Please wait...
| ID | PMID | YEAR | Sequence | Name | Length | Linear/Cyclic | Chirality | Chem-MOD | C-ter MOD | N-ter MOD | Nature | Origin | Cell Line | Cancer Type | Assay | Activity | Testing Time | Tissue Affected | Patents |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 38464729 | 2024 | U7 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | HepG-2 | Liver Cancer | MTT assay | IC50 = 523 µM | 48-h | Liver | None | ||
| 38464729 | 2024 | U7 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | MCF-7 | Breast Cancer | MTT assay | IC50 = 554 µM | 48-h | Breast | None | ||
| 38464729 | 2024 | U7 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | T-47D | Breast Cancer | MTT assay | IC50 = 584 ± 29.99 µM | 48-h | Breast | None | ||
| 38464729 | 2024 | U3 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | HepG-2 | Liver Cancer | MTT assay | IC50 = 561 µM | 48-h | Liver | None | ||
| 38464729 | 2024 | U3 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | T-47D | Breast Cancer | MTT assay | IC50 = 517.6 ± 34.86 µM | 48-h | Breast | None | ||
| 38464729 | 2024 | U3 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | MCF-7 | Breast Cancer | MTT assay | IC50 = 555 µM | 48-h | Breast | None | ||
| 37298595 | 2023 | BK-7 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (D)Pip—(D)-piperidine-2-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-8 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (D)Pip—(D)-piperidine-2-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-5 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (L)Pip—(L)-piperidine-2-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-6 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (L)Pip—(L)-piperidine-2-carboxylic acid;(D)Pip—(D)-piperidine-2-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-3 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Acc = 1-aminocyclohexane-1-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-4 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Acc = 1-aminocyclohexane-1-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-1 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Apc =1-aminocyclopentyl-1-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-2 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Apc =1-aminocyclopentyl-1-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37001908 | 2023 | A11 | 11 | Linear | L | None | Free | Free | Anticancer | Annexin A1 | A-375 | Skin Cancer | Biotin Pull Down assay | Not Available | 24-h | Skin | None | ||
| 37001908 | 2023 | A11 | 11 | Linear | L | None | Free | Free | Anticancer | Annexin A1 | MDA-MB-231 | Breast Cancer | Biotin Pull Down assay | Not Available | 24-h | Breast | None | ||
| 37001908 | 2023 | A11 | 11 | Linear | L | None | Free | Free | Anticancer | Annexin A1 | H-460 | Lung Cancer | Biotin Pull Down assay | Not Available | 24-h | Lung | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HepG-2 | Liver Cancer | Cell Viability assay | IC50 = 34.05 ± 0.53 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HT-29 | Colon Cancer | Cell Viability assay | IC50 = 42.6 ± 4.0 μM | 48-h | Colon | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HeLa | Cervical Cancer | HDAC inhibition assay | IC50 = 0.446±0.095 µM | Not Available | Cervix | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | Huh-7 | Liver Cancer | Cell Viability assay | IC50 = 28.12 ± 1.5 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | Huh-7 | Liver Cancer | Cell Viability assay | IC50 = 43.74 ± 5.4 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HepG-2 | Liver Cancer | Cell Viability assay | IC50 = 52.23 ± 0.9 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HT-29 | Colon Cancer | Cell Viability assay | IC50 = 54.6 ± 2.1 μM | 48-h | Colon | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HeLa | Cervical Cancer | HDAC inhibition assay | IC50 = 0.310±0.064 µM | Not Available | Cervix | None | ||
| 37764521 | 2023 | GE18 | 18 | Linear | L | None | Free | Free | Antimicrobial | Aphanomyces invadans | MCF-7 | Breast Cancer | MTT assay | IC50 = 35.34 µM | 24-h | Breast | None | ||
| 36626098 | 2023 | LFampin265–284 | 20 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | Jurkat | Blood Cancer | MTT assay | cell viability ~ 47% at 10 µM | 6-h | Blood | None | ||
| 36626098 | 2023 | LFampin265–284 | 20 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 50% at 1 µM | 12-h | Liver | None | ||
| 36626098 | 2023 | LFcin17–30 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | Jurkat | Blood Cancer | MTT assay | cell viability ~ 70% at 20 µM | 6-h | Blood | None | ||
| 36626098 | 2023 | LFcin17–30 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 50% at 1 µM | 12-h | Liver | None | ||
| 36509220 | 2023 | KM8-Aib | 18 | Linear | L | Aib = 2-Aminoisobutyric acid | Amidation | Free | Antimicrobial | Synthetic derivative of KM8 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 36509220 | 2023 | KM8 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic derivative of Mastoparan | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 36509220 | 2023 | Mastoparan | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Wasp venom | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 36567478 | 2023 | mtp1 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTS assay | 17.4% decrease in cell viability at 10 μM | 24-h | Lung | None | ||
| 36567478 | 2023 | mtp1 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTS assay | 33.6% decrease in cell viability at 10 μM | 24-h | Breast | None | ||
| 36567478 | 2023 | mtp1 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTS assay | 30.2 % decrease in cell viability at 10 μM | 24-h | Cervix | None | ||
| 37514049 | 2023 | Salamandrin - I | 12 | Linear | L | None | Amidation | Free | Antioxidant | Salamandra salamandra | HL-60 | Leukemia Cancer | LDH leakage assay | Absorbance ~ 2 at 490 nm at 27 27 µM | 48-h | Blood | None | ||
| 37514049 | 2023 | Salamandrin - I | 12 | Linear | L | None | Amidation | Free | Antioxidant | Salamandra salamandra | HL-60 | Leukemia Cancer | MTT assay | IC50 = 27 µM | 48-h | Blood | None | ||
| 36730301 | 2023 | Lasioglossin - III | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Lasioglossum laticeps | HepG-2 | Liver Cancer | Not Available | IC50 = 7.75 μM | Not Available | Liver | None | ||
| 36730301 | 2023 | Lasioglossin - III | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Lasioglossum laticeps | A-549 | Lung Cancer | Not Available | IC50 = 26.36 μM | Not Available | Lung | None | ||
| 36910465 | 2023 | ALA-A2 | 13 | Linear | L | None | Free | Free | Anticancer | Alpha-Lactalbumin | HT-29 | Colon Cancer | MTT assay | ~50% cell viability | 24-h | Colon | None | ||
| 36910465 | 2023 | ALA-A2 | 13 | Linear | L | None | Free | Free | Anticancer | Alpha-Lactalbumin | A-549 | Lung Cancer | MTT assay | ~50% cell viability | 24-h | Lung | None | ||
| 37183466 | 2023 | CM11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Cecropin-Melittin Hybrid Peptide | Raji | Blood Cancer | MTT assay | Survival rate = 51% at 32 μg/ml | 24-h | Blood | None | ||
| 37183466 | 2023 | CM11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Cecropin-Melittin Hybrid Peptide | Jurkat | Blood Cancer | MTT assay | Survival rate = 47% at 32 μg/ml | 24-h | Blood | None | ||
| 36982610 | 2023 | K2-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 9 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K56-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =12 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K6-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =8 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K259-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =10 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K25-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =9 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K259-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =13 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | Leu4-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 > 20 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K2569-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 12 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | Api8-NH2 | 10 | Linear | L | Z =4-aminopiperidine-4-carboxylic acid , U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 > 20 µM | 24-h | Breast | None | ||
| 36678914 | 2023 | trichoderin A analogue 4 | 10 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.5 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A | 10 | Linear | L | MDA = 2-methyl decanoic acid; AHMOD = 2-amino-6-hydroxy-4-methyl-8-oxodecanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderma sp. fungus, strain 05FI48 | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.3 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A | 10 | Linear | L | MDA = 2-methyl decanoic acid; AHMOD = 2-amino-6-hydroxy-4-methyl-8-oxodecanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderma sp. fungus, strain 05FI48 | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.4 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 4 | 10 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.4 μM | 24-h | Pancreas | None | ||
| 36687035 | 2023 | RR-1-R | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 68 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-R | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 73 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | R-1-RR | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 95 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-RR | 11 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 67 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | R-1-RR | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 122 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-RR | 11 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 58 µM | 24-h | Breast | None | ||
| 37818062 | 2023 | P10 | 13 | Linear | L | None | Free | Free | Anticancer | 40S ribosomal protein fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.01 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P09 | 13 | Linear | L | None | Free | Free | Anticancer | Eukaryotic Translation Elongation Factor 1 Gamma (Eef1G) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.07 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P10 | 13 | Linear | L | None | Free | Free | Anticancer | 40S ribosomal protein fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 1.08 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P09 | 13 | Linear | L | None | Free | Free | Anticancer | Eukaryotic Translation Elongation Factor 1 Gamma (Eef1G) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.85 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P08 | 16 | Linear | L | None | Free | Free | Anticancer | Lamin A/C (LMNA) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.92 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P08 | 16 | Linear | L | None | Free | Free | Anticancer | Lamin A/C (LMNA) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.06 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P07 | 13 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.96 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P07 | 13 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.96 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P06 | 18 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.92 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P06 | 18 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.17 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P03 | 13 | Linear | L | None | Free | Free | Anticancer | Triosephosphate Isomerase (TPI) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.98 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P01 | 16 | Linear | L | None | Free | Free | Anticancer | Histone H1.4 (H1-4) Fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.13 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P03 | 13 | Linear | L | None | Free | Free | Anticancer | Triosephosphate Isomerase (TPI) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 1.04 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P04 | 20 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.83 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P01 | 16 | Linear | L | None | Free | Free | Anticancer | Histone H1.4 (H1-4) Fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.84 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P04 | 20 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.86 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P02 | 15 | Linear | L | None | Free | Free | Anticancer | Rho GDP Dissociation Inhibitor Alpha fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.88 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P02 | 15 | Linear | L | None | Free | Free | Anticancer | Rho GDP Dissociation Inhibitor Alpha fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.93 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P05 | 12 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.98 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P05 | 12 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.85 at 50 μg/ml | 48-h | Bone | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant_R5 (R5-Aurm) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | HT-29 | Colon Cancer | MTT assay | 54.22% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant_R5 (R5-Aurm) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | SW-480 | Colon Cancer | MTT assay | 40.62% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_R5 (R5-Aur) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | HT-29 | Colon Cancer | MTT assay | 61.56% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant (Aurm) | 13 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | HT-29 | Colon Cancer | MTT assay | 66.10% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_R5 (R5-Aur) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | SW-480 | Colon Cancer | MTT assay | 43.89% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant (Aurm) | 13 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | SW-480 | Colon Cancer | MTT assay | 51.63% cell viability | 24-h | Colon | None | ||
| 37867694 | 2023 | CH3CO-Ahx-[Pal] | 10 | Linear | L | Ahx = Amino Hexanoic Acid | Amidation | Acetylation | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 31 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | Ahx-[Pal] | 10 | Linear | L | Ahx = Amino Hexanoic Acid | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT assay | IC50 = 119 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | Ahx-[Pal] | 10 | Linear | L | Ahx = Amino Hexanoic Acid | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 40 μM | 24-h | Colon | None | ||
| 36410436 | 2023 | 6F (I113-P122) | 20 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-D | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D5(G45-Y51) | 17 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | IC50 = 19.4 μM | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D3(G45-N52) | 18 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D2(Q44-Y51) | 18 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 12.29 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 16.29 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 17.70 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 22.37 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 32.32 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 29.90 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 32.51 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 52.01 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 28.78 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 41.31 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 33.85 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 30.29 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 15.87 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 62.17 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 31.51 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.459 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.810 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 12.40 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.944 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 23.18 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 4.637 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 42.88 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 23.51 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 20.58 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 20.26 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 22.55 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 47.02 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 25.09 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 17.98 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | MCF-7 | Breast Cancer | MTT assay | IC50 = 26.49 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 11.40 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | HCT-116 | Colon Cancer | MTT assay | IC50 = 8.539 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | U-251-MG | Brain Tumor | MTT assay | IC50 = 20.13 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | H-838 | Lung Cancer | MTT assay | IC50 = 27.71 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | PC-3 | Prostate Cancer | MTT assay | IC50 = 32.13 μM | 24-h | Prostate | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | EJ | Bladder Cancer | MTS assay | 89.6% apoptotic cells at 50 μg/mL | 24-h | Bladder | None | ||
| None | 2022 | MP12 | 12 | Linear | L | None | Free | Free | Antiproliferative | Aphanomyces invadans | Hep-2 | Larynx Cancer | MTT assay | IC50 = 24.7 ± 0.34 μM | Not Available | Larynx | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | EC-109 | Esophageal Cancer | MTS assay | 57.1% apoptotic cells at 50 μg/mL | 24-h | Esophagus | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | HepG-2 | Liver Cancer | MTS assay | 44.2% apoptotic cells at 50 μg/mL | 24-h | Liver | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | HeLa | Cervical cancer | MTS assay | 65.1% apoptotic cells at 50 μg/mL | 24-h | Cervix | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | SW-620 | Colon Cancer | MTT assay | IC50 >27 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | L02 | Colorectal Cancer | MTT assay | IC50 >150 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 10.88 ± 0.72 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | DLD-1 | Colorectal Cancer | MTT assay | IC50 = 2.14 ± 0.28 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | HT-29 | Colorectal Cancer | MTT assay | IC50 = 4.43 ± 0.15 μg/mL | 48-h | Colon | None | ||
| 36212827 | 2022 | Lt-MAP2 | 13 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Derivative of Lataracin-3a | C1498 | Blood Cancer | Cytotoxicity assay | EC50 = 43.9 ± 0.5 µg/mL | 24-h | Blood | None | ||
