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IDPMIDYEARSequenceNameLengthLinear/CyclicChiralityChem-MODC-ter MODN-ter MODNatureOriginCell LineCancer TypeAssayActivityTesting TimeTissue AffectedPatents
7722
None2020
LKKWWKKVKGLLGGLLGKVKKVIK
Seq ID No. 17 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticNCI-H460Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7721
None2020
LKKWWKKVKGLLGGLLGKVKKVIK
Seq ID No. 17 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticHOP-062Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7720
None2020
LKKWWKKVKGLLGGLLGKVKSVIK
Seq ID No. 16 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticCalu-1Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7719
None2020
LKKWWKKVKGLLGGLLGKVKSVIK
Seq ID No. 16 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticNCI-H460Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7718
None2020
LKKWWKKVKGLLGGLLGKVKSVIK
Seq ID No. 16 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticHOP-062Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7717
None2020
LKKWWKKVKGLLGGLLGKVTSVIK
Seq ID No. 15 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticCalu-1Lung CancerTetrazolium-based assayCell viability < 50% at 20 μM2-hLungUS20200079827A1
7716
None2020
LKKWWKKVKGLLGGLLGKVTSVIK
Seq ID No. 15 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticNCI-H460Lung CancerTetrazolium-based assayCell viability < 25% at 20 μM2-hLungUS20200079827A1
7715
None2020
LKKWWKKVKGLLGGLLGKVTSVIK
Seq ID No. 15 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticHOP-062Lung CancerTetrazolium-based assayCell viability ~ 50% at 20 μM2-hLungUS20200079827A1
7714
None2022
RRWKRFFKRWKGGVIGVTFPF
ATRA1-R3W2 - HYD21LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticH-358Lung CancerCytotoxicity assayLD50 ~24.5 μM6-hLungUS011447533B2
7709
378538142024
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerMTT assay52.5 ± 5.0% cell viability at 150 µM24-hBreastNone
7708
378538142024
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerMTT assay14.0 ± 3.0% cell viability at 150 µM24-hBreastNone
7642
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
MC–FA27LinearLNoneFolic AcidFreeAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 12.63 µg/mL24-hBreastNone
7640
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
MC–FA27LinearLNoneFolic AcidFreeAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 66.43 µg/mL24-hCervixNone
7641
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
MC–FA27LinearLNoneFolic AcidFreeAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 35.22 µg/ mL24-hCervixNone
7638
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
CM–FA27LinearLNoneAmidationFolic AcidAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 35.75 µg/mL24-hCervixNone
7639
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
CM–FA27LinearLNoneAmidationFolic AcidAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 10.38 µg/mL24-hBreastNone
7637
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
CM–FA27LinearLNoneAmidationFolic AcidAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 67.34 µg/mL24-hCervixNone
7636
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
Mel-C27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 160.62 µg/mL24-hBreastNone
7635
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
Mel-C27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 58.63 µg/mL24-hCervixNone
7634
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
Mel-C27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 50.72 µg/mL24-hCervixNone
7633
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
C-Mel27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 110.59 µg/mL24-hBreastNone
7632
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
C-Mel27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 44.76 µg/mL24-hCervixNone
7631
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
C-Mel27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 64.15 µg/mL24-hCervixNone
7628
368730172023
CLKKLLKLLKKLLKLCLEELLHHLEELLHH
LK-LE330CyclicLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 10.2 µM at pH 624-hCervixNone
7627
368730172023
CLKKLLKLLKKLLKLCLEHLLEHLEHLLEH
LK-LE230CyclicLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 12.9 µM at pH 624-hCervixNone
7626
368730172023
CLKKLLKLLKKLLKLCLHELLEHLHELLEH
LK-LE130Cyclic(C1-C16)LNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 11.3 µM at pH 624-hCervixNone
7611
377346502023
KLKSKLMVVANKIGLLKSLARKFVKSH
NKL-MUT27LinearLNoneFreeFreeAntimicrobialTrematomus bernacchiiB16-F10Skin Cancerluciferase-based ATPlite assayATP level = 0.023 ± 0.007 at 40 μM12-hSkinNone
7610
377346502023
KLKSKLMVVCNKIGLLKSLCRKFVKSH
NKL-WT27LinearLNoneFreeFreeAntimicrobialTrematomus bernacchiiB16-F10Skin Cancerluciferase-based ATPlite assayATP level = 0.753 ± 0.254 at 40 μM12-hSkinNone
7608
368404532023
FLKSLWRGVKAIFNGARQGYKEHKN
AMP-WF325LinearLNoneFreeFreeAnticancerPoecilia Mexicana fishJurkatBlood CancerMTT assayIC50 = 50 µM24-hBloodNone
7595
366260982023
FKCRRWQWRMKKLGAPSITCVRRAF
bLF25LinearLNoneFreeFreeAntimicrobialBos TaurusJurkatBlood CancerMTT assaycell viability ~ 17.5% at 20 µM4-hBloodNone
7594
366260982023
FKCRRWQWRMKKLGAPSITCVRRAF
bLF25LinearLNoneFreeFreeAntimicrobialBos TaurusHepG-2Liver CancerMTT assaycell viability ~ 21% at 10 µM24-hLiverNone
7583
370985302023
GIGAVLKVLTTGLPALISWIKRKRQQ
Mellitin26LinearLNoneAmidationFreeAnticancerMain component of honey bee venomK-562Leukemia CancerSulforhodamine B assayIC50 = 1.84 ± 0.75 μg/ml96-hBloodNone
7580
368307252023
CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK
Pep-1-Phor2130LinearLNoneFreeFreeAnticancerHybrid peptide PEP1 and Phor 21PC-3Prostrate CancerAlamarBlue assayIC50 ≤ 0.6 μM24-hProstateNone
7579
368307252023
CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK
Pep-1-Phor2130LinearLNoneFreeFreeAnticancerHybrid peptide PEP1 and Phor 21DU-145Prostrate CancerAlamarBlue assayIC50 = 2.57 ± 2.02 µM24-hProstateNone
7578
368307252023
CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK
Pep-1-Phor2130LinearLNoneFreeFreeAnticancerHybrid peptide PEP1 and Phor 21LNCaPLiver CancerAlamarBlue assayIC50 = 55.13 ± 13.56 µM24-hLiverNone
7573
375809092023
QETFSDLWKLLVQRKRQKLMP
mPNC-NLS21LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerCytotoxicity assayIC50 = 45 μM24-hLungNone
7572
375809092023
QETFSDLWKLLVQRKRQKLMP
mPNC-NLS21LinearLNoneFreeFreeAnticancerSyntheticU-87Brain TumorMTT assayIC50 = 56.9 μM24-hBrainNone
7571
375809092023
QETFSDLWKLLVQRKRQKLMP
mPNC-NLS21LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 44.9 μM24-hLungNone
7568
374839712023
THPPTTTTTTTTTTTYTAAPATTT
ATMP124LinearLNoneFreeFreeAntimicrobialAnabas testudineusMDA-MB-231Breast CancerMTT assayIC50 = 8.25 ± 0.14 μg/ml48-hBreastNone
7567
374839712023
THPPTTTTTTTTTTTYTAAPATTT
ATMP524LinearLNoneFreeFreeAnticancer; AntimicrobialSynthetic Analog of ATMP1MDA-MB-231Breast CancerMTT assayIC50 = 64.04 ± 0.021 μg /ml24-hBreastNone
7566
None2023
AWLDKLKSIGKVVGKVAIGVAKNLLNPQ
Raniseptin-328LinearLNoneFreeFreeAntimicrobial and AntitumorBoana ranicepsB16-F10Skin CancerMTT assayIC50 = 6.56 uM3-hSkinNone
7565
None2023
ALLDKLKSLGKVVGKVALGVVQNYLNPRQ
Raniseptin-629LinearLNoneFreeFreeAntimicrobial and AntitumorBoana ranicepsB16-F10Skin CancerMTT assayIC50 = 8.69 uM3-hSkinNone
7562
373105332023
RIIDRLWLVRRPQKPKFVLVWVL
PMAP-NC23LinearLNoneFreeFreeAntimicrobialSynthetic Analgog of PMAP-24A-549Lung CancerMTT assayIC50 = 7.1 μM4-hLungNone
7561
373105332023
RIIDRLWLVRRPQKPKFVLVWVL
PMAP-NC23LinearLNoneFreeFreeAntimicrobialSynthetic Analgog of PMAP-23MDA-MB-361Breast CancerMTT assayIC50 = 6.4 μM4-hBreastNone
7558
377643342023
ALWKSILKNAGKAVLNEINQIV
14VL2323LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 16.4 µM24-hLungNone
7557
377643342023
ALWKSILKNAGKAVLNEINQIV
14VL2323LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 5.7 µM24-hLungNone
7556
377643342023
ALWKKILKNAGKAVLNEINQIVQ
14V5K23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 6.1 µM24-hLungNone
7555
377643342023
ALWKKILKNAGKAVLNEINQIVQ
14V5K23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 8.1 µM24-hLungNone
7554
377643342023
ALWKSILKNVGKVLNEINQIVQ
L2V22LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 0.6 µM24-hLungNone
7553
377643342023
ALWKSILKNVGKVLNEINQIVQ
L2V22LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 2.2 µM24-hLungNone
7552
377643342023
ALWKSILKNAGKAGLNEINQIVQ
14G23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 31.7 µM24-hLungNone
7551
377643342023
ALWKSILKNAGKAGLNEINQIVQ
14G23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 48.7 µM24-hLungNone
7550
377643342023
ALWKSILKNAGKAVLNEINQIVQ
14V23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 4.1 µM24-hLungNone
7549
377643342023
ALWKSILKNAGKAVLNEINQIVQ
14V23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 7.0 µM24-hLungNone
7548
377643342023
ALWKSILKNAGKALNEINQIVQ
L1422LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 20.1 µM24-hLungNone
7547
377643342023
ALWKSILKNAGKALNEINQIVQ
L1422LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 64.4 µM24-hLungNone
7546
377643342023
ALWKSILKNAGKAALNEINQIV
Dermaseptin-SS123LinearLNoneAmidationFreeAntimicrobial and AnticancerBrown-belly leaf frog, Phyllomedusa TarsiusH-460Lung CancerMTT assayIC50 = 1.3 µM24-hLungNone
7545
377643342023
ALWKSILKNAGKAALNEINQIV
Dermaseptin-SS123LinearLNoneAmidationFreeAntimicrobial and AnticancerBrown-belly leaf frog, Phyllomedusa TarsiusH-838Lung CancerMTT assayIC50 = 7.7 µM24-hLungNone
7515
372287022023
FLPLLAGLAANFLPKIICKIARKC
B1AW-K24LinearLNoneAmidationFreeAntimicrobial and Antitumoranalogue of B1AWU251-MGBrain TumorMTT assayIC50 = 3.860 µM24-hBrainNone
7514
372287022023
FLPLLAGLAANFLPKIICKIARKC
B1AW-K24LinearLNoneAmidationFreeAntimicrobial and Antitumoranalogue of B1AWH-838Lung CancerMTT assayIC50 = 5.15 µM24-hLungNone
7513
372287022023
FLPLLAGLAANFLPKIICKIARKC
B1AW-K24LinearLNoneAmidationFreeAntimicrobial and Antitumoranalogue of B1AWPC-3Prostate CancerMTT assayIC50 = 4.283 µM24-hProstateNone
7512
372287022023
FLPLLAGLAANFLPQIICKIARKC
B1AW24LinearLNoneAmidationFreeAntimicrobial and AntitumorWuyi torrent frog, Amolops wuyiensisU251-MGBrain TumorMTT assayIC50 = 33.56 µM24-hBrainNone
7511
372287022023
FLPLLAGLAANFLPQIICKIARKC
B1AW24LinearLNoneAmidationFreeAntimicrobial and AntitumorWuyi torrent frog, Amolops wuyiensisH-838Lung CancerMTT assayIC50 = 32.15 µM24-hLungNone
7510
372287022023
FLPLLAGLAANFLPQIICKIARKC
B1AW24LinearLNoneAmidationFreeAntimicrobial and AntitumorWuyi torrent frog, Amolops wuyiensisPC-3Prostate CancerMTT assayIC50 = 33.46 µM24-hProstateNone
7509
375081982023
FLGVALKLGKVLGKALLPLASSLLHSQ
Figanin 2BN27LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)HT-29Colon CancerMTT assayLC50 = 14.1 uM24-hColonNone
7508
375081982023
FLGVALKLGKVLGKALLPLASSLLHSQ
Figanin 2BN27LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)MDA-MB-231Breast CancerMTT assayLC50 = 8.1 uM24-hBreastNone
7507
375081982023
FLGVALKLGKVLGKALLPLASSLLHSQ
Figanin 2BN27LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)A-549Lung CancerMTT assayLC50 = 6.7 uM24-hLungNone
7506
375081982023
GIFKDTLKKVVAAVLTTVADNIHPK
Picturin 1BN25LinaerLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)HT-29Colon CancerMTT assayLC50 = 84.9 uM24-hColonNone
7505
375081982023
GIFKDTLKKVVAAVLTTVADNIHPK
Picturin 1BN25LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)MDA-MB-231Breast CancerMTT assayLC50 = 64.2 uM24-hBreastNone
7504
375081982023
GIFKDTLKKVVAAVLTTVADNIHPK
Picturin 1BN25LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)A-549Lung CancerMTT assayLC50 = 30.7 µM24-hLungNone
7503
375081982023
GLMDMLKKVGKVALTVAKSALLP
Picturin 2BN23LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)HT-29Colon CancerMTT assayLC50 52.2 uM24-hColonNone
7502
375081982023
GLMDMLKKVGKVALTVAKSALLP
Picturin 2BN23LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)MDA-MB-231Breast CancerMTT assayLC50 26.3 uM24-hBreastNone
7501
375081982023
GLMDMLKKVGKVALTVAKSALLP
Picturin 2BN23LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)A-549Lung CancerMTT assayLC50 = 23 µM24-hLungNone
7500
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticA-549Lung CancerCCK-8 assayIC50 = 32.47 µM36-hLungNone
7499
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticU-2 OSBone CancerCCK-8 assayIC50 = 25.65 µM36-hBoneNone
7498
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticHeLaCervical CancerCCK-8 assayIC50 = 42.95 µM36-hCervixNone
7497
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticZR-75-30Breast CancerCCK-8 assayIC50 = 23.57 µM36-hBreastNone
7496
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerCCK-8 assayIC50 = 31.05 µM36-hBreastNone
7495
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerCCK-8 assayIC50 = 18.15 µM36-hBreastNone
7480
373969452023
LSTAADMQGVVTDGMASGLDKDYLKPDD
p2828LinearLNoneFreeFreeAntitumorPseudomonas aeruginosaCT-26Colorectal CancerMTT assayIC50 ~ 150 μg/ml24-hColonNone
7479
373969452023
LSTAADMQGVVTDGMASGLDKDYLKPDD
p2828LinearLNoneFreeFreeAntitumorPseudomonas aeruginosaHT-29Colon CancerMTT assayIC50 ~ 200 μg/ml24-hColonNone
7421
364104362023
RRRRNRTRRNRRRVRGGLTIYFY
FHV-2D523LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-G48-hLiverNone
7420
364104362023
TRRQRTRRARRNRGGLTIYFY
HTLV-II-Rex-2D521LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-G48-hLiverNone
7419
364104362023
GRKKRRQRRRPPQGGLTIYFY
TAT-2D521LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-G48-hLiverNone
7417
364104362023
RRRRRRRRGGVVELRVPTDLTLLPGHLYMM
6E(V116-M135)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-D48-hLiverNone
7413
364104362023
RRRRRRRRGGQGLTIYFYNSNR
2D(Q44-R55)22LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7412
364104362023
RRRRRRRRGGQGLTIYFYNSNRDFQ
2C(Q44-Q58)25LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7411
364104362023
RRRRRRRRGGFWAGLQGLTIYFYNSNRDFQ
2A(F39-Q58)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7410
364104362023
RRRRRRRRGGMWKGFILTVVELRVPTDLTL
#6(M108-L127)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideMCF-7Breast CancerCellTiter-Glo assayGraph figure 1-B48-hBreastNone
7409
364104362023
RRRRRRRRGGMWKGFILTVVELRVPTDLTL
#6(M108-L127)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-B48-hLiverNone
7408
364104362023
RRRRRRRRGGDQEIKFKVETLECREMWKGF
#5(D93-F112)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-B48-hLiverNone
7407
364104362023
RRRRRRRRGGDRDYKKFWAGLQGLTIYFYN
#2(D33-N52)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideMCF-7Breast CancerCellTiter-Glo assayGraph figure 1-B48-hBreastNone
7406
364104362023
RRRRRRRRGGDRDYKKFWAGLQGLTIYFYN
#2(D33-N52)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-B48-hLiverNone
7355
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1MCF-7Breast CancerMTT assayIC50 = 24.60 μM24-hBreastNone
7354
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1U-251-MGBrain TumorMTT assayIC50 = 25.06 μM24-hBrainNone
7352
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1H-157Non-small cell lung cancerMTT assayIC50 = 24 μM24-hLungNone
7353
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1PC-3Prostate cancerMTT assayIC50 = 31.27 μM24-hProstateNone
7350
356064682022
GLLGKILGAGKKVLCGVSGLC
Nigrocin-PN21LinearLNoneFreeFreeAntimicrobial and AntitumorPelophylax nigromaculatusPC-3Prostate cancerMTT assayIC50 = 53.03 μM24-hProstateNone
7351
356064682022
GLLGKILGAGKKVLCGVSGLC
Nigrocin-PN21LinearLNoneFreeFreeAntimicrobial and AntitumorPelophylax nigromaculatusU-251-MGBrain TumorMTT assayIC50 = 73.65 μM24-hBrainNone
7349
356064682022
GLLGKILGAGKKVLCGVSGLC
Nigrocin-PN21LinearLNoneFreeFreeAntimicrobial and AntitumorPelophylax nigromaculatusH-157Non-small cell lung cancerMTT assayIC50 = 18.04 μM24-hLungNone
7307
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticHCC-827Lung AdenocarcinomaMTT assayIC50 between 4.0 and 5.5 μM72-hLungNone
7306
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticH-1975Non Small Cell Lung Cancer (NSCLC)MTT assayIC50 between 4.0 and 5.5 μM72-hLungNone
7305
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticH-358Non Small Cell Lung Cancer (NSCLC)MTT assayIC50 = 4.00 ± 0.20 μM72-hLungNone
7304
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 5.55 ± 0.13 μM72-hLungNone
7303
362879852022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusHepG-2Liver CancerMTT assayIC50 = 5.524 µM24-hLiverNone
7302
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusH-460Lung CancerMTT assayIC50 = 7.07 ± 0.81 µM24-hLungNone
7301
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusPC-9Lung CancerMTT assayIC50 = 6.34 ± 0.53 µM24-hLungNone
7300
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusH-3122Lung CancerMTT assayIC50 = 4.64 ± 0.18 µM24-hLungNone
7299
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusA-549Lung CancerMTT assayIC50 = 4.06 ± 0.60 µM24-hLungNone
7276
356018272022
IWLTALKFLGKNLGKLAKQQLAKL
LyeTx-I-b24LinearLNoneAmidatedAcetylationAntimicrobialSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 2.47 µM48-hBreastNone
7275
350138812022
KLKNFAKGVAQSLLNKASCKLSGQC
Brevinin-2R25LinearLNoneFreeFreeAntimicrobialRana ridibundaHeLaCervical CancerMTT assayIC50 = 131.5 μg/ml24-hCervixNone
7274
364658442022
GVKFAKRFWRFAKKAFKRFEK
HAZ21LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 5.44 μM4-hLungNone
7254
357741632022
flgvlallgylavrpflpkkkqqk
D-NAF-124LinearDNoneFreeFreeAnticancerNAF-1/CISD2MDA-MB-231Breast CancerNot AvailableIC50 = 12.8 ± 0.2 μMNABreastNone
7253
357741632022
FLGVLALLGYLAVRPFLPKKKQQK
NAF-124LinearLNoneFreeFreeAnticancerNAF-1/CISD2MDA-MB-231Breast CancerNot AvailableIC50 = 18.3 ± 0.4 μMNABreastNone
7250
366725512022
GRKKRRQRRRPPQ-X-CWMSPRHLGTC
CIGB-30025CyclicLX = Beta- AlanineFreeBiotinylatedAnticancerSyntheticNCI-H-460Lung CancerCrystal Violet assayIC50 = 30 ± 5.3 µM48-hLungNone
7249
357456432022
FKWQFEMLIMKIAKTSGFMFYSSY
BmPLA224LinearLNoneFreeFreeAnticancerphospholipase A2 isoform from B. moojeni venomRDRhabdomyosarcomaMTT assay60% reduction in cell viability24-hMuscleNone
7248
357456432022
FKWQFEMLIMKIAKTSGFMFYSSY
BmPLA224LinearLNoneFreeFreeAnticancerphospholipase A2 isoform from B. moojeni venomCaCo-2Colorectal CancerMTT assayIC50 = 0.6 µM24-hColonNone
7223
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2MCF-7Breast CancerMTT assayEC50 = 0.724 ± 0.340 mol/L × 10-324-hBreastNone
7222
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2A-2058Skin CancerMTT assayEC50 = 0.744 ± 0.208 mol/L × 10-324-hSkinNone
7221
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2U-87Brain TumorMTT assayEC50 = 0.427 ± 0.053 mol/L × 10-324-hBrainNone
7220
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2HeLaCervical CancerMTT assayEC50 = 0.525 ± 0.160 mol/L × 10-324-hCervixNone
7219
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2B16-F10-Nex 2Skin CancerMTT assayEC50 = 0.263 ± 0.585 mol/L × 10-324-hSkinNone
7218
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinWiDrColon CancerMTT assayIC50 = 197.3 μM24-hColonNone
7217
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinAGSStomach CancerMTT assayIC50 = 29.8 μM24-hStomachNone
7216
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinA-549Lung CancerMTT assayIC50 = 42.1 μM24-hLungNone
7215
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinHep3BLiver CancerMTT assayIC50 = 77.5 μM24-hLiverNone
7214
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinHuh-7Liver CancerMTT assayIC50 = 60 μM24-hLiverNone
7213
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinJ5Liver CancerMTT assayIC50 = 11 μM24-hLiverNone
7212
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusAGSStomach CancerMTT assayIC50 = 186.5 μM24-hStomachNone
7211
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusA-549Lung CancerMTT assayIC50 = 300.8 μM24-hLungNone
7210
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusHep3BLiver CancerMTT assayIC50 = 340.9 μM24-hLiverNone
7209
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusJ5Liver CancerMTT assayIC50 = 54.9 μM24-hLiverNone
7195
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticSNB-19Brain TumorCCK-8 assayIC50 = 12.0 ± 0.6 μM72-hBrainNone
7194
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticSF-268Brain TumorCCK-8 assayIC50 = 4.8 ± 0.1 μM72-hBrainNone
7193
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-138Brain TumorCCK-8 assayIC50 = 7.5 ± 0.3 μM72-hBrainNone
7192
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticLN229Brain TumorCCK-8 assayIC50 = 4.7 ± 0.2 μM72-hBrainNone
7191
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticSW-1783Brain TumorCCK-8 assayIC50 = 4.8 ± 0.2 μM72-hBrainNone
7190
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticD54Brain TumorCCK-8 assayIC50 = 8.4 ± 0.1 μM72-hBrainNone
7189
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-118Brain TumorCCK-8 assayIC50 = 6.8 ± 0.2 μM72-hBrainNone
7188
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-373Brain TumorCCK-8 assayIC50 = 5.0 ± 0.2 μM72-hBrainNone
7187
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticT98GBrain TumorCCK-8 assayIC50 = 7.1 ± 0.2 μM96-hBrainNone
7186
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticA-172Brain TumorCCK-8 assayIC50 = 6.4 ± 0.4 μM96-hBrainNone
7185
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-251Brain TumorCCK-8 assayIC50 = 4.9 ± 0.3 μM96-hBrainNone
7184
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU87-MGBrain TumorCCK-8 assayIC50 = 4.3 ± 0.3 μM96-hBrainNone
7183
356606292022
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationFreeAntimicrobialskin mucous secretions of winter flounderSCC-9Oral CancerCCK-8 assayIC50 = 45 μg/ml24-hTongueNone
7182
356606292022
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationFreeAntimicrobialskin mucous secretions of winter flounderCAL-27Oral CancerCCK-8 assayIC50 = 45 μg/ml24-hTongueNone
7089
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMNT-1Skin CancerResazurin dye assayIC50 = 57.03 ± 6.09 µM48-hSkinUS_10550155_B2
7088
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaPC-3Prostate CancerResazurin dye assayIC50 = 57.99 ± 5.04 µM48-hProstateUS_10550155_B2
7086
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-2780Ovarian CancerResazurin dye assayIC50 = 33.92 ± 5.90 µM48-hOvaryUS_10550155_B2
7087
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMiaPaCa.2Pancreatic CancerResazurin dye assayIC50 = 57.45 ± 6.03 µM48-hPancreasUS_10550155_B2
7084
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMCF-7Breast CancerResazurin dye assayIC50 = 35.71 ± 8.50 µM48-hBreastUS_10550155_B2
7085
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-549Lung CancerResazurin dye assayIC50 = 70.71 ± 5.39 µM48-hLungUS_10550155_B2
7076
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMNT-1Skin CancerResazurin dye assayIC50 = 4.72 ± 0.36 µM48-hSkinUS_10550155_B2
7075
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaPC-3Prostate CancerResazurin dye assayIC50 = 6.31 ± 0.66 µM48-hProstateUS_10550155_B2
7074
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMiaPaCa.2Pancreatic CancerResazurin dye assayIC50 = 8.71 ± 0.35 µM48-hPancreasUS_10550155_B2
7073
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-2780Ovarian CancerResazurin dye assayIC50 = 4.42 ± 0.06 µM48-hOvaryUS_10550155_B2
7072
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-549Lung CancerResazurin dye assayIC50 = 3.79 ± 1.61 µM48-hLungUS_10550155_B2
7071
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaHepG-2Liver CancerResazurin dye assayIC50 = 14.31 ± 1.37 µM48-hLiverUS_10550155_B2
7070
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMCF-7Breast CancerResazurin dye assayIC50 = 5.69 ± 1.46 µM48-hBreastUS_10550155_B2
6904
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisB16-F10Skin CancerMTS assayIC50 = 6.65 ± 0.33 μM48-hSkinNone
6903
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisSMMC-7721Liver CancerMTS assayIC50 = 6.87 ± 0.51 μM48-hLiverNone
6902
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisA-549Lung CancerMTS assayIC50 = 5.81 ± 0.23 μM48-hLungNone
6901
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisSW-480Blood CancerMTS assayIC50 = 10.37 ± 0.40 μM48-hBloodNone
6900
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisMDA-MB-231Breast CancerMTS assayIC50 = 5.44 ± 0.33 μM48-hBreastNone
6899
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisHCT-116Colon CancerMTS assayIC50 = 5.87 ± 0.15 μM48-hColonNone
6885
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisHeLaCervical CancerMTT assayIC50 = 1.97 µM24-hCervixNone
6884
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisHeLaCervical CancerMTT assayIC50 = 18.1 µM24-hCervixNone
6883
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisA-549Lung CancerMTT assayIC50 = 2.99 µM24-hLungNone
6882
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisA-549Lung CancerMTT assayIC50 = 21.6 µM24-hLungNone
6881
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 5.25 µM24-hBreastNone
6880
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 17.5 µM24-hBreastNone
6879
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 5.52 µM24-hNot AvailableNone
6878
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 26.01 µM24-hNot AvailableNone
6877
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisHeLaCervical CancerMTT assayIC50 = 2.17 µM24-hCervixNone
6876
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisHeLaCervical CancerMTT assayIC50 = 2.22 µM24-hCervixNone
6875
