumor | CCK-8 assay | IC50 = 7.5 ± 0.3 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | LN229 | Brain Tumor | CCK-8 assay | IC50 = 4.7 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | SW-1783 | Brain Tumor | CCK-8 assay | IC50 = 4.8 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | D54 | Brain Tumor | CCK-8 assay | IC50 = 8.4 ± 0.1 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-118 | Brain Tumor | CCK-8 assay | IC50 = 6.8 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-373 | Brain Tumor | CCK-8 assay | IC50 = 5.0 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | T98G | Brain Tumor | CCK-8 assay | IC50 = 7.1 ± 0.2 μM | 96-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | A-172 | Brain Tumor | CCK-8 assay | IC50 = 6.4 ± 0.4 μM | 96-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-251 | Brain Tumor | CCK-8 assay | IC50 = 4.9 ± 0.3 μM | 96-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U87-MG | Brain Tumor | CCK-8 assay | IC50 = 4.3 ± 0.3 μM | 96-h | Brain | None | ||
| 35660629 | 2022 | NRC-03 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | skin mucous secretions of winter flounder | SCC-9 | Oral Cancer | CCK-8 assay | IC50 = 45 μg/ml | 24-h | Tongue | None | ||
| 35660629 | 2022 | NRC-03 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | skin mucous secretions of winter flounder | CAL-27 | Oral Cancer | CCK-8 assay | IC50 = 45 μg/ml | 24-h | Tongue | None | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 57.03 ± 6.09 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 57.99 ± 5.04 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 33.92 ± 5.90 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 57.45 ± 6.03 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 35.71 ± 8.50 µM | 48-h | Breast | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 70.71 ± 5.39 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 4.72 ± 0.36 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 6.31 ± 0.66 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 8.71 ± 0.35 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 4.42 ± 0.06 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 3.79 ± 1.61 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | HepG-2 | Liver Cancer | Resazurin dye assay | IC50 = 14.31 ± 1.37 µM | 48-h | Liver | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 5.69 ± 1.46 µM | 48-h | Breast | US_10550155_B2 | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | B16-F10 | Skin Cancer | MTS assay | IC50 = 6.65 ± 0.33 μM | 48-h | Skin | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | SMMC-7721 | Liver Cancer | MTS assay | IC50 = 6.87 ± 0.51 μM | 48-h | Liver | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | A-549 | Lung Cancer | MTS assay | IC50 = 5.81 ± 0.23 μM | 48-h | Lung | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | SW-480 | Blood Cancer | MTS assay | IC50 = 10.37 ± 0.40 μM | 48-h | Blood | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 5.44 ± 0.33 μM | 48-h | Breast | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | HCT-116 | Colon Cancer | MTS assay | IC50 = 5.87 ± 0.15 μM | 48-h | Colon | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 1.97 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 18.1 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 2.99 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 21.6 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 5.25 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 17.5 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 5.52 µM | 24-h | Not Available | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 26.01 µM | 24-h | Not Available | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 2.17 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 2.22 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 2.15 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 4.2 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 3.92 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 5.83 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 5.31 µM | 24-h | Not Available | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 5.58 µM | 24-h | Not Available | None | ||
| 33677023 | 2021 | Pep | 21 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 2 µM | 24-h | Breast | None | ||
| 33677023 | 2021 | Pep | 21 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4 µM | 24-h | Lung | None | ||
| 33690977 | 2021 | NMTP-5 | 24 | Linear | D | Z = C10H7CH2C(O), M, 4-(Trifluoromethyl)-D-phenylalanine | Free | Free | Anticancer | Not Available | SK-HEP-1 | Liver Cancer | MTT assay | IC50 = 53.84 ± 4.35 µM | 48-h | Liver | None | ||
| 34309373 | 2021 | Pal-N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | MCF-7 | Breast Cancer | MTT assay | IC50 = 27.26 μM | 24-h | Breast | None | ||
| 34309373 | 2021 | Pal-N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-549 | Lung Cancer | MTT assay | IC50 = 44.98 μM | 24-h | Lung | None | ||
| 34309373 | 2021 | Pal-N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-375 | Skin Cancer | MTT assay | IC50 = 36.67(Supplementary material)/15.2 ± 0.7 μM(Published paper) | 24-h | Skin | None | ||
| 34848729 | 2021 | AtMP2 | 22 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 6.97 ± 0.24 μg/ml | 48-h | Breast | None | ||
| 34848729 | 2021 | AtMP2 | 22 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.89 ± 0.14 μg/ml | 48-h | Breast | None | ||
| 34848729 | 2021 | AtMP1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 9.35 ± 0.25 μg/ml | 48-h | Breast | None | ||
| 34848729 | 2021 | AtMP1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.25 ± 0.14 μg/ml | 48-h | Breast | None | ||
| 33562681 | 2021 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | Aska-SS | Synovial Sarcoma | MTS assay | IC50 = 32.41 μg/mL | NA | Muscle | None | ||
| 33562681 | 2021 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | SW982 | Synovial Sarcoma | MTS assay | IC50 = 29.20 μg/mL | NA | Muscle | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | MDA-MB-435 DOX-R | Breast Cancer | MTS assay | IC50 = 3.4 µM | 24-h | Breast | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | MDA-MB-435 WT | Breast Cancer | MTS assay | IC50 = 3.5 µM | 24-h | Breast | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | CT-26 | Colorectal Cancer | MTS assay | IC50 = 2.2 µM | 24-h | Colon | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTS assay | IC50 = 4.5 µM | 24-h | Lung | None | ||
| 34309373 | 2021 | N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTT assay | IC50 > 50.0 μM | 24-h | Skin | None | ||
| 33582221 | 2021 | Dermaseptin-TO | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tomopterna | PC-3 | Prostate Cancer | MTT assay | Graph Figure-7 | 24-h | Prostate | None | ||
| 33582221 | 2021 | Dermaseptin-TO | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tomopterna | H-157 | Lung Cancer | MTT assay | Graph Figure-7 | 24-h | Lung | None | ||
| 33582221 | 2021 | Dermaseptin-TO | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tomopterna | U251-MG | Brain Tumor | MTT assay | Graph Figure-7 | 24-h | Brain | None | ||
| 34572719 | 2021 | LyeTxI-b | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 5.77 ± 0.83 µM | 48-h | Breast | None | ||
| 34572719 | 2021 | LyeTxI-b | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.34 ± 3.09 µM | 48-h | Breast | None | ||
| 34572719 | 2021 | LyeTxI-b | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | 4T1 | Breast Cancer | MTT assay | IC50 = 6.5 ± 5.30 µM | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | MDA-MB-231 | Breast Cancer | Annexin V-FITC assay | ~80% cell death at 200 µg/ml | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | MCF-7 | Breast Cancer | Annexin V-FITC assay | ~50% cell death at 300 µg/ml | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | SK-BR-3 | Breast Cancer | Annexin V-FITC assay | ~80% cell death at 100 µg/ml | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | MDA-MB-468 | Breast Cancer | Annexin V-FITC assay | ~60% cell death at 300 µg/ml | 48-h | Breast | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.721 µM | 24-h | Colon | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.17 µM | 24-h | Breast | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | U251-MG | Brain Tumor | MTT assay | IC50 = 3.492 µM | 24-h | Brain | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | PC-3 | Prostate Cancer | MTT assay | IC50 = 2.629 µM | 24-h | Prostate | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | H-838 | Lung Cancer | MTT assay | IC50 = 2.553 µM | 24-h | Lung | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | HCT-116 | Colon Cancer | MTT assay | IC50 = 11.03 µM | 24-h | Colon | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.883 µM | 24-h | Breast | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | U251-MG | Brain Tumor | MTT assay | IC50 = 8.629 µM | 24-h | Brain | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.473 µM | 24-h | Prostate | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | H-838 | Lung Cancer | MTT assay | IC50 = 3.976 µM | 24-h | Lung | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | HCT-116 | Colon Cancer | MTT assay | IC50 = 33.69 µM | 24-h | Colon | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | MCF-7 | Breast Cancer | MTT assay | IC50 = 112 µM | 24-h | Breast | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | U251-MG | Brain Tumor | MTT assay | IC50 = 233.0 µM | 24-h | Brain | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | PC-3 | Prostate Cancer | MTT assay | IC50 = 95.94 µM | 24-h | Prostate | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | H-838 | Lung Cancer | MTT assay | IC50 = 36.84 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.583 µM | 24-h | Colon | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | H-157 | Lung Cancer | MTT assay | IC50 = 2.811 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 2.243 µM | 24-h | Breast | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.425 µM | 24-h | Prostate | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | HCT-116 | Colon Cancer | MTT assay | IC50 = 342.8 µM | 24-h | Colon | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | H-157 | Lung Cancer | MTT assay | IC50 = 278.9 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 214.7 µM | 24-h | Breast | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | PC-3 | Prostate Cancer | MTT assay | IC50 = 186.9 µM | 24-h | Prostate | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.599 µM | 24-h | Colon | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | H-157 | Lung Cancer | MTT assay | IC50 = 3.37 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 3.47 µM | 24-h | Breast | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.87 µM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 1499 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 427.3 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 180.8 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 118.4 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 593.7 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 88.28 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 186.1 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 55.65 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 2.679 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 1.546 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 1.796 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 2.605 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 32.18 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 6.143 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 10.11 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 18.99 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | U251-MG | Brain Tumor | MTT assay | IC50 = 34.25 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | H-157 | Lung Cancer | MTT assay | IC50 = 10.20 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | H-838 | Lung Cancer | MTT assay | IC50 = 23.51 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | PC-3 | Prostate Cancer | MTT assay | IC50 = 14.67 μM | 24-h | Prostate | None | ||
| None | 2020 | D(KLAKLAK)2-TAT | 25 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 5.3 μM | 24-h | Lung | None | ||
| 32443921 | 2020 | Figainin 2 | 28 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Boana raniceps | MCF-7 | Breast Cancer | MTT assay | IC50= 15.3 µM | 24-h | Breast | None | ||
| 32443921 | 2020 | Figainin 2 | 28 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Boana raniceps | B16-F10 | Skin Cancer | MTT assay | IC50 = 12.8 µM | 24-h | Skin | None | ||
| 32498425 | 2020 | LVTX-8 | 25 | Linear | L | None | Amidation | Acetylation | Anticancer | Lycosa vittata | H-460 | Lung Cancer | CCK-8 assay | IC50 = 19 μM | 24-h | Lung | None | ||
| 32498425 | 2020 | LVTX-8 | 25 | Linear | L | None | Amidation | Acetylation | Anticancer | Lycosa vittata | A-549 | Lung Cancer | CCK-8 assay | IC50 = 8 μM | 24-h | Lung | None | ||
| 32256172 | 2020 | NMANF2 | 21 | Linear | L | None | Free | Free | Anticancer | Staphylococcus hominis strain MANF2 | HT-29 | Colon Cancer | MTT assay | IC50 = 48.9 µg/mL | NA | Colon | None | ||
| 32256172 | 2020 | NMANF2 | 21 | Linear | L | None | Free | Free | Anticancer | Staphylococcus hominis strain MANF2 | A-549 | Lung Cancer | MTT assay | IC50 = 46.6 µg/mL | NA | Lung | None | ||
| 34508563 | 2020 | Brevinin-1HL | 24 | Linear | L | None | Free | Free | Antimicrobial | Hylarana latouchii | NCI-H23 | Lung Cancer | MTT assay | IC50 = 8.52 ± 1.02 μM | 24-h | Lung | None | ||
| 32151609 | 2020 | R-DIM-LF11-334-LF11-334 | 24 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 3.6 ± 0.7 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-LF11-334-LF11-334 | 24 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 < 1 ± 0.1 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-LF11-334-LF11-334 | 24 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 < 1 ± 0.1 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11 | 23 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 20.9 ± 3.9 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11 | 23 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 10.7 ± 0.2 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11 | 23 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 125.0 ± 16.8 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32462055 | 2020 | AEM-28–2 | 28 | Linear | L | Aha= α-aminohenoic acid | Amidation | Acetylation | Anti-inflammatory and Anticancer | Synthetic | OV-2008 | Ovarian Cancer | MTS assay | ~40% cell viability at 10 μg/mL | 24-h | Ovary | None | ||
| 32462055 | 2020 | AEM-28–2 | 28 | Linear | L | Aha= α-aminohenoic acid | Amidation | Acetylation | Anti-inflammatory and Anticancer | Synthetic | SK-OV-3 | Ovarian Cancer | MTS assay | ~30% cell viability at 10 μg/mL | 24-h | Ovary | None | ||
| 32462055 | 2020 | AEM-28–2 | 28 | Linear | L | Aha= α-aminohenoic acid | Amidation | Acetylation | Anti-inflammatory and Anticancer | Synthetic | CaCo-2 | Colon Cancer | MTS assay | ~60% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32462055 | 2020 | AEM-28–2 | 28 | Linear | L | Aha= α-aminohenoic acid | Amidation | Acetylation | Anti-inflammatory and Anticancer | Synthetic | CT-26 | Colorectal Cancer | MTS assay | ~30% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32462055 | 2020 | AEM-28–2 | 28 | Linear | L | Aha= α-aminohenoic acid | Amidation | Acetylation | Anti-inflammatory and Anticancer | Synthetic | ID8 | Colon Cancer | MTS assay | ~20% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32462055 | 2020 | AEM-28 | 28 | Linear | L | None | Free | Free | Anti-inflammatory and Anticancer | Synthetic | CaCo-2 | Colon Cancer | MTS assay | ~70% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32462055 | 2020 | AEM-28 | 28 | Linear | L | None | Free | Free | Anti-inflammatory and Anticancer | Synthetic | SK-OV-3 | Ovarian Cancer | MTS assay | ~50% cell viability at 10 μg/mL | 24-h | Ovary | None | ||
| 32462055 | 2020 | AEM-28 | 28 | Linear | L | None | Free | Free | Anti-inflammatory and Anticancer | Synthetic | OV-2008 | Ovarian Cancer | MTS assay | ~60% cell viability at 10 μg/mL | 24-h | Ovary | None | ||
| 32462055 | 2020 | AEM-28 | 28 | Linear | L | None | Free | Free | Anti-inflammatory and Anticancer | Synthetic | ID8 | Colon Cancer | MTS assay | ~60% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32462055 | 2020 | AEM-28 | 28 | Linear | L | None | Free | Free | Anti-inflammatory and Anticancer | Synthetic | CT-26 | Colorectal Cancer | MTS assay | ~20% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32126228 | 2020 | MPG | 27 | Linear | L | None | Cysteamidation | Acetylation | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 15.8 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | MagaininF5W-Arg | 23 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 16.8 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | MagaininF5W-Lys | 23 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 16.8 μM | 24-h | Blood | None | ||
| 32582642 | 2020 | Dermaseptin-PP | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa palliata | H-157 | Lung Cancer | LDH leakage assay | 80% LDH release at 10−4 M | 24-h | Lung | None | ||
| 32582642 | 2020 | Dermaseptin-PP | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa palliata | U-251 | Brain Tumor | MTT assay | IC50 = 2.47 μM | 24-h | Brain | None | ||
| 32582642 | 2020 | Dermaseptin-PP | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa palliata | PC-3 | Prostate Cancer | MTT assay | IC50 = 4.15 μM | 24-h | Prostate | None | ||
| 32582642 | 2020 | Dermaseptin-PP | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa palliata | MCF-7 | Breast Cancer | MTT assay | IC50 = 2.92 μM | 24-h | Breast | None | ||
| 32582642 | 2020 | Dermaseptin-PP | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa palliata | H-157 | Lung Cancer | MTT assay | IC50 = 1.55 μM | 24-h | Lung | None | ||
| 32347293 | 2020 | Brevinin-1GHd | 24 | Linear | L | None | Free | Free | Antimicrobial | Hylarana guentheri | PC-3 | Prostate Cancer | MTT assay | IC50 = 9.854 µM | 24-h | Prostate | None | ||
| 32347293 | 2020 | Brevinin-1GHd | 24 | Linear | L | None | Free | Free | Antimicrobial | Hylarana guentheri | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 1.197 µM | 24-h | Skin | None | ||
| 32347293 | 2020 | Brevinin-1GHd | 24 | Linear | L | None | Free | Free | Antimicrobial | Hylarana guentheri | U-251-MG | Brain Tumor | MTT assay | IC50 = 7.985 µM | 24-h | Brain | None | ||