| 36212827 | 2022 | Lt-MAP2 | 13 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Derivative of Lataracin-3a | K-562 | Blood Cancer | Cytotoxicity assay | EC50 = 44 ± 3 µg/mL | 24-h | Blood | None | ||
| 36426386 | 2022 | [D4K,A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 46 ± 12 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | [D4K,A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 25 ± 1 μM | 24-h | Lung | None | ||
| 36426386 | 2022 | [D4K,A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 31 ± 1 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | [D4K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 20 ± 1 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | [D4K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 12 ± 1 μM | 24-h | Lung | None | ||
| 36426386 | 2022 | [D4K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 15 ± 1 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | Ocellatin-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Leptodactylus nesiotus | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 69 ± 10 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | Ocellatin-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Leptodactylus nesiotus | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 35 ± 1 μM | 24-h | Lung | None | ||
| 36426386 | 2022 | Ocellatin-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Leptodactylus nesiotus | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 51 ± 16 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | [A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 69 ± 18 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | [A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 59 ± 4 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | [A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 30 ± 1 μM | 24-h | Lung | None | ||
| 35209215 | 2022 | RT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Crocodylus siamensis | CaCo-2 | Colon Cancer | MTT assay | IC50 = 29.74 μM | 24-h | Colon | None | ||
| 34999227 | 2022 | LA-C1b | 18 | Linear | L | Lauric acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | LA-C1b | 18 | Linear | L | Lauric acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | OA-C1b | 18 | Linear | L | Octanoic acid acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | OA-C1b | 18 | Linear | L | Octanoic acid acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | LA-C1b | 18 | Linear | L | Lauric acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 34999227 | 2022 | PA-C1b | 18 | Linear | L | Palmitic acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | OA-C1b | 18 | Linear | L | Octanoic acid acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 34999227 | 2022 | PA-C1b | 18 | Linear | L | Palmitic acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 34999227 | 2022 | PA-C1b | 18 | Linear | L | Palmitic acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | Chensinin-1b | 18 | Linear | L | None | Amidation | Free | Antmicrobial and Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | Chensinin-1b | 18 | Linear | L | None | Amidation | Free | Antmicrobial and Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | Chensinin-1b | 18 | Linear | L | None | Amidation | Free | Antmicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 36555235 | 2022 | AC-P19 | 19 | Linear | L | None | Free | Free | Anticancer | Synthetic | H-460 | Lung Cancer | WST-8 assay | IC50 = 49.08 µM | 24-h | Lung | None | ||
| 36483599 | 2022 | Q7 | 15 | Linear | L | None | Free | Free | Anticancer | Pisum sativum | HEC-1-A | Endometrial Cancer | MTT assay | IC50 = 129.82 ± 7.53 μM | 48-h | Endometrium | None | ||
| 36555235 | 2022 | AC-P19 | 19 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | WST-8 assay | IC50 = 52.14 µM | 24-h | Lung | None | ||
| None | 2022 | RF13 | 13 | Linear | L | None | Free | Free | Anticancer | VSP26B of C. striatus | HEp-2 | Larynx Cancer | MTT assay | IC50 = 49.65 µM | 24-h | Larynx | None | ||
| 36555235 | 2022 | AC-P19M | 19 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Synthetic analogue of AC-P19 | H-460 | Lung Cancer | WST-8 assay | IC50 = 6.29 µM | 24-h | Lung | None | ||
| 36555235 | 2022 | AC-P19M | 19 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Synthetic analogue of AC-P19 | A-549 | Lung Cancer | WST-8 assay | IC50 = 9.84 µM | 24-h | Lung | None | ||
| 36183673 | 2022 | GV1001 | 16 | Linear | L | None | Free | Free | Anticancer | Human telomerase reverse transcriptase (hTERT) | A-549 | Lung Cancer | Cell Viability assay | Graph Fig 2A | 24-h | Lung | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | AlamarBlue assay | 75% cell viability at 20 μM | Not Available | Breast | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | AlamarBlue assay | IC50 = 9 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-480 | Colon Cancer | AlamarBlue assay | IC50 = 8 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-620 | Colon Cancer | AlamarBlue assay | IC50 = 9 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | AlamarBlue assay | 80% cell viability at 20 μM | Not Available | Breast | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-620 | Colon Cancer | AlamarBlue assay | IC50 = 40 ± 3 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | AlamarBlue assay | IC50 = 50 ± 3 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-480 | Colon Cancer | AlamarBlue assay | IC50 = 34 ± 2 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | AlamarBlue assay | 50% cell viability at 20 μM | Not Available | Breast | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-620 | Colon Cancer | AlamarBlue assay | IC50 = 10 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | AlamarBlue assay | IC50 = 11 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-480 | Colon Cancer | AlamarBlue assay | IC50 = 12 ± 4 μM | 24-h | Colon | None | ||
| 35094208 | 2022 | CIGB-552 | 20 | Linear | Mix | None | Free | Acetylation | Antitumor | Synthetic | A-549 | Lung Cancer | Sulforhodamine B assay | IC50 = 44.6 μM | 48-h | Lung | None | ||
| 35094208 | 2022 | CIGB-552 | 20 | Linear | Mix | None | Free | Acetylation | Antitumor | Synthetic | NCI-H-460 | Lung Cancer | Sulforhodamine B assay | IC50 = 287.9 μM | 48-h | Lung | None | ||
| 36174494 | 2022 | At12 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 14.0 µM | NA | Lung | None | ||
| 36174494 | 2022 | At12 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 13.4 µM | NA | Liver | None | ||
| 36174494 | 2022 | At11 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 7.6 µM | NA | Liver | None | ||
| 36174494 | 2022 | At11 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 7.9 µM | NA | Lung | None | ||
| 36174494 | 2022 | At10 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.2 µM | NA | Liver | None | ||
| 36174494 | 2022 | At10 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4.4 µM | NA | Lung | None | ||
| 36174494 | 2022 | At9 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 51.7 µM | NA | Liver | None | ||
| 36174494 | 2022 | At9 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 100 µM | NA | Lung | None | ||
| 36174494 | 2022 | At8 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 8.9 µM | NA | Liver | None | ||
| 36174494 | 2022 | At8 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 13.4 µM | NA | Lung | None | ||
| 36174494 | 2022 | At7 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 8.8 µM | NA | Liver | None | ||
| 36174494 | 2022 | At7 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 10.3 µM | NA | Lung | None | ||
| 36174494 | 2022 | At6 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 70.8 µM | NA | Liver | None | ||
| 36174494 | 2022 | At6 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 > 100 µM | NA | Lung | None | ||
| 36174494 | 2022 | At5 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 3.6 µM | NA | Lung | None | ||
| 36174494 | 2022 | At5 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.5 µM | NA | Liver | None | ||
| 36174494 | 2022 | At4 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.5 µM | NA | Liver | None | ||
| 36174494 | 2022 | At4 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 7.2 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; K13L; Q15K], At3 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4.3 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; K13L; Q15K], At3 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.2 µM | NA | Liver | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; Q15K], At2 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 >100 µM | NA | Liver | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; Q15K], At2 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 >100 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25), At1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 > 100 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25), At1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 >100 µM | NA | Liver | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 14.0 ± 1.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-474 | Breast Cancer | MTT assay | IC50 = 15.7 ± 1.5 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 4.2 ± 2.2 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 4.5 ± 0.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 21.1 ± 2.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-474 | Breast Cancer | MTT assay | IC50 = 37.5 ± 1.7 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 3.5 ± 1.5 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 9.0 ± 0.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0667 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 71.2 ± 1.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0667 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-474 | Breast Cancer | MTT assay | IC50 = 92.8 ± 1.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0667 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 88.8 ± 1.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0275 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 34.0 ± 1.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0275 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 44.8 ± 1.1 μM | 24-h | Breast | None | ||
| 34509120 | 2022 | GI-15 | 17 | Linear | L | None | Amidation | LC-Propargylglycine | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 16.6 ± 0.8 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | GI-15 | 17 | Linear | L | None | Amidation | LC-Propargylglycine | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 13.6 ± 0.2 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | CI-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 7.7 ± 0.2 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | CI-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 2.7 ± 0.5 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 26.7 ± 1.3 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 15.6 ± 1.0 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | IR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 > 100 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | IR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 > 100 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 83 ± 9 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | IK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 47±5 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 23 ± 2 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | IK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 29 ± 6 µM | 72-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 72.06 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 71.18 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 193.4 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 167 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 120.6 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 2.94 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 5.28 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 3.07 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.35 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 4.46 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 27.76 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 99.36 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 49.50 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 35.28 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 85.52 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 3.29 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 0.38 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.01 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 0.51 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 2.83 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 22.09 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 24.03 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 22.67 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 27.32 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 25.75 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 2.78 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 2.84 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 3.07 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 2.64 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 2.49 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | H-157 | Lung Cancer | MTT assay | IC50 = 17.40 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 21.31 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | H-838 | Lung Cancer | MTT assay | IC50 = 16.38 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | PC-3 | Prostate Cancer | MTT assay | IC50 = 7.29 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | U251-MG | Brain Tumor | MTT assay | IC50 = 23.24 μM | 24-h | Brain | None | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 15.25 ± 0.80 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 13.04 ± 1.99 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 22.36 ± 6.07 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 14.75 ± 7.35 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 14.52 ± 1.44 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | HepG-2 | Liver Cancer | Resazurin dye assay | IC50 = 31.63 ± 1.56 µM | 48-h | Liver | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 15.05 ± 8.51 µM | 48-h | Breast | US_10550155_B2 | ||
| 35631515 | 2022 | K4F6K4 | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | AnnexinV-FITC/PI double staining assay | apoptotic cells (early and late) increased from 9.59 ± 1.00% to 43.03 ± 2.13% | 12-h | Lung | None | ||
| 35631515 | 2022 | K4F8K4 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 571.87 ± 66.23 μg/mL | 48-h | Lung | None | ||
| 35631515 | 2022 | K4F6K4 | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 62.64 ± 9.55 μg/mL | 48-h | Lung | None | ||
| 35631515 | 2022 | K2F6K2 | 10 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 1146.23 ± 346.83 μg/mL | 48-h | Lung | None | ||
| 35631515 | 2022 | K3F6K3 | 12 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 123.10 ± 35.19 μg/mL | 48-h | Lung | None | ||
| 36364156 | 2022 | PS14 | 14 | Linear | L | None | Free | Free | Anticancer and Anti-inflammatory | Aphanomyces invadans | Hep-2 | Larynx Cancer | LDH leakage assay | 45.56 ± 2% LDH release at 20 µM | 24-h | Larynx | None | ||
| 36364155 | 2022 | PS14 | 14 | Linear | L | None | Free | Free | Anticancer and Anti-inflammatory | Aphanomyces invadans | Hep-2 | Larynx Cancer | MTT assay | IC50 = 21 µM | 24-h | Larynx | None | ||
| 35246961 | 2022 | d-EEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 4.78 ± 0.02 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | d-EEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.29 ± 0.01 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-EEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 0.29 ± 0.01 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 5.84 ± 0.04 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | d-DEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.36 ± 0 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 0.44 ± 0.10 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DHK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 1.24 ± 0.03 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | d-DHK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 0.32 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DHK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.23 ± 0.04 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 9.65 ± 1.20 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.35 ± 0.40 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.23 ± 0.11 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.57 ± 0.24 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.60 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.20 ± 1.84 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.40 ± 0.71 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.19 ± 0.40 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.72 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.20 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 10.40 ± 1.70 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.95 ± 0.35 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.88 ± 1.24 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.59 ± 0.92 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.40 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.65 ± 1.91 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.15 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.75 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 25.00 ± 0 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.35 ± 0.35 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.71 ± 0.13 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 20.45 ± 2.05 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.75 ±0.49 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.02 ± 0.12 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 8.15 ± 0.49 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.60 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.35 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 143.20 ± 80.33 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.45 ± 2.19 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.35 ± 1.06 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 32.88 ± 4.07 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.08 ± 0.18 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.10 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 19.88 ± 2.65 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.70 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.14 ± 0.52 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 13.30 ± 0.99 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.20 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.40 ± 0.85 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 18.88 ± 1.24 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.10 ± 0.57 