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisA-549Lung CancerMTT assayIC50 = 2.15 µM24-hLungNone
6874
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisA-549Lung CancerMTT assayIC50 = 4.2 µM24-hLungNone
6873
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 3.92 µM24-hBreastNone
6872
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 5.83 µM24-hBreastNone
6871
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 5.31 µM24-hNot AvailableNone
6870
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 5.58 µM24-hNot AvailableNone
6861
336770232021
GKLRLIKKLWVKKWKKKGWKA
Pep21LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 2 µM24-hBreastNone
6860
336770232021
GKLRLIKKLWVKKWKKKGWKA
Pep21LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 4 µM24-hLungNone
6857
336909772021
zffygwyggmekllrggrgerppr
NMTP-524LinearDZ = C10H7CH2C(O), M, 4-(Trifluoromethyl)-D-phenylalanineFreeFreeAnticancerNot AvailableSK-HEP-1Liver CancerMTT assayIC50 = 53.84 ± 4.35 µM48-hLiverNone
6809
343093732021
Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
Pal-N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acidAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinMCF-7Breast CancerMTT assayIC50 = 27.26 μM24-hBreastNone
6808
343093732021
Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
Pal-N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acidAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-549Lung CancerMTT assayIC50 = 44.98 μM24-hLungNone
6807
343093732021
Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
Pal-N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acidAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50 = 36.67(Supplementary material)/15.2 ± 0.7 μM(Published paper)24-hSkinNone
6801
348487292021
TGIATSGLATFTLHTGSLAPAT
AtMP222LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MDA-MB-231Breast CancerMTT assayIC50 = 6.97 ± 0.24 μg/ml48-hBreastNone
6800
348487292021
TGIATSGLATFTLHTGSLAPAT
AtMP222LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MCF-7Breast CancerMTT assayIC50 = 5.89 ± 0.14 μg/ml48-hBreastNone
6799
348487292021
THPPTTTTTTTTTTTTTAAPATTT
AtMP124LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MDA-MB-231Breast CancerMTT assayIC50 = 9.35 ± 0.25 μg/ml48-hBreastNone
6798
348487292021
THPPTTTTTTTTTTTTTAAPATTT
AtMP124LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MCF-7Breast CancerMTT assayIC50 = 8.25 ± 0.14 μg/ml48-hBreastNone
6785
335626812021
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusAska-SSSynovial SarcomaMTS assayIC50 = 32.41 μg/mLNAMuscleNone
6784
335626812021
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusSW982Synovial SarcomaMTS assayIC50 = 29.20 μg/mLNAMuscleNone
6778
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticMDA-MB-435 DOX-RBreast CancerMTS assayIC50 = 3.4 µM24-hBreastNone
6777
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticMDA-MB-435 WTBreast CancerMTS assayIC50 = 3.5 µM24-hBreastNone
6776
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticCT-26Colorectal CancerMTS assayIC50 = 2.2 µM24-hColonNone
6775
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticA-549Lung CancerMTS assayIC50 = 4.5 µM24-hLungNone
6730
343093732021
RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATFreeAnticancerSyntheticA-375Skin CancerMTT assayIC50 > 50.0 μM24-hSkinNone
6728
335822212021
ALWKDLLKNVGIAAGKAALNKVTDMVNQ
Dermaseptin-TO28LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tomopternaPC-3Prostate CancerMTT assayGraph Figure-724-hProstateNone
6727
335822212021
ALWKDLLKNVGIAAGKAALNKVTDMVNQ
Dermaseptin-TO28LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tomopternaH-157Lung CancerMTT assayGraph Figure-724-hLungNone
6726
335822212021
ALWKDLLKNVGIAAGKAALNKVTDMVNQ
Dermaseptin-TO28LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tomopternaU251-MGBrain TumorMTT assayGraph Figure-724-hBrainNone
6725
345727192021
IWLTALKFLGKNLGKLAKQQLAKL
LyeTxI-b24LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 5.77 ± 0.83 µM48-hBreastNone
6724
345727192021
IWLTALKFLGKNLGKLAKQQLAKL
LyeTxI-b24LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 7.34 ± 3.09 µM48-hBreastNone
6723
345727192021
IWLTALKFLGKNLGKLAKQQLAKL
LyeTxI-b24LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic4T1Breast CancerMTT assayIC50 = 6.5 ± 5.30 µM48-hBreastNone
6722
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkMDA-MB-231Breast CancerAnnexin V-FITC assay~80% cell death at 200 µg/ml48-hBreastNone
6721
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkMCF-7Breast CancerAnnexin V-FITC assay~50% cell death at 300 µg/ml48-hBreastNone
6720
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkSK-BR-3Breast CancerAnnexin V-FITC assay~80% cell death at 100 µg/ml48-hBreastNone
6719
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkMDA-MB-468Breast CancerAnnexin V-FITC assay~60% cell death at 300 µg/ml48-hBreastNone
6718
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSHCT-116Colon CancerMTT assayIC50 = 3.721 µM24-hColonNone
6717
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSMCF-7Breast CancerMTT assayIC50 = 3.17 µM24-hBreastNone
6716
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSU251-MGBrain TumorMTT assayIC50 = 3.492 µM24-hBrainNone
6715
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSPC-3Prostate CancerMTT assayIC50 = 2.629 µM24-hProstateNone
6714
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSH-838Lung CancerMTT assayIC50 = 2.553 µM24-hLungNone
6713
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSHCT-116Colon CancerMTT assayIC50 = 11.03 µM24-hColonNone
6712
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSMCF-7Breast CancerMTT assayIC50 = 8.883 µM24-hBreastNone
6711
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSU251-MGBrain TumorMTT assayIC50 = 8.629 µM24-hBrainNone
6710
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSPC-3Prostate CancerMTT assayIC50 = 5.473 µM24-hProstateNone
6709
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSH-838Lung CancerMTT assayIC50 = 3.976 µM24-hLungNone
6708
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriHCT-116Colon CancerMTT assayIC50 = 33.69 µM24-hColonNone
6707
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriMCF-7Breast CancerMTT assayIC50 = 112 µM24-hBreastNone
6706
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriU251-MGBrain TumorMTT assayIC50 = 233.0 µM24-hBrainNone
6705
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriPC-3Prostate CancerMTT assayIC50 = 95.94 µM24-hProstateNone
6704
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriH-838Lung CancerMTT assayIC50 = 36.84 µM24-hLungNone
6703
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HHCT-116Colon CancerMTT assayIC50 = 3.583 µM24-hColonNone
6702
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HH-157Lung CancerMTT assayIC50 = 2.811 µM24-hLungNone
6701
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HMDA-MB-435SBreast CancerMTT assayIC50 = 2.243 µM24-hBreastNone
6700
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HPC-3Prostate CancerMTT assayIC50 = 5.425 µM24-hProstateNone
6699
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HHCT-116Colon CancerMTT assayIC50 = 342.8 µM24-hColonNone
6698
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HH-157Lung CancerMTT assayIC50 = 278.9 µM24-hLungNone
6697
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HMDA-MB-435SBreast CancerMTT assayIC50 = 214.7 µM24-hBreastNone
6696
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HPC-3Prostate CancerMTT assayIC50 = 186.9 µM24-hProstateNone
6695
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisHCT-116Colon CancerMTT assayIC50 = 2.599 µM24-hColonNone
6694
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisH-157Lung CancerMTT assayIC50 = 3.37 µM24-hLungNone
6693
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisMDA-MB-435SBreast CancerMTT assayIC50 = 3.47 µM24-hBreastNone
6692
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisPC-3Prostate CancerMTT assayIC50 = 5.87 µM24-hProstateNone
6679
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 1499 μM24-hBrainNone
6678
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 427.3 μM24-hLungNone
6677
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 180.8 μM24-hLungNone
6676
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 118.4 μM24-hProstateNone
6675
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 593.7 μM24-hBrainNone
6674
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 88.28 μM24-hLungNone
6673
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 186.1 μM24-hLungNone
6672
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 55.65 μM24-hProstateNone
6671
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 2.679 μM24-hBrainNone
6670
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 1.546 μM24-hLungNone
6669
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 1.796 μM24-hLungNone
6668
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 2.605 μM24-hProstateNone
6667
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 32.18 μM24-hBrainNone
6666
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 6.143 μM24-hLungNone
6665
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 10.11 μM24-hLungNone
6664
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 18.99 μM24-hProstateNone
6663
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisU251-MGBrain TumorMTT assayIC50 = 34.25 μM24-hBrainNone
6662
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisH-157Lung CancerMTT assayIC50 = 10.20 μM24-hLungNone
6661
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisH-838Lung CancerMTT assayIC50 = 23.51 μM24-hLungNone
6660
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisPC-3Prostate CancerMTT assayIC50 = 14.67 μM24-hProstateNone
6582
None2020
klaklakklaklakGGRKKRRQRRR
D(KLAKLAK)2-TAT25LinearMixNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 5.3 μM24-hLungNone
6556
324439212020
FLGAILKIGHALAKTVLPMVTNAFKPKQ
Figainin 228LinearLNoneFreeFreeAntimicrobial and AnticancerBoana ranicepsMCF-7Breast CancerMTT assayIC50= 15.3 µM24-hBreastNone
6555
324439212020
FLGAILKIGHALAKTVLPMVTNAFKPKQ
Figainin 228LinearLNoneFreeFreeAntimicrobial and AnticancerBoana ranicepsB16-F10Skin CancerMTT assayIC50 = 12.8 µM24-hSkinNone
6551
324984252020
IWLTALKFLGKNLGKHLAKQQLSKL
LVTX-825LinearLNoneAmidationAcetylationAnticancerLycosa vittataH-460Lung CancerCCK-8 assayIC50 = 19 μM24-hLungNone
6550
324984252020
IWLTALKFLGKNLGKHLAKQQLSKL
LVTX-825LinearLNoneAmidationAcetylationAnticancerLycosa vittataA-549Lung CancerCCK-8 assayIC50 = 8 μM24-hLungNone
6546
322561722020
KAIGLVIPEIDGKLDGGAQRV
NMANF221LinearLNoneFreeFreeAnticancerStaphylococcus hominis strain MANF2HT-29Colon CancerMTT assayIC50 = 48.9 µg/mLNAColonNone
6545
322561722020
KAIGLVIPEIDGKLDGGAQRV
NMANF221LinearLNoneFreeFreeAnticancerStaphylococcus hominis strain MANF2A-549Lung CancerMTT assayIC50 = 46.6 µg/mLNALungNone
6544
345085632020
FLGALFKVASKLVPAAICSISKKC
Brevinin-1HL24LinearLNoneFreeFreeAntimicrobialHylarana latouchiiNCI-H23Lung CancerMTT assayIC50 = 8.52 ± 1.02 μM24-hLungNone
6527
321516092020
PWRIRIRRRRIRIRWPPWRIRIRR
R-DIM-LF11-334-LF11-33424LinearLNoneAmidationFreeAnticancerSyntheticWM164Skin CancerMTS assayLC50 = 3.6 ± 0.7 μM24-hSkinEP_2943215_B1
6526
321516092020
PWRIRIRRRRIRIRWPPWRIRIRR
R-DIM-LF11-334-LF11-33424LinearLNoneAmidationFreeAnticancerSyntheticSBcl2Skin CancerMTS assayLC50 < 1 ± 0.1 μM24-hSkinEP_2943215_B1
6525
321516092020
PWRIRIRRRRIRIRWPPWRIRIRR
R-DIM-LF11-334-LF11-33424LinearLNoneAmidationFreeAnticancerSyntheticA-375Skin CancerMTS assayLC50 < 1 ± 0.1 μM24-hSkinEP_2943215_B1
6512
321516092020
FQWQRNIRKVRPRVKRINRQWQF
R-DIM-P-LF1123LinearLNoneAmidationFreeAnticancerSyntheticWM164Skin CancerMTS assayLC50 = 20.9 ± 3.9 μM24-hSkinEP_2943215_B1
6511
321516092020
FQWQRNIRKVRPRVKRINRQWQF
R-DIM-P-LF1123LinearLNoneAmidationFreeAnticancerSyntheticSBcl2Skin CancerMTS assayLC50 = 10.7 ± 0.2 μM24-hSkinEP_2943215_B1
6510
321516092020
FQWQRNIRKVRPRVKRINRQWQF
R-DIM-P-LF1123LinearLNoneAmidationFreeAnticancerSyntheticA-375Skin CancerMTS assayLC50 = 125.0 ± 16.8 μM24-hSkinEP_2943215_B1
6505
324620552020
Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF
AEM-28–228LinearLAha= α-aminohenoic acidAmidationAcetylationAnti-inflammatory and AnticancerSyntheticOV-2008Ovarian CancerMTS assay~40% cell viability at 10 μg/mL24-hOvaryNone
6506
324620552020
Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF
AEM-28–228LinearLAha= α-aminohenoic acidAmidationAcetylationAnti-inflammatory and AnticancerSyntheticSK-OV-3Ovarian CancerMTS assay~30% cell viability at 10 μg/mL24-hOvaryNone
6507
324620552020
Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF
AEM-28–228LinearLAha= α-aminohenoic acidAmidationAcetylationAnti-inflammatory and AnticancerSyntheticCaCo-2Colon CancerMTS assay~60% cell viability at 10 μg/mL24-hColonNone
6503
324620552020
Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF
AEM-28–228LinearLAha= α-aminohenoic acidAmidationAcetylationAnti-inflammatory and AnticancerSyntheticCT-26Colorectal CancerMTS assay~30% cell viability at 10 μg/mL24-hColonNone
6504
324620552020
Aha-LRRLRRRLLRDWLKAFYDKVAEKLKEAF
AEM-28–228LinearLAha= α-aminohenoic acidAmidationAcetylationAnti-inflammatory and AnticancerSyntheticID8Colon CancerMTS assay~20% cell viability at 10 μg/mL24-hColonNone
6501
324620552020
LRKLRKRLLRDWLKAFYDKVAEKLKEAF
AEM-2828LinearLNoneFreeFreeAnti-inflammatory and AnticancerSyntheticCaCo-2Colon CancerMTS assay~70% cell viability at 10 μg/mL24-hColonNone
6500
324620552020
LRKLRKRLLRDWLKAFYDKVAEKLKEAF
AEM-2828LinearLNoneFreeFreeAnti-inflammatory and AnticancerSyntheticSK-OV-3Ovarian CancerMTS assay~50% cell viability at 10 μg/mL24-hOvaryNone
6499
324620552020
LRKLRKRLLRDWLKAFYDKVAEKLKEAF
AEM-2828LinearLNoneFreeFreeAnti-inflammatory and AnticancerSyntheticOV-2008Ovarian CancerMTS assay~60% cell viability at 10 μg/mL24-hOvaryNone
6498
324620552020
LRKLRKRLLRDWLKAFYDKVAEKLKEAF
AEM-2828LinearLNoneFreeFreeAnti-inflammatory and AnticancerSyntheticID8Colon CancerMTS assay~60% cell viability at 10 μg/mL24-hColonNone
6497
324620552020
LRKLRKRLLRDWLKAFYDKVAEKLKEAF
AEM-2828LinearLNoneFreeFreeAnti-inflammatory and AnticancerSyntheticCT-26Colorectal CancerMTS assay~20% cell viability at 10 μg/mL24-hColonNone
6496
321262282020
GALFLGFLGAAGSTMGAWSQPKKKRKV
MPG27LinearLNoneCysteamidationAcetylationAntimicrobialSyntheticJurkatBlood CancerMTT assayIC50 = 15.8 μM24-hBloodNone
6491
321262282020
GIGRWLHSARRFGRAFVGEIMNS
MagaininF5W-Arg23LinearLNoneFreeFreeAntimicrobialSyntheticJurkatBlood CancerMTT assayIC50 = 16.8 μM24-hBloodNone
6490
321262282020
GIGKWLHSAKKFGKAFVGEIMNS
MagaininF5W-Lys23LinearLNoneFreeFreeAntimicrobialSyntheticJurkatBlood CancerMTT assayIC50 = 16.8 μM24-hBloodNone
6451
325826422020
ALWKDMLKGIGKLAGKAALGAVKTLV
Dermaseptin-PP26LinearLNoneAmidationFreeAntimicrobialPhyllomedusa palliataH-157Lung CancerLDH leakage assay80% LDH release at 10−4 M24-hLungNone
6450
325826422020
ALWKDMLKGIGKLAGKAALGAVKTLV
Dermaseptin-PP26LinearLNoneAmidationFreeAntimicrobialPhyllomedusa palliataU-251Brain TumorMTT assayIC50 = 2.47 μM24-hBrainNone
6449
325826422020
ALWKDMLKGIGKLAGKAALGAVKTLV
Dermaseptin-PP26LinearLNoneAmidationFreeAntimicrobialPhyllomedusa palliataPC-3Prostate CancerMTT assayIC50 = 4.15 μM24-hProstateNone
6448
325826422020
ALWKDMLKGIGKLAGKAALGAVKTLV
Dermaseptin-PP26LinearLNoneAmidationFreeAntimicrobialPhyllomedusa palliataMCF-7Breast CancerMTT assayIC50 = 2.92 μM24-hBreastNone
6447
325826422020
ALWKDMLKGIGKLAGKAALGAVKTLV
Dermaseptin-PP26LinearLNoneAmidationFreeAntimicrobialPhyllomedusa palliataH-157Lung CancerMTT assayIC50 = 1.55 μM24-hLungNone
6408
323472932020
FLGALFKVASKLVPAAICSISKKC
Brevinin-1GHd24LinearLNoneFreeFreeAntimicrobialHylarana guentheriPC-3Prostate CancerMTT assayIC50 = 9.854 µM24-hProstateNone
6407
323472932020
FLGALFKVASKLVPAAICSISKKC
Brevinin-1GHd24LinearLNoneFreeFreeAntimicrobialHylarana guentheriMDA-MB-435SSkin CancerMTT assayIC50 = 1.197 µM24-hSkinNone
6406
323472932020
FLGALFKVASKLVPAAICSISKKC
Brevinin-1GHd24LinearLNoneFreeFreeAntimicrobialHylarana guentheriU-251-MGBrain TumorMTT assayIC50 = 7.985 µM24-hBrainNone
6405
323472932020
FLGALFKVASKLVPAAICSISKKC
Brevinin-1GHd24LinearLNoneFreeFreeAntimicrobialHylarana guentheriNCI-H-157Lung CancerMTT assayIC50 = 2.987 µM24-hLungNone
6261
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8b23LinearLNoneFree3′-Aminopropyl Beta-D-GalactopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IPC-3Prostate CancerCCK-8 assayIC50 = 4.9 ± 0.2 µM24-hProstateNone
6259
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8b23LinearLNoneFree3′-Aminopropyl Beta-D-GalactopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IH-1437Lung CancerCCK-8 assayIC50 = 5.3 ± 0.2 µM24-hLungNone
6260
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8b23LinearLNoneFree3′-Aminopropyl Beta-D-GalactopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IHGC-27Gastric CancerCCK-8 assayIC50 = 5.3 ± 0.2 µM24-hNot AvailableNone
6257
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8b23LinearLNoneFree3′-Aminopropyl Beta-D-GalactopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IA-549Lung CancerCCK-8 assayIC50 = 7.0 ± 0.3 µM24-hLungNone
6258
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8b23LinearLNoneFree3′-Aminopropyl Beta-D-GalactopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IH-460Lung CancerCCK-8 assayIC50 = 4.9 ± 0.9 µM24-hLungNone
6255
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8a23LinearLNoneFree3′-Aminopropyl-D-glucopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IPC-3Prostate CancerCCK-8 assayIC50 = 6.9 ± 0.4 µM24-hProstateNone
6256
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8b23LinearLNoneFree3′-Aminopropyl Beta-D-GalactopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IMDA-MB-231Breast CancerCCK-8 assayIC50 = 6.0 ± 0.2 µM24-hBreastNone
6254
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8a23LinearLNoneFree3′-Aminopropyl-D-glucopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IHGC-27Gastric CancerCCK-8 assayIC50 = 12.6 ± 0.6 µM24-hNot AvailableNone
6253
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8a23LinearLNoneFree3′-Aminopropyl-D-glucopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IH-1437Lung CancerCCK-8 assayIC50 = 13.0 ± 0.2 µM24-hLungNone
6252
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8a23LinearLNoneFree3′-Aminopropyl-D-glucopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IH-460Lung CancerCCK-8 assayIC50 = 8.5 ± 0.4 µM24-hLungNone
6250
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8a23LinearLNoneFree3′-Aminopropyl-D-glucopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IMDA-MB-231Breast CancerCCK-8 assayIC50 = 10.1 ± 0.2 µM24-hBreastNone
6251
312763992019
RGWFRAMRSIARFIARERLRGHL
R-Lycosin I derivative 8a23LinearLNoneFree3′-Aminopropyl-D-glucopyranosideAnticancerMonosaccharide Analogue of Anticancer Peptide R-Lycosin-IA-549Lung CancerCCK-8 assayIC50 = 9.6 ± 0.3 µM24-hLungNone
6227
311616862019
GIXXWLHSAXXFGXXFVXXIZNS
8Dap23LinearLX = 2,3-Diaminopropionic Acid , Z = norleucineAmidationFreeAnticancerSyntheticPANC-1Pancreatic CancerWST-1 assayEC50 = 61.4±0.7 μM24-hPancreasNone
6226
311616862019
GIKXWLHSAXXFGXKFVXXIZNS
6Dap23LinearLX = 2,3-Diaminopropionic Acid , Z = norleucineAmidationFreeAnticancerSyntheticPANC-1Pancreatic CancerWST-1 assayEC50 = 55.0±1.8 μM24-hPancreasNone
6225
311616862019
GIKXWLHSAXKFGXKFVKXIZNS
4Dap23LinearLX = 2,3-Diaminopropionic Acid , Z = norleucineAmidationFreeAnticancerSyntheticPANC-1Pancreatic CancerWST-1 assayEC50 = 35.7±0.7 μM24-hPancreasNone
6224
311616862019
GIKXWLHSAKKFGXKFVKKIZNS
2Dap23LinearLX = 2,3-Diaminopropionic Acid , Z = norleucineAmidationFreeAnticancerSyntheticPANC-1Pancreatic CancerWST-1 assayEC50 = 14.7±0.6 μM24-hPancreasNone
6223
311616862019
GIKKWLHSAKKFGKKFVKKIZNS
0Dap23LinearLZ = norleucineAmidationFreeAnticancerSyntheticPANC-1Pancreatic CancerWST-1 assayEC50 = 9.1±0.3 μM24-hPancreasNone
6207
None2019
CQYSVNPKIKRFELYFKGRMW
LPSBD-021LinearLNoneFreeFreeAnticancerSyntheticTHP-1Leukemia CancerNot AvailableNot Available24-hBloodNone
6206
None2019
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialScorpio maurus palmatusKG-1aLeukemia CancerLDH leakage assayFig 2NABloodNone
6205
None2019
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialScorpio maurus palmatusCCRF-CEMLeukemia CancerLDH leakage assayFig 2NABloodNone
6204
None2019
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialScorpio maurus palmatusKG-1aLeukemia CancerCellTiter-Glo assayLC50 = 16 ± 1.3 µg/mL24-hBloodNone
6203
None2019
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialScorpio maurus palmatusCCRF-CEMLeukemia CancerCellTiter-Glo assayLC50 = 16 ± 0.9 µg/mL24-hBloodNone
6198
312520472019
SRSSRAGLQFPVGRIHRLLRK
Fi-Histin1-2121LinearLNoneAmidationAcetylationAntimicrobialFenneropenaeus indicusHep-2Liver CancerXTT assayIC50 = 31.274 ± 24.531 μM24-hLiverNone
6197
312520472019
SRSSRAGLQFPVGRIHRLLRK
Fi-Histin1-2121LinearLNoneAmidationAcetylationAntimicrobialFenneropenaeus indicusNCI-H-460Lung CancerXTT assayIC50 = 22.670 ± 13.939 μM24-hLungNone
6196
303778402019
MTVVLLLIVLPLLGGVHSSGIL
TC2222LinearLNoneFreeFreeAnticancerTribolium castaneumMCF-7Breast CancerMTT assayFig 4a24-hBreastNone
6195
303778402019
MTVVLLLIVLPLLGGVHSSGIL
TC2222LinearLNoneFreeFreeAnticancerTribolium castaneumHeLaCervical CancerMTT assayFig 4a24-hCervixNone
6194
304490022019
IWLTALKFLGKNLGKLAKQQLAKL
LyeTx-I-b24LinearLNoneAmidationAcetylationAntimicrobialSyntheticSH-SY5YBrain TumorMTT/Resazurin dye assayIC50 = 93.80 ± 2.17 µM48-hBrainNone
6193
304490022019
IWLTALKFLGKNLGKLAKQQLAKL
LyeTx-I-b24LinearLNoneAmidationAcetylationAntimicrobialSyntheticU-373-MGBrain TumorMTT/Resazurin dye assayIC50 = 20.94 ± 5.18 µM48-hBrainNone
6192
304490022019
IWLTALKFLGKNLGKLAKQQLAKL
LyeTx-I-b24LinearLNoneAmidationAcetylationAntimicrobialSyntheticU-87-MGBrain TumorMTT/Resazurin dye assayIC50 = 29.20 ± 7.96 µM48-hBrainNone
6190
307173092019
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusU-251Brain TumorMTS/PMS assayLD50 = 20 μg/mL24-hBrainNone
6189
307173092019
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusU87-MGBrain TumorMTS/PMS assayLD50 = 20 μg/mL24-hBrainNone
6187
316334002019
FALGAVTKLLPSLLCMITRKC
HN-121LinearLNoneFreeFreeHost DefenseAmolops hainanensisPC-3Prostate CancerMTT assayNot Available12-hProstateNone
6188
316334002019
FALGAVTKLLPSLLCMITRKC
HN-121LinearLNoneFreeFreeHost DefenseAmolops hainanensis4T1Breast CancerMTT assayNot Available12-hBreastNone
6186
316334002019
FALGAVTKLLPSLLCMITRKC
HN-121LinearLNoneFreeFreeHost DefenseAmolops hainanensisMDA-MB-453Breast CancerMTT assayNot Available12-hBreastNone
6185
316334002019
FALGAVTKLLPSLLCMITRKC
HN-121LinearLNoneFreeFreeHost DefenseAmolops hainanensisSGC-7901Stomach CancerMTT assayNot Available12-hStomachNone
6184
316334002019
FALGAVTKLLPSLLCMITRKC
HN-121LinearLNoneFreeFreeHost DefenseAmolops hainanensisA-549Lung CancerMTT assayNot Available12-hLungNone
6183
316334002019
FALGAVTKLLPSLLCMITRKC
HN-121LinearLNoneFreeFreeHost DefenseAmolops hainanensisMCF-7Breast CancerMTT assayIC50 = 6.9 μM12-hBreastNone
6181
312263502019
GRFKRFRKKFKKLFKKLSPVIPLLHL
BMAP-2727LinearLNoneAmidationFreeAntimicrobialCathelicidinMDA-MB-361Breast CancerMTT assayIC50 = 4.2 μM48-hBreastNone
6182
312263502019
GRFKRFRKKFKKLFKKLSPVIPLLHL
BMAP-2727LinearLNoneAmidationFreeAntimicrobialCathelicidinA-549Lung CancerMTT assayIC50 = 5.3 μM48-hLungNone
6159
308854382019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
Hymenochirin - 1B29LinearLNoneAmidationFreeHost Defense PeptideHymenochirus boettgeriHepG-2Liver CancerMTT assay30% cell viability at 20 μM24-hLiverNone
6158
308854382019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
Hymenochirin - 1B29LinearLNoneAmidationFreeHost Defense PeptideHymenochirus boettgeriNCI-H-460Lung CancerMTT assay10% cell viability at 50 μM24-hLungNone
6157
308854382019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
Hymenochirin - 1B29LinearLNoneAmidationFreeHost Defense PeptideHymenochirus boettgeriA-549Lung CancerMTT assay40% cell viability at 10 μM24-hLungNone
6156
308854382019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
Hymenochirin - 1B29LinearLNoneAmidationFreeHost Defense PeptideHymenochirus boettgeriNCI-H-1299Lung CancerMTT assay20% cell viability at 10 μM24-hLungNone
6103
314263232019
ALWKTLLKHVGKAAGKAALNAVTDMVNQ
Dermaseptin-PS428LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvagiiMCF-7Breast CancerMTT assayIC50 = 0.67 µM24-hBreastNone
6102
314263232019
ALWKTLLKHVGKAAGKAALNAVTDMVNQ
Dermaseptin-PS428LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvagiiPC-3Prostate CancerMTT assayIC50 = 0.44 μM24-hProstateNone
6101
314263232019
ALWKTLLKHVGKAAGKAALNAVTDMVNQ
Dermaseptin-PS428LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvagiiH-157Lung CancerMTT assayIC50 = 0.19 μM24-hLungNone
6100
314263232019
ALWKTLLKHVGKAAGKAALNAVTDMVNQ
Dermaseptin-PS428LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvagiiMDA-MB-435SBreast CancerMTT assayIC50 = 0.11 μM24-hBreastNone
6099
314263232019
ALWKTLLKHVGKAAGKAALNAVTDMVNQ
Dermaseptin-PS428LinearLNoneAmidationFreeAntimicrobialPhyllomedusa sauvagiiU251-MGBrain TumorMTT assayIC50 = 57.66 nM24-hBrainNone
6098
307896952019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
H-029LinearLNoneAmidationFreeAntimicrobial and AnticancerHymenochirus boettgeriHepG-2Liver CancerMTT assayIC50 = 8.07 ± 0.21 μM48-hLiverNone