| 32347293 | 2020 | Brevinin-1GHd | 24 | Linear | L | None | Free | Free | Antimicrobial | Hylarana guentheri | NCI-H-157 | Lung Cancer | MTT assay | IC50 = 2.987 µM | 24-h | Lung | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8b | 23 | Linear | L | None | Free | 3′-Aminopropyl Beta-D-Galactopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | PC-3 | Prostate Cancer | CCK-8 assay | IC50 = 4.9 ± 0.2 µM | 24-h | Prostate | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8b | 23 | Linear | L | None | Free | 3′-Aminopropyl Beta-D-Galactopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | H-1437 | Lung Cancer | CCK-8 assay | IC50 = 5.3 ± 0.2 µM | 24-h | Lung | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8b | 23 | Linear | L | None | Free | 3′-Aminopropyl Beta-D-Galactopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | HGC-27 | Gastric Cancer | CCK-8 assay | IC50 = 5.3 ± 0.2 µM | 24-h | Not Available | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8b | 23 | Linear | L | None | Free | 3′-Aminopropyl Beta-D-Galactopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | A-549 | Lung Cancer | CCK-8 assay | IC50 = 7.0 ± 0.3 µM | 24-h | Lung | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8b | 23 | Linear | L | None | Free | 3′-Aminopropyl Beta-D-Galactopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | H-460 | Lung Cancer | CCK-8 assay | IC50 = 4.9 ± 0.9 µM | 24-h | Lung | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8a | 23 | Linear | L | None | Free | 3′-Aminopropyl-D-glucopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | PC-3 | Prostate Cancer | CCK-8 assay | IC50 = 6.9 ± 0.4 µM | 24-h | Prostate | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8b | 23 | Linear | L | None | Free | 3′-Aminopropyl Beta-D-Galactopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | MDA-MB-231 | Breast Cancer | CCK-8 assay | IC50 = 6.0 ± 0.2 µM | 24-h | Breast | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8a | 23 | Linear | L | None | Free | 3′-Aminopropyl-D-glucopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | HGC-27 | Gastric Cancer | CCK-8 assay | IC50 = 12.6 ± 0.6 µM | 24-h | Not Available | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8a | 23 | Linear | L | None | Free | 3′-Aminopropyl-D-glucopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | H-1437 | Lung Cancer | CCK-8 assay | IC50 = 13.0 ± 0.2 µM | 24-h | Lung | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8a | 23 | Linear | L | None | Free | 3′-Aminopropyl-D-glucopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | H-460 | Lung Cancer | CCK-8 assay | IC50 = 8.5 ± 0.4 µM | 24-h | Lung | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8a | 23 | Linear | L | None | Free | 3′-Aminopropyl-D-glucopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | MDA-MB-231 | Breast Cancer | CCK-8 assay | IC50 = 10.1 ± 0.2 µM | 24-h | Breast | None | ||
| 31276399 | 2019 | R-Lycosin I derivative 8a | 23 | Linear | L | None | Free | 3′-Aminopropyl-D-glucopyranoside | Anticancer | Monosaccharide Analogue of Anticancer Peptide R-Lycosin-I | A-549 | Lung Cancer | CCK-8 assay | IC50 = 9.6 ± 0.3 µM | 24-h | Lung | None | ||
| 31161686 | 2019 | 8Dap | 23 | Linear | L | X = 2,3-Diaminopropionic Acid , Z = norleucine | Amidation | Free | Anticancer | Synthetic | PANC-1 | Pancreatic Cancer | WST-1 assay | EC50 = 61.4±0.7 μM | 24-h | Pancreas | None | ||
| 31161686 | 2019 | 6Dap | 23 | Linear | L | X = 2,3-Diaminopropionic Acid , Z = norleucine | Amidation | Free | Anticancer | Synthetic | PANC-1 | Pancreatic Cancer | WST-1 assay | EC50 = 55.0±1.8 μM | 24-h | Pancreas | None | ||
| 31161686 | 2019 | 4Dap | 23 | Linear | L | X = 2,3-Diaminopropionic Acid , Z = norleucine | Amidation | Free | Anticancer | Synthetic | PANC-1 | Pancreatic Cancer | WST-1 assay | EC50 = 35.7±0.7 μM | 24-h | Pancreas | None | ||
| 31161686 | 2019 | 2Dap | 23 | Linear | L | X = 2,3-Diaminopropionic Acid , Z = norleucine | Amidation | Free | Anticancer | Synthetic | PANC-1 | Pancreatic Cancer | WST-1 assay | EC50 = 14.7±0.6 μM | 24-h | Pancreas | None | ||
| 31161686 | 2019 | 0Dap | 23 | Linear | L | Z = norleucine | Amidation | Free | Anticancer | Synthetic | PANC-1 | Pancreatic Cancer | WST-1 assay | EC50 = 9.1±0.3 μM | 24-h | Pancreas | None | ||
| None | 2019 | LPSBD-0 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | THP-1 | Leukemia Cancer | Not Available | Not Available | 24-h | Blood | None | ||
| None | 2019 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Scorpio maurus palmatus | KG-1a | Leukemia Cancer | LDH leakage assay | Fig 2 | NA | Blood | None | ||
| None | 2019 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Scorpio maurus palmatus | CCRF-CEM | Leukemia Cancer | LDH leakage assay | Fig 2 | NA | Blood | None | ||
| None | 2019 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Scorpio maurus palmatus | KG-1a | Leukemia Cancer | CellTiter-Glo assay | LC50 = 16 ± 1.3 µg/mL | 24-h | Blood | None | ||
| None | 2019 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Scorpio maurus palmatus | CCRF-CEM | Leukemia Cancer | CellTiter-Glo assay | LC50 = 16 ± 0.9 µg/mL | 24-h | Blood | None | ||
| 31252047 | 2019 | Fi-Histin1-21 | 21 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Fenneropenaeus indicus | Hep-2 | Liver Cancer | XTT assay | IC50 = 31.274 ± 24.531 μM | 24-h | Liver | None | ||
| 31252047 | 2019 | Fi-Histin1-21 | 21 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Fenneropenaeus indicus | NCI-H-460 | Lung Cancer | XTT assay | IC50 = 22.670 ± 13.939 μM | 24-h | Lung | None | ||
| 30377840 | 2019 | TC22 | 22 | Linear | L | None | Free | Free | Anticancer | Tribolium castaneum | MCF-7 | Breast Cancer | MTT assay | Fig 4a | 24-h | Breast | None | ||
| 30377840 | 2019 | TC22 | 22 | Linear | L | None | Free | Free | Anticancer | Tribolium castaneum | HeLa | Cervical Cancer | MTT assay | Fig 4a | 24-h | Cervix | None | ||
| 30449002 | 2019 | LyeTx-I-b | 24 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | SH-SY5Y | Brain Tumor | MTT/Resazurin dye assay | IC50 = 93.80 ± 2.17 µM | 48-h | Brain | None | ||
| 30449002 | 2019 | LyeTx-I-b | 24 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | U-373-MG | Brain Tumor | MTT/Resazurin dye assay | IC50 = 20.94 ± 5.18 µM | 48-h | Brain | None | ||
| 30449002 | 2019 | LyeTx-I-b | 24 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | U-87-MG | Brain Tumor | MTT/Resazurin dye assay | IC50 = 29.20 ± 7.96 µM | 48-h | Brain | None | ||
| 30717309 | 2019 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | U-251 | Brain Tumor | MTS/PMS assay | LD50 = 20 μg/mL | 24-h | Brain | None | ||
| 30717309 | 2019 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | U87-MG | Brain Tumor | MTS/PMS assay | LD50 = 20 μg/mL | 24-h | Brain | None | ||
| 31633400 | 2019 | HN-1 | 21 | Linear | L | None | Free | Free | Host Defense | Amolops hainanensis | PC-3 | Prostate Cancer | MTT assay | Not Available | 12-h | Prostate | None | ||
| 31633400 | 2019 | HN-1 | 21 | Linear | L | None | Free | Free | Host Defense | Amolops hainanensis | 4T1 | Breast Cancer | MTT assay | Not Available | 12-h | Breast | None | ||
| 31633400 | 2019 | HN-1 | 21 | Linear | L | None | Free | Free | Host Defense | Amolops hainanensis | MDA-MB-453 | Breast Cancer | MTT assay | Not Available | 12-h | Breast | None | ||
| 31633400 | 2019 | HN-1 | 21 | Linear | L | None | Free | Free | Host Defense | Amolops hainanensis | SGC-7901 | Stomach Cancer | MTT assay | Not Available | 12-h | Stomach | None | ||
| 31633400 | 2019 | HN-1 | 21 | Linear | L | None | Free | Free | Host Defense | Amolops hainanensis | A-549 | Lung Cancer | MTT assay | Not Available | 12-h | Lung | None | ||
| 31633400 | 2019 | HN-1 | 21 | Linear | L | None | Free | Free | Host Defense | Amolops hainanensis | MCF-7 | Breast Cancer | MTT assay | IC50 = 6.9 μM | 12-h | Breast | None | ||
| 31226350 | 2019 | BMAP-27 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Cathelicidin | MDA-MB-361 | Breast Cancer | MTT assay | IC50 = 4.2 μM | 48-h | Breast | None | ||
| 31226350 | 2019 | BMAP-27 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Cathelicidin | A-549 | Lung Cancer | MTT assay | IC50 = 5.3 μM | 48-h | Lung | None | ||
| 30885438 | 2019 | Hymenochirin - 1B | 29 | Linear | L | None | Amidation | Free | Host Defense Peptide | Hymenochirus boettgeri | HepG-2 | Liver Cancer | MTT assay | 30% cell viability at 20 μM | 24-h | Liver | None | ||
| 30885438 | 2019 | Hymenochirin - 1B | 29 | Linear | L | None | Amidation | Free | Host Defense Peptide | Hymenochirus boettgeri | NCI-H-460 | Lung Cancer | MTT assay | 10% cell viability at 50 μM | 24-h | Lung | None | ||
| 30885438 | 2019 | Hymenochirin - 1B | 29 | Linear | L | None | Amidation | Free | Host Defense Peptide | Hymenochirus boettgeri | A-549 | Lung Cancer | MTT assay | 40% cell viability at 10 μM | 24-h | Lung | None | ||
| 30885438 | 2019 | Hymenochirin - 1B | 29 | Linear | L | None | Amidation | Free | Host Defense Peptide | Hymenochirus boettgeri | NCI-H-1299 | Lung Cancer | MTT assay | 20% cell viability at 10 μM | 24-h | Lung | None | ||
| 31426323 | 2019 | Dermaseptin-PS4 | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa sauvagii | MCF-7 | Breast Cancer | MTT assay | IC50 = 0.67 µM | 24-h | Breast | None | ||
| 31426323 | 2019 | Dermaseptin-PS4 | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa sauvagii | PC-3 | Prostate Cancer | MTT assay | IC50 = 0.44 μM | 24-h | Prostate | None | ||
| 31426323 | 2019 | Dermaseptin-PS4 | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa sauvagii | H-157 | Lung Cancer | MTT assay | IC50 = 0.19 μM | 24-h | Lung | None | ||
| 31426323 | 2019 | Dermaseptin-PS4 | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa sauvagii | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 0.11 μM | 24-h | Breast | None | ||
| 31426323 | 2019 | Dermaseptin-PS4 | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa sauvagii | U251-MG | Brain Tumor | MTT assay | IC50 = 57.66 nM | 24-h | Brain | None | ||
| 30789695 | 2019 | H-0 | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Hymenochirus boettgeri | HepG-2 | Liver Cancer | MTT assay | IC50 = 8.07 ± 0.21 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-0 | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Hymenochirus boettgeri | HCT-116 | Colon Cancer | MTT assay | IC50 = 12.76 ± 0.43 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-2 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.60 ± 0.24 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-0 | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Hymenochirus boettgeri | A-549 | Lung Cancer | MTT assay | IC50 = 15.22 ± 0.21 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-2 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.54 ± 0.72 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-2 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4.26 ± 0.52 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-5 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 4.16 ± 0.21 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-5 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.82 ± 0.23 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-5 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 7.35 ± 0.22 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-10 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.50 ± 0.21 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-10 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.51 ± 0.37 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-10 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 3.59 ± 0.12 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-14 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 4.54 ± 0.25 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-14 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.841 ± 0.34 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-14 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 0.98 ± 0.11 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-15 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.95 ± 0.25 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-15 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.20 ± 0.27 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-15 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 2.26 ± 0.24 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-16 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.65 ± 0.35 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-16 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.14 ± 0.46 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-16 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 1.85 ± 0.31 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-17 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.49 ± 0.45 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-17 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.64 ± 0.47 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-18 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.61 ± 0.21 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-17 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 0.96 ± 0.33 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-18 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 0.89 ± 0.21 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-18 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.11 ± 0.21 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-19 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.64 ± 0.36 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-19 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 1.00 ± 0.36 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-19 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.78 ± 0.35 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-20 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 4.93 ± 0.53 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-20 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.63 ± 0.35 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-20 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 2.10 ± 0.32 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-21 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.50 ± 0.28 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-21 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 3.26 ± 0.36 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-21 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.05 ± 0.21 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-57 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.13 ± 0.07 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-57 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.29 ± 0.08 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-57 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 0.62 ± 0.12 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | H-58 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.29 ± 0.08 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | H-58 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.13 ± 0.07 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | H-58 | 29 | Cyclic | L | S5 = (S)-N-Fmoc-2-(4′-pentenyl)alanine | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 0.62 ± 0.12 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | [P5K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 4.28 ± 0.38 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | [P5K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 8.09 ± 0.40 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | [P5K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 2.35 ± 0.31 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | [D9K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 4.96 ± 0.43 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | [D9K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 6.50 ± 0.32 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | [D9K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 1.82 ± 0.23 μM | 48-h | Lung | None | ||
| 30789695 | 2019 | [P5K,D9K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.46 ± 0.32 μM | 48-h | Liver | None | ||
| 30789695 | 2019 | [P5K,D9K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | IC50 = 4.93 ± 0.51 μM | 48-h | Colon | None | ||
| 30789695 | 2019 | [P5K,D9K]Hymenochirin-1B | 29 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 1.17 ± 0.23 μM | 48-h | Lung | None | ||
| 31635388 | 2019 | K8, 23-DPT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PANC-1 | Pancreatic Cancer | MTT assay | IC50 = 11.17 µM | 24-h | Pancreas | None | ||
| 31635388 | 2019 | K8, 23-DPT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 9.97 µM | 24-h | Prostate | None | ||
| 31635388 | 2019 | K8, 23-DPT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 9.88 µM | 24-h | Lung | None | ||
| 31635388 | 2019 | K8, 23-DPT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 18.51 µM | 24-h | Brain | None | ||
| 31635388 | 2019 | K8, 23-DPT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.64 µM | 24-h | Breast | None | ||
| 31635388 | 2019 | Dermaseptin-PT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tarsius | PANC-1 | Pancreatic Cancer | MTT assay | IC50 = 28.95 µM | 24-h | Pancreas | None | ||
| 31635388 | 2019 | Dermaseptin-PT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tarsius | PC-3 | Prostate Cancer | MTT assay | IC50 = 21.78 µM | 24-h | Prostate | None | ||
| 31635388 | 2019 | Dermaseptin-PT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tarsius | H-157 | Lung Cancer | MTT assay | IC50 = 25.51 µM | 24-h | Lung | None | ||
| 31635388 | 2019 | Dermaseptin-PT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tarsius | U251-MG | Brain Tumor | MTT assay | IC50 = 49.51 µM | 24-h | Brain | None | ||
| 31635388 | 2019 | Dermaseptin-PT9 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tarsius | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.44 µM | 24-h | Breast | None | ||
| 29043494 | 2018 | NK-pro | 27 | Linear | Mix | None | Amidated | Free | Antimicrobial | Synthetic analog of NK-2 | HL-60 | Leukemia Cancer | MTT assay | IC50 = 26.1 μM | 24-h | Blood | None | ||
| 29043494 | 2018 | NK-pro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | T-24 | Bladder Cancer | MTT assay | IC50 = 33.0 μM | 24-h | Bladder | None | ||
| 29043494 | 2018 | NK-pro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | EJ | Bladder Cancer | MTT assay | IC50 = 23.3 μM | 24-h | Bladder | None | ||
| 29043494 | 2018 | NK-pro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | PC-3 | Prostate Cancer | MTT assay | IC50 = 9.3 μM | 24-h | Prostate | None | ||
| 29043494 | 2018 | NK-dpro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | HL-60 | Leukemia Cancer | MTT assay | IC50 = 48.4 μM | 24-h | Blood | None | ||
| 29043494 | 2018 | NK-dpro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | T-24 | Bladder Cancer | MTT assay | IC50 = 39.6 μM | 24-h | Bladder | None | ||
| 29043494 | 2018 | NK-dpro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | EJ | Bladder Cancer | MTT assay | IC50 = 28.7 μM | 24-h | Bladder | None | ||
| 29043494 | 2018 | NK-dpro | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analog of NK-2 | PC-3 | Prostate Cancer | MTT assay | IC50 = 9.6 μM | 24-h | Prostate | None | ||
| 30183307 | 2018 | R-C16 | 23 | Linear | L | None | Amidation | Fatty acid :C16H31O | Anticancer | R-Lycosin-I | A-549 | Lung Cancer | CCK-8 assay | IC50 ~ 5 µM | 24-h | Lung | None | ||
| 29667478 | 2018 | D-FP21-PEG-PEI/pGRO-α | 21 | Linear | D | conjugated to polyethylenimine (PEI) and methoxy polyethylene glycol (mPEG) | Free | Free | Anti-caner, anti-proliferative, anti-tumor | Synthetic | HO-8910 | Ovarian Cancer | CCK-8 assay | IC50 = 21.6 μg/mL | 24-h | Ovary | None | ||
| 29667478 | 2018 | L-FP21-PEG-PEI/pGRO-α | 21 | Linear | L | conjugated to polyethylenimine (PEI) and methoxy polyethylene glycol (mPEG) | Free | Free | Anti-caner, anti-proliferative, anti-tumor | Synthetic | HO-8910 | Ovarian Cancer | CCK-8 assay | IC50 = 23.4 μg/mL | 24-h | Ovary | None | ||
| 29757646 | 2018 | CyO4 | 30 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial,Cytotoxic | Viola odorata | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 9.8 μM | 24-h | Breast | None | ||
| 29757646 | 2018 | Poca B | 28 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial,Cytotoxic | Pombalia calceolaria | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 2.7 μM | 24-h | Breast | None | ||
| 29757646 | 2018 | Poca A | 30 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial,Cytotoxic | Pombalia calceolaria | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 1.8 μM | 24-h | Breast | None | ||