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.45 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 23.83 ± 0.81 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.18 ± 0.31 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.75 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 21.13 ± 3.01 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.80 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.45 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 39.75 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 4.45 ± 0.49 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 5.20 ± 0.71 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 185 ± 7 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 9.50 ± 0.99 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 117 ± 7 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 21.10 ± 6.93 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 16.05 ± 3.18 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 25.35 ± 2.76 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 11.90 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 55.85 ± 18.88 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 21.45 ± 2.47 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 49.25 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.35 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.30 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 106 ± 14 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 10.95 ± 1.06 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 19.60 ± 3.96 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 28.60 ± 10.75 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.30 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.60 ± 0.85 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 36.48 ± 3.92 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.60 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 5.35 ± 1.91 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.75 ± 1.20 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.70 ± 0 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.05 ± 0.64 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 15.95 ± 0.78 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.90 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.70 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 8.00 ± 0.71 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.30 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.80 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 9.93 ± 0.25 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.57 ± 0.33 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.10 ± 0 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 53 ± 2.83 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.92 ± 0.17 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.70 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 53.25 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 10.75 ± 0.78 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 16.70 ± 2.26 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 18.25 ± 1.06 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.55 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.90 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 17.25 ± 1.06 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.80 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.75 ± 0.92 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 49.38 ± 13.26 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.05 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.75 ± 0.78 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 47.50 ± 11 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 4.95 ± 0.49 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 6.50 ± 0.71 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 78.75 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 10.55 ± 3.46 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 6.25 ± 1.77 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 61.00 ± 1.41 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 6.05 ± 2.76 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 5.55 ± 0.35 µM | 72-h | Breast | None | ||
| 33603033 | 2021 | L. squarrosulus purifed fraction | 19 | Linear | L | None | Free | Free | Anticancer | Lentinus squarrosulus (Mont.) | H-460 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 34531430 | 2021 | PCC-1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Poecilocoris lewisi | G361 | Skin Cancer | MTS assay | IC50 = 57.8 µM | 48-h | Skin | None | ||
| 34531430 | 2021 | PCC-1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Poecilocoris lewisi | SK-Mel-28 | Skin Cancer | MTS assay | IC50 = 50.8 µM | 48-h | Skin | None | ||
| 33981363 | 2021 | 17BIPHE2 | 17 | Linear | L | None | Free | Free | Antimicrobial | Derivative of LL-37 | NCI-H-1975 | Lung Cancer | MTT assay | IC50 = 71.42 µmol/L | 24-h | Lung | None | ||
| 33981363 | 2021 | 17BIPHE2 | 17 | Linear | L | None | Free | Free | Antimicrobial | Derivative of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 34.33 µmol | 24-h | Lung | None | ||
| 33567789 | 2021 | Si1 | 14 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 746.5 ± 7.6 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si1 | 14 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 124.1 ± 8.12 µM | 72-h | Breast | None | ||
| 33428507 | 2021 | L8H6 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 16.4 µM | 24-h | Cervix | None | ||
| 33428507 | 2021 | L9H5-1 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 5.4 µM | 24-h | Cervix | None | ||
| None | 2021 | SKACP003 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-453 | Breast Cancer | MTT assay | IC50 = 156 ± 0.5 µM | 24-h | Breast | None | ||
| None | 2021 | SKACP003 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 212 ± 0.5 µM | 24-h | Breast | None | ||
| None | 2021 | SKACP003 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 193 ± 0.5 µM | 24-h | Breast | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | Sup-B15 | Blood Cancer | Trypan blue assay | IC50 = 90 ± 14 µM | 24-h | Blood | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | RS4;11 | Blood Cancer | Trypan blue assay | IC50 = 184 ± 23 µM | 24-h | Blood | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | Raji | Lymphoma Cancer | Trypan blue assay | IC50 = 89 ± 24 µM | 24-h | Blood | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | Jurkat | Blood Cancer | Trypan blue assay | IC50 = 186 ± 37 µM | 24-h | Blood | None | ||
| 33442881 | 2021 | [Arg]11-VmCT1 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 25.8 ± 5.2 μmol/L | 24-h | Breast | None | ||
| 33442881 | 2021 | [Arg]7-VmCT1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 18.0 ± 2.7 μmol/L | 24-h | Breast | None | ||
| 33442881 | 2021 | [Arg]3-VmCT1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 20.6 ± 3.1 μmol/L | 24-h | Breast | None | ||
| 33442881 | 2021 | VmCT1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Vaejovis mexicanus smithi | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.3 ± 1.4 μmol/L | 24-h | Breast | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | HepG-2 | Liver Cancer | CCK-8 assay | IC50 = 7.0 ± 1.0 µM | 24-h | Liver | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | HeLa | Cervical Cancer | CCK-8 assay | IC50 = 4.7 ± 1.4 µM | 24-h | Cervix | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 6.2 ± 1.4 µM | 24-h | Lung | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | 4T1 | Breast Cancer | CCK-8 assay | IC50 = 7.6 ± 1.3 µM | 24-h | Breast | None | ||
| 34941705 | 2021 | LVTX-9 | 19 | Linear | L | None | Amidation | Free | Anticancer | Lycosa vittata | A-549 | Lung Cancer | CCK-8 assay | IC50 = 51.7 ± 4.3 µM | 24-h | Lung | None | ||
| 33244888 | 2021 | Protonectin-F | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Protonoectin | HCT-116 | Colon Cancer | Resazurin dye assay | CC50 = 9.8 ± 1.2 µM | 24-h | Colon | None | ||
| 33244888 | 2021 | Protonectin-F | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Protonoectin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 16.0 ± 1.2 µM | 24-h | Skin | None | ||
| 33244888 | 2021 | Protonectin | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Parachartergus fraternus | HCT-116 | Colon Cancer | Resazurin dye assay | CC50 = 8.0 ± 0.5 µM | 24-h | Colon | None | ||
| 33244888 | 2021 | Protonectin | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Parachartergus fraternus | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 14.8 ± 0.9 µM | 24-h | Skin | None | ||
| 34309373 | 2021 | N-Ter | 12 | Linear | L | None | Free | Free | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-375 | Skin Cancer | MTT assay | IC50(A-375)> 50.0 μM | 24-h | Skin | None | ||
| 34117917 | 2021 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | N-terminal region of Helicobacter pylori ribosomal protein L1 | HT-29 | Colon Cancer | MTT assay | IC50 ~ 0.5 µg/mL | 24-h | Colon | None | ||
| 34117917 | 2021 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | N-terminal region of Helicobacter pylori ribosomal protein L1 | CT-26 | Colorectal Cancer | MTT assay | IC50 between 0.5 and 1 µg/mL | 24-h | Colon | None | ||
| 33517264 | 2021 | Hepcidin | 20 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Homo sapiens | U-266 | Lymphoma Cancer | MTT assay | NA | NA | Blood | None | ||
| 34796903 | 2021 | A4W-GGN5 | 11 | Linear | L | None | Amidation | Free | Anticancer | Gaegurin 5 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 22.07 ± 1.63 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | A4W-GGN5 | 11 | Linear | L | None | Amidation | Free | Anticancer | Gaegurin 5 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 98.63 ± 1.17 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop2-PS2Aa | 12 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 15.95 ± 0.69 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop1-HCoV-229E | 11 | Linear | L | None | Amidation | Free | Anticancer | Alphacoronavirus (HCoV-229E) | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 125.0 ± 1.32 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop2-PS2Aa | 12 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 92.99 ± 0.98 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop1-PS2Aa | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 106.2 ± 1.67 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop1-PS2Aa | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 23.76 ± 1.25 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | P264-G274 | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 11.28 ± 0.52 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | P264-G274 | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 90.98 ± 0.75 µM | 48-h | Colon | None | ||
| 33245189 | 2021 | Tachyplesin | 17 | Linear | L | None | Amidation | Free | Antibacterial | Horseshoe crab | H-460 | Lung Cancer | MTT assay | IC50 = 25 µg/ml | 24-h | Lung | None | ||
| 33245189 | 2021 | Tachyplesin | 17 | Linear | L | None | Amidation | Free | Antibacterial | Horseshoe crab | A-549 | Lung Cancer | MTT assay | IC50 = 35 µg/ml | 24-h | Lung | None | ||
| 33919639 | 2021 | Pugnin B | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | PC-3 | Prostate Cancer | MTT assay | 90% Cytotoxicity at 100 µM | 24-h | Prostate | None | ||
| 33919639 | 2021 | Pugnin B | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | MCF-7 | Breast Cancer | MTT assay | 5% Cytotoxicity at 100 µM | 24-h | Breast | None | ||
| 33919639 | 2021 | Pugnin A | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | PC-3 | Prostate Cancer | MTT assay | 74% Cytotoxicity at 100 µM | 24-h | Prostate | None | ||
| 33919639 | 2021 | Pugnin A | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | MCF-7 | Breast Cancer | MTT assay | 12% Cytotoxicity at 100 µM | 24-h | Breast | None | ||
| 34867962 | 2021 | SSTP1 | 18 | Linear | L | None | Free | Free | Host Defense Peptide | Indosylvirana aurantiaca | HSC-4 | Tongue Squamous Cell Carcinoma | MTT assay | IC50 = 10.22 μM | 48-h | Tongue | None | ||
| 34867962 | 2021 | SSTP1 | 18 | Linear | L | None | Free | Free | Host Defense Peptide | Indosylvirana aurantiaca | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 4.5 μM | 48-h | Breast | None | ||
| None | 2021 | DN4 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | 191.67 ± 12.02 μM | 24-h | Liver | None | ||
| None | 2021 | DN1 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | 152.17 ± 7.73 μM | 24-h | Liver | None | ||
| 33029595 | 2020 | 2-arm branched peptide | 18 | Linear | L | Branched amide bond in the branching point was formed by the primary amine of lysine. | Free | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | Cell Viability (%) ~ 73.5 ± 2.2 at 30 µg/mL | 48-h | Prostate | None | ||
| 33029595 | 2020 | 2-arm branched peptide | 18 | Linear | L | Branched amide bond in the branching point was formed by the primary amine of lysine. | Free | Free | Antimicrobial | Synthetic | HCT-116 | Colon Cancer | MTT assay | Cell Viability (%) ~ 78.6 ± 10.5 at 30 µg/mL | 48-h | Colon | None | ||
| 33029595 | 2020 | 2-arm branched peptide | 18 | Linear | L | Branched amide bond in the branching point was formed by the primary amine of lysine. | Free | Free | Antimicrobial | Synthetic | Bcap-37 | Breast Cancer | MTT assay | Cell Viability (%) ~ 81.8 ± 8.8 at 30 µg/mL | 48-h | Breast | None | ||
| 33029595 | 2020 | 2-arm branched peptide | 18 | Linear | L | Branched amide bond in the branching point was formed by the primary amine of lysine. | Free | Free | Antimicrobial | Synthetic | SK-HEP-1 | Liver Cancer | MTT assay | Cell Viability (%) ~ 85.7 ± 4.3 at 30 µg/mL | 48-h | Liver | None | ||
| 33029595 | 2020 | (LLKK)4 linear peptide | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | Cell Viability (%) ~ 17.1 ± 5.0 at 30 µg/mL | 48-h | Prostate | None | ||
| 33029595 | 2020 | (LLKK)4 linear peptide | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Bcap-37 | Breast Cancer | MTT assay | Cell Viability (%) ~ 15.07 ± 0.5 at 30 µg/mL | 48-h | Breast | None | ||
| 33029595 | 2020 | (LLKK)4 linear peptide | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colon Cancer | MTT assay | Cell Viability (%) ~ 10.73 ± 2.4 at 30 µg/mL | 48-h | Colon | None | ||
| 33029595 | 2020 | (LLKK)4 linear peptide | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | SK-HEP-1 | Liver Cancer | MTT assay | Cell Viability (%) ~ 14.1 ± 0.8 at 30 µg/mL | 48-h | Liver | None | ||
| 32716104 | 2020 | YT12 | 12 | Linear | L | None | Free | Free | Anticancer | Arthrospira platensis | HT-29 | Colon Cancer | MTT assay | IC50 = 12.5 μM | NA | Colon | None | ||
| 32971958 | 2020 | Gramicidin A | 15 | Linear | Mix | None | NCH2CH2OH | Formylation | Antimicrobial | Aneurinibacillus migulanus | HT-29 | Colon Cancer | MTT assay | IC50 = 9.78 μM | 48-h | Colon | None | ||
| 32567085 | 2020 | LL-37 Analogue 18 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 29.2 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 17 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 19.2 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 16 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 9.8 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 15 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 12.8 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 14 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 12.9 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 13 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 20.0 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 11 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 75 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 12 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 45.5 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 10 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 13.9 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 9 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 18.9 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 8 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 145 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 7 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 12.5 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 6 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 56 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 5 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 10.7 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 4 | 13 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 3.9 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 3 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 29.8 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 33.7 µg/mL | 48-h | Lung | None | ||
| 32567085 | 2020 | LL-37 Analogue 1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic Analog of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 20.1 µg/mL | 48-h | Lung | None | ||
| 33276536 | 2020 | ΔM4 | 20 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | IC50 = 9.31 μM | NA | Skin | None | ||
| 37300579 | 2020 | MP1-Q12K | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analog of Polybia MP1 | A-549 | Lung Cancer | MTT assay | IC50 = 12.5 μM | 24-h | Lung | None | ||
| 37300579 | 2020 | Polybia-MP1 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Polybia paulista | A-549 | Lung Cancer | MTT assay | IC50 = 12.5 μM | 24-h | Lung | None | ||
| 32967114 | 2020 | Figainin 1 | 18 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Boana raniceps | B16-F10 | Skin Cancer | MTT assay | IC50 = 10.5 µM | NA | Skin | None | ||
| 32967114 | 2020 | Figainin 1 | 18 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Boana raniceps | HeLa | Cervical Cancer | MTT assay | IC50 = 11.1 µM | NA | Cervix | None | ||
| 32967114 | 2020 | Figainin 1 | 18 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Boana raniceps | MCF-7 | Breast Cancer | MTT assay | IC50 = 13.7 µM | NA | Breast | None | ||
| 34508563 | 2020 | Temporin-HLa | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Hylarana latouchii | H-460 | Lung Cancer | MTT assay | IC50 = 1.64 ± 0.41 μM | 24-h | Lung | None | ||
| 34508563 | 2020 | Temporin-HLa | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Hylarana latouchii | H-157 | Lung Cancer | MTT assay | IC50 = 15.18 ± 2.98 μM | 24-h | Lung | None | ||
| 34508563 | 2020 | Temporin-HLa | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Hylarana latouchii | NCI-H23 | Lung Cancer | MTT assay | IC50 = 4.96 ± 0.94 μM | 24-h | Lung | None | ||
| 32903706 | 2020 | HX-12C | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic derivative of Temporin-Pta | KB-C2 | Cervical Cancer | MTT assay | IC50 = 6.06 μM | 72-h | Cervix | None | ||
| 32903706 | 2020 | HX-12B | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic derivative of Temporin-Pta | KB-C2 | Cervical Cancer | MTT assay | IC50 = 7.61 μM | 72-h | Cervix | None | ||