6097
307896952019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
H-029LinearLNoneAmidationFreeAntimicrobial and AnticancerHymenochirus boettgeriHCT-116Colon CancerMTT assayIC50 = 12.76 ± 0.43 μM48-hColonNone
6095
307896952019
IKLSPS5TKDS5LKKVLKGAIKGAIAVAKMV
H-229CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 1.60 ± 0.24 μM48-hLiverNone
6096
307896952019
IKLSPETKDNLKKVLKGAIKGAIAVAKMV
H-029LinearLNoneAmidationFreeAntimicrobial and AnticancerHymenochirus boettgeriA-549Lung CancerMTT assayIC50 = 15.22 ± 0.21 μM48-hLungNone
6094
307896952019
IKLSPS5TKDS5LKKVLKGAIKGAIAVAKMV
H-229CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 3.54 ± 0.72 μM48-hColonNone
6093
307896952019
IKLSPS5TKDS5LKKVLKGAIKGAIAVAKMV
H-229CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 4.26 ± 0.52 μM48-hLungNone
6091
307896952019
IKLSPETKDNLKKVLKGS5IKGS5IAVAKMV
H-529CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 4.16 ± 0.21 μM48-hColonNone
6092
307896952019
IKLSPETKDNLKKVLKGS5IKGS5IAVAKMV
H-529CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 2.82 ± 0.23 μM48-hLiverNone
6090
307896952019
IKLSPETKDNLKKVLKGS5IKGS5IAVAKMV
H-529CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 7.35 ± 0.22 μM48-hLungNone
6089
307896952019
IKLSPS5TKDS5LKKVLKGS5IKGS5IAVAKMV
H-1029CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 1.50 ± 0.21 μM48-hLiverNone
6088
307896952019
IKLSPS5TKDS5LKKVLKGS5IKGS5IAVAKMV
H-1029CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 3.51 ± 0.37 μM48-hColonNone
6087
307896952019
IKLSPS5TKDS5LKKVLKGS5IKGS5IAVAKMV
H-1029CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 3.59 ± 0.12 μM48-hLungNone
6086
307896952019
IKLSKKTKKNLKKVLKGAIKGAIAVAKMV
H-1429LinearLNoneAmidationFreeAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 4.54 ± 0.25 μM48-hLiverNone
6085
307896952019
IKLSKKTKKNLKKVLKGAIKGAIAVAKMV
H-1429LinearLNoneAmidationFreeAnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 1.841 ± 0.34 μM48-hColonNone
6084
307896952019
IKLSKKTKKNLKKVLKGAIKGAIAVAKMV
H-1429LinearLNoneAmidationFreeAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 0.98 ± 0.11 μM48-hLungNone
6082
307896952019
IKLSKS5TKDS5LKKVLKGAIKGAIAVAKMV
H-1529CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 2.95 ± 0.25 μM48-hColonNone
6083
307896952019
IKLSKS5TKDS5LKKVLKGAIKGAIAVAKMV
H-1529CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 2.20 ± 0.27 μM48-hLiverNone
6081
307896952019
IKLSKS5TKDS5LKKVLKGAIKGAIAVAKMV
H-1529CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 2.26 ± 0.24 μM48-hLungNone
6079
307896952019
IKLSPS5TKKS5LKKVLKGAIKGAIAVAKMV
H-1629CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 2.65 ± 0.35 μM48-hColonNone
6080
307896952019
IKLSPS5TKKS5LKKVLKGAIKGAIAVAKMV
H-1629CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 3.14 ± 0.46 μM48-hLiverNone
6078
307896952019
IKLSPS5TKKS5LKKVLKGAIKGAIAVAKMV
H-1629CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 1.85 ± 0.31 μM48-hLungNone
6076
307896952019
IKLSKS5TKKS5LKKVLKGAIKGAIAVAKMV
H-1729CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 1.49 ± 0.45 μM48-hColonNone
6077
307896952019
IKLSKS5TKKS5LKKVLKGAIKGAIAVAKMV
H-1729CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 1.64 ± 0.47 μM48-hLiverNone
6074
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-1829CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 1.61 ± 0.21 μM48-hLiverNone
6075
307896952019
IKLSKS5TKKS5LKKVLKGAIKGAIAVAKMV
H-1729CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 0.96 ± 0.33 μM48-hLungNone
6072
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-1829CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 0.89 ± 0.21 μM48-hLungNone
6073
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-1829CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 1.11 ± 0.21 μM48-hColonNone
6071
307896952019
IKLSKETKKNLKKVLKGS5IKGS5IAVAKMV
H-1929CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 1.64 ± 0.36 μM48-hLiverNone
6069
307896952019
IKLSKETKKNLKKVLKGS5IKGS5IAVAKMV
H-1929CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 1.00 ± 0.36 μM48-hLungNone
6070
307896952019
IKLSKETKKNLKKVLKGS5IKGS5IAVAKMV
H-1929CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 1.78 ± 0.35 μM48-hColonNone
6068
307896952019
IKLSPS5TKKS5LKKVLKGS5IKGS5IAVAKMV
H-2029CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 4.93 ± 0.53 μM48-hLiverNone
6067
307896952019
IKLSPS5TKKS5LKKVLKGS5IKGS5IAVAKMV
H-2029CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 2.63 ± 0.35 μM48-hColonNone
6066
307896952019
IKLSPS5TKKS5LKKVLKGS5IKGS5IAVAKMV
H-2029CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 2.10 ± 0.32 μM48-hLungNone
6065
307896952019
IKLSKS5TKKS5LKKVLKGS5IKGS5IAVAKMV
H-2129CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 1.50 ± 0.28 μM48-hLiverNone
6063
307896952019
IKLSKS5TKKS5LKKVLKGS5IKGS5IAVAKMV
H-2129CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 3.26 ± 0.36 μM48-hLungNone
6064
307896952019
IKLSKS5TKKS5LKKVLKGS5IKGS5IAVAKMV
H-2129CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 3.05 ± 0.21 μM48-hColonNone
6062
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-5729CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 2.13 ± 0.07 μM48-hLiverNone
6061
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-5729CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 1.29 ± 0.08 μM48-hColonNone
6060
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-5729CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 0.62 ± 0.12 μM48-hLungNone
6058
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-5829CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 1.29 ± 0.08 μM48-hColonNone
6059
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-5829CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 2.13 ± 0.07 μM48-hLiverNone
6057
307896952019
IKLSKKTKKNLKKVLKGS5IKGS5IAVAKMV
H-5829CyclicLS5 = (S)-N-Fmoc-2-(4′-pentenyl)alanineAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 0.62 ± 0.12 μM48-hLungNone
6056
307896952019
IKLSKETKDNLKKVLKGAIKGAIAVAKMV
[P5K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 4.28 ± 0.38 μM48-hLiverNone
6055
307896952019
IKLSKETKDNLKKVLKGAIKGAIAVAKMV
[P5K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 8.09 ± 0.40 μM48-hColonNone
6054
307896952019
IKLSKETKDNLKKVLKGAIKGAIAVAKMV
[P5K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 2.35 ± 0.31 μM48-hLungNone
6053
307896952019
IKLSPETKKNLKKVLKGAIKGAIAVAKMV
[D9K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 4.96 ± 0.43 μM48-hLiverNone
6052
307896952019
IKLSPETKKNLKKVLKGAIKGAIAVAKMV
[D9K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 6.50 ± 0.32 μM48-hColonNone
6051
307896952019
IKLSPETKKNLKKVLKGAIKGAIAVAKMV
[D9K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 1.82 ± 0.23 μM48-hLungNone
6050
307896952019
IKLSKETKKNLKKVLKGAIKGAIAVAKMV
[P5K,D9K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 2.46 ± 0.32 μM48-hLiverNone
6049
307896952019
IKLSKETKKNLKKVLKGAIKGAIAVAKMV
[P5K,D9K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticHCT-116Colon CancerMTT assayIC50 = 4.93 ± 0.51 μM48-hColonNone
6048
307896952019
IKLSKETKKNLKKVLKGAIKGAIAVAKMV
[P5K,D9K]Hymenochirin-1B29LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 1.17 ± 0.23 μM48-hLungNone
6047
316353882019
GLWSKIKKAAKTAGKAALGFVNKMV
K8, 23-DPT925LinearLNoneAmidationFreeAntimicrobialSyntheticPANC-1Pancreatic CancerMTT assayIC50 = 11.17 µM24-hPancreasNone
6046
316353882019
GLWSKIKKAAKTAGKAALGFVNKMV
K8, 23-DPT925LinearLNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 9.97 µM24-hProstateNone
6045
316353882019
GLWSKIKKAAKTAGKAALGFVNKMV
K8, 23-DPT925LinearLNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 9.88 µM24-hLungNone
6044
316353882019
GLWSKIKKAAKTAGKAALGFVNKMV
K8, 23-DPT925LinearLNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 18.51 µM24-hBrainNone
6043
316353882019
GLWSKIKKAAKTAGKAALGFVNKMV
K8, 23-DPT925LinearLNoneAmidationFreeAntimicrobialSyntheticMCF-7Breast CancerMTT assayIC50 = 8.64 µM24-hBreastNone
6042
316353882019
GLWSKIKDAAKTAGKAALGFVNEMV
Dermaseptin-PT925LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tarsiusPANC-1Pancreatic CancerMTT assayIC50 = 28.95 µM24-hPancreasNone
6041
316353882019
GLWSKIKDAAKTAGKAALGFVNEMV
Dermaseptin-PT925LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tarsiusPC-3Prostate CancerMTT assayIC50 = 21.78 µM24-hProstateNone
6040
316353882019
GLWSKIKDAAKTAGKAALGFVNEMV
Dermaseptin-PT925LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tarsiusH-157Lung CancerMTT assayIC50 = 25.51 µM24-hLungNone
6039
316353882019
GLWSKIKDAAKTAGKAALGFVNEMV
Dermaseptin-PT925LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tarsiusU251-MGBrain TumorMTT assayIC50 = 49.51 µM24-hBrainNone
6038
316353882019
GLWSKIKDAAKTAGKAALGFVNEMV
Dermaseptin-PT925LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tarsiusMCF-7Breast CancerMTT assayIC50 = 7.44 µM24-hBreastNone
6026
290434942018
KILRGVCKKIMRpFLRRISKDILTGKK
NK-pro27LinearMixNoneAmidatedFreeAntimicrobialSynthetic analog of NK-2HL-60Leukemia CancerMTT assayIC50 = 26.1 μM24-hBloodNone
6025
290434942018
KILRGVCKKIMRpFLRRISKDILTGKK
NK-pro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2T-24Bladder CancerMTT assayIC50 = 33.0 μM24-hBladderNone
6024
290434942018
KILRGVCKKIMRpFLRRISKDILTGKK
NK-pro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2EJBladder CancerMTT assayIC50 = 23.3 μM24-hBladderNone
6023
290434942018
KILRGVCKKIMRpFLRRISKDILTGKK
NK-pro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2PC-3Prostate CancerMTT assayIC50 = 9.3 μM24-hProstateNone
6022
290434942018
KILpGVCKKIMRpFLRRISKDILTGKK
NK-dpro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2HL-60Leukemia CancerMTT assayIC50 = 48.4 μM24-hBloodNone
6021
290434942018
KILpGVCKKIMRpFLRRISKDILTGKK
NK-dpro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2T-24Bladder CancerMTT assayIC50 = 39.6 μM24-hBladderNone
6020
290434942018
KILpGVCKKIMRpFLRRISKDILTGKK
NK-dpro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2EJBladder CancerMTT assayIC50 = 28.7 μM24-hBladderNone
6019
290434942018
KILpGVCKKIMRpFLRRISKDILTGKK
NK-dpro27LinearMixNoneAmidationFreeAntimicrobialSynthetic analog of NK-2PC-3Prostate CancerMTT assayIC50 = 9.6 μM24-hProstateNone
6018
301833072018
RGWFRAMRSIARFIARERLREHL
R-C1623LinearLNoneAmidationFatty acid :C16H31OAnticancerR-Lycosin-IA-549Lung CancerCCK-8 assayIC50 ~ 5 µM24-hLungNone
5984
296674782018
ytrdlvygdparpgiqgtgtf
D-FP21-PEG-PEI/pGRO-α21LinearDconjugated to polyethylenimine (PEI) and methoxy polyethylene glycol (mPEG)FreeFreeAnti-caner, anti-proliferative, anti-tumorSyntheticHO-8910Ovarian CancerCCK-8 assayIC50 = 21.6 μg/mL24-hOvaryNone
5983
296674782018
YTRDLVYGDPARPGIQGTGTF
L-FP21-PEG-PEI/pGRO-α21LinearLconjugated to polyethylenimine (PEI) and methoxy polyethylene glycol (mPEG)FreeFreeAnti-caner, anti-proliferative, anti-tumorSyntheticHO-8910Ovarian CancerCCK-8 assayIC50 = 23.4 μg/mL24-hOvaryNone
5974
297576462018
GIPCGESCVWIPCISSAIGCSCKNKVCYRN
CyO430CyclicLNoneCyclizedCyclizedAntimicrobial,CytotoxicViola odorataMDA-MB-231Breast CancerMTS assayIC50 = 9.8 μM24-hBreastNone
5973
297576462018
GIPCAESCVFIPCVTAILGCSCKDVCYN
Poca B28CyclicLNoneCyclizedCyclizedAntimicrobial,CytotoxicPombalia calceolariaMDA-MB-231Breast CancerMTS assayIC50 = 2.7 μM24-hBreastNone
5972
297576462018
GLPCAESCVFIPCTITAILGCSCRDRVCYD
Poca A30CyclicLNoneCyclizedCyclizedAntimicrobial,CytotoxicPombalia calceolariaMDA-MB-231Breast CancerMTS assayIC50 = 1.8 μM24-hBreastNone
5971
293013082018
FIHHIIGGLFSAGKAIHRLIRRRRR
MSP-425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusMG-63Bone CancerMTT assayCell viability = 26.78 ± 1.75% at 10 µM24-hBoneNone
5970
301239402018
Ahx-(KAVPIAQKE)GG(KRRRRRRRRE)
SmacN7-Arg8 fused peptide P722CyclicLAhx = aminohexanoic acid; Lactam Bridge between K2 and E10 and between K13 and E22AmidationFreeAnticancerSyntheticU-266Skin CancerCell Titer Blue Cell Viability assayCell viability < 50% at 50 μM48-hSkinNone
5963
298007252018
GIGAVLKKLTTGLKALISWIKRKRQQ
MEL-Pep26LinearLNoneAmidationFreeAnticancerSynthetic analog of MelittinBEL-7402/5-FULiver CancerCCK-8 assayIC50 = 4.36 μM24-hLiverNone
5943
299931852018
NDADKDEMQSVYRGKANDDNSRGSKTNHRF
Peptide10 Gonearrestide30LinearLNoneFreeFreeAnticancerAndroctonus mauritanicusU-251Brain tumorMTT assayNot Available24-hBrainNone
5942
299931852018
NDADKDEMQSVYRGKANDDNSRGSKTNHRF
Peptide10 Gonearrestide30LinearLNoneFreeFreeAnticancerAndroctonus mauritanicusDks8Colon CancerMTT assayNot Available24-hColonNone
5941
299931852018
NDADKDEMQSVYRGKANDDNSRGSKTNHRF
Peptide10 Gonearrestide30LinearLNoneFreeFreeAnticancerAndroctonus mauritanicusHKe-3Colon CancerMTT assayNot Available24-hColonNone
5940
299931852018
NDADKDEMQSVYRGKANDDNSRGSKTNHRF
Peptide10 Gonearrestide30LinearLNoneFreeFreeAnticancerAndroctonus mauritanicusDLD-1Colon CancerMTT assayNot Available24-hColonNone
5939
299931852018
NDADKDEMQSVYRGKANDDNSRGSKTNHRF
Peptide10 Gonearrestide30LinearLNoneFreeFreeAnticancerAndroctonus mauritanicusHCT-116Colon CancerMTT assayNot Available24-hColonNone
5918
302792102018
GIMDTVKNAAKNLAGQLLDKLK
R2PLx-2222LinearLNoneFreeFreeAntimicrobialSyntheticMCF-7Breast CancerMTT assayIC50 = 109.30 µM24-hBreastNone
5917
302792102018
GIMDTVKNAAKNLAGQLLDKLK
R2PLx-2222LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxU-251-MGBrain TumorMTT assayIC50 = 104.10 µM24-hBrainNone
5916
302792102018
GIMDTVKNAAKNLAGQLLDKLK
R2PLx-2222LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxPC-3Prostate CancerMTT assayIC50 = 283.90 µM24-hProstateNone
5914
302792102018
GIMDTVKNAAKNLAGQLLDKLK
R2PLx-2222LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxH-157Lung CancerMTT assayIC50 = 843.40 µM24-hLungNone
5915
302792102018
GIMDTVKNAAKNLAGQLLDKLK
R2PLx-2222LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxMDA-MB-435SSkin CancerMTT assayIC50 = 872.70 µM24-hSkinNone
5913
302792102018
GIMDTVKNAAKNLAGQLLDKLKCKITAC
Ranatuerin-2PLx28LinearLNoneFreeFreeAntimicrobialRana palustrisMCF-7Breast CancerMTT assayIC50 = 20.19 µM24-hBreastNone
5912
302792102018
GIMDTVKNAAKNLAGQLLDKLKCKITAC
Ranatuerin-2PLx28LinearLNoneFreeFreeAntimicrobialRana palustrisU-251-MGBrain TumorMTT assayIC50 = 16.14 µM24-hBrainNone
5911
302792102018
GIMDTVKNAAKNLAGQLLDKLKCKITAC
Ranatuerin-2PLx28LinearLNoneFreeFreeAntimicrobialRana palustrisPC-3Prostate CancerMTT assayIC50 = 5.79 µM24-hProstateNone
5910
302792102018
GIMDTVKNAAKNLAGQLLDKLKCKITAC
Ranatuerin-2PLx28LinearLNoneFreeFreeAntimicrobialRana palustrisMDA-MB-435SSkin CancerMTT assayIC50 = 15.44 µM24-hSkinNone
5909
302792102018
GIMDTVKNAAKNLAGQLLDKLKCKITAC
Ranatuerin-2PLx28LinearLNoneFreeFreeAntimicrobialRana palustrisH-157Lung CancerMTT assayIC50 = 5.90 µM24-hLungNone
5908
302792102018
GIMDTVKNAAKNLAGQLLDKLKCSITAC
S-24-R2PLx28LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxMCF-7Breast CancerMTT assayIC50 = 316.90 µM24-hBreastNone
5907
302792102018
GIMDTVKNAAKNLAGQLLDKLKCSITAC
S-24-R2PLx28LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxU-251-MGBrain TumorMTT assayIC50 = 278.30 µM24-hBrainNone
5906
302792102018
GIMDTVKNAAKNLAGQLLDKLKCSITAC
S-24-R2PLx28LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxMDA-MB-435SSkin CancerMTT assayIC50 = 179.00 µM24-hSkinNone
5905
302792102018
GIMDTVKNAAKNLAGQLLDKLKCSITAC
S-24-R2PLx28LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxH-157Lung CancerMTT assayIC50 = 58.18 µM24-hLungNone
5904
302792102018
GIMDTVKNAAKNLAGQLLDKLKCSITAC
S-24-R2PLx28LinearLNoneFreeFreeAntimicrobialSynthetic Analogue of Ranatuerin-2PLxPC-3Prostate CancerMTT assayIC50 = 792.60 µM24-hProstateNone
5885
300261682018
FLSGIVGMLaKLFLFKQYAELW
[G10a]SHa-BCTP22LinearMixNoneAmidationFreeAntimicrobialSynthetic analogue of Temporin-1SHaNCI-H-460Lung CancerMTT assayIC50 >100 µM24-hLungNone
5884
300261682018
FLSGIVGMLaKLFLFKQYAELW
[G10a]SHa-BCTP22LinearMixNoneAmidationFreeAntimicrobialSynthetic analogue of Temporin-1SHaHeLaCervical CancerMTT assayIC50 >100 µM24-hCervixNone
5883
300261682018
FLSGIVGMLaKLFLFKQYAELW
[G10a]SHa-BCTP22LinearMixNoneAmidationFreeAntimicrobialSynthetic analogue of Temporin-1SHaMCF-7Breast CancerMTT assayIC50 = 26.85 ± 1.85 µM24-hBreastNone
5876
299042742018
RKKRRQRRRLNLKALLAVAKKIL
tMP-C23LinearLNoneAmidationFreeAntimicrobialSyntheticU-251-MGBrain tumorMTT assayIC50 = 3.36 μM24-hBrainNone
5877
299042742018
RKKRRQRRRLNLKALLAVAKKIL
tMP-C23LinearLNoneAmidationFreeAntimicrobialSyntheticMCF-7Breast CancerMTT assayIC50 = 3.70 μM24-hBreastNone
5874
299042742018
RKKRRQRRRLNLKALLAVAKKIL
tMP-C23LinearLNoneAmidationFreeAntimicrobialSyntheticMDA-MB-435SSkin CancerMTT assayIC50 = 3.86 μM24-hSkinNone
5875
299042742018
RKKRRQRRRLNLKALLAVAKKIL
tMP-C23LinearLNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 3.86 μM24-hProstateNone
5873
299042742018
RKKRRQRRRLNLKALLAVAKKIL
tMP-C23LinearLNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 2.79 μM24-hLungNone
5861
300872682018
ALWKDILKNLLKAALNEINQIVQ
L10, 11-DPS323LinearLNoneAmidationFreeAntimicrobial and AnticancerAnalogue of Dermaseptin-PS3H-157Lung CancerMTT assayIC50 = 0.12 μMNot AvailableLungNone
5862
300872682018
ALWKDILKNLLKAALNEINQIVQ
L10, 11-DPS323LinearLNoneAmidationFreeAntimicrobial and AnticancerAnalogue of Dermaseptin-PS3PC-3Prostate CancerMTT assayIC50 = 1.85 μMNot AvailableProstateNone
5859
300872682018
ALWKKILKNAGKAALNKINQIVQ
K5, 17-DPS323LinearLNoneAmidationFreeAntimicrobial and AnticancerAnalogue of Dermaseptin-PS3H-157Lung CancerMTT assayIC50 = 18.20 μMNot AvailableLungNone
5860
300872682018
ALWKKILKNAGKAALNKINQIVQ
K5, 17-DPS323LinearLNoneAmidationFreeAntimicrobial and AnticancerAnalogue of Dermaseptin-PS3PC-3Prostate CancerMTT assayIC50 = 18.20 μMNot AvailableProstateNone
5857
300872682018
ALWKDILKNAGKAALNEINQIVQ
Dermaseptin-PS323LinearLNoneAmidationFreeAntimicrobial and AnticancerPhyllomedusa sauvagiiH-157Lung CancerMTT assayIC50 = 15.67 μMNot AvailableLungNone
5858
300872682018
ALWKDILKNAGKAALNEINQIVQ
Dermaseptin-PS323LinearLNoneAmidationFreeAntimicrobial and AnticancerPhyllomedusa sauvagiiPC-3Prostate CancerMTT assayIC50 = 18.20 μMNot AvailableProstateNone
5855
302587242018
GRKKRRQRRRGALWKSLLKNVGKA
DP-224LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticH-157Lung CancerMTT assayIC50 = 3.21 μM24-hLungNone
5856
302587242018
GRKKRRQRRRGALWKSLLKNVGKA
DP-224LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticPC-3Prostate CancerMTT assayIC50 = 6.75 μM24-hProstateNone
5854
302587242018
ALWKSLLKNVGKAAGKAALNAVTDMVNQ
DRS-DU-128LinearLNoneAmidationFreeAntimicrobial and AnticancerCallimedusa (Phyllomedusa) duellmaniPC-3Prostate CancerMTT assayIC50 = 21.6 μM24-hProstateNone
5852
291916582018
FLPIVAKLLSGLLGRKKRRQRRR
temporin-PEb23LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of Temporin-PEMDA-MB-435SSkin CancerMTT assayIC50 = 3.483 μMNot AvailableSkinNone
5853
302587242018
ALWKSLLKNVGKAAGKAALNAVTDMVNQ
DRS-DU-128LinearLNoneAmidationFreeAntimicrobial and AnticancerCallimedusa (Phyllomedusa) duellmaniH-157Lung CancerMTT assayIC50 = 8.43 μM24-hLungNone
5850
291916582018
FLPIVAKLLSGLLGRKKRRQRRR
temporin-PEb23LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of Temporin-PEU251-MGBrain TumorMTT assayIC50 = 3.087 μMNot AvailableBrainNone
5851
291916582018
FLPIVAKLLSGLLGRKKRRQRRR
temporin-PEb23LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of Temporin-PEPC-3Prostate CancerMTT assayIC50 = 3.051 μMNot AvailableProstateNone
5849
291916582018
FLPIVAKLLSGLLGRKKRRQRRR
temporin-PEb23LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic analog of Temporin-PENCI-H-157Lung CancerMTT assayIC50 = 3.464 μMNot AvailableLungNone
5840
286367812018
GIGGALLSAGKSALKGLAKGLAEHFAN
BLP-727LinearLNoneAmidationFreeAntimicrobialBombina orientaliA-375Skin CancerMTT assayCell Viability < 20% at 10 μM48-hSkinNone
5839
286367812018
GIGGALLSAGKSALKGLAKGLAEHFAN
BLP-727LinearLNoneAmidationFreeAntimicrobialBombina orientaliA-549Lung CancerMTT assayCell Viability ~ 20% at 2.5 μM48-hLungNone
5838
286367812018
GIGGALLSAGKSALKGLAKGLAEHFAN
BLP-727LinearLNoneAmidationFreeAntimicrobialBombina orientaliPC-3Prostate CancerMTT assayCell Viability ~ 20% at 2.5 μM48-hProstateNone
5837
286367812018
GIGGALLSAGKSALKGLAKGLAEHFAN
BLP-727LinearLNoneAmidationFreeAntimicrobialBombina orientaliHuh-7Liver CancerMTT assayIC50 = 1.81 μM48-hLiverNone
5836
286367812018
GIGGALLSAGKSALKGLAKGLAEHFAN
BLP-727LinearLNoneAmidationFreeAntimicrobialBombina orientaliHepG-2Liver CancerMTT assayIC50 = 2.83 μM48-hLiverNone
5835
286367812018
GIGGALLSAGKSALKGLAKGLAEHFAN
BLP-727LinearLNoneAmidationFreeAntimicrobialBombina orientaliSK-HEP-1Liver CancerMTT assayIC50 = 0.61 μM48-hLiverNone
5828
306224712018
GRFKRFRKKLKRLWHKVGPFVGPILHY
ChMAP-2827LinearLNoneFreeFreeAntimicrobialleucocytes of the goat Capra hircusB16-F10Skin CancerMTT assayIC50 = 4.82 ± 1.01 μM48-hSkinNone
5827
306224712018
GRFKRFRKKLKRLWHKVGPFVGPILHY
ChMAP-2827LinearLNoneFreeFreeAntimicrobialleucocytes of the goat Capra hircusSK-BR-3Breast CancerMTT assayIC50 = 5.63 ± 1.05 μM48-hBreastNone
5826
306224712018
GRFKRFRKKLKRLWHKVGPFVGPILHY
ChMAP-2827LinearLNoneFreeFreeAntimicrobialleucocytes of the goat Capra hircusHEK-293TRenal CancerMTT assayIC50 = 5.09 ± 0.40 μM48-hRenalNone
5825
306224712018
GRFKRFRKKLKRLWHKVGPFVGPILHY
ChMAP-2827LinearLNoneFreeFreeAntimicrobialleucocytes of the goat Capra hircusA-431Skin CancerMTT assayIC50 = 6.49 ± 0.09 μM48-hSkinNone
5824
306224712018
GRFKRFRKKLKRLWHKVGPFVGPILHY
ChMAP-2927LinearLNoneFreeFreeAntimicrobialleucocytes of the goat Capra hircusHL-60Leukemia CancerLDH leakage assay~60% LDH Release at 2.5 μM1-hBloodNone
5823
306224712018
GRFKRFRKKLKRLWHKVGPFVGPILHY
ChMAP-2827LinearLNoneFreeFreeAntimicrobialleucocytes of the goat Capra hircusHL-60Leukemia CancerMTT assayIC50 = 3.39 ± 0.15 μM48-hBloodNone
5808
290984062018
GIGSAILSAGKSIIKGLAKGLAEHF
Bombinin-BO125LinearLNoneAmidationFreeAntimicrobialBombina orientalisHuh-7Liver CancerMTT assayIC50 = 3.91 μM48-hLiverNone
5807
290984062018
GIGSAILSAGKSIIKGLAKGLAEHF
Bombinin-BO125LinearLNoneAmidationFreeAntimicrobialBombina orientalisHepG-2Liver CancerMTT assayIC50 = 3.75 μM48-hLiverNone
5806
290984062018
GIGSAILSAGKSIIKGLAKGLAEHF
Bombinin-BO125LinearLNoneAmidationFreeAntimicrobialBombina orientalisSK-HEP-1Liver CancerMTT assayIC50 = 0.76 μM48-hLiverNone
5720
292639232017
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSynthetic4T1Breast CancerCCK-8 assay49% cell viability at 100 μM24-hBreastNone
5713
None2017
VLLVTLTRLHQRGVIYEKWRHFSGRKYR
VLL-2828LinearLNoneFreeAcetylationAntibacterial and AnticancerSulfolobus islandicusHEK-293TRenal CancerMTT assayIC50 = 10 μM72-hRenalNone
5705
292809482017
KWKSFLKTfKSaKKTvLHTALKAISS
F9D/A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 125.0 ± 1.8 μM24-hPancreasNone
5704
292809482017
KWKSFLKTfKSaKKTvLHTALKAISS
F9D/A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 95.6 ± 1.8 μM24-hPancreasNone
5703
292809482017
KWKSFLKTfKSaKKTvLHTALKAISS
F9D/A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 57.9 ± 2.8 μM24-hPancreasNone
5702
292809482017
KWKSFLKTfKSaKKTvLHTALKAISS
F9D/A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 125.0 ± 3.4 μM24-hCervixNone
5701
292809482017
KWKSFLKTFKSaKKTvLHTALKAISS
A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 125.0 ± 5.9 μM24-hPancreasNone
5700
292809482017
KWKSFLKTFKSaKKTvLHTALKAISS
A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 41.4 ± 1.4 μM24-hPancreasNone
5699
292809482017
KWKSFLKTFKSaKKTvLHTALKAISS
A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 46.2 ± 3.0 μM24-hPancreasNone
5698
292809482017
KWKSFLKTFKSaKKTvLHTALKAISS
A12D/V16D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 60.1 ± 1.2 μM24-hCervixNone
5697
292809482017
KWKSFLKTfKSaKKTVLHTALKAISS
F9D/A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 125.0 ± 3.7 μM24-hPancreasNone
5696
292809482017
KWKSFLKTfKSaKKTVLHTALKAISS
F9D/A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 42.4 ± 3.0 μM24-hPancreasNone
5695
292809482017
KWKSFLKTfKSaKKTVLHTALKAISS
F9D/A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 38.8 ± 2.9 μM24-hPancreasNone
5694
292809482017
KWKSFLKTfKSaKKTVLHTALKAISS
F9D/A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 59.8 ± 0.5 μM24-hCervixNone
5693
292809482017
KWKSFLKTFKSaKKTVLHTALKAISS
A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 45.1 ± 1.0 μM24-hPancreasNone
5692
292809482017
KWKSFLKTFKSaKKTVLHTALKAISS
A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 15.5 ± 1.7 μM24-hPancreasNone
5691
292809482017
KWKSFLKTFKSaKKTVLHTALKAISS
A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 29.9 ± 4.8 μM24-hPancreasNone
5690
292809482017
KWKSFLKTFKSaKKTVLHTALKAISS
A12D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 28.8 ± 0.8 μM24-hCervixNone
5689
292809482017
KWKSFLKTFKsAKktVLHTALKAISS
S11D/K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 45.5 ± 5.6 μM24-hPancreasNone
5688
292809482017
KWKSFLKTFKsAKktVLHTALKAISS
S11D/K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 54.2 ± 1.2 μM24-hPancreasNone
5687
292809482017
KWKSFLKTFKsAKktVLHTALKAISS
S11D/K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 56.8 ± 3.3 μM24-hPancreasNone
5686
292809482017
KWKSFLKTFKsAKktVLHTALKAISS
S11D/K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 41.1 ± 0.5 μM24-hCervixNone
5685
292809482017
KWKSFLKTFKSAKktVLHTALKAISS
K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 24.1 ± 5.5 μM24-hPancreasNone
5684
292809482017
KWKSFLKTFKSAKktVLHTALKAISS
K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 22.5 ± 0.5 μM24-hPancreasNone
5683
292809482017
KWKSFLKTFKSAKktVLHTALKAISS