| 29301308 | 2018 | MSP-4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | MG-63 | Bone Cancer | MTT assay | Cell viability = 26.78 ± 1.75% at 10 µM | 24-h | Bone | None | ||
| 30123940 | 2018 | SmacN7-Arg8 fused peptide P7 | 22 | Cyclic | L | Ahx = aminohexanoic acid; Lactam Bridge between K2 and E10 and between K13 and E22 | Amidation | Free | Anticancer | Synthetic | U-266 | Skin Cancer | Cell Titer Blue Cell Viability assay | Cell viability < 50% at 50 μM | 48-h | Skin | None | ||
| 29800725 | 2018 | MEL-Pep | 26 | Linear | L | None | Amidation | Free | Anticancer | Synthetic analog of Melittin | BEL-7402/5-FU | Liver Cancer | CCK-8 assay | IC50 = 4.36 μM | 24-h | Liver | None | ||
| 29993185 | 2018 | Peptide10 Gonearrestide | 30 | Linear | L | None | Free | Free | Anticancer | Androctonus mauritanicus | U-251 | Brain tumor | MTT assay | Not Available | 24-h | Brain | None | ||
| 29993185 | 2018 | Peptide10 Gonearrestide | 30 | Linear | L | None | Free | Free | Anticancer | Androctonus mauritanicus | Dks8 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide10 Gonearrestide | 30 | Linear | L | None | Free | Free | Anticancer | Androctonus mauritanicus | HKe-3 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide10 Gonearrestide | 30 | Linear | L | None | Free | Free | Anticancer | Androctonus mauritanicus | DLD-1 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide10 Gonearrestide | 30 | Linear | L | None | Free | Free | Anticancer | Androctonus mauritanicus | HCT-116 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 30279210 | 2018 | R2PLx-22 | 22 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 109.30 µM | 24-h | Breast | None | ||
| 30279210 | 2018 | R2PLx-22 | 22 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | U-251-MG | Brain Tumor | MTT assay | IC50 = 104.10 µM | 24-h | Brain | None | ||
| 30279210 | 2018 | R2PLx-22 | 22 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | PC-3 | Prostate Cancer | MTT assay | IC50 = 283.90 µM | 24-h | Prostate | None | ||
| 30279210 | 2018 | R2PLx-22 | 22 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | H-157 | Lung Cancer | MTT assay | IC50 = 843.40 µM | 24-h | Lung | None | ||
| 30279210 | 2018 | R2PLx-22 | 22 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 872.70 µM | 24-h | Skin | None | ||
| 30279210 | 2018 | Ranatuerin-2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Rana palustris | MCF-7 | Breast Cancer | MTT assay | IC50 = 20.19 µM | 24-h | Breast | None | ||
| 30279210 | 2018 | Ranatuerin-2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Rana palustris | U-251-MG | Brain Tumor | MTT assay | IC50 = 16.14 µM | 24-h | Brain | None | ||
| 30279210 | 2018 | Ranatuerin-2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Rana palustris | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.79 µM | 24-h | Prostate | None | ||
| 30279210 | 2018 | Ranatuerin-2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Rana palustris | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 15.44 µM | 24-h | Skin | None | ||
| 30279210 | 2018 | Ranatuerin-2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Rana palustris | H-157 | Lung Cancer | MTT assay | IC50 = 5.90 µM | 24-h | Lung | None | ||
| 30279210 | 2018 | S-24-R2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | MCF-7 | Breast Cancer | MTT assay | IC50 = 316.90 µM | 24-h | Breast | None | ||
| 30279210 | 2018 | S-24-R2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | U-251-MG | Brain Tumor | MTT assay | IC50 = 278.30 µM | 24-h | Brain | None | ||
| 30279210 | 2018 | S-24-R2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 179.00 µM | 24-h | Skin | None | ||
| 30279210 | 2018 | S-24-R2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | H-157 | Lung Cancer | MTT assay | IC50 = 58.18 µM | 24-h | Lung | None | ||
| 30279210 | 2018 | S-24-R2PLx | 28 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analogue of Ranatuerin-2PLx | PC-3 | Prostate Cancer | MTT assay | IC50 = 792.60 µM | 24-h | Prostate | None | ||
| 30026168 | 2018 | [G10a]SHa-BCTP | 22 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 >100 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G10a]SHa-BCTP | 22 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 >100 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G10a]SHa-BCTP | 22 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 = 26.85 ± 1.85 µM | 24-h | Breast | None | ||
| 29904274 | 2018 | tMP-C | 23 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U-251-MG | Brain tumor | MTT assay | IC50 = 3.36 μM | 24-h | Brain | None | ||
| 29904274 | 2018 | tMP-C | 23 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.70 μM | 24-h | Breast | None | ||
| 29904274 | 2018 | tMP-C | 23 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 3.86 μM | 24-h | Skin | None | ||
| 29904274 | 2018 | tMP-C | 23 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.86 μM | 24-h | Prostate | None | ||
| 29904274 | 2018 | tMP-C | 23 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 2.79 μM | 24-h | Lung | None | ||
| 30087268 | 2018 | L10, 11-DPS3 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of Dermaseptin-PS3 | H-157 | Lung Cancer | MTT assay | IC50 = 0.12 μM | Not Available | Lung | None | ||
| 30087268 | 2018 | L10, 11-DPS3 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of Dermaseptin-PS3 | PC-3 | Prostate Cancer | MTT assay | IC50 = 1.85 μM | Not Available | Prostate | None | ||
| 30087268 | 2018 | K5, 17-DPS3 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of Dermaseptin-PS3 | H-157 | Lung Cancer | MTT assay | IC50 = 18.20 μM | Not Available | Lung | None | ||
| 30087268 | 2018 | K5, 17-DPS3 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of Dermaseptin-PS3 | PC-3 | Prostate Cancer | MTT assay | IC50 = 18.20 μM | Not Available | Prostate | None | ||
| 30087268 | 2018 | Dermaseptin-PS3 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Phyllomedusa sauvagii | H-157 | Lung Cancer | MTT assay | IC50 = 15.67 μM | Not Available | Lung | None | ||
| 30087268 | 2018 | Dermaseptin-PS3 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Phyllomedusa sauvagii | PC-3 | Prostate Cancer | MTT assay | IC50 = 18.20 μM | Not Available | Prostate | None | ||
| 30258724 | 2018 | DP-2 | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 3.21 μM | 24-h | Lung | None | ||
| 30258724 | 2018 | DP-2 | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 6.75 μM | 24-h | Prostate | None | ||
| 30258724 | 2018 | DRS-DU-1 | 28 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Callimedusa (Phyllomedusa) duellmani | PC-3 | Prostate Cancer | MTT assay | IC50 = 21.6 μM | 24-h | Prostate | None | ||
| 29191658 | 2018 | temporin-PEb | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 3.483 μM | Not Available | Skin | None | ||
| 30258724 | 2018 | DRS-DU-1 | 28 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Callimedusa (Phyllomedusa) duellmani | H-157 | Lung Cancer | MTT assay | IC50 = 8.43 μM | 24-h | Lung | None | ||
| 29191658 | 2018 | temporin-PEb | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | U251-MG | Brain Tumor | MTT assay | IC50 = 3.087 μM | Not Available | Brain | None | ||
| 29191658 | 2018 | temporin-PEb | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.051 μM | Not Available | Prostate | None | ||
| 29191658 | 2018 | temporin-PEb | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | NCI-H-157 | Lung Cancer | MTT assay | IC50 = 3.464 μM | Not Available | Lung | None | ||
| 28636781 | 2018 | BLP-7 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientali | A-375 | Skin Cancer | MTT assay | Cell Viability < 20% at 10 μM | 48-h | Skin | None | ||
| 28636781 | 2018 | BLP-7 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientali | A-549 | Lung Cancer | MTT assay | Cell Viability ~ 20% at 2.5 μM | 48-h | Lung | None | ||
| 28636781 | 2018 | BLP-7 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientali | PC-3 | Prostate Cancer | MTT assay | Cell Viability ~ 20% at 2.5 μM | 48-h | Prostate | None | ||
| 28636781 | 2018 | BLP-7 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientali | Huh-7 | Liver Cancer | MTT assay | IC50 = 1.81 μM | 48-h | Liver | None | ||
| 28636781 | 2018 | BLP-7 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientali | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.83 μM | 48-h | Liver | None | ||
| 28636781 | 2018 | BLP-7 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientali | SK-HEP-1 | Liver Cancer | MTT assay | IC50 = 0.61 μM | 48-h | Liver | None | ||
| 30622471 | 2018 | ChMAP-28 | 27 | Linear | L | None | Free | Free | Antimicrobial | leucocytes of the goat Capra hircus | B16-F10 | Skin Cancer | MTT assay | IC50 = 4.82 ± 1.01 μM | 48-h | Skin | None | ||
| 30622471 | 2018 | ChMAP-28 | 27 | Linear | L | None | Free | Free | Antimicrobial | leucocytes of the goat Capra hircus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 5.63 ± 1.05 μM | 48-h | Breast | None | ||
| 30622471 | 2018 | ChMAP-28 | 27 | Linear | L | None | Free | Free | Antimicrobial | leucocytes of the goat Capra hircus | HEK-293T | Renal Cancer | MTT assay | IC50 = 5.09 ± 0.40 μM | 48-h | Renal | None | ||
| 30622471 | 2018 | ChMAP-28 | 27 | Linear | L | None | Free | Free | Antimicrobial | leucocytes of the goat Capra hircus | A-431 | Skin Cancer | MTT assay | IC50 = 6.49 ± 0.09 μM | 48-h | Skin | None | ||
| 30622471 | 2018 | ChMAP-29 | 27 | Linear | L | None | Free | Free | Antimicrobial | leucocytes of the goat Capra hircus | HL-60 | Leukemia Cancer | LDH leakage assay | ~60% LDH Release at 2.5 μM | 1-h | Blood | None | ||
| 30622471 | 2018 | ChMAP-28 | 27 | Linear | L | None | Free | Free | Antimicrobial | leucocytes of the goat Capra hircus | HL-60 | Leukemia Cancer | MTT assay | IC50 = 3.39 ± 0.15 μM | 48-h | Blood | None | ||
| 29098406 | 2018 | Bombinin-BO1 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | Huh-7 | Liver Cancer | MTT assay | IC50 = 3.91 μM | 48-h | Liver | None | ||
| 29098406 | 2018 | Bombinin-BO1 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.75 μM | 48-h | Liver | None | ||
| 29098406 | 2018 | Bombinin-BO1 | 25 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | SK-HEP-1 | Liver Cancer | MTT assay | IC50 = 0.76 μM | 48-h | Liver | None | ||
| 29263923 | 2017 | E5 | 22 | Linear | L | None | Free | Free | Anticancer | Synthetic | 4T1 | Breast Cancer | CCK-8 assay | 49% cell viability at 100 μM | 24-h | Breast | None | ||
| None | 2017 | VLL-28 | 28 | Linear | L | None | Free | Acetylation | Antibacterial and Anticancer | Sulfolobus islandicus | HEK-293T | Renal Cancer | MTT assay | IC50 = 10 μM | 72-h | Renal | None | ||
| 29280948 | 2017 | F9D/A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 125.0 ± 1.8 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | F9D/A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 95.6 ± 1.8 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | F9D/A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 57.9 ± 2.8 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | F9D/A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 125.0 ± 3.4 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 125.0 ± 5.9 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 41.4 ± 1.4 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 46.2 ± 3.0 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | A12D/V16D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 60.1 ± 1.2 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | F9D/A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 125.0 ± 3.7 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | F9D/A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 42.4 ± 3.0 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | F9D/A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 38.8 ± 2.9 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | F9D/A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 59.8 ± 0.5 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 45.1 ± 1.0 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 15.5 ± 1.7 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 29.9 ± 4.8 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | A12D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 28.8 ± 0.8 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | S11D/K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 45.5 ± 5.6 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | S11D/K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 54.2 ± 1.2 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | S11D/K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 56.8 ± 3.3 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | S11D/K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 41.1 ± 0.5 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 24.1 ± 5.5 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 22.5 ± 0.5 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 47.1 ± 5.3 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | K14D/T15D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 31.6 ± 2.1 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | S11D/K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 22.4 ± 2.3 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | S11D/K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 25.5 ± 0.5 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | S11D/K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 41.3 ± 2.6 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | S11D/K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 30.6 ± 0.5 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 20.0 ± 0.8 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HPAC | Pancreatic Cancer | MTT assay | IC50 = 7.2 ± 5.2 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 17.9 ± 2.3 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analogue of V13K | HeLa | Cervical Cancer | MTT assay | IC50 = 15.6 ± 4.1 μM | 24-h | Cervix | None | ||
| 29280948 | 2017 | V13K | 26 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | BxPC-3 | Pancreatic Cancer | MTT assay | IC50 = 12.5 ± 1.2 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | V13K | 26 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | HPAC | Pancreatic Cancer | MTT assay | IC50 = 7.6 ± 4.0 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | V13K | 26 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MIA PaCa-2 | Pancreatic Cancer | MTT assay | IC50 = 24.8 ± 0.6 μM | 24-h | Pancreas | None | ||
| 29280948 | 2017 | V13K | 26 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 16 ± 0.5 μM | 24-h | Cervix | None | ||
| None | 2017 | BR-C | 25 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 75.44 μg/ml | 24-h | Lung | None | ||
| None | 2017 | BR-C | 25 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 45.72 μg/ml | 24-h | Breast | None | ||
| None | 2017 | BR-D | 25 | Linear | Mix | None | Free | Free | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 67.52 μg/ml | 24-h | Breast | None | ||
| None | 2017 | BR-D | 25 | Linear | Mix | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 94.74 μg/ml | 24-h | Lung | None | ||
| 29064402 | 2017 | Dermaseptin-PH | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pithecopus (Phyllomedusa) hypochondrialis | PC-3 | Prostate Cancer | MTT assay | IC50 = 11.8 μM | Not Available | Prostate | None | ||
| 29064402 | 2017 | Dermaseptin-PH | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pithecopus (Phyllomedusa) hypochondrialis | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 9.94 μM | Not Available | Breast | None | ||
| 29064402 | 2017 | Dermaseptin-PH | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pithecopus (Phyllomedusa) hypochondrialis | U251-MG | Brain Tumor | MTT assay | IC50 = 2.36 μM | Not Available | Brain | None | ||
| 29064402 | 2017 | Dermaseptin-PH | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pithecopus (Phyllomedusa) hypochondrialis | H-157 | Lung Cancer | MTT assay | IC50 = 2.01 μM | Not Available | Lung | None | ||
| 29064402 | 2017 | Dermaseptin-PH | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pithecopus (Phyllomedusa) hypochondrialis | MCF-7 | Breast Cancer | MTT assay | IC50 = 0.69 μM | Not Available | Breast | None | ||
| 27248170 | 2016 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | MDA-MB-231 | Breast Cancer | LDH leakage assay | LDH activity = 1.5mU/mL at 10 μg/mL | 3-h | Breast | None | ||
| 27248170 | 2016 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | MCF-7 | Breast Cancer | MTS assay | IC50 = 5.03 μM | 6-h | Breast | None | ||
| 27248170 | 2016 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | MDA-MB-453 | Breast Cancer | MTS assay | IC50 = 5.03 μM | 6-h | Breast | None | ||
| 27248170 | 2016 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 5.03 μM | 6-h | Breast | None | ||
| None | 2015 | LPSBD-0 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Hep3B | Liver Cancer | Cell Proliferation assay | ~40% cell survival at 60 µg/ml | 24-h | Liver | None | ||
| None | 2015 | LPSBD-0 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | Cell Proliferation assay | ~20% cell survival at 60 µg/ml | 24-h | Lung | None | ||
| 25447543 | 2015 | Human neutrophil peptide-1 (HNP-1) | 30 | Cyclic(C2-C30, C4-C19,C9-C29) | L | None | Free | Free | Antimicrobial | Homo sapiens | PC-3 | Prostate Cancer | Cytotoxicity assay (LIVE/DEAD® Viability/Cytotoxicity Assay Kit (L-3224)) | IC50 = 2.2 ± 0.3 μM | 4h | Prostate | None | ||
| 26322745 | 2015 | Cyclotide mela-6 | 29 | Cyclic | L | None | Cyclized | Cyclized | Antibacterial and Anticancer | Melicytus latifolius | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 11.42 ±1.00 µM | Not Available | Cervix | None | ||
| 26322745 | 2015 | Cyclotide mela-6 | 29 | Cyclic | L | None | Cyclized | Cyclized | Antibacterial and Anticancer | Melicytus latifolius | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.58 ±0.48 µM | Not Available | Skin | None | ||
| 26399495 | 2015 | Mra30 | 30 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial and Anticancer | Viola tricolor, Melicytus ramiflorus, Viola philippica | BGC-823 | Gastric Cancer | Resazurin dye assay | IC50 = 1.75 ±0.05 µM | Not Available | Stomach | None | ||
| 26399495 | 2015 | Mra30 | 30 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial and Anticancer | Viola tricolor, Melicytus ramiflorus, Viola philippica | HeLa | Cervical Cancer | Resazurin dye assay | IC50 = 15.5 ±0.06 µM | Not Available | Cervix | None | ||
| 26399495 | 2015 | Mra30 | 30 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial and Anticancer | Viola tricolor, Melicytus ramiflorus, Viola philippica | MM96L | Skin Cancer | Resazurin dye assay | IC50 = 4.91 ±0.04 µM | Not Available | Skin | None | ||
| 26322745 | 2015 | Mela3 | 29 | Cyclic | L | None | Cyclized | Cyclized | Antibacterial and Anticancer | Melicytus latifolius | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 18.73 ±1.82 µM | Not Available | Cervix | None | ||
| 26322745 | 2015 | Mela3 | 29 | Cyclic | L | None | Cyclized | Cyclized | Antibacterial and Anticancer | Melicytus latifolius | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 2.04 ±0.26 µM | Not Available | Skin | None | ||
| 26751970 | 2015 | Vigno 5 | 29 | Cyclic(C5-C19,C9-C21,C14-C21) | L | None | Free | Free | Anticancer | Viola ignobilis | HeLa | Cervical Cancer | MTT assay | 24% cell viability at 7.5 μM | 24-h | Cervix | None | ||
| 26064310 | 2015 | DC3 | 30 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Hedyotis diffusa | DU-145 | Liver Cancer | CCK-8 assay | IC50 = 0.55 μM | 72-h | Liver | None | ||
| 26064310 | 2015 | DC3 | 30 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Hedyotis diffusa | PC-3 | Prostate Cancer | CCK-8 assay | IC50 = 0.76 μM | 72-h | Prostate | None | ||