| 32903706 | 2020 | HX-12A | 12 | Linear | L | None | Free | Free | Antimicrobial | Synthetic derivative of Temporin-Pta | KB-C2 | Cervical Cancer | MTT assay | IC50 = 6.45 μM | 72-h | Cervix | None | ||
| 32959810 | 2020 | RA-3 | 20 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 44.14 μM | 48-h | Breast | None | ||
| 32959810 | 2020 | RA-3 | 20 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 28.4 μM | 48-h | Breast | None | ||
| 32959810 | 2020 | RA-3 | 20 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U87-MG | Brain Tumor | MTT assay | IC50 = 32.27 μM | 48-h | Brain | None | ||
| 32151609 | 2020 | DIM-LF11-339 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 3.8 ± 0.3 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | DIM-LF11-339 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 4.7 ± 0.3 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | DIM-LF11-339 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 4.8 ± 0.4 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-334 | 16 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 5.0 ± 0.1 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-334 | 16 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 3.4 ± 0.4 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-334 | 16 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 6.6 ± 0.3 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-215 | 17 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 4.6 ± 0.1 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-215 | 17 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 < 1 ± 0.0 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-215 | 17 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 2.7 ± 0.9 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | DIM-LF11-322 | 18 | Linear | L | None | Free | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 4.6 ± 0.1 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | DIM-LF11-322 | 18 | Linear | L | None | Free | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 < 1 ± 0.0 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | DIM-LF11-322 | 18 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 6.3 ± 0.3 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | WM164 | Skin Cancer | MTS assay | LC50 = 4.7 ± 0.2 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 2.5 ± 0.1 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32151609 | 2020 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 4.2 ± 0.2 μM | 24-h | Skin | EP_2943215_B1 | ||
| 32462055 | 2020 | HM-10/10 | 20 | Linear | L | None | Amidation | Acetylation | Anti-inflammatory and Anticancer | Synthetic | CT-26 | Colorectal Cancer | MTS assay | ~60% cell viability at 10 μg/mL | 24-h | Colon | None | ||
| 32126228 | 2020 | Indolicidin-Lys | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 9.5 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Indolicidin-Arg | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 13.7 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | PuroA-Lys | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 12.0 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | PuroA-Arg | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 10.0 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp DiSu | 15 | Cyclic(C1-15) | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 12.3 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W78Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 25.6 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W678Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≥ 65 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W68Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 35.4 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W67Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 32.2 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W8Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 12.0 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W7Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 11.4 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W6Y | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 19.3 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W678A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≥ 65 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W78A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≥ 65 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W68A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≥ 65 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W67A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≥ 65 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W8A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 22.8 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W7A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 48.2 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W6A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 36.5 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W789hW | 13 | Linear | L | 5-hydroxytryptophan | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 44.8 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W7hW | 13 | Linear | L | 5-hydroxytryptophan | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 15.1 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W8hW | 13 | Linear | L | 5-hydroxytryptophan | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 10.7 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W678F | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 24.6 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W678bTA | 13 | Linear | L | β-3-benzothienyl-1-Ala | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 9.6 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-W6hW | 13 | Linear | L | 5-hydroxytryptophan | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 16.1 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-P9A-Lys | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 15.1 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-P9A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 6.8 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-P5A-Lys | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 27.6 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-P5A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 16.2 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-P59A-Lys | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 27.6 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-P59A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 12.5 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-Orn | 13 | Linear | L | Orn = Ornithine | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≤ 6.5 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-Dab | 13 | Linear | L | Dab = 2,4-diaminobutyric acid | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≤ 6.5 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-Lys | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 11.5 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-Dap | 13 | Linear | L | Dap = 2,3-diaminopropionic acid | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 ≥ 65 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-Agb | 13 | Linear | L | Agb = (S)-2-amino-4 guanidinobutyric acid | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 9.6 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-hArg | 13 | Linear | L | Homo-arginine | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 13.3 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrp-Arg | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | Jurkat | Blood Cancer | MTT assay | IC50 = 9.4 μM | 24-h | Blood | None | ||
| 32126228 | 2020 | Tritrpticin | 13 | Linear | L | None | Free | Free | Antimicrobial | Jurkat | Blood Cancer | MTT assay | IC50 = 18.3 μM | 24-h | Blood | None | |||
| 33363118 | 2020 | A4K14 - Citropin 1.1 | 16 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 14.16 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 | 16 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 14.8 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 | 16 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 29.05 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 | 16 | Linear | L | None | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 14.97 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 1 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 11.26 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 1 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 12.48 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 1 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 11.88 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 1 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 8.94 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 2 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 12.55 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 2 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 14.76 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 2 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 12.65 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 2 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 10.14 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 3 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 11.92 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 3 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 12.11 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 3 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 11.93 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 3 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 17.89 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 4 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 10.49 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 4 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 10.51 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 4 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 7.277 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 4 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 8.9 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 5 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 12.42 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 5 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 9.899 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 5 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 8.229 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 5 | 16 | Cyclic | L | S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 11.9 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 6 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 23.78 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 6 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 30.19 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 6 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 34.49 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 6 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 35.84 µM | 24-h | Prostate | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 7 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 12.1 µM | 24-h | Breast | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 7 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | U-87 | Brain Tumor | CCK-8 assay | IC50 = 14.72 µM | 24-h | Brain | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 7 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 16.37 µM | 24-h | Lung | None | ||
| 33363118 | 2020 | A4K14 - Citropin 1.1 - Sp 7 | 16 | Cyclic | L | R8=(R)-2-(7-octenyl)alanine; S5= (S)-2-(4-pentenyl)alanine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | C4-2B | Prostate Cancer | CCK-8 assay | IC50 = 10.23 µM | 24-h | Prostate | None | ||
| 32630734 | 2020 | Kassiniatuerin-3 | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Kassina senegalensis | NCI-H23 | Lung Cancer | MTT assay | IC50 = 4.52 µM | 24-h | Lung | None | ||
| 32630734 | 2020 | Kassiniatuerin-3 | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Kassina senegalensis | H-157 | Lung Cancer | MTT assay | IC50 = 21.54 µM | 24-h | Lung | None | ||
| 32630734 | 2020 | Kassiniatuerin-3 | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Kassina senegalensis | H-460 | Lung Cancer | MTT assay | IC50 = 1.67 µM | 24-h | Lung | None | ||
| 32630734 | 2020 | Kassiniatuerin-3 | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Kassina senegalensis | H-838 | Lung Cancer | MTT assay | IC50 = 10.03 µM | 24-h | Lung | None | ||
| 32630734 | 2020 | Kassiniatuerin-3 | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Kassina senegalensis | LNCaP | Prostate Cancer | MTT assay | IC50 = 3.79 µM | 24-h | Prostate | None | ||
| 32630734 | 2020 | Kassiniatuerin-3 | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Kassina senegalensis | U251-MG | Brain Tumor | MTT assay | IC50 = 13.20 µM | 24-h | Brain | None | ||
| 30862544 | 2019 | GM15 | 15 | Linear | L | None | Free | Free | Antioxidant | Arthrospira platensis | KB | Oral Cancer | MTT assay | ~ 35% cell viability at 25 μM | 24-h | Not Available | None | ||
| None | 2019 | LPSBD-2 | 20 | Linear | L | None | Free | Free | Anticancer | Synthetic | THP-1 | Leukemia Cancer | Not Available | Not Available | 24-h | Blood | None | ||
| 31909181 | 2019 | AP1-Z9 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 2A | 24-h | Breast | None | ||
| 31909181 | 2019 | AP1-Z9 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | A-375 | Skin Cancer | MTT assay | Graph Figure 2B | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z9 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | U-87 | Brain Tumor | MTT assay | Graph Figure 2C | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z7 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | A-375 | Skin Cancer | MTT assay | Graph Figure 2B | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z7 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | U-87 | Brain Tumor | MTT assay | Graph Figure 2C | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z3b | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | A-375 | Skin Cancer | MTT assay | Graph Figure 2B | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z3b | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | U-87 | Brain Tumor | MTT assay | Graph Figure 2C | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z7 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 2A | 24-h | Breast | None | ||
| 31909181 | 2019 | AP1-Z3a | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | A-375 | Skin Cancer | MTT assay | Graph Figure 2B | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z3a | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | U-87 | Brain Tumor | MTT assay | Graph Figure 2C | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z3b | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 2A | 24-h | Breast | None | ||
| 31909181 | 2019 | AP1-Z5b | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | U-87 | Brain Tumor | MTT assay | IC50 = 3.115 μM | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z3a | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 2A | 24-h | Breast | None | ||
| 31909181 | 2019 | AP1-Z5a | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | U-87 | Brain Tumor | MTT assay | Graph Figure 2C | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z5b | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 1.037 μM | 24-h | Breast | None | ||
| 31909181 | 2019 | AP1-Z5b | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | A-375 | Skin Cancer | MTT assay | IC50 = 2.607 μM | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z5a | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 2A | 24-h | Breast | None | ||
| 31909181 | 2019 | AP1-Z5a | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | Mutant of APR-Z1 | A-375 | Skin Cancer | MTT assay | Graph Figure 2B | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z1 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | AcrAP1 from the venom of the Arabian scorpion | A-375 | Skin Cancer | MTT assay | IC50 = 9.478 μM | 24-h | Skin | None | ||
| 31909181 | 2019 | AP1-Z1 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | AcrAP1 from the venom of the Arabian scorpion | U-87 | Brain Tumor | MTT assay | IC50 = 10.21 μM | 24-h | Brain | None | ||
| 31909181 | 2019 | AP1-Z1 | 18 | Linear | L | None | Amidation | Amidation | Antimicrobial | AcrAP1 from the venom of the Arabian scorpion | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.222 μM | 24-h | Breast | None | ||