K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 47.1 ± 5.3 μM24-hPancreasNone
5682
292809482017
KWKSFLKTFKSAKktVLHTALKAISS
K14D/T15D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 31.6 ± 2.1 μM24-hCervixNone
5681
292809482017
KWKSFLKTFKsAKkTVLHTALKAISS
S11D/K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 22.4 ± 2.3 μM24-hPancreasNone
5680
292809482017
KWKSFLKTFKsAKkTVLHTALKAISS
S11D/K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 25.5 ± 0.5 μM24-hPancreasNone
5679
292809482017
KWKSFLKTFKsAKkTVLHTALKAISS
S11D/K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 41.3 ± 2.6 μM24-hPancreasNone
5678
292809482017
KWKSFLKTFKsAKkTVLHTALKAISS
S11D/K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 30.6 ± 0.5 μM24-hCervixNone
5677
292809482017
KWKSFLKTFKSAKkTVLHTALKAISS
K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KBxPC-3Pancreatic CancerMTT assayIC50 = 20.0 ± 0.8 μM24-hPancreasNone
5676
292809482017
KWKSFLKTFKSAKkTVLHTALKAISS
K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHPACPancreatic CancerMTT assayIC50 = 7.2 ± 5.2 μM24-hPancreasNone
5675
292809482017
KWKSFLKTFKSAKkTVLHTALKAISS
K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KMIA PaCa-2Pancreatic CancerMTT assayIC50 = 17.9 ± 2.3 μM24-hPancreasNone
5674
292809482017
KWKSFLKTFKSAKkTVLHTALKAISS
K14D26LinearMixNoneAmidationAcetylationAntimicrobial and AnticancerSynthetic Analogue of V13KHeLaCervical CancerMTT assayIC50 = 15.6 ± 4.1 μM24-hCervixNone
5673
292809482017
KWKSFLKTFKSAKKTVLHTALKAISS
V13K26LinearLNoneAmidationAcetylationAntimicrobial and AnticancerSyntheticBxPC-3Pancreatic CancerMTT assayIC50 = 12.5 ± 1.2 μM24-hPancreasNone
5672
292809482017
KWKSFLKTFKSAKKTVLHTALKAISS
V13K26LinearLNoneAmidationAcetylationAntimicrobial and AnticancerSyntheticHPACPancreatic CancerMTT assayIC50 = 7.6 ± 4.0 μM24-hPancreasNone
5671
292809482017
KWKSFLKTFKSAKKTVLHTALKAISS
V13K26LinearLNoneAmidationAcetylationAntimicrobial and AnticancerSyntheticMIA PaCa-2Pancreatic CancerMTT assayIC50 = 24.8 ± 0.6 μM24-hPancreasNone
5670
292809482017
KWKSFLKTFKSAKKTVLHTALKAISS
V13K26LinearLNoneAmidationAcetylationAntimicrobial and AnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 16 ± 0.5 μM24-hCervixNone
5593
None2017
CKLKNFAKGVAQSLLNKASKLSGQC
BR-C25CyclicLNoneCyclizedCyclizedAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 75.44 μg/ml24-hLungNone
5592
None2017
CKLKNFAKGVAQSLLNKASKLSGQC
BR-C25CyclicLNoneCyclizedCyclizedAntimicrobialSyntheticMCF-7Breast CancerMTT assayIC50 = 45.72 μg/ml24-hBreastNone
5590
None2017
KlKNFAKGVAQSllNKASCKlSGQC
BR-D25LinearMixNoneFreeFreeAntimicrobialSyntheticMCF-7Breast CancerMTT assayIC50 = 67.52 μg/ml24-hBreastNone
5591
None2017
KlKNFAKGVAQSllNKASCKlSGQC
BR-D25LinearMixNoneFreeFreeAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 94.74 μg/ml24-hLungNone
5589
290644022017
ALWKEVLKNAGKAALNEINNLV
Dermaseptin-PH22LinearLNoneAmidationFreeAntimicrobial and AnticancerPithecopus (Phyllomedusa) hypochondrialisPC-3Prostate CancerMTT assayIC50 = 11.8 μMNot AvailableProstateNone
5588
290644022017
ALWKEVLKNAGKAALNEINNLV
Dermaseptin-PH22LinearLNoneAmidationFreeAntimicrobial and AnticancerPithecopus (Phyllomedusa) hypochondrialisMDA-MB-435SBreast CancerMTT assayIC50 = 9.94 μMNot AvailableBreastNone
5587
290644022017
ALWKEVLKNAGKAALNEINNLV
Dermaseptin-PH22LinearLNoneAmidationFreeAntimicrobial and AnticancerPithecopus (Phyllomedusa) hypochondrialisU251-MGBrain TumorMTT assayIC50 = 2.36 μMNot AvailableBrainNone
5586
290644022017
ALWKEVLKNAGKAALNEINNLV
Dermaseptin-PH22LinearLNoneAmidationFreeAntimicrobial and AnticancerPithecopus (Phyllomedusa) hypochondrialisH-157Lung CancerMTT assayIC50 = 2.01 μMNot AvailableLungNone
5585
290644022017
ALWKEVLKNAGKAALNEINNLV
Dermaseptin-PH22LinearLNoneAmidationFreeAntimicrobial and AnticancerPithecopus (Phyllomedusa) hypochondrialisMCF-7Breast CancerMTT assayIC50 = 0.69 μMNot AvailableBreastNone
5301
272481702016
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusMDA-MB-231Breast CancerLDH leakage assayLDH activity = 1.5mU/mL at 10 μg/mL3-hBreastNone
5300
272481702016
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusMCF-7Breast CancerMTS assayIC50 = 5.03 μM6-hBreastNone
5299
272481702016
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusMDA-MB-453Breast CancerMTS assayIC50 = 5.03 μM6-hBreastNone
5298
272481702016
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusMDA-MB-231Breast CancerMTS assayIC50 = 5.03 μM6-hBreastNone
5270
None2015
CQYSVNPKIKRFELYFKGRMW
LPSBD-021LinearLNoneFreeFreeAnticancerSyntheticHep3BLiver CancerCell Proliferation assay~40% cell survival at 60 µg/ml24-hLiverNone
5269
None2015
CQYSVNPKIKRFELYFKGRMW
LPSBD-021LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerCell Proliferation assay~20% cell survival at 60 µg/ml24-hLungNone
5214
254475432015
ACYCRIPACIAGERRYGTCIYQGRLWAFCC
Human neutrophil peptide-1 (HNP-1)30Cyclic(C2-C30, C4-C19,C9-C29)LNoneFreeFreeAntimicrobialHomo sapiensPC-3Prostate CancerCytotoxicity assay (LIVE/DEAD® Viability/Cytotoxicity Assay Kit (L-3224))IC50 = 2.2 ± 0.3 μM4hProstateNone
5182
263227452015
GLPTCGETCFKGKCYTPGCSCSYPICKKD
Cyclotide mela-629CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusHeLaCervical CancerResazurin dye assayCC50 = 11.42 ±1.00 µMNot AvailableCervixNone
5181
263227452015
GLPTCGETCFKGKCYTPGCSCSYPICKKD
Cyclotide mela-629CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusMM96LSkin CancerResazurin dye assayCC50 = 1.58 ±0.48 µMNot AvailableSkinNone
5180
263994952015
GIPCGESCVFIPCLTSAIGCSCKSKVCYRN
Mra3030CyclicLNoneCyclizedCyclizedAntimicrobial and AnticancerViola tricolor, Melicytus ramiflorus, Viola philippicaBGC-823Gastric CancerResazurin dye assayIC50 = 1.75 ±0.05 µMNot AvailableStomachNone
5179
263994952015
GIPCGESCVFIPCLTSAIGCSCKSKVCYRN
Mra3030CyclicLNoneCyclizedCyclizedAntimicrobial and AnticancerViola tricolor, Melicytus ramiflorus, Viola philippicaHeLaCervical CancerResazurin dye assayIC50 = 15.5 ±0.06 µMNot AvailableCervixNone
5178
263994952015
GIPCGESCVFIPCLTSAIGCSCKSKVCYRN
Mra3030CyclicLNoneCyclizedCyclizedAntimicrobial and AnticancerViola tricolor, Melicytus ramiflorus, Viola philippicaMM96LSkin CancerResazurin dye assayIC50 = 4.91 ±0.04 µMNot AvailableSkinNone
5177
263227452015
GKPICGETCFKGKCYTPGCTCSYPICKKD
Mela329CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusHeLaCervical CancerResazurin dye assayCC50 = 18.73 ±1.82 µMNot AvailableCervixNone
5176
263227452015
GKPICGETCFKGKCYTPGCTCSYPICKKD
Mela329CyclicLNoneCyclizedCyclizedAntibacterial and AnticancerMelicytus latifoliusMM96LSkin CancerResazurin dye assayCC50 = 2.04 ±0.26 µMNot AvailableSkinNone
5162
267519702015
GLPLCGETCVGGTCNTPGCSCGWPVCVRN
Vigno 529Cyclic(C5-C19,C9-C21,C14-C21)LNoneFreeFreeAnticancerViola ignobilisHeLaCervical CancerMTT assay24% cell viability at 7.5 μM24-hCervixNone
5152
260643102015
GTSCGETCVLLPCLSSVLGCTCQNKRCYKD
DC330CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaDU-145Liver CancerCCK-8 assayIC50 = 0.55 μM72-hLiverNone
5151
260643102015
GTSCGETCVLLPCLSSVLGCTCQNKRCYKD
DC330CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaPC-3Prostate CancerCCK-8 assayIC50 = 0.76 μM72-hProstateNone
5150
260643102015
GTSCGETCVLLPCLSSVLGCTCQNKRCYKD
DC330CyclicLNoneCyclizedCyclizedAnticancerHedyotis diffusaLNCaPProstate CancerCCK-8 assayIC50 = 0.21 μM72-hProstateNone
5139
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 1.8 ± 0.02 μM24-hCervixNone
5138
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticB-16Skin CancerMTT assayIC50 = 3.9 ± 0.02 μM24-hSkinNone
5137
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 5.8 ± 0.36 μM24-hLiverNone
5136
264058062015
FKKLKKLFSKLWNWKRKKRRQRRR
HPRP-A1-TAT24LinearLNoneAmidationAcetylationAnticancerSyntheticSGC-7901Gastric cancerMTT assayIC50 = 4.8 ± 0.08 μM24-hStomachNone
5128
262395372015
FWQRRIRRWRRFWQRRIRRWRR
DIM-LF11-31822LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerMTS assayLC50 = 9.4 ± 0.5 μM24-hSkinNone
5127
262395372015
FWQRRIRRWRRFWQRRIRRWRR
DIM-LF11-31822LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerMTS assayLC50 = 9.3 ± 0.8 μM24-hSkinNone
5126
262395372015
FWQRRIRRWRRFWQRRIRRWRR
DIM-LF11-31822LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerPI uptake assayLC50 = 3.8 ± 0.5 μM8-hSkinNone
5125
262395372015
PFWRRRIRIRRRRIRIRRRWFP
R-DIM-LF11-33722LinearLNoneAmidationFreeHost Defence PeptideSyntheticSBcl2Skin CancerMTS assayLC50 = 5.0 ± 0.4 μM24-hSkinNone
5124
262395372015
PFWRRRIRIRRRRIRIRRRWFP
R-DIM-LF11-33722LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerMTS assayLC50 = 12.3 ± 1.3 μM24-hSkinNone
5123
262395372015
PFWRRRIRIRRRRIRIRRRWFP
R-DIM-LF11-33722LinearLNoneAmidationFreeHost Defence PeptideSyntheticA-375Skin CancerPI uptake assayLC50 = 3.5 ± 0.4 μM8-hSkinNone
5093
253122532014
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSyntheticU-937Leukemia CancerFITC-Annexin V/PI double staining and flow cytometry assay>20% apoptosis rate at 80 μM24-hBloodNone
5092
253122532014
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSyntheticHL-60Leukemia CancerFITC-Annexin V/PI double staining and flow cytometry assay>20% apoptosis rate at 80 μM24-hBloodNone
5091
253122532014
GGRSFFLLRRIQGCRFRNTVDD
E522LinearLNoneFreeFreeAnticancerSyntheticNB-4Leukemia CancerFITC-Annexin V/PI double staining and flow cytometry assay60% apoptosis rate at 80 μM24-hBloodNone
5054
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC107Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5053
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC107Colorectal CancerCell Viability assayCell viability >65% at 12.5μM approx24-hColonNone
5052
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC107Colorectal CancerCell Viability assayCell viability >50% at 12.5μM approx24-hColonNone
5051
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >85% at 12.5μM approx24-hColonNone
5050
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >80% at 12.5μM approx24-hColonNone
5049
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5048
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC113Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5047
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC113Colorectal CancerCell Viability assayCell viability >65% at 12.5μM approx24-hColonNone
5046
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC113Colorectal CancerCell Viability assayCell viability >80% at 12.5μM approx24-hColonNone
5045
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5044
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >60% at 12.5μM approx24-hColonNone
5043
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5042
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >85% at 12.5μM approx24-hColonNone
5041
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >80% at 12.5μM approx24-hColonNone
5040
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >45% at 12.5μM approx24-hColonNone
5039
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >70% at 12.5μM approx24-hColonNone
5038
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5037
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5036
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC18Colorectal CancerCell Viability assayCell viability >75% at 12.5μM approx24-hColonNone
5035
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC18Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5034
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC18Colorectal CancerCell Viability assayCell viability >55% at 12.5μM approx24-hColonNone
5033
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >50% at 12.5μM approx24-hColonNone
5032
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >40% at 12.5μM approx24-hColonNone
5031
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >40% at 12.5μM approx24-hColonNone
5030
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability =50% at 12.5μM approx.1-hColonNone
5029
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability =50% at 12.5μM approx.1-hColonNone
5028
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC32Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5027
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5026
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5025
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC60Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5024
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5023
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5022
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC40Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5021
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5020
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5019
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHROC24Colorectal CancerCell Viability assayCell viability >60% at 25μM approx1-hColonNone
5018
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A-Δ27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >50% at 12.5μM approx.1-hColonNone
5017
249629502014
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability =50% at 12.5μM approx.1-hColonNone
5016
249629502014
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntitumorNK-2 peptide based derivativesHCT-116Colorectal CancerCell Viability assayCell viability >50% at 25μM approx1-hColonNone
5011
246610242014
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneFreeFreeAntimicrobialMain component of honey bee venomSCC25Skin CancerCell Viability assay102.9 ± 4.1% cell growth inhibition at 1 µM24-hSkinNone
5005
245873502014
GIGKFLKKAKKFGKAFVKILKK
Pexiganan22LinearLNoneAmidationFreeAntimicrobialAnalog of magainin 2OVRCAR-3Ovarian CancerMTT/MTS assayLC50= 13 at 100 µM72-hOvaryNone
5003
245873502014
GIGKFLKKAKKFGKAFVKILKK
Pexiganan22LinearLNoneAmidationFreeAntimicrobialAnalog of magainin 2LNCaPProstate cancerMTT/MTS assayLC50= 6 at 100 µM72-hProstateNone
5001
245873502014
GIGKFLKKAKKFGKAFVKILKK
Pexiganan22LinearLNoneAmidationFreeAntimicrobialAnalog of magainin 2MCF-7Breast CancerMTT/MTS assayLC50= 8 at 100 µM72-hBreastNone
4674
152798992004
FRKSKEKIGKEFKRIVQRIKDFLRNLV
HCAP18(109-135)27LinearLNoneFreeFreeAntimicrobialhCAP18 synthetic peptideSAS-H1Oral CancerNot AvailableNot AvailableNot AvailableOral mucosaNone
4673
228851722012
GLFGKLIKKFARKAISYAVKKARGKH
ltc2aG11A26LinearLNoneFreeFreeAntimicrobialCentral Asian spider, Lachesana tarabaeviProstate tumor celllineProstate CancerLDH leakage assaygraph fig 8 ANot AvailableProstateNone
4672
228851722012
GLFGKLIKKFGRKAISYAVKKARGKH
Latarcin 2a26LinearLNoneFreeFreeAntimicrobialCentral Asian spider, Lachesana tarabaeviBreast tumor celllineBreast CancerLDH leakage assaygraph fig 8 ANot AvailableBreastNone
4607
124175872003
TRSSRAGLQWPVGRVHRLLRKGGC
BF2d24LinearLNoneAmidationFreeAntimicrobialSyntheticHeLaCervical CancerMTT/MTS assayat 100 µM 90-100% viablity6-hCervixNone
4605
124175872003
TRSSRAGLQWPVGRVHRLLRKGGC
BF2d24LinearLNoneAmidationFreeAntimicrobialSyntheticHeLaCervical CancerMTT/MTS assayat 10 µM 90-95% viablity6-hCervixNone
4603
124175872003
TRSSRAGLQWPVGRVHRLLRKGGC
BF2d24LinearLNoneAmidationFreeAntimicrobialSyntheticHeLaCervical CancerMTT/MTS assayat 1 µM 90-100% viablity6-hCervixNone
4602
124175872003
GIGKFLHSAKKWGKAFVGQIMNC
MG2d23LinearLNoneAmidationFreeAntimicrobialSyntheticHeLaCervical CancerMTT/MTS assayat 1 µM 90-100% viablity6-hCervixNone
4592
214039172011
TRSSRAGLQFPVGRVHRLLRK
Buforin 221LinearLNoneFreeFreeAntimicrobialBufo Bufo GargarizansU-937Lymphoma CancerMTT/MTS assayIC50 =90-95 µg/mlNot AvailableBloodNone
4575
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7-TX400Breast CancerMTT/MTS assay~5% cytotoxic at 50 µM24-hBreastNone
4574
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7-TX400Breast CancerMTT/MTS assay60-70% cytotoxic at 50 µM24-hBreastNone
4571
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7Breast CancerMTT/MTS assay70% cytotoxic at 50 µM24-hBreastNone
4572
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7Breast CancerMTT/MTS assay0% cytotoxic at 50 µM24-hBreastNone
4573
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7-TX400Breast CancerMTT/MTS assay60-70% cytotoxic at 50 µM24-hBreastNone
4567
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay~0% cytotoxic at 10 µM24-hBreastNone
4568
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay5-10% cytotoxic at 25 µM24-hBreastNone
4569
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay20% cytotoxic at 50 µM24-hBreastNone
4570
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMCF-7Breast CancerMTT/MTS assay70% cytotoxic at 50 µM24-hBreastNone
4564
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay5% cytotoxic at 25 µM24-hBreastNone
4565
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay10-15% cytotoxic at 50 µM24-hBreastNone
4566
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4561
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay15-20% cytotoxic at 50 µM24-hBreastNone
4562
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay~5% cytotoxic at 5 µM24-hBreastNone
4563
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay~5% cytotoxic at 10 µM24-hBreastNone
4559
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay10% cytotoxic at 10 µM24-hBreastNone
4560
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay10-15% cytotoxic at 25 µM24-hBreastNone
4557
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10-15% cytotoxic at 50 µM24-hBreastNone
4558
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay10% cytotoxic at 5 µM24-hBreastNone
4555
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay~0% cytotoxic at 10 µM24-hBreastNone
4556
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10% cytotoxic at 25 µM24-hBreastNone
4552
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay10% cytotoxic at 25 µM24-hBreastNone
4553
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay10-15% cytotoxic at 50 µM24-hBreastNone
4554
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4549
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay80-90% cytotoxic at 25 µM24-hBreastNone
4550
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay85-90% cytotoxic at 50 µM24-hBreastNone
4551
220237342011
GWRTLLKKAEVKTVGKLALKHYL
NRC-1323LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay~5% cytotoxic at 10 µM24-hBreastNone
4546
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay80-90% cytotoxic at 50 µM24-hBreastNone
4547
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay30-40% cytotoxic at 5 µM24-hBreastNone
4548
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay60-70% cytotoxic at 10 µM24-hBreastNone
4544
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay50% cytotoxic at 10 µM24-hBreastNone
4545
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay80% cytotoxic at 25 µM24-hBreastNone
4543
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay10% cytotoxic at 5 µM24-hBreastNone
4540
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay20% cytotoxic at 10 µM24-hBreastNone
4541
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay70-80% cytotoxic at 25 µM24-hBreastNone
4542
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay80-85% cytotoxic at 50 µM24-hBreastNone
4538
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay40-50% cytotoxic at 50 µM24-hBreastNone
4539
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4537
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay20% cytotoxic at 25 µM24-hBreastNone
4534
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay40-50% cytotoxic at 50 µM24-hBreastNone
4535
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4536
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10% cytotoxic at 10 µM24-hBreastNone
4532
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay5% cytotoxic at 10 µM24-hBreastNone
4533
220237342011
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay20-30% cytotoxic at 25 µM24-hBreastNone
4530
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay85-90% cytotoxic at 50 µM24-hBreastNone
4531
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0725LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay~0% cytotoxic at 5 µM24-hBreastNone
4528
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay40-50% cytotoxic at 10 µM24-hBreastNone
4529
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay80% cytotoxic at 25 µM24-hBreastNone
4525
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay60-70% cytotoxic at 25 µM24-hBreastNone
4526
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay80-85% cytotoxic at 50 µM24-hBreastNone
4527
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-family4T1Breast CancerMTT/MTS assay15-20% cytotoxic at 5 µM24-hBreastNone
4524
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay40-50% cytotoxic at 10 µM24-hBreastNone
4521
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay70% cytotoxic at 25 µM24-hBreastNone
4522
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay80-85% cytotoxic at 50 µM24-hBreastNone
4523
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-468Breast CancerMTT/MTS assay30% cytotoxic at 5 µM24-hBreastNone
4520
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay50% cytotoxic at 10 µM24-hBreastNone
4518
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay60% cytotoxic at 50 µM24-hBreastNone
4519
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familySKBR-3Breast CancerMTT/MTS assay30% cytotoxic at 5 µM24-hBreastNone
4517
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay30-35% cytotoxic at 25 µM24-hBreastNone
4515
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay5-10% cytotoxic at 5 µM24-hBreastNone
4516
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyT-47DBreast CancerMTT/MTS assay10% cytotoxic at 10 µM24-hBreastNone
4514
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay60% cytotoxic at 50 µM24-hBreastNone
4511
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay5% cytotoxic at 5 µM24-hBreastNone
4512
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay5% cytotoxic at 10 µM24-hBreastNone
4513
220237342011
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationBiotinylatedAntimicrobialPleurocidin-familyMDA-MB-231Breast CancerMTT/MTS assay30-35% cytotoxic at 25 µM24-hBreastNone
4504
220572782011
AAKKWAKAKWAKAKKWAKAA
Z1021LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4503
220572782011
AAWKWAWAKKWAKAKKWAKAA
Z921LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =13 µMNot AvailableColonNone
4501
220572782011
KAAKKAWKAAKKAWKAAKKAA
Z721LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =21 µMNot AvailableColonNone
4502
220572782011
AWKKWAKAWKWAKAKWWAKAA
Z821LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =23 µMNot AvailableColonNone
4500
220572782011
KWWKKAAKAAKKAAKAAKKWA
Z621LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =31 µMNot AvailableColonNone
4499
220572782011
KAAKKAWKWAKKAAKWAKKAA
Z521LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =67 µMNot AvailableColonNone
4498
220572782011
KAAKKAWKAAKKAAKWWKKAA
Z421LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 =173 µMNot AvailableColonNone
4497
220572782011
KAAKKAWKAWKKAAKAAWKKAA
Z321LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4496
220572782011
KAAKKWAKAWKKAAKAWKKAA
Z221LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4495
220572782011
KAAKKWAKAAKKWAKAWKKAA
Z121LinearLNoneFreeFreeAnticancerSyntheticHT-29Colon CancerMTT/MTS assayEC50 >211 µMNot AvailableColonNone
4494
220572782011
AAKKWAKAKWAKAKKWAKAA
Z1021LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 >211 µMNot AvailableBreastNone
4493
220572782011
AAWKWAWAKKWAKAKKWAKAA
Z921LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =16 µMNot AvailableBreastNone
4492
220572782011
AWKKWAKAWKWAKAKWWAKAA
Z821LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =14 µMNot AvailableBreastNone
4491
220572782011
KAAKKAWKAAKKAWKAAKKAA
Z721LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =15 µMNot AvailableBreastNone
4490
220572782011
KWWKKAAKAAKKAAKAAKKWA
Z621LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =16 µMNot AvailableBreastNone
4489
220572782011
KAAKKAWKWAKKAAKWAKKAA
Z521LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =28 µMNot AvailableBreastNone
4488
220572782011
KAAKKAWKAAKKAAKWWKKAA
Z421LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =68 µMNot AvailableBreastNone
4487
220572782011
KAAKKAWKAWKKAAKAAWKKAA
Z321LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =128 µMNot AvailableBreastNone
4486
220572782011
KAAKKWAKAWKKAAKAWKKAA
Z221LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =173 µMNot AvailableBreastNone
4485
220572782011
KAAKKWAKAAKKWAKAWKKAA
Z121LinearLNoneFreeFreeAnticancerSyntheticMT-1Breast CancerMTT/MTS assayEC50 =186 µMNot AvailableBreastNone
4484
220572782011
AAKKWAKAKWAKAKKWAKAA
Z1021LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4483
220572782011
AAWKWAWAKKWAKAKKWAKAA
Z921LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =9 µMNot AvailableSkinNone
4482
220572782011
AWKKWAKAWKWAKAKWWAKAA
Z821LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =19 µMNot AvailableSkinNone
4481
220572782011
KAAKKAWKAAKKAWKAAKKAA
Z721LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =15 µMNot AvailableSkinNone
4480
220572782011
KWWKKAAKAAKKAAKAAKKWA
Z621LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =17 µMNot AvailableSkinNone
4479
220572782011
KAAKKAWKWAKKAAKWAKKAA
Z521LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =42 µMNot AvailableSkinNone
4478
220572782011
KAAKKAWKAAKKAAKWWKKAA