| 26064310 | 2015 | DC3 | 30 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Hedyotis diffusa | LNCaP | Prostate Cancer | CCK-8 assay | IC50 = 0.21 μM | 72-h | Prostate | None | ||
| 26405806 | 2015 | HPRP-A1-TAT | 24 | Linear | L | None | Amidation | Acetylation | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 1.8 ± 0.02 μM | 24-h | Cervix | None | ||
| 26405806 | 2015 | HPRP-A1-TAT | 24 | Linear | L | None | Amidation | Acetylation | Anticancer | Synthetic | B-16 | Skin Cancer | MTT assay | IC50 = 3.9 ± 0.02 μM | 24-h | Skin | None | ||
| 26405806 | 2015 | HPRP-A1-TAT | 24 | Linear | L | None | Amidation | Acetylation | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 5.8 ± 0.36 μM | 24-h | Liver | None | ||
| 26405806 | 2015 | HPRP-A1-TAT | 24 | Linear | L | None | Amidation | Acetylation | Anticancer | Synthetic | SGC-7901 | Gastric cancer | MTT assay | IC50 = 4.8 ± 0.08 μM | 24-h | Stomach | None | ||
| 26239537 | 2015 | DIM-LF11-318 | 22 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 9.4 ± 0.5 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | DIM-LF11-318 | 22 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 9.3 ± 0.8 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | DIM-LF11-318 | 22 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | PI uptake assay | LC50 = 3.8 ± 0.5 μM | 8-h | Skin | None | ||
| 26239537 | 2015 | R-DIM-LF11-337 | 22 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 5.0 ± 0.4 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | R-DIM-LF11-337 | 22 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 12.3 ± 1.3 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | R-DIM-LF11-337 | 22 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | PI uptake assay | LC50 = 3.5 ± 0.4 μM | 8-h | Skin | None | ||
| 25312253 | 2014 | E5 | 22 | Linear | L | None | Free | Free | Anticancer | Synthetic | U-937 | Leukemia Cancer | FITC-Annexin V/PI double staining and flow cytometry assay | >20% apoptosis rate at 80 μM | 24-h | Blood | None | ||
| 25312253 | 2014 | E5 | 22 | Linear | L | None | Free | Free | Anticancer | Synthetic | HL-60 | Leukemia Cancer | FITC-Annexin V/PI double staining and flow cytometry assay | >20% apoptosis rate at 80 μM | 24-h | Blood | None | ||
| 25312253 | 2014 | E5 | 22 | Linear | L | None | Free | Free | Anticancer | Synthetic | NB-4 | Leukemia Cancer | FITC-Annexin V/PI double staining and flow cytometry assay | 60% apoptosis rate at 80 μM | 24-h | Blood | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC107 | Colorectal Cancer | Cell Viability assay | Cell viability >70% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC107 | Colorectal Cancer | Cell Viability assay | Cell viability >65% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC107 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC32 | Colorectal Cancer | Cell Viability assay | Cell viability >85% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC32 | Colorectal Cancer | Cell Viability assay | Cell viability >80% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC32 | Colorectal Cancer | Cell Viability assay | Cell viability >55% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC113 | Colorectal Cancer | Cell Viability assay | Cell viability >70% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC113 | Colorectal Cancer | Cell Viability assay | Cell viability >65% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC113 | Colorectal Cancer | Cell Viability assay | Cell viability >80% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC60 | Colorectal Cancer | Cell Viability assay | Cell viability >70% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC60 | Colorectal Cancer | Cell Viability assay | Cell viability >60% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC60 | Colorectal Cancer | Cell Viability assay | Cell viability >70% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC40 | Colorectal Cancer | Cell Viability assay | Cell viability >85% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC40 | Colorectal Cancer | Cell Viability assay | Cell viability >80% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC40 | Colorectal Cancer | Cell Viability assay | Cell viability >45% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC24 | Colorectal Cancer | Cell Viability assay | Cell viability >70% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC24 | Colorectal Cancer | Cell Viability assay | Cell viability >55% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC24 | Colorectal Cancer | Cell Viability assay | Cell viability >55% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC18 | Colorectal Cancer | Cell Viability assay | Cell viability >75% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC18 | Colorectal Cancer | Cell Viability assay | Cell viability >55% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC18 | Colorectal Cancer | Cell Viability assay | Cell viability >55% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HCT-116 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HCT-116 | Colorectal Cancer | Cell Viability assay | Cell viability >40% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HCT-116 | Colorectal Cancer | Cell Viability assay | Cell viability >40% at 12.5μM approx | 24-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC32 | Colorectal Cancer | Cell Viability assay | Cell viability =50% at 12.5μM approx. | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC32 | Colorectal Cancer | Cell Viability assay | Cell viability =50% at 12.5μM approx. | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC32 | Colorectal Cancer | Cell Viability assay | Cell viability >60% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC60 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC60 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC60 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC40 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC40 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC40 | Colorectal Cancer | Cell Viability assay | Cell viability >60% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC24 | Colorectal Cancer | Cell Viability assay | Cell viability >60% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC24 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HROC24 | Colorectal Cancer | Cell Viability assay | Cell viability >60% at 25μM approx | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-Δ | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HCT-116 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 12.5μM approx. | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HCT-116 | Colorectal Cancer | Cell Viability assay | Cell viability =50% at 12.5μM approx. | 1-h | Colon | None | ||
| 24962950 | 2014 | C7A | 27 | Linear | L | None | Amidation | Free | Antitumor | NK-2 peptide based derivatives | HCT-116 | Colorectal Cancer | Cell Viability assay | Cell viability >50% at 25μM approx | 1-h | Colon | None | ||
| 24661024 | 2014 | Melittin | 26 | Linear | L | None | Free | Free | Antimicrobial | Main component of honey bee venom | SCC25 | Skin Cancer | Cell Viability assay | 102.9 ± 4.1% cell growth inhibition at 1 µM | 24-h | Skin | None | ||
| 24587350 | 2014 | Pexiganan | 22 | Linear | L | None | Amidation | Free | Antimicrobial | Analog of magainin 2 | OVRCAR-3 | Ovarian Cancer | MTT/MTS assay | LC50= 13 at 100 µM | 72-h | Ovary | None | ||
| 24587350 | 2014 | Pexiganan | 22 | Linear | L | None | Amidation | Free | Antimicrobial | Analog of magainin 2 | LNCaP | Prostate cancer | MTT/MTS assay | LC50= 6 at 100 µM | 72-h | Prostate | None | ||
| 24587350 | 2014 | Pexiganan | 22 | Linear | L | None | Amidation | Free | Antimicrobial | Analog of magainin 2 | MCF-7 | Breast Cancer | MTT/MTS assay | LC50= 8 at 100 µM | 72-h | Breast | None | ||
| 15279899 | 2004 | HCAP18(109-135) | 27 | Linear | L | None | Free | Free | Antimicrobial | hCAP18 synthetic peptide | SAS-H1 | Oral Cancer | Not Available | Not Available | Not Available | Oral mucosa | None | ||
| 22885172 | 2012 | ltc2aG11A | 26 | Linear | L | None | Free | Free | Antimicrobial | Central Asian spider, Lachesana tarabaevi | Prostate tumor cellline | Prostate Cancer | LDH leakage assay | graph fig 8 A | Not Available | Prostate | None | ||
| 22885172 | 2012 | Latarcin 2a | 26 | Linear | L | None | Free | Free | Antimicrobial | Central Asian spider, Lachesana tarabaevi | Breast tumor cellline | Breast Cancer | LDH leakage assay | graph fig 8 A | Not Available | Breast | None | ||
| 12417587 | 2003 | BF2d | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 100 µM 90-100% viablity | 6-h | Cervix | None | ||
| 12417587 | 2003 | BF2d | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 10 µM 90-95% viablity | 6-h | Cervix | None | ||
| 12417587 | 2003 | BF2d | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 1 µM 90-100% viablity | 6-h | Cervix | None | ||
| 12417587 | 2003 | MG2d | 23 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 1 µM 90-100% viablity | 6-h | Cervix | None | ||
| 21403917 | 2011 | Buforin 2 | 21 | Linear | L | None | Free | Free | Antimicrobial | Bufo Bufo Gargarizans | U-937 | Lymphoma Cancer | MTT/MTS assay | IC50 =90-95 µg/ml | Not Available | Blood | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MCF-7-TX400 | Breast Cancer | MTT/MTS assay | ~5% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MCF-7-TX400 | Breast Cancer | MTT/MTS assay | 60-70% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MCF-7 | Breast Cancer | MTT/MTS assay | 70% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MCF-7 | Breast Cancer | MTT/MTS assay | 0% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MCF-7-TX400 | Breast Cancer | MTT/MTS assay | 60-70% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 5-10% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 20% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MCF-7 | Breast Cancer | MTT/MTS assay | 70% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 5% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 10-15% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 15-20% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | ~5% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | ~5% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 10-15% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 10-15% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 10-15% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 80-90% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 85-90% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-13 | 23 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | ~5% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 80-90% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 30-40% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 60-70% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 50% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 80% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 20% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 70-80% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 80-85% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 40-50% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 20% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 40-50% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 5% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 20-30% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 85-90% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-07 | 25 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | ~0% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 40-50% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 80% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 60-70% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 80-85% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | 4T1 | Breast Cancer | MTT/MTS assay | 15-20% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 40-50% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 70% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 80-85% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-468 | Breast Cancer | MTT/MTS assay | 30% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 50% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 60% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | SKBR-3 | Breast Cancer | MTT/MTS assay | 30% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 30-35% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 5-10% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | T-47D | Breast Cancer | MTT/MTS assay | 10% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 60% cytotoxic at 50 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 5% cytotoxic at 5 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 5% cytotoxic at 10 µM | 24-h | Breast | None | ||
| 22023734 | 2011 | NRC-03 | 26 | Linear | L | None | Amidation | Biotinylated | Antimicrobial | Pleurocidin-family | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 30-35% cytotoxic at 25 µM | 24-h | Breast | None | ||
| 22057278 | 2011 | Z10 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z9 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 =13 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z7 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 =21 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z8 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 =23 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z6 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 =31 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z5 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 =67 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z4 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 =173 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z3 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z2 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z1 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Colon | None | ||
| 22057278 | 2011 | Z10 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z9 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =16 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z8 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =14 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z7 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =15 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z6 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =16 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z5 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =28 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z4 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =68 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z3 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =128 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z2 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =173 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z1 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | MT-1 | Breast Cancer | MTT/MTS assay | EC50 =186 µM | Not Available | Breast | None | ||
| 22057278 | 2011 | Z10 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z9 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 =9 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z8 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 =19 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z7 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 =15 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z6 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 =17 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z5 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 =42 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z4 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 =155 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z3 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z2 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Skin | None | ||
| 22057278 | 2011 | Z1 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | Meth A | Skin Cancer | MTT/MTS assay | EC50 >211 µM | Not Available | Skin | None | ||
| 17067680, 18957441 | 2007 | hepcidin TH1-5 | 22 | Not Available | L | None | Free | Free | Anticancer | Tilapia, Oreochromis mossambicus | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 8245827, 18957441 | 1993 | Plantaricin A | 26 | Not Available | L | None | Free | Free | Antibacterial | Lactobacillus plantarumC11, WCFS1, V90 | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 11713517, 18957441 | 2001 | Piscidin 1 | 22 | Not Available | L | None | Free | Free | Antibacterial | Hybrid striped bass (Morone saxatilis x M. chrysops) | Not Available | Breast Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 12581207, 18957441 | 2003 | Chrysophsin-1 | 25 | Not Available | L | None | Free | Free | Antibacterial | Red sea bream,Chrysophrys majororPagrus major | Not Available | Breast Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 12804591, 19923233 | 2003 | Prepromelittin-related peptide | 23 | Not Available | L | None | Free | Free | Antibacterial | Rana tagoi [Tago frog] | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 4056036, 18957441 | 1985 | HNP-3 | 30 | Not Available | L | None | Free | Free | Anticancer | Homo sapiens | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 4056036, 18957441 | 1985 | HNP-2 | 29 | Not Available | L | None | Free | Free | Anticancer | Homo sapiens | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 4056036, 18957441 | 1985 | HNP-1 | 30 | Not Available | L | None | Free | Free | Anticancer | Homo sapiens | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 9548831, 18957441 | 1998 | Varv peptide A | 29 | Not Available | L | None | Free | Free | Anticancer | Viola arvensis,Viola odorata, Viola tricolor, Viola baoshanensis, Viola yedoensis, and Viola biflora | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 21434649, 18957441 | 2011 | Vaby D | 30 | Not Available | L | None | Free | Free | Anticancer | African, the Ethiopian highlands, Viola abyssinica | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 21434649, 18957441 | 2011 | Vaby A | 29 | Not Available | L | None | Free | Free | Anticancer | African, the Ethiopian highlands, Viola abyssinica | Not Available | Fibrosarcoma | Not Available | Not Available | Not Available | Fibrous connective tissue | None | ||