| 31714739 | 2019 | [I11F-G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 5.1 ± 0.3 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | [I11F-G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 1.9 ± 0.1 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | [I11F-G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 2.9 ± 0.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [I11F-G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 3.2 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [I11F-G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.3 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 6.7 ± 1.1 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | [G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 1.7 ± 0.1 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | [G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 3.2 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [G18K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.0 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R9S-R14S-R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 4.8 ± 0.3 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | [R9S-R14S-R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 11.1 ± 0.9 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R9S-R14S-R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 11.8 ± 0.9 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 12.2 ± 0.4 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | [R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 4.5 ± 0.3 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 1.8 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 1.2 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R17S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.8 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R14S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 7.5 ± 0.3 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | [R14S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 3.5 ± 0.3 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R14S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R14S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 2.3 ± 0.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R14S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.7 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R9S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 5.3 ± 0.6 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [Y8S-I11S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 13.2 ± 0.9 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | [Y8S-I11S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 28.2 ± 2.0 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [Y8S-I11S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 27.8 ± 2.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [Y8S-I11S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 17.3 ± 1.0 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [W2S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 22.5 ± 2.1 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | [W2S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.2 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | [W2S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 18.9 ± 0.9 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [W2S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 3.9 ± 0.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [W2S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 3.0 ± 0.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [W2S]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 2.0 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R/K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 13.4 ± 1.9 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | [R/K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 2.5 ± 0.1 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | [R/K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 3.5 ± 0.4 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | [R/K]cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 4.3 ± 0.3 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 6.7 ± 0.6 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 6.4 ± 0.6 µM | 24-h | Breast | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 2.0 ± 0.1 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.3 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 1.4 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | cT1 | 18 | Cyclic | L | None | Cyclized | Cyclized | Host Defense Peptide | Synthetic | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.3 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 13.1 ± 1.2 µM | 24-h | Cervix | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 16.0 ± 2.0 µM | 24-h | Breast | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 1.7 ± 0.1 µM | 24-h | Blood | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | MDA-MB-435S | Skin Cancer | Resazurin dye assay | CC50 = 8.0 ± 0.6 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | WM164 | Skin Cancer | Resazurin dye assay | CC50 = 2.5 ± 0.1 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | HT-144 | Skin Cancer | Resazurin dye assay | CC50 = 1.7 ± 0.2 µM | 24-h | Skin | None | ||
| 31714739 | 2019 | T1 | 17 | Linear | L | None | Amidation | Free | Host Defense Peptide | Horseshoe Crab | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.5 ± 0.1 µM | 24-h | Skin | None | ||
| 30612735 | 2019 | Phylloseptin-PBa3 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | H-838 | Lung Cancer | MTT assay | Cell viability ~ 65% at 10-5 M | 72-h | Lung | None | ||
| 30612735 | 2019 | Phylloseptin-PBa3 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 208 µM | 72-h | Breast | None | ||
| 30612735 | 2019 | Phylloseptin-PBa1 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | H-838 | Lung Cancer | MTT assay | Cell viability ~ 65% at 10-5 M | 72-h | Lung | None | ||
| 30612735 | 2019 | Phylloseptin-PBa1 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | H-460 | Lung Cancer | MTT assay | Cell viability < 50% at 10-5 M | 72-h | Lung | None | ||
| 30612735 | 2019 | Phylloseptin-PBa1 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | DU-145 | Prostate Cancer | MTT assay | Cell viability ~ 50% at 10-5 M | 72-h | Prostate | None | ||
| 30612735 | 2019 | Phylloseptin-PBa1 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | U251-MG | Brain Tumor | MTT assay | Cell viability ~ 40% at 10-5 M | 72-h | Brain | None | ||
| 30612735 | 2019 | Phylloseptin-PBa1 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 0.50 µM | 72-h | Breast | None | ||
| 30612735 | 2019 | Phylloseptin-PBa3 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | H-838 | Lung Cancer | MTT assay | Cell viability ~ 65% at 10-5 M | 72-h | Lung | None | ||
| 30612735 | 2019 | Phylloseptin-PBa3 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | H-460 | Lung Cancer | MTT assay | Cell viability ~ 60% at 10-5 M | 72-h | Lung | None | ||
| 30612735 | 2019 | Phylloseptin-PBa2 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | U251-MG | Brain Tumor | MTT assay | Cell viability ~ 60% at 10-5 M | 72-h | Brain | None | ||
| 30612735 | 2019 | Phylloseptin-PBa2 | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa burmeisteri | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 0.29 µM | 72-h | Breast | None | ||
| 30563041 | 2018 | B11 | 15 | Linear | L | None | Free | Free | Antimicrobial | Litopenaeus vannamei hemocyanin-derived peptide | EC-109 | Esophageal Cancer | MTS assay | Decreased cell viability by 13% at 50 μg/mL | 24-h | Esophagus | None | ||
| 30563041 | 2018 | B11 | 15 | Linear | L | None | Free | Free | Antimicrobial | Litopenaeus vannamei hemocyanin-derived peptide | HepG-2 | Liver Cancer | MTS assay | Decreased cell viability by 23% at 50 μg/mL | 24-h | Liver | None | ||
| 30563041 | 2018 | B11 | 15 | Linear | L | None | Free | Free | Antimicrobial | Litopenaeus vannamei hemocyanin-derived peptide | HeLa | Cervical Cancer | MTS assay | Decreased cell viability by 20% at 50 μg/mL | 24-h | Cervix | None | ||
| 30031283 | 2018 | RT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Crocodylus siamensis | HCT-116 | Colon Cancer | MTT assay | IC50 = 90.25 μg/mL | 24-h | Colon | None | ||
| 30031283 | 2018 | KT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Crocodylus siamensis | HCT-116 | Colon Cancer | MTT assay | IC50 = 90.25 μg/mL | 24-h | Colon | None | ||
| 28254375 | 2018 | TP | 16 | Linear | L | None | Free | Free | Antimicrobial | Tibetan swine | NB-4 | Leukemia Cancer | MTT assay | IC50 = 11.479 μM | 48-h | Blood | None | ||
| 28254375 | 2018 | TP | 16 | Linear | L | None | Free | Free | Antimicrobial | Tibetan swine | MKN-45 | Gastric Cancer | MTT assay | IC50 = 4.686 μM | 48-h | Stomach | None | ||
| 30123940 | 2018 | SmacN7-Arg8 fused peptide P5 | 18 | Cyclic | L | Ahx = aminohexanoic acid; Lactam Bridge between K2 and E10 | Amidation | Free | Anticancer | Synthetic | U-266 | Skin Cancer | Cell Titer Blue Cell Viability assay | Cell viability < 50% at 50 μM | 48-h | Skin | None | ||
| 30123940 | 2018 | SmacN7-Arg8 fused peptide P4 | 18 | Cyclic | L | Ahx = aminohexanoic acid; Lactam Bridge between K6 and E18 | Amidation | Free | Anticancer | Synthetic | U-266 | Skin Cancer | Cell Titer Blue Cell Viability assay | Cell viability < 50% at 50 μM | 48-h | Skin | None | ||
| 29993185 | 2018 | Peptide13 Gonearrestide | 18 | Linear | L | None | Amidation | Free | Anticancer | Androctonus mauritanicus | U-251 | Brain tumor | MTT assay | Not Available | 24-h | Brain | None | ||
| 29993185 | 2018 | Peptide13 Gonearrestide | 18 | Linear | L | None | Amidation | Free | Anticancer | Androctonus mauritanicus | Dks8 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide13 Gonearrestide | 18 | Linear | L | None | Amidation | Free | Anticancer | Androctonus mauritanicus | DLD-1 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide13 Gonearrestide | 18 | Linear | L | None | Amidation | Free | Anticancer | Androctonus mauritanicus | HKe-3 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide13 Gonearrestide | 18 | Linear | L | None | Amidation | Free | Anticancer | Androctonus mauritanicus | HCT-116 | Colon Cancer | MTT assay | IC50 ~ 100 μM/L | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide6 Gonearrestide | 12 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | U-251 | Brain tumor | MTT assay | Not Available | 24-h | Brain | None | ||
| 29993185 | 2018 | Peptide6 Gonearrestide | 12 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | Dks8 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide6 Gonearrestide | 12 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | HKe-3 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide6 Gonearrestide | 12 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | DLD-1 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide6 Gonearrestide | 12 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | HCT-116 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide4 Gonearrestide | 18 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | U-251 | Brain tumor | MTT assay | Not Available | 24-h | Brain | None | ||
| 29993185 | 2018 | Peptide4 Gonearrestide | 18 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | Dks8 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide4 Gonearrestide | 18 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | HKe-3 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide4 Gonearrestide | 18 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | DLD-1 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 29993185 | 2018 | Peptide4 Gonearrestide | 18 | Linear | L | None | Free | Free | Anticancer | Androctonus australis | HCT-116 | Colon Cancer | MTT assay | Not Available | 24-h | Colon | None | ||
| 30409511 | 2018 | Pantinin-3 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | DU-145 | Prostate Cancer | MTS assay | IC50 = 17.3 ± 1.0 µM | 24-h | Prostate | None | ||
| 30409511 | 2018 | Pantinin-3 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 13.5 ± 2.0 µM | 24-h | Breast | None | ||
| 30409511 | 2018 | Pantinin-2 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | DU-145 | Prostate Cancer | MTS assay | IC50 = 16.5 ± 1.0 µM | 24-h | Prostate | None | ||
| 30409511 | 2018 | Pantinin-2 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 12.5 ± 1.0 µM | 24-h | Breast | None | ||
| 30409511 | 2018 | Pantinin-1 | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | DU-145 | Prostate Cancer | MTS assay | IC50 = 47.5 ± 2.0 µM | 24-h | Prostate | None | ||
| 30318506 | 2018 | IL13Rα2 D1 peptide | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | U-118 | Brain Cancer | MTT assay | inhibited IL13-stimulated cell adhesion | 48-h | Brain | None | ||
| 30409511 | 2018 | Pantinin-1 | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 28.5 ± 1.0 µM | 24-h | Breast | None | ||
| 30318506 | 2018 | IL13Rα2 D1 peptide | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | U-87 | Brain Cancer | MTT assay | inhibited IL13-stimulated cell adhesion | 48-h | Brain | None | ||
| 30318506 | 2018 | IL13Rα2 D1 peptide | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | SW-620 | Colorectal Cancer | MTT assay | inhibited IL13-stimulated cell adhesion | 48-h | Colon | None | ||
| 30318506 | 2018 | IL13Rα2 D1 peptide | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | KM12SM | Colorectal Cancer | MTT assay | inhibited IL13-stimulated cell adhesion | 48-h | Colon | None | ||
| 30026168 | 2018 | [G7,10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 >100 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G7,10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 = 21.3 ± 1.13 µM | 24-h | Breast | None | ||
| 30026168 | 2018 | [G7,10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 >100 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G4,7,10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 >100 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G4,7,10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 >100 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G4,7,10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 = 26.33 ± 5.8 µM | 24-h | Breast | None | ||
| 30026168 | 2018 | [G4,7a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 >100 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G4,7a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 = 37.3 ± 3.5 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 =24.3 ± 0.8 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G4,7a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 = 29.5 ± 6.03 µM | 24-h | Breast | None | ||
| 30026168 | 2018 | [G10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 = 16.2 ± 2.2 µM | 24-h | Breast | None | ||
| 30026168 | 2018 | [G10a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 = 22.7 ± 0.86 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G7a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 >100 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G7a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 >100 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G7a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 =22.4 ± 2.2 µM | 24-h | Breast | None | ||
| 30026168 | 2018 | [G4a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | NCI-H-460 | Lung Cancer | MTT assay | IC50 >100 µM | 24-h | Lung | None | ||
| 30026168 | 2018 | [G4a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | HeLa | Cervical Cancer | MTT assay | IC50 >100 µM | 24-h | Cervix | None | ||
| 30026168 | 2018 | [G4a]SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic analogue of Temporin-1SHa | MCF-7 | Breast Cancer | MTT assay | IC50 = 17.9 ± 1.1 µM | 24-h | Breast | None | ||
| 29842923 | 2018 | Temporin-CPa | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | 4T1 | Breast Cancer | MTS assay | LC50 = 80 μM | Not Available | Breast | None | ||
| 29842923 | 2018 | Temporin-1Oc | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTS assay | LC50 = 50 μM | Not Available | Cervix | None | ||
| 29842923 | 2018 | Temporin-1Ga | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | 4T1 | Breast Cancer | MTS assay | LC50 = 20 μM | Not Available | Breast | None | ||
| 29842923 | 2018 | Temporin-1OLa | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTS assay | LC50 = 25 μM | Not Available | Cervix | None | ||
| 29842923 | 2018 | Temporin-1Oc | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | 4T1 | Breast Cancer | MTS assay | LC50 = 65 μM | Not Available | Breast | None | ||
| 29904274 | 2018 | cMP-C | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 13.66 μM | 24-h | Breast | None | ||
| 29904274 | 2018 | cMP-C | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 13.87 μM | 24-h | Skin | None | ||
| 29904274 | 2018 | cMP-C | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 13.87 μM | 24-h | Prostate | None | ||
| 29904274 | 2018 | cMP-C | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U-251-MG | Brain tumor | MTT assay | IC50 = 8.56 μM | 24-h | Brain | None | ||
| 29904274 | 2018 | Mastoparan-C | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Vespa crabro | U-251-MG | Brain tumor | MTT assay | IC50 = 36.65 μM | 24-h | Brain | None | ||
| 29904274 | 2018 | Mastoparan-C | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Vespa crabro | MCF-7 | Breast Cancer | MTT assay | IC50 = 25.27 μM | 24-h | Breast | None | ||
| 29904274 | 2018 | cMP-C | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 7.02 μM | 24-h | Lung | None | ||
| 29904274 | 2018 | Mastoparan-C | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Vespa crabro | H-157 | Lung Cancer | MTT assay | IC50 = 13.57 μM | 24-h | Lung | None | ||
| 29904274 | 2018 | Mastoparan-C | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Vespa crabro | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 27.70 μM | 24-h | Skin | None | ||
| 29904274 | 2018 | Mastoparan-C | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Vespa crabro | PC-3 | Prostate Cancer | MTT assay | IC50 = 6.29 μM | 24-h | Prostate | None | ||
| 29191658 | 2018 | temporin-PEa | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | PC-3 | Prostate Cancer | MTT assay | IC50 = 27.62 μM | Not Available | Prostate | None | ||
| 29191658 | 2018 | temporin-PEa | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 9.864 μM | Not Available | Skin | None | ||
| 29191658 | 2018 | temporin-PEa | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | U251-MG | Brain Tumor | MTT assay | IC50 = 3.520 μM | Not Available | Brain | None | ||
| 29191658 | 2018 | temporin-PEa | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of Temporin-PE | NCI-H-157 | Lung Cancer | MTT assay | IC50 = 3.398 μM | Not Available | Lung | None | ||
| 29191658 | 2018 | Temporin-PE | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pelophylax kl. esculentus | MDA-MB-435S | Skin Cancer | MTT assay | IC50 = 33.23 μM | Not Available | Skin | None | ||
| 29191658 | 2018 | Temporin-PE | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pelophylax kl. esculentus | PC-3 | Prostate Cancer | MTT assay | IC50 = 38.56 μM | Not Available | Prostate | None | ||
| 29191658 | 2018 | Temporin-PE | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pelophylax kl. esculentus | U251-MG | Brain Tumor | MTT assay | IC50 = 25.13 μM | Not Available | Brain | None | ||
| 29191658 | 2018 | Temporin-PE | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pelophylax kl. esculentus | NCI-H-157 | Lung Cancer | MTT assay | IC50 = 34.56 μM | Not Available | Lung | None | ||
| 28636781 | 2018 | Bombinin H-BO | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | A-549 | Lung Cancer | MTT assay | Cell Viability ~ 20% at 5 μM | 48-h | Lung | None | ||
| 28636781 | 2018 | Bombinin H-BO | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | A-375 | Skin Cancer | MTT assay | Cell Viability < 20% at 5 μM | 48-h | Skin | None | ||
| 28636781 | 2018 | Bombinin H-BO | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | Huh-7 | Liver Cancer | MTT assay | IC50 = 3.87 μM | 48-h | Liver | None | ||
| 28636781 | 2018 | Bombinin H-BO | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | PC-3 | Prostate Cancer | MTT assay | Cell Viability ~ 40% at 2.5 μM | 48-h | Prostate | None | ||
| 28636781 | 2018 | Bombinin H-BO | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | SK-HEP-1 | Liver Cancer | MTT assay | IC50 = 0.99 μM | 48-h | Liver | None | ||
| 28636781 | 2018 | Bombinin H-BO | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.88 μM | 48-h | Liver | None | ||
| 29515106 | 2018 | TAT-327 | 18 | Linear | L | None | Free | Free | Anticancer | Peptide-327 | SW-620 | Colorectal Cancer | CCK-8 assay | EC50 = 64.61 ± 1.63 μM | 12-h | Colon | None | ||
| 29515106 | 2018 | TAT-327 | 18 | Linear | L | None | Free | Free | Anticancer | Peptide-327 | HT-29 | Colon Cancer | CCK-8 assay | EC50 = 74.08 ± 0.63 μM | 12-h | Colon | None | ||
| 29515106 | 2018 | TAT-327 | 18 | Linear | L | None | Free | Free | Anticancer | Peptide-327 | HepG-2 | Liver Cancer | CCK-8 assay | EC50 = 68.52 ± 2.96 μM | 12-h | Liver | None | ||
| 29515106 | 2018 | TAT-327 | 18 | Linear | L | None | Free | Free | Anticancer | Peptide-327 | Colo-320 | Colon Cancer | CCK-8 assay | EC50 = 68.40 ± 0.42 μM | 12-h | Colon | None | ||
| 29515106 | 2018 | TAT-327 | 18 | Linear | L | None | Free | Free | Anticancer | Peptide-327 | A-549 | Lung Cancer | CCK-8 assay | EC50 = 55.42 ± 0.84 μM | 12-h | Lung | None | ||