Z421LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 =155 µMNot AvailableSkinNone
4477
220572782011
KAAKKAWKAWKKAAKAAWKKAA
Z321LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4476
220572782011
KAAKKWAKAWKKAAKAWKKAA
Z221LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4475
220572782011
KAAKKWAKAAKKAAKAWKKAA
Z121LinearLNoneFreeFreeAnticancerSyntheticMeth ASkin CancerMTT/MTS assayEC50 >211 µMNot AvailableSkinNone
4454
17067680, 189574412007
GIKCRFCCGCCTPGICGVCCRF
hepcidin TH1-522Not AvailableLNoneFreeFreeAnticancerTilapia, Oreochromis mossambicusNot AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4448
8245827, 189574411993
KSSAYSLQMGATAIKQVKKLFKKWGW
Plantaricin A26Not AvailableLNoneFreeFreeAntibacterialLactobacillus plantarumC11, WCFS1, V90Not AvailableColorectal CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4437
11713517, 189574412001
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 122Not AvailableLNoneFreeFreeAntibacterialHybrid striped bass (Morone saxatilis x M. chrysops)Not AvailableBreast CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4436
12581207, 189574412003
FFGWLIKGAIHAGKAIHGLIHRRRH
Chrysophsin-125Not AvailableLNoneFreeFreeAntibacterialRed sea bream,Chrysophrys majororPagrus majorNot AvailableBreast CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4433
12804591, 199232332003
AIGSILGALAKGLPTLISWIKNR
Prepromelittin-related peptide23Not AvailableLNoneFreeFreeAntibacterialRana tagoi [Tago frog]Not AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4432
4056036, 189574411985
DCYCRIPACIAGERRYGTCIYQGRLWAFCC
HNP-330Not AvailableLNoneFreeFreeAnticancerHomo sapiensNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4431
4056036, 189574411985
CYCRIPACIAGERRYGTCIYQGRLWAFCC
HNP-229Not AvailableLNoneFreeFreeAnticancerHomo sapiensNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4430
4056036, 189574411985
ACYCRIPACIAGERRYGTCIYQGRLWAFCC
HNP-130Not AvailableLNoneFreeFreeAnticancerHomo sapiensNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4428
9548831, 189574411998
GLPVCGETCVGGTCNTPGCSCSWPVCTRN
Varv peptide A29Not AvailableLNoneFreeFreeAnticancerViola arvensis,Viola odorata, Viola tricolor, Viola baoshanensis, Viola yedoensis, and Viola bifloraNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4427
21434649, 189574412011
GLPVCGETCFGGTCNTPGCTCDPWPVCTRN
Vaby D30Not AvailableLNoneFreeFreeAnticancerAfrican, the Ethiopian highlands, Viola abyssinicaNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4426
21434649, 189574412011
GLPVCGETCAGGTCNTPGCSCSWPICTRN
Vaby A29Not AvailableLNoneFreeFreeAnticancerAfrican, the Ethiopian highlands, Viola abyssinicaNot AvailableFibrosarcomaNot AvailableNot AvailableNot AvailableFibrous connective tissue None
4425
10601876, 189574412000
GLLSVLGSVAKHVLPHVVPVIAEKL
Caerin 1.1025Not AvailableLNoneFreeFreeAnticancerMagnificent treefrog Litoria splendida, AustraliaNot AvailableLung CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4424
9266696, 189574411997
GLLSVLGSVAKHVLPHVVPVIAEHL
Caerin 1.125Not AvailableLNoneFreeFreeAnticancerAustralian green tree frogLitoria splendida; Litoria rothiiNot AvailableLung CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4422
18191970, 189574412008
GIPCAESCVWIPCTVTALIGCGCSNKVCYN
Vibi E30Not AvailableLNoneFreeFreeAnticancerAlpine violetViola bifloraNot AvailableLeukemia CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4421
10075760, 189574411999
GVPICGETCTLGTCYTAGCSCSWPVCTRN
Varv peptide F29Not AvailableLNoneFreeFreeAnticancerViola arvensisNot AvailableLeukemia CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4416
22771617, 189574412012
GLLGLLGSVVSHVVPAIVGHF
Maculatin 1.321Not AvailableLNoneFreeFreeAnticancerBlue-thighed frog,Litoria chloris, AustraliaNot AvailableSkin CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4415
22771617, 189574412012
GLLGLLGSVVSHVLPAITQHL
Maculatin 1.421Not AvailableLNoneFreeFreeAnticancerBlue-thighed frog,Litoria chloris, AustraliaNot AvailableSkin CancerNot AvailableNot AvailableNot AvailableNot AvailableNone
4413
9230483, 189574411997
GLFSVLGAVAKHVLPHVVPVIAEK
Caerin 1.624Not AvailableLNoneFreeFreeAnticancerBlue-thighed frog,Litoria chloris, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4412
9230483, 189574411997
GLFKVLGSVAKHLLPHVVPVIAEK
Caerin 1.824Not AvailableLNoneFreeFreeAnticancerBlue-thighed frog,Litoria chloris, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4411
9230483, 189574411997
GLFKVLGSVAKHLLPHVAPVIAEK
Caerin 1.724Not AvailableLNoneFreeFreeAnticancerOrange-thighed frog,Litoria xanthomera, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4410
9516047, 189574411998
GLFGVLGSIAKHVLPHVVPVIAEK
Caerin 1.924Not AvailableLNoneFreeFreeAnticancerLitoria chloris, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4401
11835991, 189574412002
GIGTKILGGVKTALKGALKELASTYAN
Maximin 127Not AvailableLNoneFreeFreeAnticancerBombina maximaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4400
11835991, 189574412002
GIGGVLLSAGKAALKGLAKVLAEKYAN
Maximin 427Not AvailableLNoneFreeFreeAnticancerBombina maximaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4399
11835991, 189574412002
GIGGKILSGLKTALKGAAKELASTYLH
Maximin 327Not AvailableLNoneFreeFreeAntibacterialBombina maximaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4398
11835991, 189574412002
ILGPVISTIGGVLGGLLKNL
Maximin H127Not AvailableLNoneFreeFreeAntibacterialBombina maximaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4397
20575512, 189574412010
GIACGESCVFLGCFIPGCSCKSKVCYFN
Psyle A28Not AvailableLNoneFreeFreeAntibacterialPsychotria leptothyrsaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4395
20575512, 189574412010
KLCGETCFKFKCYTPGCSCSYPFCK
Psyle C25Not AvailableLNoneFreeFreeAntibacterialPsychotria leptothyrsaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4394
8910461, 189574411996
GGLRSLGRKILRAWKKYGPIIVPIIRIG
BMAP-2828Not AvailableLNoneFreeFreeAntibacterialCowBos taurusNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4393
8910461, 189574411996
GRFKRFRKKFKKLFKKLSPVIPLLHLG
BMAP-2727Not AvailableLNoneFreeFreeAntibacterialCowBos taurusNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4392
9620615, 189574411998
GLLQTIKEKLESLESLAKGIVSGIQA
Maculatin 3.126Not AvailableLNoneFreeFreeAnticancerLitoria genimaculate, Litoria eucnemis, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4391
9620615, 189574411998
GLFVGVLAKVAAHVVPAIAEHF
Maculatin 1.122Not AvailableLNoneFreeFreeAntibacterialLitoria genimaculate, Litoria eucnemis, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4390
9620615, 189574411998
GLFVGLAKVAAHNNPAIAEHFQA
Maculatin 1.223Not AvailableLNoneFreeFreeAntibacterialLitoria genimaculate, Litoria eucnemis, AustraliaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4384
21596752, 189574412011
GEFLKCGESCVQGECYTPGCSCDWPICKKN
Cliotide T230Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4383
21596752, 189574412011
GIPCGESCVFIPCITAAIGCSCKSKVCYRN
Cliotide T430Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4382
21596752, 189574412011
GIPCGESCVFIPCITGAIGCSCKSKVCYRN
Cliotide T130Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4381
21596752, 189574412011
GLPTCGETCTLGTCYVPDCSCSWPICMKN
Cliotide T329Not AvailableLNoneFreeFreeAntibacterialClitoria ternateaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4380
10600388, 189574411999
GIPCGESCVWIPCISSAIGCSCKSKVCYRN
Cycloviolacin O230Not AvailableLNoneFreeFreeAntibacterialViola odorataNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4378
21723349, 189574412011
GLPVCGETCVGGTCNTPGCGCSWPVCTRN
Viba1729Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4377
21723349, 189574412011
GLPVCGETCVGGTCNTPGCACSWPVCTRN
Viba 1529Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4376
21723349, 189574412011
GIPCGESCVFIPCLTSAIDCSCKSKVCYRN
Mram 830Not AvailableLNoneFreeFreeAntibacterialViola philippicaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4371
22467870, 189574412012
GEYCGESCYLIPCFTPGCYCVSRQCVNKN
Chassatide C1029Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4370
22467870, 189574412012
GDACGETCFTGICFTAGCSCNPWPTCTRN
Chassatide C429Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4369
22467870, 189574412012
GASCGETCFTGICFTAGCSCNPWPTCTRN
Chassatide C429Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4368
22467870, 189574412012
IPCGESCVWIPCISGMFGCSCKDKVCYS
ChaC1129Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4367
22467870, 189574412012
AIPCGESCVWIPCISTVIGCSCSNKVCYR
Chassatide C829Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4366
22467870, 189574412012
IPCGESCVWIPCITAIAGCSCKNKVCYT
ChaC729Not AvailableLNoneFreeFreeAntibacterialChassalia chartaceaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4364
16713189, 189574412006
FLPILASLAAKFGPKLFCLVTKKC
Brevinin-1BYa24Not AvailableLNoneFreeFreeAntibacterialRana boylii, North AmericaNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4362
19254736, 189574412009
GLMDTIKGVAKTVAASWLDKLKCKITGC
Ranatuerin-2Ya28Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates yavapaiensisNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4361
19254736, 189574412009
FLPVIAGVAANFLPKLFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4360
19254736, 189574412009
FLPIIAGVAAKVLPKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4359
19254736, 189574412009
FLPIIAGIAAKFLPKIFCTISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4358
19254736, 189574412009
FLPIIAGAAAKVVQKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4357
19254736, 189574412009
FLPIIAGAAAKVVEKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4356
19254736, 189574412009
FLPAIVGAAAKFLPKIFCAISKKC
Brevinin-1BLa24Not AvailableLNoneFreeFreeAntibacterialNorth America, leopard frog, Lithobates blairiNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
4354
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptideSU.86.86Pancreatic CancerWST-1 assayIC50= 8.0 µM48-hPancreaticWO_2010_064207_A2
4353
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptidePane- 1Breast CancerWST-1 assayIC50= 14.1 µM48-hBreastWO_2010_064207_A2
4352
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptideCFPAC-IPancreatic CancerWST-1 assayIC50= 9.2 µM48-hPancreaticWO_2010_064207_A2
4351
None2009
GRVPYPRGGLLkLLKklLKKLlKL
Sema3A(aa371-377) -nLytic24LinearMixNoneFreeFreeAnticancerSynthetic PeptideBxPC-3Pancreatic CancerWST-1 assayIC50= 14.7 µM48-hPancreaticWO_2010_064207_A2
4262
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay2% apoptosis at 50 µM8-hNot AvailableNone
4261
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay1% apoptosis at 20 µM8-hNot AvailableNone
4260
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay0% apoptosis at 10 µM8-hNot AvailableNone
4259
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay3% apoptosis at 50 µM8-hNot AvailableNone
4258
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay2% apoptosis at 20 µM8-hNot AvailableNone
4257
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay1% apoptosis at 10 µM8-hNot AvailableNone
4256
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay5% apoptosis at 50 µM8-hBrainNone
4255
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay1% apoptosis at 20 µM8-hBrainNone
4254
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay2% apoptosis at 10 µM8-hBrainNone
4253
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay3% apoptosis at 50 µM8-hBrainNone
4252
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay2% apoptosis at 20 µM8-hBrainNone
4251
165680932006
rrrrrrrrGEDIIRNIARHAAQVGASMDR
r8-BidBH3Alt29LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay1% apoptosis at 10 µM8-hBrainNone
4250
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay55% apoptosis at 50 µM8-hNot AvailableNone
4249
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay35% apoptosis at 20 µM8-hNot AvailableNone
4248
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideIMR5TumorMTT/MTS assay23% apoptosis at 10 µM8-hNot AvailableNone
4247
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay79% apoptosis at 50 µM8-hNot AvailableNone
4246
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay46% apoptosis at 20 µM8-hNot AvailableNone
4245
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNGPTumorMTT/MTS assay43% apoptosis at 10 µM8-hNot AvailableNone
4244
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay68% apoptosis at 50 µM8-hBrainNone
4243
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay66% apoptosis at 20 µM8-hBrainNone
4242
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideNB69Brain TumorMTT/MTS assay25% apoptosis at 10 µM8-hBrainNone
4241
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay65% apoptosis at 50 µM8-hBrainNone
4240
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay45% apoptosis at 20 µM8-hBrainNone
4239
165680932006
rrrrrrrrGEDIIRNIARHLAQVGDSMDR
r8-BidBH329LinearMixNoneFreeFreeAntitumorSynthetic PeptideSK-N-ASBrain TumorMTT/MTS assay8% apoptosis at 10 µM8-hBrainNone
4207
158673602005
LGQSAASAHHAYIVLAIENSFMTASKKK
hP828LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel AssayNo inhibition at 7 mg/kg/d672-hPancreaticNone
4206
158673602005
ETWRTEAPSATGQASSLLGGRLLGQ
hP725LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel AssayNo inhibition at 7 mg/kg/d672-hPancreaticNone
4205
158673602005
HPTWPQKSVWHGSDPNGRRLTESY
hP624LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel AssayNo inhibition at 7 mg/kg/d672-hPancreaticNone
4204
158673602005
GSEGPLKPGARIFSFDGKDVLRHPT
hP525LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel Assay29% inhibition at 7 mg/kg/d672-hPancreaticNone
4203
158673602005
AAVPIVNLKDELLFPSWEALFSGSE
hP425LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel AssayNo inhibition at 7 mg/kg/d672-hPancreaticNone
4202
158673602005
TFRAFLSSRLQDLYSIVRRADRAAV
hP325LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel AssayNo inhibition at 7 mg/kg/d672-hPancreaticNone
4201
158673602005
MRGIRGADFQAFQQARAVGLAGTFR
hP225LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel Assay19% inhibition at 7 mg/kg/d672-hPancreaticNone
4200
158673602005
HSHRDFQPVLHLVALNSPLSGGMRG
hP125LinearLNoneFreeFreeAntiangiogenesisHuman endostatin peptidesBxPC-3Pancreatic CancerMatrigel Assay39% inhibition at 7 mg/kg/d672-hPancreaticNone
4198
154677502004
GRKKRRQRRRGGWMWVTNLRTD
TAT-Ras-GAP317-32622LinearLNoneFreeFreeAnticancerNot AvailableHeLaCervical CancerLDH leakage assay79% apoptosis at 50 µM16 to 24-hCervixNone
4197
154677502004
GRKKRRQRRRGGWMWVTNLRTD
TAT-Ras-GAP317-32622LinearLNoneFreeFreeAnticancerNot AvailableHeLaCervical CancerLDH leakage assay72% apoptosis at 30 µM16 to 24-hCervixNone
4196
154677502004
GRKKRRQRRRGGWMWVTNLRTD
TAT-Ras-GAP317-32622LinearLNoneFreeFreeAnticancerNot AvailableHeLaCervical CancerLDH leakage assay47% apoptosis at 20 µM16 to 24-hCervixNone
4195
154677502004
GRKKRRQRRRGGWMWVTNLRTD
TAT-Ras-GAP317-32622LinearLNoneFreeFreeAnticancerNot AvailableHeLaCervical CancerLDH leakage assay15% apoptosis at 10 µM16 to 24-hCervixNone
3842
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP(O)25Cyclic(C2-C10,CLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay52% inhibition at 10µg/mlNANot AvailableNone
3841
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP(O)25Cyclic(C2-C10,CLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay42% inhibition at 5µg/mlNANot AvailableNone
3840
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP(O)25Cyclic(C2-C10,CLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay40% inhibition at 2.5µg/mlNANot AvailableNone
3839
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP25LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay75% inhibition at 10µg/mlNANot AvailableNone
3838
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP25LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay40% inhibition at 5µg/mlNANot AvailableNone
3837
205150452010
ACDCRGDCFCGGGGIVRRADRAAVP
AP25LinearLNoneFreeFreeAntitumorEndostatin derived synthetic peptideBAETumorMTT/MTS assay50% inhibition at 2.5µg/mlNANot AvailableNone
3815
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 1.4±0.1 µM24-hSkinNone
3813
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 13.1±0.9 µM24-hSkinNone
3812
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 12.3±1.0 µM24-hSkinNone
3811
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 3.7± 4.3 µM24-hSkinNone
3810
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 40 µM (approx)24-hSkinNone
3809
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 1.8±0.1 µM4-hSkinNone
3807
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 9.3±1.5 µM4-hSkinNone
3806
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 8.3±0.5 µM4-hSkinNone
3805
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 12.1±1.6 µM4-hSkinNone
3804
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 50 µM (approx)4-hSkinNone
3803
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 2.1±0.1 µM2-hSkinNone
3801
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 13.8±2.0 µM2-hSkinNone
3800
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 12.3±2.0 µM2-hSkinNone
3799
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 13.0±1.0 µM2-hSkinNone
3798
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 50 µM (approx)2-hSkinNone
3797
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 3.2±0.1 µM30-MinSkinNone
3795
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A- Δ23LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 7.5±0.4 µM30-MinSkinNone
3794
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21k27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 8.4±0.2 µM30-MinSkinNone
3793
238936052013
KILRGVAKKILRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAnticancerNK-2 variantsE42/02Skin CancerMTT/MTS assayIC50= 10.6±0.4 µM30-MinSkinNone
3792
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 70 µM (approx)30-MinSkinNone
3791
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAnticancerNatural component of bee venomE42/02Skin CancerMTT/MTS assayIC50= 1.4±0.1 µM4-hSkinNone
3789
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAnticancerResidue of 39-65 of porcine NK-lysineE42/02Skin CancerMTT/MTS assayIC50= 4.3±0.3 µM4-hSkinNone
3772
228376672012
KWKSFlKTFKSlKKTVlHTllKAISS
Peptide L6D/L12D/L17D/L20D/L21D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 12.88±0.15 µMol/L1-hCervixNone
3771
228376672012
KWKSFlKTFKSlKKTVlHTlLKAISS
Peptide L6D/L12D/L17D/L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 9.69±0.38 µMol/L1-hCervixNone
3769
228376672012
KWKSFLKTFKSlKKTVLHTlLKAISS
Peptide L12D/L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 3.14±0.06 µMol/L1-hCervixNone
3770
228376672012
KWKSFlKTFKSlKKTVLHTlLKAISS
Peptide L6D/L12D/L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 7.80±0.26 µMol/L1-hCervixNone
3767
228376672012
KWKSFLKTFKSLKKTVLHTlLKAISS
Peptide L20D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.33±0.06 µMol/L1-hCervixNone
3768
228376672012
KWKSFlKTFKSlKKTVLHTLLKAISS
Peptide L6D/L12D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 3.01±0.08 µMol/L1-hCervixNone
3766
228376672012
KWKSFLKTFKSlKKTVLHTLLKAISS
Peptide L12D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.63±0.07 µMol/L1-hCervixNone
3765
228376672012
KWKSFlKTFKSLKKTVLHTLLKAISS
Peptide L6D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.23±0.10 µMol/L1-hCervixNone
3764
228376672012
kWkSFLkTFkSLKkTVLHTLLkAISS
Peptide K1D/K3D/K7D /K10D/K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 18.07±0.48 µMol/L1-hCervixNone
3762
228376672012
KWKSFLkTFkSLKkTVLHTLLkAISS
Peptide K7D /K10D/K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 4.79±0.23 µMol/L1-hCervixNone
3763
228376672012
KWkSFLkTFkSLKkTVLHTLLkAISS
Peptide K3D/K7D /K10D/K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 20.41±0.64 µMol/L1-hCervixNone
3761
228376672012
KWKSFLkTFKSLKkTVLHTLLKAISS
Peptide K7D /K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 4.45±0.19 µMol/L1-hCervixNone
3760
228376672012
KWKSFLKTFKSLKkTVLHTLLkAISS
Peptide K14D/K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.40±0.09 µMol/L1-hCervixNone
3759
228376672012
KWKSFLkTFKSLKkTVLHTLLKAISS
Peptide K7D /K14D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 2.06±0.01 µMol/L1-hCervixNone
3758
228376672012
KWKSFLKTFKSLKKTVLHTLLkAISS
Peptide K22D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.39±0.02 µMol/L1-hCervixNone
3757
228376672012
KWKSFLKTFKSLKkTVLHTLLKAISS
Peptide K14D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.52±0.05 µMol/L1-hCervixNone
3756
228376672012
KWKSFLkTFKSLKKTVLHTLLKAISS
Peptide K7D26LinearMixNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.29±0.03 µMol/L1-hCervixNone
3755
228376672012
KWKSFLKTFKSLKKTVLHTLLKAISS
Peptide P26LinearLNoneAmidationAcetylationAnticancerA12L/A20LHeLaCervical CancerMTT/MTS assayIC50= 1.71±0.07 µMol/L1-hCervixNone
3718
241768522013
YGRKKRRQRRRREADFFWSLCTADMS
KilerFLIP26linearLNoneFreeFreeNANAJurkatBlood CancerNot AvailableNANABloodNone
3468
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay~30% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3469
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay>40% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3466
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay<20% cytotoxicity at 1 µM48-hBladderWO_2012042540_A2
3467
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay20% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3464
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay40% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3465
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHTB-9Bladder CancerMTT/MTS assay~50% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3462
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3463
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3460
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<5% cytotoxicity at 1 µM48-hBladderWO2012042540A2
3461
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<3% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3458
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay<15% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3459
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHTB-9Bladder CancerMTT/MTS assay~15% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3450
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3451
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~45% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3449
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~55% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3447
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~40% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3448
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3445
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay>20% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3446
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCaSkiCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3443
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3444
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~15% cytotoxicity at 1 µM72-hCervixWO2012042540A2
3441
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~15% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3442
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay<3% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3440
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCaSkiCervical CancerMTT/MTS assay~5% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3433
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay~45% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3432
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3431
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay~50% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3430
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay<20% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3429
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay>40% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3428
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinSiHaCervical CancerMTT/MTS assay>20% cytotoxicity at 1 µM24-hCervixWO2012042540A2
3427
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay~40% cytotoxicity at 10 µM72-hCervixWO_2012042540_A2
3426
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay~20% cytotoxicity at 1 µM72-hCervixWO_2012042540_A2
3425
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hCervixWO_2012042540_A2
3424
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay<3% cytotoxicity at 1 µM48-hCervixWO_2012042540_A2
3423
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay>10% cytotoxicity at 10 µM24-hCervixWO_2012042540_A2
3422
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiSiHaCervical CancerMTT/MTS assay5% cytotoxicity at 1 µM24-hCervixWO_2012042540_A2
3415
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay~40% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3414
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay>30% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3413
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay>20% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3412
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay<20% cytotoxicity at 1 µM48-hColonWO2012042540A2
3411
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay50% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3410