| 10601876, 18957441 | 2000 | Caerin 1.10 | 25 | Not Available | L | None | Free | Free | Anticancer | Magnificent treefrog Litoria splendida, Australia | Not Available | Lung Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 9266696, 18957441 | 1997 | Caerin 1.1 | 25 | Not Available | L | None | Free | Free | Anticancer | Australian green tree frogLitoria splendida; Litoria rothii | Not Available | Lung Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 18191970, 18957441 | 2008 | Vibi E | 30 | Not Available | L | None | Free | Free | Anticancer | Alpine violetViola biflora | Not Available | Leukemia Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 10075760, 18957441 | 1999 | Varv peptide F | 29 | Not Available | L | None | Free | Free | Anticancer | Viola arvensis | Not Available | Leukemia Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 22771617, 18957441 | 2012 | Maculatin 1.3 | 21 | Not Available | L | None | Free | Free | Anticancer | Blue-thighed frog,Litoria chloris, Australia | Not Available | Skin Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 22771617, 18957441 | 2012 | Maculatin 1.4 | 21 | Not Available | L | None | Free | Free | Anticancer | Blue-thighed frog,Litoria chloris, Australia | Not Available | Skin Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 9230483, 18957441 | 1997 | Caerin 1.6 | 24 | Not Available | L | None | Free | Free | Anticancer | Blue-thighed frog,Litoria chloris, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9230483, 18957441 | 1997 | Caerin 1.8 | 24 | Not Available | L | None | Free | Free | Anticancer | Blue-thighed frog,Litoria chloris, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9230483, 18957441 | 1997 | Caerin 1.7 | 24 | Not Available | L | None | Free | Free | Anticancer | Orange-thighed frog,Litoria xanthomera, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9516047, 18957441 | 1998 | Caerin 1.9 | 24 | Not Available | L | None | Free | Free | Anticancer | Litoria chloris, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 11835991, 18957441 | 2002 | Maximin 1 | 27 | Not Available | L | None | Free | Free | Anticancer | Bombina maxima | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 11835991, 18957441 | 2002 | Maximin 4 | 27 | Not Available | L | None | Free | Free | Anticancer | Bombina maxima | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 11835991, 18957441 | 2002 | Maximin 3 | 27 | Not Available | L | None | Free | Free | Antibacterial | Bombina maxima | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 11835991, 18957441 | 2002 | Maximin H1 | 27 | Not Available | L | None | Free | Free | Antibacterial | Bombina maxima | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20575512, 18957441 | 2010 | Psyle A | 28 | Not Available | L | None | Free | Free | Antibacterial | Psychotria leptothyrsa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20575512, 18957441 | 2010 | Psyle C | 25 | Not Available | L | None | Free | Free | Antibacterial | Psychotria leptothyrsa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 8910461, 18957441 | 1996 | BMAP-28 | 28 | Not Available | L | None | Free | Free | Antibacterial | CowBos taurus | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 8910461, 18957441 | 1996 | BMAP-27 | 27 | Not Available | L | None | Free | Free | Antibacterial | CowBos taurus | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9620615, 18957441 | 1998 | Maculatin 3.1 | 26 | Not Available | L | None | Free | Free | Anticancer | Litoria genimaculate, Litoria eucnemis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9620615, 18957441 | 1998 | Maculatin 1.1 | 22 | Not Available | L | None | Free | Free | Antibacterial | Litoria genimaculate, Litoria eucnemis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9620615, 18957441 | 1998 | Maculatin 1.2 | 23 | Not Available | L | None | Free | Free | Antibacterial | Litoria genimaculate, Litoria eucnemis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21596752, 18957441 | 2011 | Cliotide T2 | 30 | Not Available | L | None | Free | Free | Antibacterial | Clitoria ternatea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21596752, 18957441 | 2011 | Cliotide T4 | 30 | Not Available | L | None | Free | Free | Antibacterial | Clitoria ternatea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21596752, 18957441 | 2011 | Cliotide T1 | 30 | Not Available | L | None | Free | Free | Antibacterial | Clitoria ternatea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21596752, 18957441 | 2011 | Cliotide T3 | 29 | Not Available | L | None | Free | Free | Antibacterial | Clitoria ternatea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10600388, 18957441 | 1999 | Cycloviolacin O2 | 30 | Not Available | L | None | Free | Free | Antibacterial | Viola odorata | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21723349, 18957441 | 2011 | Viba17 | 29 | Not Available | L | None | Free | Free | Antibacterial | Viola philippica | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21723349, 18957441 | 2011 | Viba 15 | 29 | Not Available | L | None | Free | Free | Antibacterial | Viola philippica | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 21723349, 18957441 | 2011 | Mram 8 | 30 | Not Available | L | None | Free | Free | Antibacterial | Viola philippica | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22467870, 18957441 | 2012 | Chassatide C10 | 29 | Not Available | L | None | Free | Free | Antibacterial | Chassalia chartacea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22467870, 18957441 | 2012 | Chassatide C4 | 29 | Not Available | L | None | Free | Free | Antibacterial | Chassalia chartacea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22467870, 18957441 | 2012 | Chassatide C4 | 29 | Not Available | L | None | Free | Free | Antibacterial | Chassalia chartacea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22467870, 18957441 | 2012 | ChaC11 | 29 | Not Available | L | None | Free | Free | Antibacterial | Chassalia chartacea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22467870, 18957441 | 2012 | Chassatide C8 | 29 | Not Available | L | None | Free | Free | Antibacterial | Chassalia chartacea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22467870, 18957441 | 2012 | ChaC7 | 29 | Not Available | L | None | Free | Free | Antibacterial | Chassalia chartacea | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 16713189, 18957441 | 2006 | Brevinin-1BYa | 24 | Not Available | L | None | Free | Free | Antibacterial | Rana boylii, North America | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Ranatuerin-2Ya | 28 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates yavapaiensis | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 19254736, 18957441 | 2009 | Brevinin-1BLa | 24 | Not Available | L | None | Free | Free | Antibacterial | North America, leopard frog, Lithobates blairi | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | SU.86.86 | Pancreatic Cancer | WST-1 assay | IC50= 8.0 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | Pane- 1 | Breast Cancer | WST-1 assay | IC50= 14.1 µM | 48-h | Breast | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | CFPAC-I | Pancreatic Cancer | WST-1 assay | IC50= 9.2 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| None | 2009 | Sema3A(aa371-377) -nLytic | 24 | Linear | Mix | None | Free | Free | Anticancer | Synthetic Peptide | BxPC-3 | Pancreatic Cancer | WST-1 assay | IC50= 14.7 µM | 48-h | Pancreatic | WO_2010_064207_A2 | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 2% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 1% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 0% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 3% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 2% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 1% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 5% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 1% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 2% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 3% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 2% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3Alt | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 1% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 55% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 35% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | IMR5 | Tumor | MTT/MTS assay | 23% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 79% apoptosis at 50 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 46% apoptosis at 20 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NGP | Tumor | MTT/MTS assay | 43% apoptosis at 10 µM | 8-h | Not Available | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 68% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 66% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | NB69 | Brain Tumor | MTT/MTS assay | 25% apoptosis at 10 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 65% apoptosis at 50 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 45% apoptosis at 20 µM | 8-h | Brain | None | ||
| 16568093 | 2006 | r8-BidBH3 | 29 | Linear | Mix | None | Free | Free | Antitumor | Synthetic Peptide | SK-N-AS | Brain Tumor | MTT/MTS assay | 8% apoptosis at 10 µM | 8-h | Brain | None | ||
| 15867360 | 2005 | hP8 | 28 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | No inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP7 | 25 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | No inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP6 | 24 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | No inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP5 | 25 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | 29% inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP4 | 25 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | No inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP3 | 25 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | No inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP2 | 25 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | 19% inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15867360 | 2005 | hP1 | 25 | Linear | L | None | Free | Free | Antiangiogenesis | Human endostatin peptides | BxPC-3 | Pancreatic Cancer | Matrigel Assay | 39% inhibition at 7 mg/kg/d | 672-h | Pancreatic | None | ||
| 15467750 | 2004 | TAT-Ras-GAP317-326 | 22 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 79% apoptosis at 50 µM | 16 to 24-h | Cervix | None | ||
| 15467750 | 2004 | TAT-Ras-GAP317-326 | 22 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 72% apoptosis at 30 µM | 16 to 24-h | Cervix | None | ||
| 15467750 | 2004 | TAT-Ras-GAP317-326 | 22 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 47% apoptosis at 20 µM | 16 to 24-h | Cervix | None | ||
| 15467750 | 2004 | TAT-Ras-GAP317-326 | 22 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 15% apoptosis at 10 µM | 16 to 24-h | Cervix | None | ||
| 20515045 | 2010 | AP(O) | 25 | Cyclic(C2-C10,C | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 52% inhibition at 10µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP(O) | 25 | Cyclic(C2-C10,C | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 42% inhibition at 5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP(O) | 25 | Cyclic(C2-C10,C | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 40% inhibition at 2.5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP | 25 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 75% inhibition at 10µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP | 25 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 40% inhibition at 5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | AP | 25 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 50% inhibition at 2.5µg/ml | NA | Not Available | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Anticancer | Natural component of bee venom | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 1.4±0.1 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | C7A- Δ | 23 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 13.1±0.9 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | C7A-D21k | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 12.3±1.0 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 3.7± 4.3 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Anticancer | Residue of 39-65 of porcine NK-lysine | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 40 µM (approx) | 24-h | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Anticancer | Natural component of bee venom | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 1.8±0.1 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | C7A- Δ | 23 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 9.3±1.5 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | C7A-D21k | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 8.3±0.5 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 12.1±1.6 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Anticancer | Residue of 39-65 of porcine NK-lysine | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 50 µM (approx) | 4-h | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Anticancer | Natural component of bee venom | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 2.1±0.1 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | C7A- Δ | 23 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 13.8±2.0 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | C7A-D21k | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 12.3±2.0 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 13.0±1.0 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Anticancer | Residue of 39-65 of porcine NK-lysine | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 50 µM (approx) | 2-h | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Anticancer | Natural component of bee venom | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 3.2±0.1 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | C7A- Δ | 23 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 7.5±0.4 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | C7A-D21k | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 8.4±0.2 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Anticancer | NK-2 variants | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 10.6±0.4 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Anticancer | Residue of 39-65 of porcine NK-lysine | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 70 µM (approx) | 30-Min | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Anticancer | Natural component of bee venom | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 1.4±0.1 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Anticancer | Residue of 39-65 of porcine NK-lysine | E42/02 | Skin Cancer | MTT/MTS assay | IC50= 4.3±0.3 µM | 4-h | Skin | None | ||
| 22837667 | 2012 | Peptide L6D/L12D/L17D/L20D/L21D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 12.88±0.15 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L6D/L12D/L17D/L20D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 9.69±0.38 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L12D/L20D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 3.14±0.06 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L6D/L12D/L20D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 7.80±0.26 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L20D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 2.33±0.06 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L6D/L12D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 3.01±0.08 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L12D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 2.63±0.07 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide L6D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 2.23±0.10 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K1D/K3D/K7D /K10D/K14D/K22D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 18.07±0.48 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K7D /K10D/K14D/K22D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 4.79±0.23 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K3D/K7D /K10D/K14D/K22D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 20.41±0.64 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K7D /K14D/K22D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 4.45±0.19 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K14D/K22D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 1.40±0.09 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K7D /K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 2.06±0.01 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K22D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 1.39±0.02 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K14D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 1.52±0.05 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide K7D | 26 | Linear | Mix | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 1.29±0.03 µMol/L | 1-h | Cervix | None | ||
| 22837667 | 2012 | Peptide P | 26 | Linear | L | None | Amidation | Acetylation | Anticancer | A12L/A20L | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 1.71±0.07 µMol/L | 1-h | Cervix | None | ||
| 24176852 | 2013 | KilerFLIP | 26 | linear | L | None | Free | Free | NA | NA | Jurkat | Blood Cancer | Not Available | NA | NA | Blood | None | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HTB-9 | Bladder Cancer | MTT/MTS assay | ~30% cytotoxicity at 1 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HTB-9 | Bladder Cancer | MTT/MTS assay | >40% cytotoxicity at 10 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HTB-9 | Bladder Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HTB-9 | Bladder Cancer | MTT/MTS assay | 20% cytotoxicity at 10 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HTB-9 | Bladder Cancer | MTT/MTS assay | 40% cytotoxicity at 1 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HTB-9 | Bladder Cancer | MTT/MTS assay | ~50% cytotoxicity at 10 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <5% cytotoxicity at 10 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 48-h | Bladder | WO2012042540A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <3% cytotoxicity at 10 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <15% cytotoxicity at 1 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | ~15% cytotoxicity at 10 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | CaSki | Cervical Cancer | MTT/MTS assay | ~20% cytotoxicity at 1 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | CaSki | Cervical Cancer | MTT/MTS assay | ~45% cytotoxicity at 10 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | CaSki | Cervical Cancer | MTT/MTS assay | ~55% cytotoxicity at 10 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | CaSki | Cervical Cancer | MTT/MTS assay | ~40% cytotoxicity at 10 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | CaSki | Cervical Cancer | MTT/MTS assay | ~20% cytotoxicity at 1 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | >20% cytotoxicity at 10 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | CaSki | Cervical Cancer | MTT/MTS assay | ~20% cytotoxicity at 1 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | >20% cytotoxicity at 10 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | ~15% cytotoxicity at 1 µM | 72-h | Cervix | WO2012042540A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | ~15% cytotoxicity at 10 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | <3% cytotoxicity at 1 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | ~5% cytotoxicity at 1 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | SiHa | Cervical Cancer | MTT/MTS assay | ~45% cytotoxicity at 10 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | SiHa | Cervical Cancer | MTT/MTS assay | ~20% cytotoxicity at 1 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | SiHa | Cervical Cancer | MTT/MTS assay | ~50% cytotoxicity at 10 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | SiHa | Cervical Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | SiHa | Cervical Cancer | MTT/MTS assay | >40% cytotoxicity at 10 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | SiHa | Cervical Cancer | MTT/MTS assay | >20% cytotoxicity at 1 µM | 24-h | Cervix | WO2012042540A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | ~40% cytotoxicity at 10 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | ~20% cytotoxicity at 1 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | >20% cytotoxicity at 10 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | <3% cytotoxicity at 1 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | >10% cytotoxicity at 10 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | 5% cytotoxicity at 1 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HCT-116 | Colon Cancer | MTT/MTS assay | ~40% cytotoxicity at 10 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HCT-116 | Colon Cancer | MTT/MTS assay | >30% cytotoxicity at 1 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HCT-116 | Colon Cancer | MTT/MTS assay | >20% cytotoxicity at 10 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HCT-116 | Colon Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 48-h | Colon | WO2012042540A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HCT-116 | Colon Cancer | MTT/MTS assay | 50% cytotoxicity at 10 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | HCT-116 | Colon Cancer | MTT/MTS assay | >40% cytotoxicity at 1 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 10 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 10 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | ~5% cytotoxicity at 1 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | 15% cytotoxicity at 10 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <15% cytotoxicity at 1 µM | 24-h | Colon | WO2012042540A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | UM-UC-3 | Bladder Cancer | MTT/MTS assay | >40% cytotoxicity at 1 µM | 72-h | Bladder | WO2012042540A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~50% cytotoxicity at 10 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~50% cytotoxicity at 10 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | UM-UC-3 | Bladder Cancer | MTT/MTS assay | <30% cytotoxicity at 1 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | UM-UC-3 | Bladder Cancer | MTT/MTS assay | <30% cytotoxicity at 10 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~30% cytotoxicity at 1 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | <45% cytotoxicity at 10 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~45% cytotoxicity at 1 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | >25% cytotoxicity at 10 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~25% cytotoxicity at 1 µM | 48-h | Bladder | WO2012042540A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~25% cytotoxicity at 10 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~25% cytotoxicity at 1 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | COLO-205 | Colon Cancer | MTT/MTS assay | ~20% cytotoxicity at 10 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | COLO-205 | Colon Cancer | MTT/MTS assay | ~35% cytotoxicity at 10 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | COLO-205 | Colon Cancer | MTT/MTS assay | >20% cytotoxicity at 1 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 10 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | MB30 | 30 | Linear | L | None | Free | Free | Anticancer | Derived from the MPT63 secreted protein | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 10 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | >10% cytotoxicity at 1 µM | 72-h | Colon | WO2012042540A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | >10% cytotoxicity at 10 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | 10% cytotoxicity at 1 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | ~10% cytotoxicity at 10 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG23 | 22 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 24-h | Colon | WO_2012042540_A2 | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =2.1 ± 0.1 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =1.8 ± 0.1 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =1.4 ± 0.1 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | C7A-Δ | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =7.5 ± 0.4 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | C7A-Δ | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =13.8 ± 2.0 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | C7A-Δ | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =9.3 ± 1.5 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | C7A-Δ | 24 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =13.1 ± 0.9 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | Melittin | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =3.2 ± 0.1 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =12.3 ± 1.0 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =8.3 ± 0.5 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =12.3 ± 2.0 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | C7A-D21K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =8.4 ± 0.2 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =37 ± 4.3 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =12.1 ± 1.6 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =13.0 ± 1.0 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | C7A | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 =10.6 ± 0.4 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 = ~40 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 = ~50 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 = ~50 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 = ~70 µM | 30-Min | Skin | None | ||
| 19527490 | 2009 | KW5 | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic peptide | HT-29 | Colon Cancer | MTT/MTS assay | IC50 =55±14 µM | NA | Colon | None | ||
| 19527490 | 2009 | KW5 | 21 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | FEMX | Skin Cancer | MTT/MTS assay | IC50 =30±3 µM | NA | Skin | None | ||
| 18815734 | 2008 | di-PST13-RK-K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =10 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | di-PST13-RK-K | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 =15 µg/ml | NA | Lung | None | ||
| 18815734 | 2008 | di-PST13-RK-C | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =17 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | di-PST13-RK-C | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 =17 µg/ml | NA | Lung | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <40% cell viability at 50 µM | NA | Stomach | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | 100% cell viability at 5 µM | NA | Stomach | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | <60% cell viability at 50 µM | NA | Blood | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | 100% cell viability at 5 µM | NA | Blood | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | 60% cell viability at 50 µM | NA | Colon | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | >100% cell viability at 5 µM | NA | Colon | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <20% cell viability at 50 µM | NA | Stomach | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <100% cell viability at 5 µM | NA | Stomach | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | <40% cell viability at 50 µM | NA | Blood | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | 100% cell viability at 5 µM | NA | Blood | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | 40% cell viability at 50 µM | NA | Colon | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | 100% cell viability at 5 µM | NA | Colon | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <100% cell viability at 5 µM | 24-h | Stomach | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <40% cell viability at 50 µM | 24-h | Stomach | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | 60% cell viability at 50 µM | 24-h | Colon | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | 100% cell viability at 5 µM | 24-h | Blood | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | <60% cell viability at 50 µM | 24-h | Blood | None | ||
| 22783018 | 2012 | N29D | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | >100% cell viability at 5 µM | 24-h | Colon | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <20% cell viability at 50 µM | 24-h | Stomach | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SNU-1 | Gastric Cancer | Cell Viability assay | <100% cell viability at 5 µM | 24-h | Stomach | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | <40% cell viability at 50 µM | 24-h | Blood | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | U-937 | Lymphoma Cancer | Cell Viability assay | 100% cell viability at 5 µM | 24-h | Blood | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | 40% cell viability at 50 µM | 24-h | Colon | None | ||
| 22783018 | 2012 | N29N | 30 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic peptide | SW-480 | Colon Cancer | Cell Viability assay | 100% cell viability at 5 µM | 24-h | Colon | None | ||
| 16004618 | 2005 | Pep27anal5 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=>70 µM | 19.17-Min | Breast | None | ||
| 16004618 | 2005 | Pep27anal4 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | MCF-7 | Breast Cancer | MTT/MTS assay | IC50= 29 µM | 19.15-Min | Breast | None | ||
| 16004618 | 2005 | Pep27anal3 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | MCF-7 | Breast Cancer | MTT/MTS assay | IC50= 38 µM | 20.08-Min | Breast | None | ||
| 16004618 | 2005 | Pep27anal2 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | MCF-7 | Breast Cancer | MTT/MTS assay | IC50= <10 µM | 22.5-Min | Breast | None | ||
| 16004618 | 2005 | Pep27anal1 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | MCF-7 | Breast Cancer | MTT/MTS assay | IC50= 55 µM | 18.67-Min | Breast | None | ||
| 16004618 | 2005 | Pep27 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | MCF-7 | Breast Cancer | MTT/MTS assay | IC50= >70 µM | 14.54-Min | Breast | None | ||
| 16004618 | 2005 | Pep27anal5 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | SNU-601 | Gastric Cancer | MTT/MTS assay | IC50=>70 µM | 19.17-Min | Stomach | None | ||
| 16004618 | 2005 | Pep27anal4 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | SNU-601 | Gastric Cancer | MTT/MTS assay | IC50= 37 µM | 19.15-Min | Stomach | None | ||
| 16004618 | 2005 | Pep27anal3 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | SNU-601 | Gastric Cancer | MTT/MTS assay | IC50= 50 µM | 20.08-Min | Stomach | None | ||
| 16004618 | 2005 | Pep27anal2 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | SNU-601 | Gastric Cancer | MTT/MTS assay | IC50= 25 µM | 22.5-Min | Stomach | None | ||
| 16004618 | 2005 | Pep27anal1 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | SNU-601 | Gastric Cancer | MTT/MTS assay | IC50= 37 µM | 18.67-Min | Stomach | None | ||
| 16004618 | 2005 | Pep27anal5 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | Jurkat | Blood Cancer | MTT/MTS assay | IC50=>70 µM | 19.17-Min | Blood | None | ||
| 16004618 | 2005 | Pep27 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | SNU-601 | Gastric Cancer | MTT/MTS assay | IC50= >70 µM | 14.54-Min | Stomach | None | ||
| 16004618 | 2005 | Pep27anal4 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | Jurkat | Blood Cancer | MTT/MTS assay | IC50= 46 µM | 19.15-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal3 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | Jurkat | Blood Cancer | MTT/MTS assay | IC50= 50 µM | 20.08-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal2 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | Jurkat | Blood Cancer | MTT/MTS assay | IC50= 23 µM | 22.5-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal1 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | Jurkat | Blood Cancer | MTT/MTS assay | IC50= 47 µM | 18.67-Min | Blood | None | ||
| 16004618 | 2005 | Pep27 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | Jurkat | Blood Cancer | MTT/MTS assay | IC50=>70 µM | 14.54-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal5 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50= >70 µM | 19.17-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal4 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50=51 µM | 19.15-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal3 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50= 52 µM | 20.08-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal2 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50= 20 µM | 22.5-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal1 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50= 53 µM | 18.67-Min | Blood | None | ||
| 16004618 | 2005 | Pep27 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50= >70 µM | 14.54-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal5 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | AML-2 | Leukemia Cancer | MTT/MTS assay | IC50= >70 µM | 19.17-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal4 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | AML-2 | Leukemia Cancer | MTT/MTS assay | IC50= 50 µM | 19.15-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal3 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | AML-2 | Leukemia Cancer | MTT/MTS assay | IC50= 67 µM | 20.08-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal2 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | AML-2 | Leukemia Cancer | MTT/MTS assay | IC50= 29 µM | 22.5-Min | Blood | None | ||
| 16004618 | 2005 | Pep27anal1 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | AML-2 | Leukemia Cancer | MTT/MTS assay | IC50= 50 µM | 18.67-Min | Blood | None | ||
| 16004618 | 2005 | Pep27 | 27 | Linear | L | None | Free | Free | Anticancer | S. pneumoniae | AML-2 | Leukemia Cancer | MTT/MTS assay | Not Available | 14.54-Min | Blood | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 10 % Cytotoxicity at 3.125 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 1 % Cytotoxicity at 6.25 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 20 % Cytotoxicity at 12.5 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 90 % Cytotoxicity at 25 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 90 % Cytotoxicity at 50 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 15 % Cytotoxicity at 3.125 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 35 % Cytotoxicity at 6.25 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 30 % Cytotoxicity at 12.5 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 85 % Cytotoxicity at 25 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 90 % Cytotoxicity at 50 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 35 % Cytotoxicity at 3.125 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 30 % Cytotoxicity at 6.25 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 48 % Cytotoxicity at 12.5 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 84% Cytotoxicity at 25 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 84 % Cytotoxicity at 50 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 25 % Cytotoxicity at 3.125 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 30 % Cytotoxicity at 6.25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 45 % Cytotoxicity at 12.5 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 85 % Cytotoxicity at 25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 80 % Cytotoxicity at 50 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 18 % Cytotoxicity at 3.125 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 18 % Cytotoxicity at 6.25 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 18 % Cytotoxicity at 12.5 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 82 % Cytotoxicity at 25 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 90 % Cytotoxicity at 50 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 10 % Cytotoxicity at 3.125 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 4 % Cytotoxicity at 6.25 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 18 % Cytotoxicity at 12.5 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 70 % Cytotoxicity at 25 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 82 % Cytotoxicity at 50 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 5 % Cytotoxicity at 3.125 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 10 % Cytotoxicity at 6.25 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 10 % Cytotoxicity at 12.5 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 70 % Cytotoxicity at 25 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 78 % Cytotoxicity at 50 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 1 % Cytotoxicity at 3.125 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 5 % Cytotoxicity at 6.25 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 4 % Cytotoxicity at 12.5 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 60 % Cytotoxicity at 25 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Pardaxin-6 | 27 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 70 % Cytotoxicity at 50 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 28 % Cytotoxicity at 3.125 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 30 % Cytotoxicity at 6.25 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 85 % Cytotoxicity at 25 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 38 % Cytotoxicity at 12.5 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 84 % Cytotoxicity at 50 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 28 % Cytotoxicity at 3.125 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 30 % Cytotoxicity at 6.25 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 46 % Cytotoxicity at 12.5 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 96 % Cytotoxicity at 25 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 95 % Cytotoxicity at 50 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 25 % Cytotoxicity at 3.125 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 25 % Cytotoxicity at 6.25 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 45 % Cytotoxicity at 12.5 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 95 % Cytotoxicity at 25 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 90 % Cytotoxicity at 50 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 41 % Cytotoxicity at 6.25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 41 % Cytotoxicity at 6.25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 41 % Cytotoxicity at 6.25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 39 % Cytotoxicity at 3.125 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 41 % Cytotoxicity at 6.25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 42 % Cytotoxicity at 12.5 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 85 % Cytotoxicity at 25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 82 % Cytotoxicity at 50 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 77 % Cytotoxicity at 25 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 83% Cytotoxicity at 50 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 65% Cytotoxicity at 25 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 75 % Cytotoxicity at 50 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 65% Cytotoxicity at 25 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 75% Cytotoxicity at 50 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 38% Cytotoxicity at 25 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-1 | 21 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 45% Cytotoxicity at 50 mg/L | 3-h | Cervix | None | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =100 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =125 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =215 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16)-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =19 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =97 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =270 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =240 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =28 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | Not Available | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | Not Available | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =20 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =145 