| 29098406 | 2018 | Bombinin-H-BO1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | Huh-7 | Liver Cancer | MTT assay | IC50 = 8.42 μM | 48-h | Liver | None | ||
| 29098406 | 2018 | Bombinin-H-BO1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | HepG-2 | Liver Cancer | MTT assay | IC50 = 8.08 μM | 48-h | Liver | None | ||
| 29098406 | 2018 | Bombinin-H-BO1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Bombina orientalis | SK-HEP-1 | Liver Cancer | MTT assay | IC50 = 3.61 μM | 48-h | Liver | None | ||
| 28811617 | 2017 | L-K6 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Temporin 1CEb analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 31 μM | 24-h | Breast | None | ||
| 28249727 | 2017 | Maximin H5 | 20 | Linear | L | None | Amidation | Free | Host defense peptide | Bombina maxima | T98G | Human glioblastoma | MTS assay | IC50 = 125 µM | 72-h | Brain | None | ||
| 28719744 | 2017 | PTP-7S | 16 | Linear | L | None | Free | Free | Anticancer | PTP-7 | A-549 | Lung Cancer | MTT assay | 65% cell viability at 10 µΜ | 6-h | Lung | None | ||
| 28719744 | 2017 | PTP-7S | 16 | Linear | L | None | Free | Free | Anticancer | PTP-7 | HeLa | Cervical Cancer | MTT assay | 55 - 60% cell viability at 75 µM | 24-h | Cervix | None | ||
| 28850103 | 2017 | Phylloseptin-PHa | 19 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Pithecopus hypochondrialis | NCI-H-157 | Lung Cancer | MTT assay | IC50 = 14.10 μM | 24-h | Lung | None | ||
| 28850103 | 2017 | Phylloseptin-PTa | 19 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Phyllomedusa tarsius | NCI-H-157 | Lung Cancer | MTT assay | IC50 = 6.73 μM | 24-h | Lung | None | ||
| 36982972 | 2017 | cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.1 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 15.3 ± 1.4 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 2.9 ± 0.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 > 64 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 39.8 ± 1.0 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [Y7W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 3.9 ± 0.2 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [Y7W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 > 64 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [Y7W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 5.1 ± 0.3 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 2.7 ± 0.1 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [Y7W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 23.3 ± 0.4 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 50.4 ± 2.4 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 4.0 ± 0.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 30.3 ± 1.1 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 3.1 ± 0.1 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 5.0 ± 0.3 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 39.4 ± 2.6 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 29.4 ± 1.1 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [Y7W, K8R, Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 3.9 ± 0.1 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [Y7W, K8R, Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 15.1 ± 1.4 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | [Y7W, K8R, Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 41.0 ± 4.2 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [Y7W, K8R, Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 31.6 ± 1.3 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [Y7W, K8R, Y14W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 5.4 ± 0.3 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [R4A, R18A]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HL-60 | Leukemia Cancer | Resazurin dye assay | CC50 = 34.1 ± 3.9 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [R4A, R18A]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 11.5 ± 0.6 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [R4A, R18A]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 48.4 ± 0.7 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | [R4A, R18A]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 10.3 ± 1.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [R4A, R18A]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 > 64 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [R4A, R18A]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 > 64 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [G1K, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HL-60 | Leukemia Cancer | Resazurin dye assay | CC50 = 9.0 ± 1.1μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [G1K, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 2.1 ± 0.2 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [G1K, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 6.7 ± 0.7 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | [G1K, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 44.2 ± 2.2μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [G1K, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 19.5 ± 0.5 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [G1K, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 1.7 ± 0.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [C/U]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 1.4 ± 0.2 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [C/U]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HL-60 | Leukemia Cancer | Resazurin dye assay | CC50 = 38.5 ± 4.8 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [C/U]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 4.6 ± 0.2 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [C/U]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 > 64 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [C/U]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 37.5 ± 3.3 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | [C/U]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 51.0 ± 4.6 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [L5W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 1.0 ± 0.1 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [L5W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 4.0 ± 0.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [L5W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 17.1 ± 0.7 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [L5W]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 18.3 ± 1.4 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [D-P L-P]cGm | 20 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 3.9 ± 0.2 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [D-P L-P]cGm | 20 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 51.5 ± 3.9 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [D-P L-P]cGm | 20 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 3.0 ± 0.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [D-P L-P]cGm | 20 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 22.5 ± 3.3 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [G1K, L5Y, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 1.3 ± 0.1 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [G1K, L5Y, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HL-60 | Leukemia Cancer | Resazurin dye assay | CC50 = 15.7 ±1.1μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [G1K, L5Y, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 15.2 ± 1.9 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | [G1K, L5Y, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 20.9 ± 1.4 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [G1K, L5Y, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 2.0 ± 0.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | [C/U, G1K, L5Y, K8R]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HL-60 | Leukemia Cancer | Resazurin dye assay | CC50 = 33.3 ±7.4μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [G1K, L5Y, K8R]cGm | 18 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 26.5 ± 2.4 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [C/U, G1K, L5Y, K8R]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | HeLa | Cervical Cancer | Resazurin dye assay | CC50 = 36.2 ± 2.8 μM | 24-h | Cervix | None | ||
| 36982972 | 2017 | [C/U, G1K, L5Y, K8R]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MCF-7 | Breast Cancer | Resazurin dye assay | CC50 = 29.0 ± 3.7 μM | 24-h | Breast | None | ||
| 36982972 | 2017 | [C/U, G1K, L5Y, K8R]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | K-562 | Leukemia Cancer | Resazurin dye assay | CC50 = 6.4 ± 0.6 μM | 24-h | Blood | None | ||
| 36982972 | 2017 | [C/U, G1K, L5Y, K8R]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | CRL-1739 | Gastric Cancer | Resazurin dye assay | CC50 = 46.2 ± 7.6 μM | 24-h | Stomach | None | ||
| 36982972 | 2017 | [C/U, G1K, L5Y, K8R]cGm | 18 | Cyclic | L | U = SelenoCys | Cyclized | Cyclized | Antimicrobial | Synthetic Analogue of Gomesin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 2.3 ± 0.2 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | Gomesin | 18 | Cyclic | L | Z= pyroglutamic acid | Amidation | Free | Antimicrobial and Anticancer | Acanthoscurria gomesiana | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 5.5 ± 1.1 μM | 24-h | Skin | None | ||
| 36982972 | 2017 | Gomesin | 18 | Cyclic | L | Z= pyroglutamic acid | Amidation | Free | Antimicrobial and Anticancer | Acanthoscurria gomesiana | K-562 | Blood Cancer | Resazurin dye assay | CC50 = 5.5 ± 1.1 μM | 24-h | Blood | None | ||
| 29183371;21530568 | 2017 | NN-32 | 10 | Linear | L | None | Free | Free | Anticancer | Indian spectacled cobra venom Naja naja | MDA-MB-231 | Breast Cancer | Anti-proliferation assay | Survival(%) = 64% at 10 μg/ml | 72-h | Breast | None | ||
| 29183371;21530568 | 2017 | NN-32 | 10 | Linear | L | None | Free | Free | Anticancer | Indian spectacled cobra venom Naja naja | MCF-7 | Breast Cancer | LDH leakage assay | 74% LDH Release at 2 μg/ml | 72-h | Breast | None | ||
| 29183371;21530568 | 2017 | NN-32 | 10 | Linear | L | None | Free | Free | Anticancer | Indian spectacled cobra venom Naja naja | MDA-MB-231 | Breast Cancer | LDH leakage assay | 66% LDH Release at 2 μg/ml | 72-h | Breast | None | ||
| 29183371;21530568 | 2017 | NN-32 | 10 | Linear | L | None | Free | Free | Anticancer | Indian spectacled cobra venom Naja naja | MCF-7 | Breast Cancer | MTT assay | IC50 = 2.5 μg/ml | 48-h | Breast | None | ||
| 29183371;21530568 | 2017 | NN-32 | 10 | Linear | L | None | Free | Free | Anticancer | Indian spectacled cobra venom Naja naja | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 6.7 μg/ml | 48-h | Breast | None | ||
| 29183371;21530568 | 2017 | NN-32 | 10 | Linear | L | None | Free | Free | Anticancer | Indian spectacled cobra venom Naja naja | MCF-7 | Breast Cancer | Anti-proliferation assay | Survival(%) = 68% at 10 μg/ml | 48-h | Breast | None | ||
| 28123590 | 2017 | LfcinB-P13 | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic analog of LFcinB | SMMC-7721 | Liver Cancer | MTT assay | IC50 = 41.8 µg/ml | 24-h | Liver | None | ||
| 28483698 | 2017 | FR8,11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HepG-2 | Liver Cancer | MTT assay | IC50 = 15 μM | 24-h | Liver | None | ||
| 28483698 | 2017 | FR8,11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HeLa | Cervical Cancer | MTT assay | IC50 = 18.9 μM | 24-h | Cervix | None | ||
| 28483698 | 2017 | FR8,11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | DLD-1 | Colon Cancer | MTT assay | IC50 = 22 μM | 24-h | Colon | None | ||
| 28483698 | 2017 | FR8,11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 27 μM | 24-h | Breast | None | ||
| 28483698 | 2017 | FR4,8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HepG-2 | Liver Cancer | MTT assay | IC50 = 5 μM | 24-h | Liver | None | ||
| 28483698 | 2017 | FR4,8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HeLa | Cervical Cancer | MTT assay | IC50 = 13.8 μM | 24-h | Cervix | None | ||
| 28483698 | 2017 | FR4,8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | DLD-1 | Colon Cancer | MTT assay | IC50 = 15.3 μM | 24-h | Colon | None | ||
| 28483698 | 2017 | FR4,8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 15.4 μM | 24-h | Breast | None | ||
| 28483698 | 2017 | FR11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | DLD-1 | Colon Cancer | MTT assay | IC50 = 12.9 μM | 24-h | Colon | None | ||
| 28483698 | 2017 | FR11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HepG-2 | Liver Cancer | MTT assay | IC50 = 4.8 μM | 24-h | Liver | None | ||
| 28483698 | 2017 | FR11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HeLa | Cervical Cancer | MTT assay | IC50 = 11 μM | 24-h | Cervix | None | ||
| 28483698 | 2017 | FR8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HepG-2 | Liver Cancer | MTT assay | IC50 = 4.2 μM | 24-h | Liver | None | ||
| 28483698 | 2017 | FR11P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 7 μM | 24-h | Breast | None | ||
| 28483698 | 2017 | FR8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | DLD-1 | Colon Cancer | MTT assay | IC50 = 10.8 μM | 24-h | Colon | None | ||
| 28483698 | 2017 | FR8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HeLa | Cervical Cancer | MTT assay | IC50 = 10.5 μM | 24-h | Cervix | None | ||
| 28483698 | 2017 | FR4P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.5 μM | 24-h | Liver | None | ||
| 28483698 | 2017 | FR8P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 6.4 μM | 24-h | Breast | None | ||
| 28483698 | 2017 | FR4P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | DLD-1 | Colon Cancer | MTT assay | IC50 = 9.4 μM | 24-h | Colon | None | ||
| 28483698 | 2017 | FR4P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 6.3 μM | 24-h | Breast | None | ||
| 28483698 | 2017 | FR4P | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Analogue of FR-15 | HeLa | Cervical Cancer | MTT assay | IC50 = 7.7 μM | 24-h | Cervix | None | ||
| 28483698 | 2017 | FR-15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.5 μM | 24-h | Liver | None | ||
| 28483698 | 2017 | FR-15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | MTT assay | IC50 = 6.7 μM | 24-h | Colon | None | ||
| 28483698 | 2017 | FR-15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 4.9 μM | 24-h | Cervix | None | ||
| 28483698 | 2017 | FR-15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 3.15 μM | 24-h | Breast | None | ||
| 27778166 | 2017 | IL-5 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | LDH leakage assay | 35% LDH release at 32 μM | 2-h | Cervix | None | ||
| 27778166 | 2017 | IL-5 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | PC-3 | Prostate Cancer | MTT assay | IC50 = 22.0 ± 2.6 μM | 4-h | Prostate | None | ||
| 27778166 | 2017 | IL-5 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | MTT assay | IC50 = 28.0 ± 4.6 μM | 4-h | Cervix | None | ||
| 27778166 | 2017 | IL-4 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | LDH leakage assay | 28% LDH release at 32 μM | 2-h | Cervix | None | ||
| 27778166 | 2017 | IL-4 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | PC-3 | Prostate Cancer | MTT assay | IC50 = 35.5 ± 3.9 μM | 4-h | Prostate | None | ||
| 27778166 | 2017 | IL-4 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | MTT assay | IC50 = 54.4 ± 3.0 μM | 4-h | Cervix | None | ||
| 27778166 | 2017 | IL-3 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | LDH leakage assay | 35% LDH release at 32 μM | 2-h | Cervix | None | ||
| 27778166 | 2017 | IL-3 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | PC-3 | Prostate Cancer | MTT assay | IC50 = 74.9 ± 13.3 μM | 4-h | Prostate | None | ||
| 27778166 | 2017 | IL-3 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | MTT assay | IC50 = 93.5 ± 19.4 μM | 4-h | Cervix | None | ||
| 27778166 | 2017 | IL-2 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | LDH leakage assay | 30% LDH release at 32 μM | 2-h | Cervix | None | ||
| 27778166 | 2017 | IL-2 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | PC-3 | Prostate Cancer | MTT assay | IC50 = 43.6 ± 7.9 μM | 4-h | Prostate | None | ||
| 27778166 | 2017 | IL-2 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | MTT assay | IC50 = 52.0 ± 5.8 μM | 4-h | Cervix | None | ||
| 27778166 | 2017 | IL-1 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | LDH leakage assay | 30% LDH release at 32 μM | 2-h | Cervix | None | ||
| 27778166 | 2017 | IL-1 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | PC-3 | Prostate Cancer | MTT assay | IC50 = 58.4 ± 13.7 μM | 4-h | Prostate | None | ||
| 27778166 | 2017 | IL-1 | 16 | Linear | L | None | Free | Free | Anticancer | Synthetic; Mutant form of ZXR-II | HeLa | Cervical Cancer | MTT assay | IC50 = 73.9 ± 13.6 μM | 4-h | Cervix | None | ||
| 27778166 | 2017 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | HeLa | Cervical Cancer | LDH leakage assay | 40% LDH release at 32 μM | 2-h | Cervix | None | ||
| 28524273 | 2017 | B8 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | LDH leakage assay | ~60-60% LDH release at 8 μM | 24-h | Blood | None | ||
| 28524273 | 2017 | B4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | LDH leakage assay | ~60-80% LDH release at 8 μM | 24-h | Blood | None | ||
| 28524273 | 2017 | BP100 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Icthyopthirius multifilis (Strain G5) | K-562 | Leukemia Cancer | LDH leakage assay | ~40-60% LDH release at 8 μM | 24-h | Blood | None | ||