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinHCT-116Colon CancerMTT/MTS assay>40% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3409
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3408
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3407
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3406
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay~5% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3405
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay15% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3404
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiHCT-116Colon CancerMTT/MTS assay<15% cytotoxicity at 1 µM24-hColonWO2012042540A2
3396
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay>40% cytotoxicity at 1 µM72-hBladderWO2012042540A2
3397
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay~50% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3395
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay~50% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3394
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay<30% cytotoxicity at 1 µM48-hBladderWO_2012042540_A2
3393
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay<30% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3392
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinUM-UC-3Bladder CancerMTT/MTS assay~30% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3391
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay<45% cytotoxicity at 10 µM72-hBladderWO_2012042540_A2
3390
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~45% cytotoxicity at 1 µM72-hBladderWO_2012042540_A2
3389
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay>25% cytotoxicity at 10 µM48-hBladderWO_2012042540_A2
3388
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 1 µM48-hBladderWO2012042540A2
3387
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 10 µM24-hBladderWO_2012042540_A2
3386
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiUM-UC-3Bladder CancerMTT/MTS assay~25% cytotoxicity at 1 µM24-hBladderWO_2012042540_A2
3379
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay~20% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3378
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM72-hColonWO_2012042540_A2
3377
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay~35% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3376
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay>20% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3375
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3374
None2012
GQVWEATATVNAIRGSVTPAVSQFNARTAD
MB3030LinearLNoneFreeFreeAnticancerDerived from the MPT63 secreted proteinCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3373
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 10 µM72-hColonWO_2012042540_A2
3372
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay>10% cytotoxicity at 1 µM72-hColonWO2012042540A2
3371
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay>10% cytotoxicity at 10 µM48-hColonWO_2012042540_A2
3370
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay10% cytotoxicity at 1 µM48-hColonWO_2012042540_A2
3369
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay~10% cytotoxicity at 10 µM24-hColonWO_2012042540_A2
3368
None2012
TAGIKLTVPIEKFPVTTQTFWG
TG2322LinearLNoneFreeFreeAnticancerDerived from the SAG1 surface protein from the parasite Toxoplasma gondiiCOLO-205Colon CancerMTT/MTS assay<5% cytotoxicity at 1 µM24-hColonWO_2012042540_A2
3338
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =2.1 ± 0.1 µM2-hSkinNone
3339
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =1.8 ± 0.1 µM4-hSkinNone
3340
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =1.4 ± 0.1 µM24-hSkinNone
3329
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =7.5 ± 0.4 µM30-MinSkinNone
3330
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =13.8 ± 2.0 µM2-hSkinNone
3331
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =9.3 ± 1.5 µM4-hSkinNone
3332
238936052013
KILRGVAKKIMRTFLRRILTGKK
C7A-Δ24LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =13.1 ± 0.9 µM24-hSkinNone
3337
238936052013
GIGAVLKVLTTGLPALISWIKRKRQQ
Melittin26LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =3.2 ± 0.1 µM30-MinSkinNone
3328
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =12.3 ± 1.0 µM24-hSkinNone
3327
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =8.3 ± 0.5 µM4-hSkinNone
3326
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =12.3 ± 2.0 µM2-hSkinNone
3325
238936052013
KILRGVAKKIMRTFLRRISKKILTGKK
C7A-D21K27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =8.4 ± 0.2 µM30-MinSkinNone
3324
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =37 ± 4.3 µM24-hSkinNone
3323
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =12.1 ± 1.6 µM4-hSkinNone
3322
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =13.0 ± 1.0 µM2-hSkinNone
3321
238936052013
KILRGVAKKIMRTFLRRISKDILTGKK
C7A27LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 =10.6 ± 0.4 µM30-MinSkinNone
3320
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~40 µM24-hSkinNone
3319
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~50 µM4-hSkinNone
3318
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~50 µM2-hSkinNone
3317
238936052013
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntimicrobialSynthetic peptideE42/02Skin CancerMTT/MTS assayIC50 = ~70 µM30-MinSkinNone
3289
195274902009
KAAKKAAKAAKKAAKAAKKAA
KW521LinearLNoneFreeFreeAnticancerSynthetic peptideHT-29Colon CancerMTT/MTS assayIC50 =55±14 µMNAColonNone
3288
195274902009
KAAKKAAKAAKKAAKAAKKAA
KW521LinearLNoneFreeFreeAnticancerBovine lactoferrin (Lf-B)FEMXSkin CancerMTT/MTS assayIC50 =30±3 µMNASkinNone
3278
188157342008
KKKFPWWWPFKKKKKKFPWWWPFKKKK
di-PST13-RK-K27LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinMDA-MB-361Breast CancerMTT/MTS assayIC50 =10 µg/mlNABreastNone
3277
188157342008
KKKFPWWWPFKKKKKKFPWWWPFKKKK
di-PST13-RK-K27LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinA-549Lung CancerMTT/MTS assayIC50 =15 µg/mlNALungNone
3275
188157342008
KKKFPWWWPFKKKCKKKFPWWWPFKKKC
di-PST13-RK-C28LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinMDA-MB-361Breast CancerMTT/MTS assayIC50 =17 µg/mlNABreastNone
3274
188157342008
KKKFPWWWPFKKKCKKKFPWWWPFKKKC
di-PST13-RK-C28LinearLNoneAmidationFreeAntimicrobialDerivative of tritrpticinA-549Lung CancerMTT/MTS assayIC50 =17 µg/mlNALungNone
3265
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<40% cell viability at 50 µMNAStomachNone
3264
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay100% cell viability at 5 µMNAStomachNone
3263
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<60% cell viability at 50 µMNABloodNone
3262
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µMNABloodNone
3261
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay60% cell viability at 50 µMNAColonNone
3260
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay>100% cell viability at 5 µMNAColonNone
3259
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<20% cell viability at 50 µMNAStomachNone
3258
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<100% cell viability at 5 µMNAStomachNone
3257
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<40% cell viability at 50 µMNABloodNone
3256
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µMNABloodNone
3255
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay40% cell viability at 50 µMNAColonNone
3254
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay100% cell viability at 5 µMNAColonNone
3112
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<100% cell viability at 5 µM24-hStomachNone
3113
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<40% cell viability at 50 µM24-hStomachNone
3109
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay60% cell viability at 50 µM24-hColonNone
3110
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µM24-hBloodNone
3111
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<60% cell viability at 50 µM24-hBloodNone
3108
227830182012
PDEDAINDALNKVCSTGRRQRSICKQLLKK
N29D30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay>100% cell viability at 5 µM24-hColonNone
3107
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<20% cell viability at 50 µM24-hStomachNone
3106
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSNU-1Gastric CancerCell Viability assay<100% cell viability at 5 µM24-hStomachNone
3105
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay<40% cell viability at 50 µM24-hBloodNone
3104
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideU-937Lymphoma CancerCell Viability assay100% cell viability at 5 µM24-hBloodNone
3103
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay40% cell viability at 50 µM24-hColonNone
3102
227830182012
PDEDAINNALNKVCSTGRRQRSICKQLLKK
N29N30LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic peptideSW-480Colon CancerCell Viability assay100% cell viability at 5 µM24-hColonNone
3101
160046182005
MWKWFHNVLSSGQLLADKWWAWWYNWW
Pep27anal527LinearLNoneFreeFreeAnticancerS. pneumoniaeMCF-7Breast CancerMTT/MTS assayIC50=>70 µM19.17-MinBreastNone
3100
160046182005
MWKEFHNVLSSGQLLADKRWARWYNRW
Pep27anal427LinearLNoneFreeFreeAnticancerS. pneumoniaeMCF-7Breast CancerMTT/MTS assayIC50= 29 µM19.15-MinBreastNone
3099
160046182005
MRKWFHNVLSSGQLLADKWPAWDYNRK
Pep27anal327LinearLNoneFreeFreeAnticancerS. pneumoniaeMCF-7Breast CancerMTT/MTS assayIC50= 38 µM20.08-MinBreastNone
3098
160046182005
MWKWFHNVLSWWWLLADKRPARDYNRK
Pep27anal227LinearLNoneFreeFreeAnticancerS. pneumoniaeMCF-7Breast CancerMTT/MTS assayIC50= <10 µM22.5-MinBreastNone
3097
160046182005
MWKWFHNVLSSWQLLADKRPARDYNRK
Pep27anal127LinearLNoneFreeFreeAnticancerS. pneumoniaeMCF-7Breast CancerMTT/MTS assayIC50= 55 µM18.67-MinBreastNone
3096
160046182005
MRKEFHNVLSSGQLLADKRPARDYNRK
Pep2727LinearLNoneFreeFreeAnticancerS. pneumoniaeMCF-7Breast CancerMTT/MTS assayIC50= >70 µM14.54-MinBreastNone
3095
160046182005
MWKWFHNVLSSGQLLADKWWAWWYNWW
Pep27anal527LinearLNoneFreeFreeAnticancerS. pneumoniaeSNU-601Gastric CancerMTT/MTS assayIC50=>70 µM19.17-MinStomachNone
3094
160046182005
MWKEFHNVLSSGQLLADKRWARWYNRW
Pep27anal427LinearLNoneFreeFreeAnticancerS. pneumoniaeSNU-601Gastric CancerMTT/MTS assayIC50= 37 µM19.15-MinStomachNone
3093
160046182005
MRKWFHNVLSSGQLLADKWPAWDYNRK
Pep27anal327LinearLNoneFreeFreeAnticancerS. pneumoniaeSNU-601Gastric CancerMTT/MTS assayIC50= 50 µM20.08-MinStomachNone
3092
160046182005
MWKWFHNVLSWWWLLADKRPARDYNRK
Pep27anal227LinearLNoneFreeFreeAnticancerS. pneumoniaeSNU-601Gastric CancerMTT/MTS assayIC50= 25 µM22.5-MinStomachNone
3091
160046182005
MWKWFHNVLSSWQLLADKRPARDYNRK
Pep27anal127LinearLNoneFreeFreeAnticancerS. pneumoniaeSNU-601Gastric CancerMTT/MTS assayIC50= 37 µM18.67-MinStomachNone
3089
160046182005
MWKWFHNVLSSGQLLADKWWAWWYNWW
Pep27anal527LinearLNoneFreeFreeAnticancerS. pneumoniaeJurkatBlood CancerMTT/MTS assayIC50=>70 µM19.17-MinBloodNone
3090
160046182005
MRKEFHNVLSSGQLLADKRPARDYNRK
Pep2727LinearLNoneFreeFreeAnticancerS. pneumoniaeSNU-601Gastric CancerMTT/MTS assayIC50= >70 µM14.54-MinStomachNone
3088
160046182005
MWKEFHNVLSSGQLLADKRWARWYNRW
Pep27anal427LinearLNoneFreeFreeAnticancerS. pneumoniaeJurkatBlood CancerMTT/MTS assayIC50= 46 µM19.15-MinBloodNone
3087
160046182005
MRKWFHNVLSSGQLLADKWPAWDYNRK
Pep27anal327LinearLNoneFreeFreeAnticancerS. pneumoniaeJurkatBlood CancerMTT/MTS assayIC50= 50 µM20.08-MinBloodNone
3086
160046182005
MWKWFHNVLSWWWLLADKRPARDYNRK
Pep27anal227LinearLNoneFreeFreeAnticancerS. pneumoniaeJurkatBlood CancerMTT/MTS assayIC50= 23 µM22.5-MinBloodNone
3085
160046182005
MWKWFHNVLSSWQLLADKRPARDYNRK
Pep27anal127LinearLNoneFreeFreeAnticancerS. pneumoniaeJurkatBlood CancerMTT/MTS assayIC50= 47 µM18.67-MinBloodNone
3084
160046182005
MRKEFHNVLSSGQLLADKRPARDYNRK
Pep2727LinearLNoneFreeFreeAnticancerS. pneumoniaeJurkatBlood CancerMTT/MTS assayIC50=>70 µM14.54-MinBloodNone
3083
160046182005
MWKWFHNVLSSGQLLADKWWAWWYNWW
Pep27anal527LinearLNoneFreeFreeAnticancerS. pneumoniaeHL-60Leukemia CancerMTT/MTS assayIC50= >70 µM19.17-MinBloodNone
3082
160046182005
MWKEFHNVLSSGQLLADKRWARWYNRW
Pep27anal427LinearLNoneFreeFreeAnticancerS. pneumoniaeHL-60Leukemia CancerMTT/MTS assayIC50=51 µM19.15-MinBloodNone
3081
160046182005
MRKWFHNVLSSGQLLADKWPAWDYNRK
Pep27anal327LinearLNoneFreeFreeAnticancerS. pneumoniaeHL-60Leukemia CancerMTT/MTS assayIC50= 52 µM20.08-MinBloodNone
3080
160046182005
MWKWFHNVLSWWWLLADKRPARDYNRK
Pep27anal227LinearLNoneFreeFreeAnticancerS. pneumoniaeHL-60Leukemia CancerMTT/MTS assayIC50= 20 µM22.5-MinBloodNone
3079
160046182005
MWKWFHNVLSSWQLLADKRPARDYNRK
Pep27anal127LinearLNoneFreeFreeAnticancerS. pneumoniaeHL-60Leukemia CancerMTT/MTS assayIC50= 53 µM18.67-MinBloodNone
3078
160046182005
MRKEFHNVLSSGQLLADKRPARDYNRK
Pep2727LinearLNoneFreeFreeAnticancerS. pneumoniaeHL-60Leukemia CancerMTT/MTS assayIC50= >70 µM14.54-MinBloodNone
3077
160046182005
MWKWFHNVLSSGQLLADKWWAWWYNWW
Pep27anal527LinearLNoneFreeFreeAnticancerS. pneumoniaeAML-2Leukemia CancerMTT/MTS assayIC50= >70 µM19.17-MinBloodNone
3076
160046182005
MWKEFHNVLSSGQLLADKRWARWYNRW
Pep27anal427LinearLNoneFreeFreeAnticancerS. pneumoniaeAML-2Leukemia CancerMTT/MTS assayIC50= 50 µM19.15-MinBloodNone
3075
160046182005
MRKWFHNVLSSGQLLADKWPAWDYNRK
Pep27anal327LinearLNoneFreeFreeAnticancerS. pneumoniaeAML-2Leukemia CancerMTT/MTS assayIC50= 67 µM20.08-MinBloodNone
3074
160046182005
MWKWFHNVLSWWWLLADKRPARDYNRK
Pep27anal227LinearLNoneFreeFreeAnticancerS. pneumoniaeAML-2Leukemia CancerMTT/MTS assayIC50= 29 µM22.5-MinBloodNone
3073
160046182005
MWKWFHNVLSSWQLLADKRPARDYNRK
Pep27anal127LinearLNoneFreeFreeAnticancerS. pneumoniaeAML-2Leukemia CancerMTT/MTS assayIC50= 50 µM18.67-MinBloodNone
3072
160046182005
MRKEFHNVLSSGQLLADKRPARDYNRK
Pep2727LinearLNoneFreeFreeAnticancerS. pneumoniaeAML-2Leukemia CancerMTT/MTS assayNot Available14.54-MinBloodNone
3071
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
3070
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay1 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
3069
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay20 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
3068
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
3067
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
3066
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay15 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
3065
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
3064
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
3063
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
3062
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
3061
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay35 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
3060
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
3059
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay48 % Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
3058
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay84% Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
3057
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay84 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
3056
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay25 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
3055
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
3054
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay45 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
3053
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
3052
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay80 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
3051
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 3.125 mg/L24-hCervixNone
3050
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 6.25 mg/L24-hCervixNone
3049
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 12.5 mg/L24-hCervixNone
3048
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay82 % Cytotoxicity at 25 mg/L24-hCervixNone
3047
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay90 % Cytotoxicity at 50 mg/L24-hCervixNone
3046
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 3.125 mg/L12-hCervixNone
3045
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 6.25 mg/L12-hCervixNone
3044
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay18 % Cytotoxicity at 12.5 mg/L12-hCervixNone
3043
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L12-hCervixNone
3042
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay82 % Cytotoxicity at 50 mg/L12-hCervixNone
3041
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 3.125 mg/L6-hCervixNone
3040
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 6.25 mg/L6-hCervixNone
3039
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay10 % Cytotoxicity at 12.5 mg/L6-hCervixNone
3038
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 25 mg/L6-hCervixNone
3037
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay78 % Cytotoxicity at 50 mg/L6-hCervixNone
3036
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay1 % Cytotoxicity at 3.125 mg/L3-hCervixNone
3035
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay5 % Cytotoxicity at 6.25 mg/L3-hCervixNone
3034
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay4 % Cytotoxicity at 12.5 mg/L3-hCervixNone
3033
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay60 % Cytotoxicity at 25 mg/L3-hCervixNone
3032
235980792013
GFFALIPKIISSPLFKTLLSAVGSALS
Pardaxin-627LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay70 % Cytotoxicity at 50 mg/L3-hCervixNone
2955
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay28 % Cytotoxicity at 3.125 mg/L24-hFibrous connective tissue None
2954
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L24-hFibrous connective tissue None
2952
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L24-hFibrous connective tissue None
2953
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay38 % Cytotoxicity at 12.5 mg/L24-hFibrous connective tissue None
2951
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay84 % Cytotoxicity at 50 mg/L24-hFibrous connective tissue None
2950
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay28 % Cytotoxicity at 3.125 mg/L12-hFibrous connective tissue None
2949
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay30 % Cytotoxicity at 6.25 mg/L12-hFibrous connective tissue None
2948
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay46 % Cytotoxicity at 12.5 mg/L12-hFibrous connective tissue None
2947
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay96 % Cytotoxicity at 25 mg/L12-hFibrous connective tissue None
2946
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay95 % Cytotoxicity at 50 mg/L12-hFibrous connective tissue None
2945
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay25 % Cytotoxicity at 3.125 mg/L6-hFibrous connective tissue None
2944
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay25 % Cytotoxicity at 6.25 mg/L6-hFibrous connective tissue None
2943
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay45 % Cytotoxicity at 12.5 mg/L6-hFibrous connective tissue None
2942
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay95 % Cytotoxicity at 25 mg/L6-hFibrous connective tissue None
2941
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay90 % Cytotoxicity at 50 mg/L6-hFibrous connective tissue None
2940
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2939
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2938
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2937
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay39 % Cytotoxicity at 3.125 mg/L3-hFibrous connective tissue None
2936
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay41 % Cytotoxicity at 6.25 mg/L3-hFibrous connective tissue None
2935
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay42 % Cytotoxicity at 12.5 mg/L3-hFibrous connective tissue None
2934
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay85 % Cytotoxicity at 25 mg/L3-hFibrous connective tissue None
2933
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHT-1080FibrosarcomaMTT/MTS assay82 % Cytotoxicity at 50 mg/L3-hFibrous connective tissue None
2932
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay77 % Cytotoxicity at 25 mg/L24-hCervixNone
2931
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay83% Cytotoxicity at 50 mg/L24-hCervixNone
2930
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay65% Cytotoxicity at 25 mg/L12-hCervixNone
2929
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75 % Cytotoxicity at 50 mg/L12-hCervixNone
2928
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay65% Cytotoxicity at 25 mg/L6-hCervixNone
2927
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay75% Cytotoxicity at 50 mg/L6-hCervixNone
2926
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay38% Cytotoxicity at 25 mg/L3-hCervixNone
2925
235980792013
GFIFHIIKGLFHAGKMIHGLV
Epinecidin-121LinearLNoneFreeFreeAntimicrobialEpinephelus nebulosusHeLaCervical CancerMTT/MTS assay45% Cytotoxicity at 50 mg/L3-hCervixNone
2809
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =100 µg/ml24-hCervixUS_06875744_B2
2805
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =170 µg/ml24-hCervixUS_06875744_B2
2804
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =125 µg/ml24-hCervixUS_06875744_B2
2783
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 = >1000 µg/ml24-hCervixUS_06875744_B2
2761
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =215 µg/ml24-hCervixUS_06875744_B2
2760
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 = >1000 µg/ml24-hCervixUS_06875744_B2
2736
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =35 µg/ml24-hCervixUS_06875744_B2
2733
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 = >1000 µg/ml24-hCervixUS_06875744_B2
2728
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =180 µg/ml24-hCervixUS_06875744_B2
2720
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =19 µg/ml24-hCervixUS_06875744_B2
2719
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16) Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =97 µg/ml24-hCervixUS_06875744_B2
2713
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =270 µg/ml24-hCervixUS_06875744_B2
2712
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =240 µg/ml24-hCervixUS_06875744_B2
2710
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =28 µg/ml24-hCervixUS_06875744_B2
2688
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayNot Available24-hCervixUS_06875744_B2
2683
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayNot Available24-hCervixUS_06875744_B2
2679
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =190 µg/ml24-hCervixUS_06875744_B2
2675
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =150 µg/ml24-hCervixUS_06875744_B2
2674
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =20 µg/ml24-hCervixUS_06875744_B2
2673
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =145 µg/ml24-hCervixUS_06875744_B2
2672
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =82 µg/ml24-hCervixUS_06875744_B2
2671
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =>1000 µg/ml24-hCervixUS_06875744_B2
2668
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =50 µg/ml24-hCervixUS_06875744_B2
2667
None2005
FALALKALKKALKKLKKALKKAL
Hecate AC23LinearLNoneFreeFreeAnticancerFLAK peptidesHeLaCervical CancerMTT/MTS assayLD50 =95 µg/ml24-hCervixUS_06875744_B2
2666
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =66 µg/ml24-hProstateUS_06875744_B2
2662
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =45 µg/ml24-hProstateUS_06875744_B2
2661
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =45 µg/ml24-hProstateUS_06875744_B2
2640
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =375 µg/ml24-hProstateUS_06875744_B2
2618
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =310 µg/ml24-hProstateUS_06875744_B2
2617
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =>1000 µg/ml24-hProstateUS_06875744_B2
2593
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =13 µg/ml24-hProstateUS_06875744_B2
2590
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayNot Available24-hProstateUS_06875744_B2
2585
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =28 µg/ml24-hProstateUS_06875744_B2
2577
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =170 µg/ml24-hProstateUS_06875744_B2
2576
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16) Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =28 µg/ml24-hProstateUS_06875744_B2
2570
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7)Shiva10(1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =97 µg/ml24-hProstateUS_06875744_B2
2569
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =63 µg/ml24-hProstateUS_06875744_B2
2567
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =82 µg/ml24-hProstateUS_06875744_B2
2545
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =66 µg/ml24-hProstateUS_06875744_B2
2540
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =64 µg/ml24-hProstateUS_06875744_B2
2536
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =65 µg/ml24-hProstateUS_06875744_B2
2532
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =125 µg/ml24-hProstateUS_06875744_B2
2531
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =12 µg/ml24-hProstateUS_06875744_B2
2530
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =38 µg/ml24-hProstateUS_06875744_B2
2529