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =82 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =50 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Hecate AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =95 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =66 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =45 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =45 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =375 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =310 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =13 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =28 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16)-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =28 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | CA(1-7)Shiva10(1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =97 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =63 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =82 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =66 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =65 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =125 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =12 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =38 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =41 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =83 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Hecate AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =61 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =77 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =315 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =25 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16) | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =22 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | CA(1-7)Shiva10(1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =63 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =125 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =84 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =37 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =72 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Hecate AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AC V | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | D2A21V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =83 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =130 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =155 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =18 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =94 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16)-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =12 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =76 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CA(1-7)Shiva10(1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =360 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =290 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =94 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =85 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =36 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =94 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =27 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =128 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =72 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AC V | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | D2A21V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =83 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =130 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =155 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =18 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =94 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16)-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =12 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =76 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CA(1-7)Shiva10(1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =360 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =290 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =94 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =94 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =36 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =85 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =27 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =128 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Hecate AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =72 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Hecate AC V | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Hecate AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | D2A21V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =73 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =76 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =80 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =740 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =23 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =120 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16)-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =13 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =70 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =82 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =11 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =34 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =57 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =62 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =8 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =12 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =38 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =5 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Hecate AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =6 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =84 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Hecate AC V | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Hecate AM V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =340 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | D2A21V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =210 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Anubis-2 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =38 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | D2A21 | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Magainin2wisc | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =22 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FAGVL | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =240 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z4 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z3 | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | MELITTIIN | 26 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | PYL-ME | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =635 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | SHIVA 11[(1-16)ME(2-9]-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =95 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | CA(1-7) Shiva10(1-16)-COOH | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =63 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 (1-16) Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =29 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | CA (1-7) Shiva10 (1-16) | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 PEPTIDE 71 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =93 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | SHIVA DERIV P69 + KWKL | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | MSI-78 AM | 22 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =31 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | HECATE 2DAc | 23 | Linear | Mix | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =14 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | KAL V | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =72 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK05 AM | 21 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =74 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK04 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =10 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK03 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =26 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK01 AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =62 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | SHIVA 10 AC | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Hecate AM | 23 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =23 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Hecate Ac | 23 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| 9614066 | 1998 | DRS B4 | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Dermaseptins B | MCF-7 | Breast Cancer | Thymidine Incorporation assay | Cytotoxicity =15 µM | 6-h | Breast | None | ||
| 9614066 | 1998 | DRS B3 | 28 | Linear | L | None | Free | Free | Antimicrobial | Dermaseptins B | MCF-7 | Breast Cancer | Thymidine Incorporation assay | Cytotoxicity =12 µM | 6-h | Breast | None | ||
| 15796184 | 2005 | Apo E | 30 | Linear | L | None | Free | Free | Antibacterial | Apoprotein E | COLO-201 | Colon Cancer | MTT/MTS assay | 65 % Cytotoxity at 40 µg/ml | 4-h | Colon | None | ||
| 15796184 | 2005 | Apo E | 30 | Linear | L | None | Free | Free | Antibacterial | Apoprotein E | MKN-7 | Gastric Cancer | MTT/MTS assay | 35 % Cytotoxity at 40 µg/ml | 4-h | Stomach | None | ||
| 15796184 | 2005 | Apo E | 30 | Linear | L | None | Free | Free | Antibacterial | Apoprotein E | MKN-1 | Gastric Cancer | MTT/MTS assay | 60 % Cytotoxity at 40 µg/ml | 4-h | Stomach | None | ||
| 15796184 | 2005 | Apo E | 30 | Linear | L | None | Free | Free | Antibacterial | Apoprotein E | Paca-2 | Pancreatic Cancer | MTT/MTS assay | 55 % Cytotoxity at 40 µg/ml | 4-h | Pancreatic | None | ||
| 15796184 | 2005 | Apo E | 30 | Linear | L | None | Free | Free | Antibacterial | Apoprotein E | PANC-1 | Pancreatic Cancer | MTT/MTS assay | 55 % Cytotoxity at 40 µg/ml | 4-h | Pancreatic | None | ||
| 11835991 | 2001 | maximin5 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | T-24 | Bladder Cancer | MTT/MTS assay | IC50=>50 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin4 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | T-24 | Bladder Cancer | MTT/MTS assay | IC50=>50 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin3 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | T-24 | Bladder Cancer | MTT/MTS assay | IC50 =18 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin1 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | T-24 | Bladder Cancer | MTT/MTS assay | IC50 =35.4 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin5 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | BIU-87 | Bladder Cancer | MTT/MTS assay | IC50 =>50 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin4 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | BIU-87 | Bladder Cancer | MTT/MTS assay | IC50 =>50 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin3 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | BIU-87 | Bladder Cancer | MTT/MTS assay | IC50=28 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin1 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | BIU-87 | Bladder Cancer | MTT/MTS assay | IC50=20.5 µg/ml | 48-h | Bladder | None | ||
| 11835991 | 2001 | maximin5 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | MOLT-4 | Leukemia Cancer | MTT/MTS assay | IC50 >50 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin4 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | MOLT-4 | Leukemia Cancer | MTT/MTS assay | IC50 =53.4 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin3 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | MOLT-4 | Leukemia Cancer | MTT/MTS assay | IC50 =25.2 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin1 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | MOLT-4 | Leukemia Cancer | MTT/MTS assay | IC50=24.3 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin5 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | C8166 | Leukemia Cancer | MTT/MTS assay | IC50=34.4 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin4 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | C8166 | Leukemia Cancer | MTT/MTS assay | IC50=24.2 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin3 | 27 | Linear | L | None | Free | Free | Antimicrobial | Bombina maxima | C8166 | Leukemia Cancer | MTT/MTS assay | IC50=11.4 µg/ml | 48-h | Blood | None | ||
| 11835991 | 2001 | maximin1 | 27 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina maxima | C8166 | Leukemia Cancer | MTT/MTS assay | IC50=15.3 µg/ml | 48-h | Blood | None | ||
| 18656352 | 2008 | Tat-a5 | 22 | Linear | L | None | Free | Free | Anticancer | HIV-Tat (49-57) | HCT-116 | Colon Cancer | MTT/MTS assay | ~80% Cytotoxicity at 100 µM | 24-h | Colon | None | ||
| 16637646 | 2006 | LL-37(13-37) | 25 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | LC50=38 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(13-37) | 25 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | LC50=40 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(13-37) | 25 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | LC50=39 µM | 24-h | Not Available | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=2.2 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=2 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=4.3 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=3.8 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=10.4 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=58.6 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=64.7 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | HeLa | Cervical Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Cervix | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=4.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=4.4 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=7.8 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=5.2 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=11.5 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=62.5 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=63.5 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | B-16 | Skin Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=2.7 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=4.1 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=2.9 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=4.4 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=4.7 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=14 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=15.6 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=16.4 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=37.7 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | H-1299 | Lung Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=5.5 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=6.4 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=9.8 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=7.5 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=25.2 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=3.5 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | RD | Rhabdomyosarcoma Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Muscle | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=4.3 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=5 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=6.4 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=11.1 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | SW-1116 | Colorectal Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Colon | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=5.7 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=6.2 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=5.1 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=5 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=15.8 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=62.3 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=70.8 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Breast | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=7.2 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=8.7 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=6.5 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=4.3 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=17.8 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=59.8 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=58.7 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-375 | Skin Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Skin | None | ||
| 21252288 | 2011 | A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=8.7 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A12L/A20L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=9.7 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A12L/A20L/A23L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=9.2 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L6A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=53 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | P | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=33 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | A12L | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=11.1 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L17A/L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L21A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=71 µMo/L | 36-h | Lung | None | ||
| 21252288 | 2011 | L6A/L17A | 26 | Linear | L | None | Free | Free | Anticancer | PeptideV13K | A-549 | Lung Cancer | MTT/MTS assay | IC50=>83.6 µMo/L | 36-h | Lung | None | ||
| 21955251 | 2011 | Cationic Amphiphilic | 21 | Cyclic | L | None | Free | Free | Antimicrobial | AMP | HL-60 | Pancreatic Cancer | WST-1 assay | IC50 = 10 µM | Not Available | Pancreatic | None | ||
| 21955251 | 2011 | Magainin 2 | 23 | Linear | L | None | Free | Free | Antimicrobial | Xenopus laevis | HeLa | Pancreatic Cancer | WST-1 assay | IC50 = >60 µM | Not Available | Pancreatic | None | ||
| 21955251 | 2011 | Cationic Amphiphilic | 21 | Cyclic | L | None | Free | Free | Antimicrobial | AMP | HeLa | Pancreatic Cancer | WST-1 assay | IC50 = 4 µM | Not Available | Pancreatic | None | ||
| 16269280 | 2005 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antibacterial | NK-lysin | SW-480 | Leukemia Cancer | PI-uptake assay | LD50=1-4 µM | Not Available | Blood | None | ||
| 16269280 | 2005 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antibacterial | NK-lysin | U-937 | Lymphoma Cancer | PI-uptake assay | LD50=30 µM | Not Available | Blood | None | ||
| 16269280 | 2005 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antibacterial | NK-lysin | SH-SY5Y | Brain Tumor | PI-uptake assay | LD50=1-4 µM | Not Available | Brain | None | ||
| 16269280 | 2005 | NK-2 | 27 | Linear | L | None | Amidation | Free | Antibacterial | NK-lysin | NB LA-N-1 | Colorectal Cancer | PI-uptake assay | LD50=1-4 µM | Not Available | Colon | None | ||