| 28524273 | 2017 | B9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 83.7 ± 5.3 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 30.6 ± 5.7 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 38.3 ± 2.5 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 60.7 ± 5.4 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B8 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 8.1 ± 0.9 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B8 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 10.9 ± 1.2 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B8 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.6 ± 1.4 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B8 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 7.7 ± 1.2 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B7 | 10 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 97.3 ± 11.4 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B7 | 10 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 73.7 ± 6.1 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B7 | 10 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 77.3 ± 5.6 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B6 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 22.7 ± 2.3 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B6 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 20.7 ± 1.6 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B6 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 18.4 ± 1.5 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B6 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 19.2 ± 2.3 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B5 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 28.3 ± 2.3 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B5 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 28.2 ± 2.7 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B5 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 27.3 ± 2.4 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B5 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 26.5 ± 1.5 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 7.7 ± 0.4 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 6.3 ± 0.4 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.9 ± 0.2 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 6.6 ± 0.5 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B3 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 25.3 ± 3.2 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B3 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 28.4 ± 3.1 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B3 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 47.4 ± 12.5 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 39.6 ± 5.7 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 36.1 ± 6.7 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 30.8 ± 3.4 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 33.6 ± 4.2 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 19.1 ± 2.1 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 18.2 ± 1.3 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | B1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | MCF-7 | Breast Cancer | MTT assay | IC50 = 15.7 ± 1.5 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | BP100 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Icthyopthirius multifilis (Strain G5) | K-562/ADM | Leukemia Cancer | MTT assay | IC50 = 32.6 ± 3.4 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | B1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of BP 100 | K-562 | Leukemia Cancer | MTT assay | IC50 = 17.9 ± 1.4 μM | 48-h | Blood | None | ||
| 28524273 | 2017 | BP100 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Icthyopthirius multifilis (Strain G5) | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 25.3 ± 2.5 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | BP100 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Icthyopthirius multifilis (Strain G5) | MCF-7 | Breast Cancer | MTT assay | IC50 = 27.6 ± 3.0 μM | 48-h | Breast | None | ||
| 28524273 | 2017 | BP100 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Icthyopthirius multifilis (Strain G5) | K-562 | Leukemia Cancer | MTT assay | IC50 = 30.4 ± 2.7 μM | 48-h | Blood | None | ||
| 27933724 | 2016 | CIGB-552 | 20 | Linear | Mix | None | Free | Acetylation | Anticancer | Synthetic | MCF-7 | Breast Cancer | Sulforhodamine B assay | IC50 = 379.1 ± 8.6 µM | 48-h | Breast | None | ||
| 27039838 | 2016 | [TOAC1, Lys5,6] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 10 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [TOAC1, Lys5,6] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 6 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [TOAC1, Api4] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, Z = 4-aminopiperidine-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 13 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [TOAC1, Arg9] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 5 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [Lys5,6] TG | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 7 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [Lys5,6] TG | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 10 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [TOAC1, Arg2] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 9 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [TOAC1, Arg9] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 8 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [Arg2] TG | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 8 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [Arg2] TG | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 4 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [TOAC1, Arg2] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 8 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [Lys6] TG | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 2 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [TOAC1, Lys6] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 1 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [TOAC1, Lys6] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 3 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [TOAC1] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 1 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | [TOAC1] TG | 10 | Linear | L | X = 2,2,6,6-tetramethylpiperidine-1-oxyl-4-amino-4-carboxylic acid, U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | HeLa | Cervical Cancer | MTT assay | EC50 = 3 µM | 24-h | Cervix | None | ||
| 27039838 | 2016 | [Lys6] TG | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichogin GA | T-67 | Brain Tumor | MTT assay | EC50 = 4 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | Trichogin GA | 10 | Linear | L | U = 2-Aminoisobutyric acid (Aib) | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichoderma longibrachiatum | T-67 | Brain Tumor | MTT assay | EC50 = 2 µM | 24-h | Brain | None | ||
| 27039838 | 2016 | Trichogin GA | 10 | Linear | L | U = 2-Aminoisobutyric acid (Aib) | Lol = leucinol | Oct = 1-octanoyl | AMP, Anticancer | Trichoderma longibrachiatum | HeLa | Cervical Cancer | MTT assay | EC50 = 8 µM | 24-h | Cervix | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 = 4.2 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 = 6.4 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 = 6.7 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 11 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 = 7.3 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 10 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid, A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 9 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Oic = octahydroindolecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 8 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid; Tic = tetrahydroisoquinolinecarboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 7 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 6 | 20 | Cyclic | L | A5c = 1-aminocyclopentane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 = 2.1 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 4.4 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 = 1.9 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 = 2.6 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 = 6.4 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 = 2.3 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 = 3.0 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 4 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Dab = diaminobutyric acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 2.7 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 3.6 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 = 4.7 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 = 6.2 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 = 3.1 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 = 5.4 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 = 3.2 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 5.9 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 3 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid, Orn = Ornithine | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 = 4.6 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 5.0 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 = 5.6 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 = 6.6 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 = 6.4 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 = 6.4 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 = 7.0 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 = 6.0 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | RL | Lymphoma Cancer | CellTiter-Glo assay | Not Available | 72-h | Blood | None | ||
| 27387357 | 2016 | Peptide - 2 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 2.6 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | PC-3 | Prostate Cancer | CellTiter-Glo assay | Not Available | 72-h | Prostate | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | CellTiter-Glo assay | Not Available | 72-h | Lung | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | NCI-H69 | Lung Cancer | CellTiter-Glo assay | Not Available | 72-h | Lung | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo assay | IC50 = 7.3 µM | 72-h | Pancreas | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | A-498 | Renal Cancer | CellTiter-Glo assay | IC50 = 3.0 µM | 72-h | Kidney | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | COLO-205 | Colon Cancer | CellTiter-Glo assay | IC50 = 5.4 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | DLD-1 | Colon Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Colon | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | UACC-62 | Skin Cancer | CellTiter-Glo assay | IC50 = 2.6 µM | 72-h | Skin | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | CellTiter-Glo assay | IC50 = 6.2 µM | 72-h | Breast | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | IGROV-1 | Ovarian Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Ovary | None | ||
| 27387357 | 2016 | Peptide - 1 | 20 | Cyclic | L | A6c = 1-aminocyclohexane carboxylic acid | Amidation | Acetylation | Antimicrobial and Anticancer | Synthetic | CPFAC-1 | Pancreatic Cancer | CellTiter-Glo assay | IC50 > 7.5 µM | 72-h | Pancreas | None | ||
| 27129462 | 2016 | RT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Crocodylus siamensis | CaSki | Cervical Cancer | Sulforhodamine B assay | IC50 = 17.28 ± 0.2 µM | 24-h | Cervix | None | ||
| 27129462 | 2016 | RT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Crocodylus siamensis | HeLa | Cervical Cancer | Sulforhodamine B assay | IC50 = 28.67 ± 0.4 µM | 24-h | Cervix | None | ||
| 27129462 | 2016 | KT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Crocodylus siamensis | CaSki | Cervical Cancer | Sulforhodamine B assay | IC50 = 30.81 ± 0.2 µM | 24-h | Cervix | None | ||
| 27129462 | 2016 | KT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Crocodylus siamensis | HeLa | Cervical Cancer | Sulforhodamine B assay | IC50 = 53.41 ± 1.0 µM | 24-h | Cervix | None | ||
| 27207743 | 2016 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | PC-3 | Prostate Cancer | MTT assay | IC50 = 14.2 ± 0.5 μM | 4-h | Prostate | None | ||
| 27207743 | 2016 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | 293T | Kidney Cancer | MTT assay | IC50 = 6.3 ± 0.7 μM | 4-h | Kidney | None | ||
| 27207743 | 2016 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | Huh-7 | Liver Cancer | MTT assay | IC50 = 8.4 ± 1.1 μM | 4-h | Liver | None | ||
| 27207743 | 2016 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | HepG-2 | Liver Cancer | MTT assay | IC50 = 7.5 ± 1.2 μM | 4-h | Liver | None | ||
| 27207743 | 2016 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | SACC-83 | Salivary Cancer | MTT assay | IC50 = 9.9 ± 1.7 μM | 4-h | Salivary gland | None | ||
| 27207743 | 2016 | ZXR-1 | 16 | Linear | L | None | Free | Free | Antimicrobial | Mauriporin | 293T | Kidney Cancer | MTT assay | IC50 = 186.7 ± 13.1 μM | 4-h | Kidney | None | ||
| 27207743 | 2016 | ZXR-2 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic; Mutant form of ZXR-I | HeLa | Cervical Cancer | MTT assay | IC50 = 8.1 ± 1.6 μM | 4-h | Cervix | None | ||
| 27207743 | 2016 | ZXR-1 | 16 | Linear | L | None | Free | Free | Antimicrobial | Mauriporin | PC-3 | Prostate Cancer | MTT assay | IC50 = 69.1 ± 1.6 μM | 4-h | Prostate | None | ||
| 27207743 | 2016 | ZXR-1 | 16 | Linear | L | None | Free | Free | Antimicrobial | Mauriporin | Huh-7 | Liver Cancer | MTT assay | IC50 = 77.9 ± 0.9 μM | 4-h | Liver | None | ||
| 27207743 | 2016 | ZXR-1 | 16 | Linear | L | None | Free | Free | Antimicrobial | Mauriporin | SACC-83 | Salivary Cancer | MTT assay | IC50 = 27.9 ± 7.7 μM | 4-h | Salivary gland | None | ||
| 27207743 | 2016 | ZXR-1 | 16 | Linear | L | None | Free | Free | Antimicrobial | Mauriporin | HepG-2 | Liver Cancer | MTT assay | IC50 = 141.7 ± 12.2 μM | 4-h | Liver | None | ||
| 27207743 | 2016 | ZXR-1 | 16 | Linear | L | None | Free | Free | Antimicrobial | Mauriporin | HeLa | Cervical Cancer | MTT assay | IC50 = 62.6 ± 8.4 μM | 4-h | Cervix | None | ||
| None | 2015 | LPSBD-2 | 20 | Linear | L | None | Free | Free | Anticancer | Synthetic | Hep3B | Liver Cancer | Cell Proliferation assay | ~40% cell survival at 60 µg/ml | 24-h | Liver | None | ||
| None | 2015 | LPSBD-2 | 20 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | Cell Proliferation assay | ~20% cell survival at 60 µg/ml | 24-h | Lung | None | ||
| 25854366 | 2015 | Bmkn-21 | 12 | Linear | L | None | Free | Free | Antimicrobial | Derivative of Bmkn-2 | HSC-4 | Tongue Squamous Cell Carcinoma | MTT assay | IC50 between 29-97 µg/ml | 24-h | Tongue | None | ||
| 25854366 | 2015 | BmKn-23 | 10 | Linear | L | None | Free | Free | Antimicrobial | Derivative of Bmkn-2 | HSC-4 | Tongue Squamous Cell Carcinoma | MTT assay | IC50 between 29-97 µg/ml | 24-h | Tongue | None | ||
| 25854366 | 2015 | BmKn2 | 13 | Linear | L | None | Free | Free | Antimicrobial | Mesobuthus martensii Karsch | HSC-4 | Tongue Squamous Cell Carcinoma | MTT assay | IC50 = 29 µg/mL | 24-h | Tongue | None | ||
| 25854366 | 2015 | Bmkn-22 | 11 | Linear | L | None | Free | Free | Antimicrobial | Derivative of Bmkn-2 | HSC-4 | Tongue Squamous Cell Carcinoma | MTT assay | IC50 between 29-97 µg/ml | 24-h | Tongue | None | ||
| 25462264 | 2015 | B1-Glu | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 36.6 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Glu | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 38.9 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Asp | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 19.9 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Asp | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 44.7 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-His | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 10.5 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-His | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.0µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Arg | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.5 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Arg | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 8.7 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Lys | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562/ADM | Leukemia cancer | MTT assay | IC50 = 5.5 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Lys | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 5.5 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Lys | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 8.6 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Lys | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.3 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Thr | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 17.0 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Gln | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 16.2 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Thr | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 19.1 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Gln | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 14.5 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Gly | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 14.8 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Phe | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 3.7 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Gly | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 15.8 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Phe | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 1.3 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Leu | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562/ADM | Leukemia cancer | MTT assay | IC50 = 3.3 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Leu | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 4.4 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Leu | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 1.1 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Val | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 5.0 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Leu | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.6 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Val | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 4.9 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1-Ala14 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | K-562 | Leukemia cancer | MTT assay | IC50 = 8.6 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1-Ala14 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic analog of B1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.9 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Cathelicidin-BF15 | MCF-7/ADM | Breast Cancer | MTT assay | IC50 = 24.1 µM | 24-h | Breast | None | ||
| 25462264 | 2015 | B1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Cathelicidin-BF15 | K-562/ADM | Leukemia cancer | MTT assay | IC50 = 31.6 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Cathelicidin-BF15 | K-562 | Leukemia cancer | MTT assay | IC50 = 26.9 µM | 24-h | Blood | None | ||
| 25462264 | 2015 | B1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Cathelicidin-BF15 | MCF-7 | Breast Cancer | MTT assay | IC50 = 21.9 µM | 24-h | Breast | None | ||
| 25626077 | 2015 | AaeAP2a | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic analog of AaeAP2 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 4 | 24-h | Breast | None | ||
| 25626077 | 2015 | AaeAP2a | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic analog of AaeAP2 | PC-3 | Prostate Cancer | MTT assay | Graph Figure 4 | 24-h | Prostate | None | ||
| 25626077 | 2015 | AaeAP2a | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic analog of AaeAP2 | MDA-MB-435S | Skin Cancer | MTT assay | Graph Figure 4 | 24-h | Skin | None | ||
| 25626077 | 2015 | AaeAP1a | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic analog of AaeAP1 | MCF-7 | Breast Cancer | MTT assay | Graph Figure 4 | 24-h | Breast | None | ||
| 25626077 | 2015 | AaeAP1a | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic analog of AaeAP1 | PC-3 | Prostate Cancer | MTT assay | Graph Figure 4 | 24-h | Prostate | None | ||
| 25626077 | 2015 | AaeAP1a | 19 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic analog of AaeAP1 | MDA-MB-435S | Skin Cancer | MTT assay | Graph Figure 4 | 24-h | Skin | None | ||