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =41 µg/ml24-hProstateUS_06875744_B2
2528
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =83 µg/ml24-hProstateUS_06875744_B2
2525
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =44 µg/ml24-hProstateUS_06875744_B2
2523
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =160 µg/ml24-hLungUS_06875744_B2
2524
None2005
FALALKALKKALKKLKKALKKAL
Hecate AC23LinearLNoneFreeFreeAnticancerFLAK peptidesPC-3Prostate CancerMTT/MTS assayLD50 =61 µg/ml24-hProstateUS_06875744_B2
2519
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =77 µg/ml24-hLungUS_06875744_B2
2518
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =60 µg/ml24-hLungUS_06875744_B2
2497
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =315 µg/ml24-hLungUS_06875744_B2
2475
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =115 µg/ml24-hLungUS_06875744_B2
2474
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =>1000 µg/ml24-hLungUS_06875744_B2
2450
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =25 µg/ml24-hLungUS_06875744_B2
2447
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =>1000 µg/ml24-hLungUS_06875744_B2
2442
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =54 µg/ml24-hLungUS_06875744_B2
2434
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)23LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =22 µg/ml24-hLungUS_06875744_B2
2433
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16)23LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =64 µg/ml24-hLungUS_06875744_B2
2427
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7)Shiva10(1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =115 µg/ml24-hLungUS_06875744_B2
2426
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =160 µg/ml24-hLungUS_06875744_B2
2424
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =63 µg/ml24-hLungUS_06875744_B2
2402
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =150 µg/ml24-hLungUS_06875744_B2
2397
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =150 µg/ml24-hLungUS_06875744_B2
2393
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =125 µg/ml24-hLungUS_06875744_B2
2389
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =84 µg/ml24-hLungUS_06875744_B2
2388
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =37 µg/ml24-hLungUS_06875744_B2
2387
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =72 µg/ml24-hLungUS_06875744_B2
2386
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =64 µg/ml24-hLungUS_06875744_B2
2385
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =>1000 µg/ml24-hLungUS_06875744_B2
2382
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =140 µg/ml24-hLungUS_06875744_B2
2381
None2005
FALALKALKKALKKLKKALKKAL
Hecate AC23LinearLNoneFreeFreeAnticancerFLAK peptidesH-1299Lung CancerMTT/MTS assayLD50 =44 µg/ml24-hLungUS_06875744_B2
2379
None2005
VALALKALKKLAKKLKKLAKKAL
FLAK04 AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2378
None2005
VALALKALKKALKKLKKALKKAL
Hecate AC V23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2377
None2005
VALALKALKKALKKLKKALKKAL
Hecate AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2373
None2005
VAKKFAKKFKKFAKKFAKFAFAF
D2A21V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2370
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =83 µg/ml24-hSkinUS_06875744_B2
2366
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =140 µg/ml24-hSkinUS_06875744_B2
2365
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =130 µg/ml24-hSkinUS_06875744_B2
2344
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =600 µg/ml24-hSkinUS_06875744_B2
2321
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =>1000 µg/ml24-hSkinUS_06875744_B2
2322
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =155 µg/ml24-hSkinUS_06875744_B2
2294
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2297
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =18 µg/ml24-hSkinUS_06875744_B2
2289
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2282
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =12 µg/ml24-hSkinUS_06875744_B2
2281
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16) Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =76 µg/ml24-hSkinUS_06875744_B2
2275
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7)Shiva10(1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =360 µg/ml24-hSkinUS_06875744_B2
2274
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =290 µg/ml24-hSkinUS_06875744_B2
2272
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2250
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =140 µg/ml24-hSkinUS_06875744_B2
2245
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =150 µg/ml24-hSkinUS_06875744_B2
2241
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =140 µg/ml24-hSkinUS_06875744_B2
2235
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =85 µg/ml24-hSkinUS_06875744_B2
2236
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =36 µg/ml24-hSkinUS_06875744_B2
2237
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2233
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2234
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =27 µg/ml24-hSkinUS_06875744_B2
2230
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =128 µg/ml24-hSkinUS_06875744_B2
2229
None2005
FALALKALKKALKKLKKALKKAL
Hecate AC23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =72 µg/ml24-hSkinUS_06875744_B2
2227
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2226
None2005
VALALKALKKALKKLKKALKKAL
Hecate AC V23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2225
None2005
VALALKALKKALKKLKKALKKAL
Hecate AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2221
None2005
VAKKFAKKFKKFAKKFAKFAFAF
D2A21V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2218
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =83 µg/ml24-hSkinUS_06875744_B2
2214
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =140 µg/ml24-hSkinUS_06875744_B2
2213
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =130 µg/ml24-hSkinUS_06875744_B2
2192
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =600 µg/ml24-hSkinUS_06875744_B2
2169
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =>1000 µg/ml24-hSkinUS_06875744_B2
2170
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =155 µg/ml24-hSkinUS_06875744_B2
2145
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =18 µg/ml24-hSkinUS_06875744_B2
2142
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2137
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2130
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =12 µg/ml24-hSkinUS_06875744_B2
2129
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16) Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =76 µg/ml24-hSkinUS_06875744_B2
2123
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7)Shiva10(1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =360 µg/ml24-hSkinUS_06875744_B2
2122
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =290 µg/ml24-hSkinUS_06875744_B2
2120
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2098
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =140 µg/ml24-hSkinUS_06875744_B2
2093
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =150 µg/ml24-hSkinUS_06875744_B2
2089
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =140 µg/ml24-hSkinUS_06875744_B2
2085
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =94 µg/ml24-hSkinUS_06875744_B2
2084
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =36 µg/ml24-hSkinUS_06875744_B2
2083
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =85 µg/ml24-hSkinUS_06875744_B2
2082
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =27 µg/ml24-hSkinUS_06875744_B2
2081
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayNot Available24-hSkinUS_06875744_B2
2078
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =128 µg/ml24-hSkinUS_06875744_B2
2077
None2005
FALALKALKKALKKLKKALKKAL
Hecate AC23LinearLNoneFreeFreeAnticancerFLAK peptidesBMKCSkin CancerMTT/MTS assayLD50 =72 µg/ml24-hSkinUS_06875744_B2
2075
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayNot Available24-hColonUS_06875744_B2
2074
None2005
VALALKALKKALKKLKKALKKAL
Hecate AC V23LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayNot Available24-hColonUS_06875744_B2
2073
None2005
VALALKALKKALKKLKKALKKAL
Hecate AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayNot Available24-hColonUS_06875744_B2
2069
None2005
VAKKFAKKFKKFAKKFAKFAFAF
D2A21V23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayNot Available24-hColonUS_06875744_B2
2066
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =73 µg/ml24-hColonUS_06875744_B2
2062
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =76 µg/ml24-hColonUS_06875744_B2
2061
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =60 µg/ml24-hColonUS_06875744_B2
2040
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =530 µg/ml24-hColonUS_06875744_B2
2018
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =80 µg/ml24-hColonUS_06875744_B2
2017
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =740 µg/ml24-hColonUS_06875744_B2
1993
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =23 µg/ml24-hColonUS_06875744_B2
1990
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =>1000 µg/ml24-hColonUS_06875744_B2
1985
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =120 µg/ml24-hColonUS_06875744_B2
1978
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =13 µg/ml24-hColonUS_06875744_B2
1977
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16) Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =35 µg/ml24-hColonUS_06875744_B2
1971
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =70 µg/ml24-hColonUS_06875744_B2
1970
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =82 µg/ml24-hColonUS_06875744_B2
1968
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =11 µg/ml24-hColonUS_06875744_B2
1946
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =34 µg/ml24-hColonUS_06875744_B2
1941
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =57 µg/ml24-hColonUS_06875744_B2
1937
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =62 µg/ml24-hColonUS_06875744_B2
1933
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =8 µg/ml24-hColonUS_06875744_B2
1932
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =12 µg/ml24-hColonUS_06875744_B2
1931
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =38 µg/ml24-hColonUS_06875744_B2
1930
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =5 µg/ml24-hColonUS_06875744_B2
1929
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayNot Available24-hColonUS_06875744_B2
1926
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =46 µg/ml24-hColonUS_06875744_B2
1925
None2005
FALALKALKKALKKLKKALKKAL
Hecate AC23LinearLNoneFreeFreeAnticancerFLAK peptidesSW-480Colon CancerMTT/MTS assayLD50 =6 µg/ml24-hColonUS_06875744_B2
1923
None2005
VALALKALKKLAKKLKKLAKKAL
FLAK04 AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =84 µg/ml24-hBreastUS_06875744_B2
1922
None2005
VALALKALKKALKKLKKALKKAL
Hecate AC V23LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =160 µg/ml24-hBreastUS_06875744_B2
1921
None2005
VALALKALKKALKKLKKALKKAL
Hecate AM V23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =340 µg/ml24-hBreastUS_06875744_B2
1917
None2005
VAKKFAKKFKKFAKKFAKFAFAF
D2A21V23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =210 µg/ml24-hBreastUS_06875744_B2
1914
None2005
FAKKLAKKLKKLAKKLAKLAKKL
Anubis-223LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =38 µg/ml24-hBreastUS_06875744_B2
1910
None2005
FAKKFAKKFKKFAKKFAKFAFAF
D2A2123LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =64 µg/ml24-hBreastUS_06875744_B2
1909
None2005
GIGKFLHAAKKFAKAFVAEIMNS
Magainin2wisc23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =22 µg/ml24-hBreastUS_06875744_B2
1888
None2005
FAVGLRAIKRALKKLRRGVRKVAKDL
FAGVL26LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =240 µg/ml24-hBreastUS_06875744_B2
1866
None2005
FAKLWAKLAFGKGIGKVGKKLL
FLAK50 Z422LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =54 µg/ml24-hBreastUS_06875744_B2
1865
None2005
FAKAIAKIAFGKGIGKVGKKLL
FLAK50 Z322LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =>1000 µg/ml24-hBreastUS_06875744_B2
1841
None2005
GIGAVLKVLTTGLPALISWIKRKRQQ
MELITTIIN26LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =9 µg/ml24-hBreastUS_06875744_B2
1838
None2005
KIAKVALAKLGIGAVLKVLTTGL
PYL-ME23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =635 µg/ml24-hBreastUS_06875744_B2
1833
None2005
FAKKLAKKLKKLAKKLIGAVLKV
SHIVA 11[(1-16)ME(2-9]-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =95 µg/ml24-hBreastUS_06875744_B2
1826
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA(1-7) Shiva10(1-16)-COOH23LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =63 µg/ml24-hBreastUS_06875744_B2
1825
None2005
KTKLFKKFAKKLAKKLKKLAKKL
SHIVA 10 (1-16) Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =29 µg/ml24-hBreastUS_06875744_B2
1819
None2005
KWKLFKKKTKLFKKFAKKLAKKL
CA (1-7) Shiva10 (1-16)23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =150 µg/ml24-hBreastUS_06875744_B2
1818
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA 10 PEPTIDE 71 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =93 µg/ml24-hBreastUS_06875744_B2
1816
None2005
FAKKLAKKLKKLAKKLAKKWKL
SHIVA DERIV P69 + KWKL22LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =44 µg/ml24-hBreastUS_06875744_B2
1794
None2005
GIGKFLKKAKKFGKAFVKILKK
MSI-78 AM22LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =31 µg/ml24-hBreastUS_06875744_B2
1789
None2005
FALALKALKKALkkLKKALKKAL
HECATE 2DAc23LinearMixNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =14 µg/ml24-hBreastUS_06875744_B2
1785
None2005
VALALKALKKALKKLKKALKKAL
KAL V23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =72 µg/ml24-hBreastUS_06875744_B2
1781
None2005
FALAKLAKKAKAKLKKALKAL
FLAK05 AM21LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =74 µg/ml24-hBreastUS_06875744_B2
1780
None2005
FALALKALKKLAKKLKKLAKKAL
FLAK04 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =10 µg/ml24-hBreastUS_06875744_B2
1779
None2005
FALALKALKKLLKKLKKLAKKAL
FLAK03 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =26 µg/ml24-hBreastUS_06875744_B2
1778
None2005
FALAAKALKKLAKKLKKLAKKAL
FLAK01 AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =62 µg/ml24-hBreastUS_06875744_B2
1777
None2005
FAKKLAKKLKKLAKKLAKLALAL
SHIVA 10 AC23LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =>1000 µg/ml24-hBreastUS_06875744_B2
1774
None2005
FALALKALKKALKKLKKALKKAL
Hecate AM23LinearLNoneAmidationFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =23 µg/ml24-hBreastUS_06875744_B2
1773
None2005
FALALKALKKALKKLKKALKKAL
Hecate Ac23LinearLNoneFreeFreeAnticancerFLAK peptidesMCF-7Breast CancerMTT/MTS assayLD50 =54 µg/ml24-hBreastUS_06875744_B2
1707
96140661998
ALWKDILKNVGKAAGKAVLNTVTDMVNQ
DRS B428LinearLNoneAmidationFreeAntimicrobialDermaseptins BMCF-7Breast CancerThymidine Incorporation assayCytotoxicity =15 µM6-hBreastNone
1706
96140661998
ALWKNMLKGIGKLAGQAALGAVKTLVGA
DRS B328LinearLNoneFreeFreeAntimicrobialDermaseptins BMCF-7Breast CancerThymidine Incorporation assayCytotoxicity =12 µM6-hBreastNone
1669
157961842005
LRVRLASHLRKLRKRLLRDADDLQKRLAVY
Apo E30LinearLNoneFreeFreeAntibacterialApoprotein ECOLO-201Colon CancerMTT/MTS assay65 % Cytotoxity at 40 µg/ml4-hColonNone
1668
157961842005
LRVRLASHLRKLRKRLLRDADDLQKRLAVY
Apo E30LinearLNoneFreeFreeAntibacterialApoprotein EMKN-7Gastric CancerMTT/MTS assay35 % Cytotoxity at 40 µg/ml4-hStomachNone
1667
157961842005
LRVRLASHLRKLRKRLLRDADDLQKRLAVY
Apo E30LinearLNoneFreeFreeAntibacterialApoprotein EMKN-1Gastric CancerMTT/MTS assay60 % Cytotoxity at 40 µg/ml4-hStomachNone
1666
157961842005
LRVRLASHLRKLRKRLLRDADDLQKRLAVY
Apo E30LinearLNoneFreeFreeAntibacterialApoprotein EPaca-2Pancreatic CancerMTT/MTS assay55 % Cytotoxity at 40 µg/ml4-hPancreaticNone
1665
157961842005
LRVRLASHLRKLRKRLLRDADDLQKRLAVY
Apo E30LinearLNoneFreeFreeAntibacterialApoprotein EPANC-1Pancreatic CancerMTT/MTS assay55 % Cytotoxity at 40 µg/ml4-hPancreaticNone
1664
118359912001
SIGAKILGGVKTFFKGALKELASTYLQ
maximin527LinearLNoneFreeFreeAntimicrobialBombina maximaT-24Bladder CancerMTT/MTS assayIC50=>50 µg/ml48-hBladderNone
1663
118359912001
GIGVLLSAGKAALKGLAKVLAEKYAN
maximin426LinearLNoneAmidationFreeAntimicrobialBombina maximaT-24Bladder CancerMTT/MTS assayIC50=>50 µg/ml48-hBladderNone
1662
118359912001
GIGGKILSGLKTALKGAAKELASTYLH
maximin327LinearLNoneFreeFreeAntimicrobialBombina maximaT-24Bladder CancerMTT/MTS assayIC50 =18 µg/ml48-hBladderNone
1661
118359912001
GIGTKILGGVKTALKGALKELASTYAN
maximin127LinearLNoneAmidationFreeAntimicrobialBombina maximaT-24Bladder CancerMTT/MTS assayIC50 =35.4 µg/ml48-hBladderNone
1660
118359912001
SIGAKILGGVKTFFKGALKELASTYLQ
maximin527LinearLNoneFreeFreeAntimicrobialBombina maximaBIU-87Bladder CancerMTT/MTS assayIC50 =>50 µg/ml48-hBladderNone
1659
118359912001
GIGVLLSAGKAALKGLAKVLAEKYAN
maximin426LinearLNoneAmidationFreeAntimicrobialBombina maximaBIU-87Bladder CancerMTT/MTS assayIC50 =>50 µg/ml48-hBladderNone
1658
118359912001
GIGGKILSGLKTALKGAAKELASTYLH
maximin327LinearLNoneFreeFreeAntimicrobialBombina maximaBIU-87Bladder CancerMTT/MTS assayIC50=28 µg/ml48-hBladderNone
1657
118359912001
GIGTKILGGVKTALKGALKELASTYAN
maximin127LinearLNoneAmidationFreeAntimicrobialBombina maximaBIU-87Bladder CancerMTT/MTS assayIC50=20.5 µg/ml48-hBladderNone
1656
118359912001
SIGAKILGGVKTFFKGALKELASTYLQ
maximin527LinearLNoneFreeFreeAntimicrobialBombina maximaMOLT-4Leukemia CancerMTT/MTS assayIC50 >50 µg/ml48-hBloodNone
1655
118359912001
GIGVLLSAGKAALKGLAKVLAEKYAN
maximin426LinearLNoneAmidationFreeAntimicrobialBombina maximaMOLT-4Leukemia CancerMTT/MTS assayIC50 =53.4 µg/ml48-hBloodNone
1654
118359912001
GIGGKILSGLKTALKGAAKELASTYLH
maximin327LinearLNoneFreeFreeAntimicrobialBombina maximaMOLT-4Leukemia CancerMTT/MTS assayIC50 =25.2 µg/ml48-hBloodNone
1653
118359912001
GIGTKILGGVKTALKGALKELASTYAN
maximin127LinearLNoneAmidationFreeAntimicrobialBombina maximaMOLT-4Leukemia CancerMTT/MTS assayIC50=24.3 µg/ml48-hBloodNone
1652
118359912001
SIGAKILGGVKTFFKGALKELASTYLQ
maximin527LinearLNoneFreeFreeAntimicrobialBombina maximaC8166Leukemia CancerMTT/MTS assayIC50=34.4 µg/ml48-hBloodNone
1651
118359912001
GIGVLLSAGKAALKGLAKVLAEKYAN
maximin426LinearLNoneAmidationFreeAntimicrobialBombina maximaC8166Leukemia CancerMTT/MTS assayIC50=24.2 µg/ml48-hBloodNone
1650
118359912001
GIGGKILSGLKTALKGAAKELASTYLH
maximin327LinearLNoneFreeFreeAntimicrobialBombina maximaC8166Leukemia CancerMTT/MTS assayIC50=11.4 µg/ml48-hBloodNone
1649
118359912001
GIGTKILGGVKTALKGALKELASTYAN
maximin127LinearLNoneAmidationFreeAntimicrobialBombina maximaC8166Leukemia CancerMTT/MTS assayIC50=15.3 µg/ml48-hBloodNone
1549
186563522008
KAQIRAMECNILGRKKRRQRRR
Tat-a522LinearLNoneFreeFreeAnticancerHIV-Tat (49-57)HCT-116Colon CancerMTT/MTS assay~80% Cytotoxicity at 100 µM24-hColonNone
1538
166376462006
IGKEFKRIVQRIKDFLRNLVPRTES
LL-37(13-37)25LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsHBMECProstate CancerMTT/MTS assayLC50=38 µM24-hNot AvailableNone
1532
166376462006
IGKEFKRIVQRIKDFLRNLVPRTES
LL-37(13-37)25LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBOral CancerMTT/MTS assayLC50=40 µM24-hNot AvailableNone
1526
166376462006
IGKEFKRIVQRIKDFLRNLVPRTES
LL-37(13-37)25LinearLNoneFreeFreeAntibacterialLL-37,a series of peptide fragmentsKBvTumorMTT/MTS assayLC50=39 µM24-hNot AvailableNone
1524
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=2.2 µMo/L36-hCervixNone
1523
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=2 µMo/L36-hCervixNone
1522
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=4.3 µMo/L36-hCervixNone
1521
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=3.8 µMo/L36-hCervixNone
1520
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=10.4 µMo/L36-hCervixNone
1519
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=58.6 µMo/L36-hCervixNone
1518
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=64.7 µMo/L36-hCervixNone
1517
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=>83.6 µMo/L36-hCervixNone
1516
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=>83.6 µMo/L36-hCervixNone
1515
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KHeLaCervical CancerMTT/MTS assayIC50=>83.6 µMo/L36-hCervixNone
1514
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=4.6 µMo/L36-hSkinNone
1513
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=4.4 µMo/L36-hSkinNone
1512
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=7.8 µMo/L36-hSkinNone
1511
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=5.2 µMo/L36-hSkinNone
1510
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=11.5 µMo/L36-hSkinNone
1509
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=62.5 µMo/L36-hSkinNone
1508
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=63.5 µMo/L36-hSkinNone
1507
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1506
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1505
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KB-16Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1504
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=2.7 µMo/L36-hLungNone
1503
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=4.1 µMo/L36-hLungNone
1502
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=2.9 µMo/L36-hLungNone
1501
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=4.4 µMo/L36-hLungNone
1500
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=4.7 µMo/L36-hLungNone
1499
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=14 µMo/L36-hLungNone
1498
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=15.6 µMo/L36-hLungNone
1497
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=16.4 µMo/L36-hLungNone
1496
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=37.7 µMo/L36-hLungNone
1495
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KH-1299Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1494
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=5.5 µMo/L36-hMuscleNone
1493
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=6.4 µMo/L36-hMuscleNone
1492
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=9.8 µMo/L36-hMuscleNone
1491
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=7.5 µMo/L36-hMuscleNone
1490
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=25.2 µMo/L36-hMuscleNone
1488
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1489
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1487
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1486
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1484
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=3.5 µMo/L36-hColonNone
1485
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KRDRhabdomyosarcoma CancerMTT/MTS assayIC50=>83.6 µMo/L36-hMuscleNone
1483
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=4.3 µMo/L36-hColonNone
1482
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=5 µMo/L36-hColonNone
1481
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=6.4 µMo/L36-hColonNone
1480
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=11.1 µMo/L36-hColonNone
1479
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1478
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1477
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1476
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1475
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KSW-1116Colorectal CancerMTT/MTS assayIC50=>83.6 µMo/L36-hColonNone
1474
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=5.7 µMo/L36-hBreastNone
1473
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=6.2 µMo/L36-hBreastNone
1472
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=5.1 µMo/L36-hBreastNone
1471
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=5 µMo/L36-hBreastNone
1470
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=15.8 µMo/L36-hBreastNone
1469
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=62.3 µMo/L36-hBreastNone
1468
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=70.8 µMo/L36-hBreastNone
1467
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=>83.6 µMo/L36-hBreastNone
1466
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=>83.6 µMo/L36-hBreastNone
1465
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KMCF-7Breast CancerMTT/MTS assayIC50=>83.6 µMo/L36-hBreastNone
1464
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=7.2 µMo/L36-hSkinNone
1463
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=8.7 µMo/L36-hSkinNone
1462
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=6.5 µMo/L36-hSkinNone
1461
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=4.3 µMo/L36-hSkinNone
1460
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=17.8 µMo/L36-hSkinNone
1458
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=59.8 µMo/L36-hSkinNone
1459
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=58.7 µMo/L36-hSkinNone
1455
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1456
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1457
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-375Skin CancerMTT/MTS assayIC50=>83.6 µMo/L36-hSkinNone
1452
212522882011
KWKSFLKTFKSAKKTVLHTLLKAISS
A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=8.7 µMo/L36-hLungNone
1453
212522882011
KWKSFLKTFKSLKKTVLHTLLKAISS
A12L/A20L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=9.7 µMo/L36-hLungNone
1454
212522882011