| 7768152, 21403917 | 1994 | PexigaNAn MSI-78 | 22 | Linear | L | None | Amidation | Free | Antimicrobial | Helical peptide with a predominance of one or more amino acids tryptophane-rich | U-937 | Lymphoma Cancer | MTT/MTS assay | 75% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 8573171, 21403917 | 1996 | Buforin2 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Bufo Bufo Gargarizans | U-937 | Lymphoma Cancer | MTT/MTS assay | 5% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | PC-3 | Prostate Cancer | Trypan blue assay | IC50 >200 µg/ml | 72-h | Prostate | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | PC-3 | Prostate Cancer | Trypan blue assay | Not Available | 72-h | Prostate | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | PC-3 | Prostate Cancer | Trypan blue assay | Not Available | 72-h | Prostate | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | PC-3 | Prostate Cancer | Trypan blue assay | IC50=53 µg/ml | 72-h | Prostate | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | PC-3 | Prostate Cancer | Trypan blue assay | IC50=47 µg/ml | 72-h | Prostate | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | PC-3 | Prostate Cancer | Trypan blue assay | IC50=41 µg/ml | 72-h | Prostate | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MCF-7 | Breast Cancer | Trypan blue assay | IC50 >200 µg/ml | 72-h | Breast | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MCF-7 | Breast Cancer | Trypan blue assay | Not Available | 72-h | Breast | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MCF-7 | Breast Cancer | Trypan blue assay | Not Available | 72-h | Breast | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | MCF-7 | Breast Cancer | Trypan blue assay | IC50=49 µg/ml | 72-h | Breast | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | MCF-7 | Breast Cancer | Trypan blue assay | IC50=42 µg/ml | 72-h | Breast | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MCF-7 | Breast Cancer | Trypan blue assay | IC50=37 µg/ml | 72-h | Breast | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | CHP-100 | Ewing sarcoma | Trypan blue assay | IC50 >200 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | CHP-100 | Ewing sarcoma | Trypan blue assay | Not Available | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | CHP-100 | Ewing sarcoma | Trypan blue assay | Not Available | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | CHP-100 | Ewing sarcoma | Trypan blue assay | IC50=45 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | CHP-100 | Ewing sarcoma | Trypan blue assay | IC50=39 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | CHP-100 | Ewing sarcoma | Trypan blue assay | IC50=32 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | K-562 | Leukemia Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | K-562 | Leukemia Cancer | Trypan blue assay | IC50=112 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | K-562 | Leukemia Cancer | Trypan blue assay | IC50=98 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | K-562 | Leukemia Cancer | Trypan blue assay | IC50=40 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | K-562 | Leukemia Cancer | Trypan blue assay | IC50=37 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | K-562 | Leukemia Cancer | Trypan blue assay | IC50=32 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Raji | Lymphoma Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Raji | Lymphoma Cancer | Trypan blue assay | IC50=72 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Raji | Lymphoma Cancer | Trypan blue assay | IC50=64 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | Raji | Lymphoma Cancer | Trypan blue assay | IC50=20 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | Raji | Lymphoma Cancer | Trypan blue assay | IC50=25 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Raji | Lymphoma Cancer | Trypan blue assay | IC50=23 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MLA | Leukemia Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MLA | Leukemia Cancer | Trypan blue assay | IC50=102 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MLA | Leukemia Cancer | Trypan blue assay | IC50=80 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | MLA | Leukemia Cancer | Trypan blue assay | IC50=34 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | MLA | Leukemia Cancer | Trypan blue assay | IC50=33 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | MLA | Leukemia Cancer | Trypan blue assay | IC50=30 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Daudi | Colon Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Daudi | Brain Tumor | Trypan blue assay | IC50=115 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Daudi | Leukemia Cancer | Trypan blue assay | IC50=143 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | Daudi | Lung Cancer | Trypan blue assay | IC50=30 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | Daudi | Renal Cancer | Trypan blue assay | IC50=38 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | Daudi | Ovarian Cancer | Trypan blue assay | IC50=28 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | SSKT-1 | Hematopoietic Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | SSKT-1 | Hematopoietic Cancer | Trypan blue assay | IC50=109 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | SSKT-1 | Hematopoietic Cancer | Trypan blue assay | IC50=107 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | SSKT-1 | Hematopoietic Cancer | Trypan blue assay | IC50=29 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | SSKT-1 | Hematopoietic Cancer | Trypan blue assay | IC50=23 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | SSKT-1 | Hematopoietic Cancer | Trypan blue assay | IC50=27 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | 8402 | Leukemia Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | 8402 | Leukemia Cancer | Trypan blue assay | IC50=83 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | 8402 | Leukemia Cancer | Trypan blue assay | IC50=60 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | 8402 | Leukemia Cancer | Trypan blue assay | IC50=18 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | 8402 | Leukemia Cancer | Trypan blue assay | IC50=16 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | 8402 | Leukemia Cancer | Trypan blue assay | IC50=12 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | U-937 | Lymphoma Cancer | Trypan blue assay | IC50 >150 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z24 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | U-937 | Lymphoma Cancer | Trypan blue assay | IC50=123 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Z44 | 24 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | U-937 | Lymphoma Cancer | Trypan blue assay | IC50=97 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | U-937 | Lymphoma Cancer | Trypan blue assay | IC50=16 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | Xenopus laevis | U-937 | Lymphoma Cancer | Trypan blue assay | IC50=19 µg/ml | 72-h | Blood | None | ||
| 1708887, 2285300 | 1990 | Magainin B | 23 | Linear | L | None | Amidation | Free | Antibacterial | Xenopus laevis | U-937 | Lymphoma Cancer | Trypan blue assay | IC50=17 µg/ml | 72-h | Blood | None | ||
| 18425992 | 2008 | mPep1 | 22 | Linear | L | None | Free | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | HL-60 | Skin Cancer | MTT/MTS assay | IC50=8 µM | 24-h | Blood | None | ||
| 18425992 | 2008 | pep1 | 22 | Linear | L | None | Free | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | HL-60 | Prostate Cancer | MTT/MTS assay | IC50=77 µM | 24-h | Blood | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 486P(G4) | Bladder Cancer | Cell Viability assay | IC50=59.4 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 647V(G2) | Bladder Cancer | Cell Viability assay | IC50=31 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | RT4(G1) | Bladder Cancer | Cell Viability assay | IC50=135.3 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 486P(G4) | Bladder Cancer | WST-1 assay | IC50=57.8 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 647V(G2) | Bladder Cancer | WST-1 assay | IC50=52.4 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 486P(G4) | Bladder Cancer | LDH leakage assay | IC50=28.6 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | RT4(G1) | Bladder Cancer | WST-1 assay | IC50=484 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | 647V(G2) | Bladder Cancer | LDH leakage assay | IC50=54.1 µM | 48-h | Bladder | None | ||
| 16476519 | 2006 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antimicrobial | African clawed frog Xenopus laevis skin | RT4(G1) | Bladder Cancer | LDH leakage assay | IC50=32.3 µM | 48-h | Bladder | None | ||
| 8319212 | 1993 | MSI-238 | 22 | Linear | D | None | Amidation | Free | Antibacterial | African clawed frog Xenopus laevis skin | A-549 | Lung Cancer | MTT/MTS assay | IC50=6 µM | 48-h | Lung | None | ||
| 8319212 | 1993 | MSI-136 | 22 | Linear | L | None | Amidation | Free | Antibacterial | African clawed frog Xenopus laevis skin | A-549 | Lung Cancer | MTT/MTS assay | IC50=10 µM | 48-h | Lung | None | ||
| 8319212 | 1993 | Magainin 2 | 23 | Linear | L | None | Amidation | Free | Antibacterial | African clawed frog Xenopus laevis skin | A-549 | Lung Cancer | MTT/MTS assay | IC50=110 µM | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | DU-145 | Prostate Cancer | MTT/MTS assay | IC50=15.3 µg/ml | 48-h | Prostate | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SW-620 | Colon Cancer | MTT/MTS assay | IC50=12.7 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | PC-3 | Prostate Cancer | MTT/MTS assay | IC50=12 µg/ml | 48-h | Prostate | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | KM12 | Colon Cancer | MTT/MTS assay | IC50=12 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HT-29 | Colon Cancer | MTT/MTS assay | IC50=17.6 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HCT-15 | Colon Cancer | MTT/MTS assay | IC50=13.2 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | COLO-205 | Colon Cancer | MTT/MTS assay | IC50=11.2 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HCT-116 | Colon Cancer | MTT/MTS assay | IC50=14.6 µg/ml | 48-h | Colon | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | Histone H2A | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50=12.6 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-8 | Ovarian Cancer | MTT/MTS assay | IC50=13 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-5 | Ovarian Cancer | MTT/MTS assay | IC50=13.8 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-4 | Ovarian Cancer | MTT/MTS assay | IC50=17.6 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | OVRCAR-3 | Ovarian Cancer | MTT/MTS assay | IC50=15.2 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | IGROV1 | Ovarian Cancer | MTT/MTS assay | IC50=9 µg/ml | 48-h | Ovary | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | UO-31 | Renal Cancer | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SN-12C | Renal Cancer | MTT/MTS assay | IC50=11.4 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | TK-10 | Renal Cancer | MTT/MTS assay | IC50=13.1 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | RFX393 | Renal Cancer | MTT/MTS assay | IC50=11 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | CAKI-1 | Renal Cancer | MTT/MTS assay | IC50=14.1 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | ACHN | Renal Cancer | MTT/MTS assay | IC50=12 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | A-498 | Renal Cancer | MTT/MTS assay | IC50=10 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | 786-0 | Renal Cancer | MTT/MTS assay | IC50=12.2 µg/ml | 48-h | Renal | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | UACC-62 | Skin Cancer | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | UACC-257 | Skin Cancer | MTT/MTS assay | IC50=12.5 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SK-MEL-5 | Skin Cancer | MTT/MTS assay | IC50=8.9 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50=11.1 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MALME-3M | Skin Cancer | MTT/MTS assay | IC50=10.9 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | M14 | Skin Cancer | MTT/MTS assay | IC50=15.1 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | LOXIMVI | Skin Cancer | MTT/MTS assay | IC50=9.5 µg/ml | 48-h | Skin | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SNB-75 | Brain Tumor | MTT/MTS assay | IC50=15.5 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | U-251 | Brain Tumor | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SNB-19 | Brain Tumor | MTT/MTS assay | IC50=13.8 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SF-539 | Brain Tumor | MTT/MTS assay | IC50=9.5 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SF-295 | Brain Tumor | MTT/MTS assay | IC50=12.9 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SF-268 | Brain Tumor | MTT/MTS assay | IC50=12.4 µg/ml | 48-h | Brain | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H522 | Lung Cancer | MTT/MTS assay | IC50=11.2 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H460 | Lung Cancer | MTT/MTS assay | IC50=12.1 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H322M | Lung Cancer | MTT/MTS assay | IC50=10.7 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H23 | Lung Cancer | MTT/MTS assay | IC50=10.8 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI-H226 | Lung Cancer | MTT/MTS assay | IC50=13.3 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HOP-92 | Lung Cancer | MTT/MTS assay | IC50=7.2 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HOP-62 | Lung Cancer | MTT/MTS assay | IC50=12.6 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | EKVX | Lung Cancer | MTT/MTS assay | IC50=12.1 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | A-549 | Lung Cancer | MTT/MTS assay | IC50=11.7 µg/ml | 48-h | Lung | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | T-47D | Breast Cancer | MTT/MTS assay | IC50=23.9 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | BT-549 | Breast Cancer | MTT/MTS assay | IC50=12.9 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MDA-N | Breast Cancer | MTT/MTS assay | IC50=10.6 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MDA-MB-435 | Breast Cancer | MTT/MTS assay | IC50=11.3 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HS578T | Breast Cancer | MTT/MTS assay | IC50=11.7 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=11.3 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | NCI/ADR-RES | Breast Cancer | MTT/MTS assay | IC50=11.5 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=15.1 µg/ml | 48-h | Breast | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | SR | Leukemia Cancer | MTT/MTS assay | IC50=20.2 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | RPMI-8226 | Leukemia Cancer | MTT/MTS assay | IC50=10.5 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | MOLT-4 | Leukemia Cancer | MTT/MTS assay | IC50=17 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=8.2 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50=11.3 µg/ml | 48-h | Blood | None | ||
| 18617323 | 2008 | Buforin IIb | 21 | Linear | L | None | Free | Free | Antibacterial | histone H2A | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50=14.7 µg/ml | 48-h | Blood | None | ||
| 1319823, 2285300 | 1992 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H889 | Lung Cancer | MTT/MTS assay | IC50=6.57 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H841 | Lung Cancer | MTT/MTS assay | IC50=11.7 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H735 | Lung Cancer | MTT/MTS assay | IC50=7.23 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H678 | Lung Cancer | MTT/MTS assay | IC50=4.44 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H526 | Lung Cancer | MTT/MTS assay | IC50=10.5 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin G | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H182 | Lung Cancer | MTT/MTS assay | IC50=12.5 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H889 | Lung Cancer | MTT/MTS assay | IC50=6.56 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H841 | Lung Cancer | MTT/MTS assay | IC50=9.7 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H735 | Lung Cancer | MTT/MTS assay | IC50=10.4 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H678 | Lung Cancer | MTT/MTS assay | IC50=6.23 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H526 | Lung Cancer | MTT/MTS assay | IC50=11.7 µM | 24-h | Lung | None | ||
| 1319823, 2285300 | 1992 | Magainin A | 23 | Linear | L | None | Amidation | Beta-alanine | Antibacterial | African clawed frog Xenopus laevis skin | NCI-H182 | Lung Cancer | MTT/MTS assay | IC50=7.28 µM | 24-h | Lung | None | ||
| 14499271 | 2003 | PTP4 | 24 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=18.1 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP1 | 21 | Cyclic(C15-C21) | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | GGN6 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=4.88 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP4 | 24 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=18.18 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | GGN6 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=4.91 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP1 | 21 | Cyclic(C15-C21) | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP4 | 24 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | PC-3 | Prostate Cancer | MTT/MTS assay | IC50=18.63 µg/ml | 96-h | Prostate | None | ||
| 14499271 | 2003 | PTP1 | 21 | Cyclic(C15-C21) | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | GGN6 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=5.75 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP4 | 24 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=26.15 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP1 | 21 | Cyclic(C15-C21) | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | GGN6 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=5.62 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP4 | 24 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=13.71 µg/ml | 96-h | Lung | None | ||
| 14499271 | 2003 | GGN6 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=6.49 µg/ml | 96-h | Lung | None | ||
| 14499271 | 2003 | PTP1 | 21 | Cyclic(C15-C21) | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50= >100 µg/ml | 96-h | Lung | None | ||
| None | 2020 | Seq ID No. 17 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | Calu-1 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 26 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | H-460 | Lung Cancer | Tetrazolium-based assay | Cell viability < 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 26 from patent ID US202000079827A1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | Calu-1 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 34 from patent ID US202000079827A1 | 24 | Linear | Mix | None | Free | Free | Antimicrobial and Anticancer | Synthetic | NCI-H460 | Lung Cancer | Tetrazolium-based assay | Cell viability < 25% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | Seq ID No. 34 from patent ID US202000079827A1 | 24 | Linear | Mix | None | Free | Free | Antimicrobial and Anticancer | Synthetic | Calu-1 | Lung Cancer | Tetrazolium-based assay | Cell viability > 50% at 20 μM | 2-h | Lung | US20200079827A1 | ||
| None | 2020 | IDP-LLCb01 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-LLCb01 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 2.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-LLCb01 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2023 | Sample Peptide 2 from EP3604345B1 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H2444 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 3.6% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 2 from EP3604345B1 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 4.9% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 2 from EP3604345B1 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 9.1% at 25 μM | 48-h | Lung | EP3604345B1 |