KWKSFLKTFKSLKKTVLHTLLKLISS
A12L/A20L/A23L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=9.2 µMo/L36-hLungNone
1449
212522882011
KWKSFAKTFKSAKKTVLHTALKAISS
L6A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=53 µMo/L36-hLungNone
1450
212522882011
KWKSFLKTFKSAKKTVLHTALKAISS
P26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=33 µMo/L36-hLungNone
1451
212522882011
KWKSFLKTFKSLKKTVLHTALKAISS
A12L26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=11.1 µMo/L36-hLungNone
1446
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L17A/L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1447
212522882011
KWKSFLKTFKSAKKTVAHTALKAISS
L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1448
212522882011
KWKSFLKTFKSAKKTVAHTAAKAISS
L21A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=71 µMo/L36-hLungNone
1445
212522882011
KWKSFAKTFKSAKKTVAHTALKAISS
L6A/L17A26LinearLNoneFreeFreeAnticancerPeptideV13KA-549Lung CancerMTT/MTS assayIC50=>83.6 µMo/L36-hLungNone
1438
219552512011
GIIKKIIIKKIIIKKIIIKKI
Cationic Amphiphilic21CyclicLNoneFreeFreeAntimicrobialAMPHL-60Pancreatic CancerWST-1 assayIC50 = 10 µMNot AvailablePancreaticNone
1435
219552512011
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneFreeFreeAntimicrobialXenopus laevisHeLaPancreatic CancerWST-1 assayIC50 = >60 µMNot AvailablePancreaticNone
1434
219552512011
GIIKKIIIKKIIIKKIIIKKI
Cationic Amphiphilic21CyclicLNoneFreeFreeAntimicrobialAMPHeLaPancreatic CancerWST-1 assayIC50 = 4 µMNot AvailablePancreaticNone
1431
162692802005
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntibacterialNK-lysinSW-480Leukemia CancerPI-uptake assayLD50=1-4 µMNot AvailableBloodNone
1430
162692802005
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntibacterialNK-lysinU-937Lymphoma CancerPI-uptake assayLD50=30 µMNot AvailableBloodNone
1429
162692802005
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntibacterialNK-lysinSH-SY5YBrain TumorPI-uptake assayLD50=1-4 µMNot AvailableBrainNone
1428
162692802005
KILRGVCKKIMRTFLRRISKDILTGKK
NK-227LinearLNoneAmidationFreeAntibacterialNK-lysinNB LA-N-1Colorectal CancerPI-uptake assayLD50=1-4 µMNot AvailableColonNone
1425
7768152, 214039171994
GIGKFLKKAKKFGKAFVKILKK
PexigaNAn MSI-7822LinearLNoneAmidationFreeAntimicrobialHelical peptide with a predominance of one or more amino acids tryptophane-richU-937Lymphoma CancerMTT/MTS assay75% Cytotoxicity at 0.5 µg/ml6-hBloodNone
1420
8573171, 214039171996
TRSSRAGLQFPVGRVHRLLRK
Buforin221LinearLNoneAmidationFreeAntimicrobialBufo Bufo GargarizansU-937Lymphoma CancerMTT/MTS assay5% Cytotoxicity at 0.5 µg/ml6-hBloodNone
1413
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisPC-3Prostate CancerTrypan blue assayIC50 >200 µg/ml72-hProstateNone
1412
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisPC-3Prostate CancerTrypan blue assayNot Available72-hProstateNone
1411
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisPC-3Prostate CancerTrypan blue assayNot Available72-hProstateNone
1410
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisPC-3Prostate CancerTrypan blue assayIC50=53 µg/ml72-hProstateNone
1409
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisPC-3Prostate CancerTrypan blue assayIC50=47 µg/ml72-hProstateNone
1408
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisPC-3Prostate CancerTrypan blue assayIC50=41 µg/ml72-hProstateNone
1407
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisMCF-7Breast CancerTrypan blue assayIC50 >200 µg/ml72-hBreastNone
1406
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisMCF-7Breast CancerTrypan blue assayNot Available72-hBreastNone
1405
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisMCF-7Breast CancerTrypan blue assayNot Available72-hBreastNone
1404
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisMCF-7Breast CancerTrypan blue assayIC50=49 µg/ml72-hBreastNone
1403
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisMCF-7Breast CancerTrypan blue assayIC50=42 µg/ml72-hBreastNone
1402
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisMCF-7Breast CancerTrypan blue assayIC50=37 µg/ml72-hBreastNone
1401
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisCHP-100Ewing sarcomaTrypan blue assayIC50 >200 µg/ml72-hBloodNone
1400
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisCHP-100Ewing sarcomaTrypan blue assayNot Available72-hBloodNone
1399
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisCHP-100Ewing sarcomaTrypan blue assayNot Available72-hBloodNone
1398
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisCHP-100Ewing sarcomaTrypan blue assayIC50=45 µg/ml72-hBloodNone
1397
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisCHP-100Ewing sarcomaTrypan blue assayIC50=39 µg/ml72-hBloodNone
1396
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisCHP-100Ewing sarcomaTrypan blue assayIC50=32 µg/ml72-hBloodNone
1395
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisK-562Leukemia CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1394
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisK-562Leukemia CancerTrypan blue assayIC50=112 µg/ml72-hBloodNone
1393
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisK-562Leukemia CancerTrypan blue assayIC50=98 µg/ml72-hBloodNone
1392
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisK-562Leukemia CancerTrypan blue assayIC50=40 µg/ml72-hBloodNone
1391
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisK-562Leukemia CancerTrypan blue assayIC50=37 µg/ml72-hBloodNone
1390
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisK-562Leukemia CancerTrypan blue assayIC50=32 µg/ml72-hBloodNone
1389
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisRajiLymphoma CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1388
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisRajiLymphoma CancerTrypan blue assayIC50=72 µg/ml72-hBloodNone
1387
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisRajiLymphoma CancerTrypan blue assayIC50=64 µg/ml72-hBloodNone
1386
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisRajiLymphoma CancerTrypan blue assayIC50=20 µg/ml72-hBloodNone
1385
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisRajiLymphoma CancerTrypan blue assayIC50=25 µg/ml72-hBloodNone
1384
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisRajiLymphoma CancerTrypan blue assayIC50=23 µg/ml72-hBloodNone
1383
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisMLALeukemia CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1382
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisMLALeukemia CancerTrypan blue assayIC50=102 µg/ml72-hBloodNone
1381
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisMLALeukemia CancerTrypan blue assayIC50=80 µg/ml72-hBloodNone
1380
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisMLALeukemia CancerTrypan blue assayIC50=34 µg/ml72-hBloodNone
1379
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisMLALeukemia CancerTrypan blue assayIC50=33 µg/ml72-hBloodNone
1378
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisMLALeukemia CancerTrypan blue assayIC50=30 µg/ml72-hBloodNone
1377
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisDaudiColon CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1375
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisDaudiBrain TumorTrypan blue assayIC50=115 µg/ml72-hBloodNone
1376
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisDaudiLeukemia CancerTrypan blue assayIC50=143 µg/ml72-hBloodNone
1374
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisDaudiLung CancerTrypan blue assayIC50=30 µg/ml72-hBloodNone
1373
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisDaudiRenal CancerTrypan blue assayIC50=38 µg/ml72-hBloodNone
1372
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisDaudiOvarian CancerTrypan blue assayIC50=28 µg/ml72-hBloodNone
1371
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisSSKT-1Hematopoietic CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1370
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisSSKT-1Hematopoietic CancerTrypan blue assayIC50=109 µg/ml72-hBloodNone
1369
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisSSKT-1Hematopoietic CancerTrypan blue assayIC50=107 µg/ml72-hBloodNone
1367
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisSSKT-1Hematopoietic CancerTrypan blue assayIC50=29 µg/ml72-hBloodNone
1368
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisSSKT-1Hematopoietic CancerTrypan blue assayIC50=23 µg/ml72-hBloodNone
1366
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisSSKT-1Hematopoietic CancerTrypan blue assayIC50=27 µg/ml72-hBloodNone
1365
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevis8402Leukemia CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1364
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevis8402Leukemia CancerTrypan blue assayIC50=83 µg/ml72-hBloodNone
1363
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevis8402Leukemia CancerTrypan blue assayIC50=60 µg/ml72-hBloodNone
1362
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevis8402Leukemia CancerTrypan blue assayIC50=18 µg/ml72-hBloodNone
1361
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevis8402Leukemia CancerTrypan blue assayIC50=16 µg/ml72-hBloodNone
1360
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevis8402Leukemia CancerTrypan blue assayIC50=12 µg/ml72-hBloodNone
1359
1708887, 22853001990
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialXenopus laevisU-937Lymphoma CancerTrypan blue assayIC50 >150 µg/ml72-hBloodNone
1358
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z2424LinearLNoneAmidationFreeAntibacterialXenopus laevisU-937Lymphoma CancerTrypan blue assayIC50=123 µg/ml72-hBloodNone
1357
1708887, 22853001990
ALSKALSKALSKALSKALSKALSK
Z4424LinearLNoneAmidationFreeAntibacterialXenopus laevisU-937Lymphoma CancerTrypan blue assayIC50=97 µg/ml72-hBloodNone
1356
1708887, 22853001990
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisU-937Lymphoma CancerTrypan blue assayIC50=16 µg/ml72-hBloodNone
1355
1708887, 22853001990
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialXenopus laevisU-937Lymphoma CancerTrypan blue assayIC50=19 µg/ml72-hBloodNone
1354
1708887, 22853001990
GIGKFLHAAKKFAKAFVAEIMNS
Magainin B23LinearLNoneAmidationFreeAntibacterialXenopus laevisU-937Lymphoma CancerTrypan blue assayIC50=17 µg/ml72-hBloodNone
1353
184259922008
RKAFRWAWRMLKKAAPSITCVR
mPep122LinearLNoneFreeFreeAntimicrobialBovine lactoferrin (Lf-B)HL-60Skin CancerMTT/MTS assayIC50=8 µM24-hBloodNone
1352
184259922008
FKCRRWQWRMKKLGAPSITCVR
pep122LinearLNoneFreeFreeAntimicrobialBovine lactoferrin (Lf-B)HL-60Prostate CancerMTT/MTS assayIC50=77 µM24-hBloodNone
1314
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin486P(G4)Bladder CancerCell Viability assayIC50=59.4 µM48-hBladderNone
1313
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin647V(G2)Bladder CancerCell Viability assayIC50=31 µM48-hBladderNone
1312
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skinRT4(G1)Bladder CancerCell Viability assayIC50=135.3 µM48-hBladderNone
1311
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin486P(G4)Bladder CancerWST-1 assayIC50=57.8 µM48-hBladderNone
1310
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin647V(G2)Bladder CancerWST-1 assayIC50=52.4 µM48-hBladderNone
1308
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin486P(G4)Bladder CancerLDH leakage assayIC50=28.6 µM48-hBladderNone
1309
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skinRT4(G1)Bladder CancerWST-1 assayIC50=484 µM48-hBladderNone
1307
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skin647V(G2)Bladder CancerLDH leakage assayIC50=54.1 µM48-hBladderNone
1306
164765192006
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntimicrobialAfrican clawed frog Xenopus laevis skinRT4(G1)Bladder CancerLDH leakage assayIC50=32.3 µM48-hBladderNone
1118
83192121993
gigkflkkakkfakafvkiinn
MSI-23822LinearDNoneAmidationFreeAntibacterialAfrican clawed frog Xenopus laevis skinA-549Lung CancerMTT/MTS assayIC50=6 µM48-hLungNone
1117
83192121993
GIGKFLKKAKKFAKAFVKIINN
MSI-13622LinearLNoneAmidationFreeAntibacterialAfrican clawed frog Xenopus laevis skinA-549Lung CancerMTT/MTS assayIC50=10 µM48-hLungNone
1116
83192121993
GIGKFLHSAKKFGKAFVGEIMNS
Magainin 223LinearLNoneAmidationFreeAntibacterialAfrican clawed frog Xenopus laevis skinA-549Lung CancerMTT/MTS assayIC50=110 µM48-hLungNone
1110
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ADU-145Prostate CancerMTT/MTS assayIC50=15.3 µg/ml48-hProstateNone
1108
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASW-620Colon CancerMTT/MTS assayIC50=12.7 µg/ml48-hColonNone
1109
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2APC-3Prostate CancerMTT/MTS assayIC50=12 µg/ml48-hProstateNone
1107
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AKM12Colon CancerMTT/MTS assayIC50=12 µg/ml48-hColonNone
1106
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHT-29Colon CancerMTT/MTS assayIC50=17.6 µg/ml48-hColonNone
1105
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHCT-15Colon CancerMTT/MTS assayIC50=13.2 µg/ml48-hColonNone
1103
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ACOLO-205Colon CancerMTT/MTS assayIC50=11.2 µg/ml48-hColonNone
1104
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHCT-116Colon CancerMTT/MTS assayIC50=14.6 µg/ml48-hColonNone
1102
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialHistone H2ASK-OV-3Ovarian CancerMTT/MTS assayIC50=12.6 µg/ml48-hOvaryNone
1101
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-8Ovarian CancerMTT/MTS assayIC50=13 µg/ml48-hOvaryNone
1100
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-5Ovarian CancerMTT/MTS assayIC50=13.8 µg/ml48-hOvaryNone
1099
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-4Ovarian CancerMTT/MTS assayIC50=17.6 µg/ml48-hOvaryNone
1098
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AOVRCAR-3Ovarian CancerMTT/MTS assayIC50=15.2 µg/ml48-hOvaryNone
1097
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AIGROV1Ovarian CancerMTT/MTS assayIC50=9 µg/ml48-hOvaryNone
1096
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AUO-31Renal CancerMTT/MTS assayIC50=10.6 µg/ml48-hRenalNone
1094
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASN-12CRenal CancerMTT/MTS assayIC50=11.4 µg/ml48-hRenalNone
1095
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ATK-10Renal CancerMTT/MTS assayIC50=13.1 µg/ml48-hRenalNone
1093
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ARFX393Renal CancerMTT/MTS assayIC50=11 µg/ml48-hRenalNone
1092
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ACAKI-1Renal CancerMTT/MTS assayIC50=14.1 µg/ml48-hRenalNone
1091
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AACHNRenal CancerMTT/MTS assayIC50=12 µg/ml48-hRenalNone
1090
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AA-498Renal CancerMTT/MTS assayIC50=10 µg/ml48-hRenalNone
1089
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2A786-0Renal CancerMTT/MTS assayIC50=12.2 µg/ml48-hRenalNone
1088
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AUACC-62Skin CancerMTT/MTS assayIC50=10.6 µg/ml48-hSkinNone
1087
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AUACC-257Skin CancerMTT/MTS assayIC50=12.5 µg/ml48-hSkinNone
1086
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASK-MEL-5Skin CancerMTT/MTS assayIC50=8.9 µg/ml48-hSkinNone
1085
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASK-MEL-2Skin CancerMTT/MTS assayIC50=11.1 µg/ml48-hSkinNone
1083
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMALME-3MSkin CancerMTT/MTS assayIC50=10.9 µg/ml48-hSkinNone
1084
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AM14Skin CancerMTT/MTS assayIC50=15.1 µg/ml48-hSkinNone
1082
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ALOXIMVISkin CancerMTT/MTS assayIC50=9.5 µg/ml48-hSkinNone
1080
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASNB-75Brain TumorMTT/MTS assayIC50=15.5 µg/ml48-hBrainNone
1081
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AU-251Brain TumorMTT/MTS assayIC50=10.6 µg/ml48-hBrainNone
1079
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASNB-19Brain TumorMTT/MTS assayIC50=13.8 µg/ml48-hBrainNone
1078
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASF-539Brain TumorMTT/MTS assayIC50=9.5 µg/ml48-hBrainNone
1077
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASF-295Brain TumorMTT/MTS assayIC50=12.9 µg/ml48-hBrainNone
1076
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASF-268Brain TumorMTT/MTS assayIC50=12.4 µg/ml48-hBrainNone
1075
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H522Lung CancerMTT/MTS assayIC50=11.2 µg/ml48-hLungNone
1074
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H460Lung CancerMTT/MTS assayIC50=12.1 µg/ml48-hLungNone
1073
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H322MLung CancerMTT/MTS assayIC50=10.7 µg/ml48-hLungNone
1072
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H23Lung CancerMTT/MTS assayIC50=10.8 µg/ml48-hLungNone
1071
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI-H226Lung CancerMTT/MTS assayIC50=13.3 µg/ml48-hLungNone
1070
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHOP-92Lung CancerMTT/MTS assayIC50=7.2 µg/ml48-hLungNone
1069
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHOP-62Lung CancerMTT/MTS assayIC50=12.6 µg/ml48-hLungNone
1068
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AEKVXLung CancerMTT/MTS assayIC50=12.1 µg/ml48-hLungNone
1067
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AA-549Lung CancerMTT/MTS assayIC50=11.7 µg/ml48-hLungNone
1066
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AT-47DBreast CancerMTT/MTS assayIC50=23.9 µg/ml48-hBreastNone
1065
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ABT-549Breast CancerMTT/MTS assayIC50=12.9 µg/ml48-hBreastNone
1064
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMDA-NBreast CancerMTT/MTS assayIC50=10.6 µg/ml48-hBreastNone
1063
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMDA-MB-435Breast CancerMTT/MTS assayIC50=11.3 µg/ml48-hBreastNone
1062
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHS578TBreast CancerMTT/MTS assayIC50=11.7 µg/ml48-hBreastNone
1061
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMDA-MB-231Breast CancerMTT/MTS assayIC50=11.3 µg/ml48-hBreastNone
1060
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ANCI/ADR-RESBreast CancerMTT/MTS assayIC50=11.5 µg/ml48-hBreastNone
1059
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMCF-7Breast CancerMTT/MTS assayIC50=15.1 µg/ml48-hBreastNone
1058
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ASRLeukemia CancerMTT/MTS assayIC50=20.2 µg/ml48-hBloodNone
1057
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ARPMI-8226Leukemia CancerMTT/MTS assayIC50=10.5 µg/ml48-hBloodNone
1056
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AMOLT-4Leukemia CancerMTT/MTS assayIC50=17 µg/ml48-hBloodNone
1055
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AK-562Leukemia CancerMTT/MTS assayIC50=8.2 µg/ml48-hBloodNone
1054
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2AHL-60Leukemia CancerMTT/MTS assayIC50=11.3 µg/ml48-hBloodNone
1053
186173232008
RAGLQFPVGRLLRRLLRRLLR
Buforin IIb21LinearLNoneFreeFreeAntibacterialhistone H2ACCRF-CEMLeukemia CancerMTT/MTS assayIC50=14.7 µg/ml48-hBloodNone
1052
1319823, 22853001992
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H889Lung CancerMTT/MTS assayIC50=6.57 µM24-hLungNone
1051
1319823, 22853001992
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H841Lung CancerMTT/MTS assayIC50=11.7 µM24-hLungNone
1050
1319823, 22853001992
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H735Lung CancerMTT/MTS assayIC50=7.23 µM24-hLungNone
1049
1319823, 22853001992
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H678Lung CancerMTT/MTS assayIC50=4.44 µM24-hLungNone
1048
1319823, 22853001992
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H526Lung CancerMTT/MTS assayIC50=10.5 µM24-hLungNone
1047
1319823, 22853001992
GIGKFLHSAKKFAKAFVAEIMNS
Magainin G23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H182Lung CancerMTT/MTS assayIC50=12.5 µM24-hLungNone
1046
1319823, 22853001992
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H889Lung CancerMTT/MTS assayIC50=6.56 µM24-hLungNone
1045
1319823, 22853001992
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H841Lung CancerMTT/MTS assayIC50=9.7 µM24-hLungNone
1044
1319823, 22853001992
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H735Lung CancerMTT/MTS assayIC50=10.4 µM24-hLungNone
1043
1319823, 22853001992
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H678Lung CancerMTT/MTS assayIC50=6.23 µM24-hLungNone
1042
1319823, 22853001992
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H526Lung CancerMTT/MTS assayIC50=11.7 µM24-hLungNone
1041
1319823, 22853001992
AIGKFLHSAKKFGKAFVGEIMNS
Magainin A23LinearLNoneAmidationBeta-alanineAntibacterialAfrican clawed frog Xenopus laevis skinNCI-H182Lung CancerMTT/MTS assayIC50=7.28 µM24-hLungNone
1036
144992712003
FLKLLKKLAAKFLPTIICKISYKC
PTP424LinearLNoneFreeFreeAntibacterialGaegurinMCF-7Breast CancerMTT/MTS assayIC50=18.1 µg/ml96-hBreastNone
1034
144992712003
LLAGLAANFLPTIICKISYKC
PTP121Cyclic(C15-C21)LNoneFreeFreeAntibacterialGaegurinMCF-7Breast CancerMTT/MTS assayIC50=>100 µg/ml96-hBreastNone
1033
144992712003
FLPLLAGLAANFLPTIICKISYKC
GGN624Cyclic(C18-C24)LNoneFreeFreeAntibacterialGaegurinMCF-7Breast CancerMTT/MTS assayIC50=4.88 µg/ml96-hBreastNone
1028
144992712003
FLKLLKKLAAKFLPTIICKISYKC
PTP424LinearLNoneFreeFreeAntibacterialGaegurinHep3BLiver CancerMTT/MTS assayIC50=18.18 µg/ml96-hLiverNone
1025
144992712003
FLPLLAGLAANFLPTIICKISYKC
GGN624Cyclic(C18-C24)LNoneFreeFreeAntibacterialGaegurinHep3BLiver CancerMTT/MTS assayIC50=4.91 µg/ml96-hLiverNone
1026
144992712003
LLAGLAANFLPTIICKISYKC
PTP121Cyclic(C15-C21)LNoneFreeFreeAntibacterialGaegurinHep3BLiver CancerMTT/MTS assayIC50=>100 µg/ml96-hLiverNone
1020
144992712003
FLKLLKKLAAKFLPTIICKISYKC
PTP424LinearLNoneFreeFreeAntibacterialGaegurinPC-3Prostate CancerMTT/MTS assayIC50=18.63 µg/ml96-hProstateNone
1018
144992712003
LLAGLAANFLPTIICKISYKC
PTP121Cyclic(C15-C21)LNoneFreeFreeAntibacterialGaegurin293Renal CancerMTT/MTS assayIC50=>100 µg/ml96-hRenalNone
1017
144992712003
FLPLLAGLAANFLPTIICKISYKC
GGN624Cyclic(C18-C24)LNoneFreeFreeAntibacterialGaegurin293Renal CancerMTT/MTS assayIC50=5.75 µg/ml96-hRenalNone
1012
144992712003
FLKLLKKLAAKFLPTIICKISYKC
PTP424LinearLNoneFreeFreeAntibacterialGaegurin293Renal CancerMTT/MTS assayIC50=26.15 µg/ml96-hRenalNone
1010
144992712003
LLAGLAANFLPTIICKISYKC
PTP121Cyclic(C15-C21)LNoneFreeFreeAntibacterialGaegurin293Renal CancerMTT/MTS assayIC50=>100 µg/ml96-hRenalNone
1009
144992712003
FLPLLAGLAANFLPTIICKISYKC
GGN624Cyclic(C18-C24)LNoneFreeFreeAntibacterialGaegurin293Renal CancerMTT/MTS assayIC50=5.62 µg/ml96-hRenalNone
1004
144992712003
FLKLLKKLAAKFLPTIICKISYKC
PTP424LinearLNoneFreeFreeAntibacterialGaegurinA-549Lung CancerMTT/MTS assayIC50=13.71 µg/ml96-hLungNone
1001
144992712003
FLPLLAGLAANFLPTIICKISYKC
GGN624Cyclic(C18-C24)LNoneFreeFreeAntibacterialGaegurinA-549Lung CancerMTT/MTS assayIC50=6.49 µg/ml96-hLungNone
1002
144992712003
LLAGLAANFLPTIICKISYKC
PTP121Cyclic(C15-C21)LNoneFreeFreeAntibacterialGaegurinA-549Lung CancerMTT/MTS assayIC50= >100 µg/ml96-hLungNone
7723
None2020
LKKWWKKVKGLLGGLLGKVKKVIK
Seq ID No. 17 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticCalu-1Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7724
None2020
RRWVRRVRRVWRRVVRVVRRWVRR
Seq ID No. 26 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticH-460Lung CancerTetrazolium-based assayCell viability < 50% at 20 μM2-hLungUS20200079827A1
7725
None2020
RRWVRRVRRVWRRVVRVVRRWVRR
Seq ID No. 26 from patent ID US202000079827A124LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticCalu-1Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7726
None2020
RRWvRRvRRvWRRvvRvvRRWvRR
Seq ID No. 34 from patent ID US202000079827A124LinearMixNoneFreeFreeAntimicrobial and AnticancerSyntheticNCI-H460Lung CancerTetrazolium-based assayCell viability < 25% at 20 μM2-hLungUS20200079827A1
7727
None2020
RRWvRRvRRvWRRvvRvvRRWvRR
Seq ID No. 34 from patent ID US202000079827A124LinearMixNoneFreeFreeAntimicrobial and AnticancerSyntheticCalu-1Lung CancerTetrazolium-based assayCell viability > 50% at 20 μM2-hLungUS20200079827A1
7754
None2020
RRRRRRRSKAPKVVILSKALEYLQA
IDP-LLCb0125LinearLNoneFreeFreeAnticancerSyntheticNCl-H187Lung CancerMTT/Alamamar-Blue/Hexosaminidase activity testEC50 ~ 5 μM48-72 hLungUS20200239547A1
7755
None2020
RRRRRRRSKAPKVVILSKALEYLQA
IDP-LLCb0125LinearLNoneFreeFreeAnticancerSyntheticNCl-H82Lung CancerMTT/Alamamar-Blue/Hexosaminidase activity testEC50 ~ 2.5 μM48-72 hLungUS20200239547A1
7756
None2020
RRRRRRRSKAPKVVILSKALEYLQA
IDP-LLCb0125LinearLNoneFreeFreeAnticancerSyntheticNCl-H510ALung CancerMTT/Alamamar-Blue/Hexosaminidase activity testEC50 ~ 5 μM48-72 hLungUS20200239547A1
7828
None2023
MQIPQAPWPVVWAVLQLGWRRKKRRQRRR
Sample Peptide 2 from EP3604345B129LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 / WST-8Cell Viability = 3.6% at 25 μM48-hLungEP3604345B1
7831
None2023
MQIPQAPWPVVWAVLQLGWRRKKRRQRRR
Sample Peptide 2 from EP3604345B129LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 4.9% at 25 μM48-hLungEP3604345B1
7835
None2023
MQIPQAPWPVVWAVLQLGWRRKKRRQRRR
Sample Peptide 2 from EP3604345B129LinearLNoneAmidationFreeAnticancerSyntheticA-549Lung CancerCCK-8 / WST-8Cell Viability = 9.1% at 25 μM48-hLungEP3604345B1