| 26402731 | 2015 | Chaxapeptin | 15 | Mix | L | None | Free | Cyclized to form macrolactam ring | Antimicrobial and Anticancer | Streptomyces leeuwenhoekii Strain C58 | A-549 | Lung Cancer | CyQUANT Direct assay | Cell invasion < 50% at 50 μM | 36-h | Lung | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-668 | Gastric cancer | LDH release assay | Cytotoxicity ~ 60-80% at 50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-638 | Gastric cancer | LDH release assay | Cytotoxicity ~ 60-80% at 50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-601 | Gastric cancer | LDH release assay | Cytotoxicity ~ 60-80% at 50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-484 | Gastric cancer | LDH release assay | Cytotoxicity ~ 60-80% at 50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-668 | Gastric cancer | MTS assay | IC50 ~ 20-50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-638 | Gastric cancer | MTS assay | IC50 ~ 20-50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-601 | Gastric cancer | MTS assay | IC50 ~ 20-50 μM | 24-h | Stomach | None | ||
| 25047444 | 2015 | CopA3 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | analogue derived from coprisin | SNU-484 | Gastric cancer | MTS assay | IC50 ~ 20-50 μM | 24-h | Stomach | None | ||
| 26405806 | 2015 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | Helicobacter pylori | HeLa | Cervical Cancer | MTT assay | IC50 = 3.5 ± 0.03 μM | 24-h | Cervix | None | ||
| 26405806 | 2015 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | Helicobacter pylori | HepG-2 | Liver Cancer | MTT assay | IC50 = 7.7 ± 0.23 μM | 24-h | Liver | None | ||
| 26405806 | 2015 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | Helicobacter pylori | SGC-7901 | Gastric cancer | MTT assay | IC50 = 5.2 ± 0.14 μM | 24-h | Stomach | None | ||
| 26405806 | 2015 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | Helicobacter pylori | B-16 | Skin Cancer | MTT assay | IC50 = 6.1 ± 0.02 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | RW-AH | 18 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 4.6 ± 0.2 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | RW-AH | 18 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 8.4 ± 0.5 μM | 24-h | Skin | None | ||
| 26239537 | 2015 | RW-AH | 18 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | PI uptake assay | LC50 = 4.5 ± 0.02 μM | 8-h | Skin | None | ||
| 26239537 | 2015 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | SBcl2 | Skin Cancer | MTS assay | LC50 = 10.4 ± 0.7 μM | 24-h | Skin | EP_2943215_B1 | ||
| 26239537 | 2015 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | MTS assay | LC50 = 23.3 ± 1.7 μM | 24-h | Skin | EP_2943215_B1 | ||
| 26239537 | 2015 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | SBcl2 | Skin Cancer | PI uptake assay | LC50 = 5.9 ± 0.3 μM | 8-h | Skin | EP_2943215_B1 | ||
| 26239537 | 2015 | R-DIM-P-LF11-322 | 19 | Linear | L | None | Amidation | Free | Host Defence Peptide | Synthetic | A-375 | Skin Cancer | PI uptake assay | LC50 = 9.5 ± 0.3 μM | 8-h | Skin | EP_2943215_B1 | ||
| 25970292 | 2015 | K6-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | SAS | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Tongue | None | ||
| 25970292 | 2015 | K6-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | OECM-1 | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Not Available | None | ||
| 25970292 | 2015 | K6-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | C9 | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Not Available | None | ||
| 25970292 | 2015 | K6-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 25970292 | 2015 | K6-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | PC-9G | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 25970292 | 2015 | K6-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | PC-9 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 25970292 | 2015 | K4R2-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | SAS | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Tongue | None | ||
| 25970292 | 2015 | K4R2-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | OECM-1 | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Not Available | None | ||
| 25970292 | 2015 | K4R2-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | C9 | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Not Available | None | ||
| 25970292 | 2015 | K4R2-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 25970292 | 2015 | K4R2-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | PC-9G | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 25970292 | 2015 | K4R2-Nal2-S1 | 18 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | PC-9 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 25970292 | 2015 | Nal2-S1 | 12 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | SAS | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Tongue | US_10093699_B2 | ||
| 25970292 | 2015 | Nal2-S1 | 12 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | OECM-1 | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Not Available | US_10093699_B2 | ||
| 25970292 | 2015 | Nal2-S1 | 12 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | C9 | Oral Cancer | MTT assay | Graph Figure 2 | 24-h | Not Available | US_10093699_B2 | ||
| 25970292 | 2015 | Nal2-S1 | 12 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | US_10093699_B2 | ||
| 25970292 | 2015 | Nal2-S1 | 12 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | PC-9G | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | US_10093699_B2 | ||
| 25970292 | 2015 | Nal2-S1 | 12 | Linear | L | Nal = beta-naphthylalanine | Amidation | Acetylation | Antimicrobial | Synthetic | PC-9 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | US_10093699_B2 | ||
| 24704757 | 2014 | Frenatin 2.1S | 16 | Linear | L | None | alpha-amidation | Free | Antimicrobial | Sphaenorhynchus lacteus | A-549 | Lung Cancer | Trypan blue assay | LC50 = 80 ± 6 μM | 24-h | Lung | None | ||
| 24704757 | 2014 | Frenatin 2.2S | 16 | Linear | L | None | alpha-amidation | Free | Antimicrobial | Sphaenorhynchus lacteus | A-549 | Lung Cancer | Trypan blue assay | LC50 = 75 ± 5 μM | 24-h | Lung | None | ||
| 24830845 | 2014 | mt_S20A/L22 W/P27A | 12 | Linear | L | None | Free | Free | Anticancer | MDM5 | MCF-7 | Breast Cancer | MTT/MTS assay | IC50= 8.7 µM | Not Available | Breast | None | ||
| 24830845 | 2014 | mt_T18S/L22 W/P27A | 12 | Linear | L | None | Free | Free | Anticancer | MDM4 | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=27 µM | Not Available | Breast | None | ||
| 24830845 | 2014 | mt_E17L/L22 W/P27A | 12 | Linear | L | None | Free | Free | Anticancer | MDM3 | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=15.1 µM | Not Available | Breast | None | ||
| 24830845 | 2014 | mt_L22 W/P27A | 12 | Linear | L | None | Free | Free | Anticancer | MDM2 | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=16.3 µM | Not Available | Breast | None | ||
| 24714081 | 2014 | T Peptide | 19 | Linear | L | None | Free | Free | Anticancer | Tuftsin derivative | BGC-823 | Gastric Cancer | MTT/MTS assay | 67.2% maximum inhibitory rate at 8 mg/kg | 48-h | Stomach | None | ||
| 24714081 | 2014 | T Peptide | 19 | Linear | L | None | Free | Free | Anticancer | Tuftsin derivative | HT-29 | Colon Cancer | MTT/MTS assay | 70% maximum inhibitory rate at 8 mg/kg | 48-h | Colon | None | ||
| 24714081 | 2014 | T Peptide | 19 | Linear | L | None | Free | Free | Anticancer | Tuftsin derivative | HepG-2 | Liver Cancer | MTT/MTS assay | 69.6% maximum inhibitory rate at 8 mg/kg | 48-h | Liver | None | ||
| 12417587 | 2003 | Tat (47-57) | 11 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 100 µM 60% viablity | 6-h | Cervix | None | ||
| 12417587 | 2003 | Tat (47-57) | 11 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 10 µM 80% viablity | 6-h | Cervix | None | ||
| 12417587 | 2003 | Tat (47-57) | 11 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HeLa | Cervical Cancer | MTT/MTS assay | at 1 µM 90-100% viablity | 6-h | Cervix | None | ||
| 21403917 | 2011 | Temporin A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Frog Rana temporaria | U-943 | Lymphoma Cancer | MTT/MTS assay | IC50 =80-90 µg/ml | Not Available | Blood | None | ||
| 21403917 | 2011 | Protegrin 1 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | alpha helical peptide without cysteines | U-942 | Lymphoma Cancer | MTT/MTS assay | IC50 =30-40 µg/ml | Not Available | Blood | None | ||
| 21403917 | 2011 | Pexiganan MSI-78 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Analog of Magainin | U-941 | Lymphoma Cancer | MTT/MTS assay | IC50 =20-30 µg/ml | Not Available | Blood | None | ||
| 21403917 | 2011 | Omiganan MBI-226 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Bovine neutrophils | U-937 | Lymphoma Cancer | MTT/MTS assay | IC50 =80-85 µg/ml | Not Available | Blood | None | ||
| 21403917 | 2011 | Demegen P-113 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Canaida albicans | U-939 | Lymphoma Cancer | MTT/MTS assay | IC50 =85-90 µg/ml | Not Available | Blood | None | ||
| 21403917 | 2011 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Australian blue mountains tree frog, Litoria citropa | U-938 | Lymphoma Cancer | MTT/MTS assay | IC50 =40 µg/ml | Not Available | Blood | None | ||
| 21423613 | 2011 | P5317-28 | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =30 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | 3A | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 >100 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =0.12 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | DI | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =1.6 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP(M11A) | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =0.4 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP(R9A) | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =0.02 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP(L10A) | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =1.14 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP(W7A) | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 >100 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP(Y6A) | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 >100 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | MIP(F3A) | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =0.57 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | 3A | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 >100 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | P5317-28 | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =4.7 µM | Not Available | Colon | None | ||
| 21423613 | 2011 | DI | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =0.29 µM | Not Available | Colon | None | ||
| 21928125 | 2012 | p776 | 15 | Linear | L | None | Free | Free | Antitumor | Synthetic Peptide | Not Available | Tumor | ELISPOT assay | Not Available | Not Available | Not Available | None | ||
| 21423613 | 2011 | MIP | 12 | Linear | L | None | Free | Free | Antitumor | E3 ubiquitin-protein ligase | HCT-116-p53+/+ | Colon Cancer | Immunoprecipitation assay | IC50 =0.01 µM | Not Available | Colon | None | ||
| 21928125 | 2012 | p85 | 10 | Linear | L | None | Free | Free | Antitumor | Synthetic Peptide | Not Available | Tumor | ELISPOT assay | Not Available | Not Available | Not Available | None | ||
| 22076954 | 2011 | Peptide-3 | 11 | Linear | L | Pem= Pemetrexed | Amidation | Free | Anticancer | Synthetic | NCI-H358 | Lung Cancer | MTT/MTS assay | IC50 = 8.41 µM | 3-h | Lung | None | ||
| 22076954 | 2011 | Peptide-2 | 20 | Linear | L | Pem= Pemetrexed | Amidation | Free | Anticancer | Synthetic | NCI-H358 | Lung Cancer | MTT/MTS assay | IC50 = 2.19 µM | 3-h | Lung | None | ||
| 22076954 | 2011 | Peptide-1 | 10 | Linear | L | Pem= Pemetrexed | Amidation | Free | Anticancer | Synthetic | NCI-H358 | Lung Cancer | MTT/MTS assay | IC50 = 4.63 mM | 3-h | Lung | None | ||
| 22076954 | 2011 | Peptide-3 | 11 | Linear | L | Pem= Pemetrexed | Amidation | Free | Anticancer | Synthetic | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50 = 6.24 µM | 3-h | Blood | None | ||
| 22076954 | 2011 | Peptide-2 | 10 | Linear | L | Pem= Pemetrexed | Amidation | Free | Anticancer | Synthetic | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50 = 2.64 µM | 3-h | Blood | None | ||
| 22076954 | 2011 | Peptide-1 | 10 | Linear | L | Pem= Pemetrexed | Amidation | Free | Anticancer | Synthetic | HL-60 | Leukemia Cancer | MTT/MTS assay | IC50 = 2.17 µM | 3-h | Blood | None | ||
| 8555423, 18957441 | 1995 | Mastoparan B | 14 | Not Available | L | None | Free | Free | Antimicrobial | Hornet,Vespa basalis | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 15949629, 18957441 | 2005 | Sesquin | 10 | Not Available | L | None | Free | Free | Antimicrobial | Seeds, Vigna sesquipedalis, ground bean | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 16269344, 18957441 | 2005 | Lunatusin | 20 | Not Available | L | None | Free | Free | Antimicrobial | Phaseolus lunatus L. (lima bean) | Not Available | Colorectal Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 19341344, 18957441 | 2009 | Temporin-1CEb | 17 | Not Available | L | None | Free | Free | Antimicrobial | Rana chensinensis, China, Asia | Not Available | Breast Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 16129513, 18957441 | 2005 | Polybia-MPI | 14 | Not Available | L | None | Free | Free | Antibacterial | venom, social wasp,Polybia paulista | Not Available | Breast Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 10942757, 18957441 | 2000 | Gomesin | 18 | Not Available | L | None | Free | Free | Antibacterial | Hemocytes, Acanthoscurria gomesiana | Not Available | Breast Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 12235362, 18957441 | 2002 | Alloferon 1 | 13 | Not Available | L | None | Free | Free | Antibacterial | Blow flyCalliphora vicina | Not Available | Skin Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 11738090, 18957441 | 2001 | CPF-ST3 | 18 | Not Available | L | None | Free | Free | Anticancer | Diploid clawed frogXenopus tropicalis, Africa | Not Available | Skin Cancer | Not Available | Not Available | Not Available | Not Available | None | ||
| 10951191, 18957441 | 2000 | Aurein 2.1 | 16 | Not Available | L | None | Free | Free | Anticancer | Southern bell frogLitoria aureaorLitoria raniformis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10951191, 18957441 | 2000 | Aurein 2.4 | 16 | Not Available | L | None | Free | Free | Anticancer | Litoria aureaandLitoria raniformis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10951191, 18957441 | 2000 | Aurein 2.2 | 16 | Not Available | L | None | Free | Free | Anticancer | Litoria aureaandLitoria raniformis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10951191, 18957441 | 2000 | Aurein 2.3 | 16 | Not Available | L | None | Free | Free | Anticancer | Litoria aureaandLitoria raniformis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10504394, 18957441 | 1999 | Citropin 1.2 | 16 | Not Available | L | None | Free | Free | Anticancer | Australian blue mountains tree frog, Litoria citropa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10504394, 18957441 | 1999 | Citropin 1.3 | 16 | Not Available | L | None | Free | Free | Anticancer | Australian blue mountains tree frog, Litoria citropa | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 10951191, 18957441 | 2000 | Aurein 1.1 | 13 | Not Available | L | None | Free | Free | Anticancer | Litoria aureaandLitoria raniformis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20198492, 18957441 | 2010 | Halictine 2 | 12 | Not Available | L | None | Free | Free | Anticancer | Venom, the eusocial bee, Halictus sexcinctus | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 20198492, 18957441 | 2010 | Halictine 1 | 12 | Not Available | L | None | Free | Free | Anticancer | venom, the eusocial bee, Halictus sexcinctus | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9620615, 18957441 | 1998 | Maculatin 2.1 | 18 | Not Available | L | None | Free | Free | Antibacterial | Litoria genimaculate, Litoria eucnemis, Australia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 15207717, 18957441 | 2004 | Ascaphin-8 | 19 | Not Available | L | None | Free | Free | Antibacterial | Coastal Tailed Frog,Ascaphus truei, Pacific Northwest, USA, North America | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22100226, 18957441 | 2012 | Macropin 1 | 13 | Not Available | L | None | Free | Free | Antibacterial | Venom, the solitary beeMacropis fulvipes | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 22100226, 18957441 | 2012 | Macropin 2 | 17 | Not Available | L | None | Free | Free | Antibacterial | Venom, the solitary beeMacropis fulvipes | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 9022710, 18957441 | 1996 | Temporin L | 13 | Not Available | L | None | Free | Free | Antibacterial | European common frog,Rana temporaria | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 17698251, 18957441 | 2007 | Dybowskin-2 | 17 | Not Available | L | None | Free | Free | Antibacterial | Rana dybowskii, Rana chensinensis, Asia | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| None | 2004 | DDA-DL6R6-25 | 15 | Linear | Mix | None | Free | Free | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | CL-1 | Tumor | MTT/MTS assay | LC50=3.125 µM | Not Available | Pancreatic | AU_2004_246909_A1 | ||
| None | 2004 | DDA-DL6R6-25 | 15 | Linear | Mix | None | Free | Free | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | 22RV1 | Prostate Cancer | MTT/MTS assay | LC50=3.125 µM | Not Available | Prostate | AU_2004_246909_A1 | ||
| None | 2004 | DL6R6 | 12 | Linear | Mix | None | Free | Free | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | 22RV1 | Prostate Cancer | MTT/MTS assay | LC50=50 µM | Not Available | Prostate | AU_2004_246909_A1 | ||
| None | 2004 | DL6R6 | 12 | Linear | Mix | None | Free | Free | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | CL-1 | Tumor | MTT/MTS assay | LC50>100 µM | Not Available | Pancreatic | AU_2004_246909_A1 | ||
| None | 2004 | PA-DL6K6-24 | 12 | Linear | Mix | None | Amidation | CH3(CH2)14CO | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | 22RV1 | Prostate Cancer | MTT/MTS assay | LC50<3.125 µM | Not Available | Prostate | AU_2004_246909_A1 | ||
| None | 2004 | PA-DL6K6-24 | 12 | Linear | Mix | None | Amidation | CH3(CH2)14CO | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | CL-1 | Tumor | MTT/MTS assay | LC50=3.125 µM | Not Available | Pancreatic | AU_2004_246909_A1 | ||
| None | 2004 | MA-DL6K6-23 | 12 | Linear | Mix | None | Amidation | CH3(CH2)12CO | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | 22RV1 | Prostate Cancer | MTT/MTS assay | LC50<3.125 µM | Not Available | Prostate | AU_2004_246909_A1 | ||
| None | 2004 | MA-DL6K6-23 | 12 | Linear | Mix | None | Amidation | CH3(CH2)12CO | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | CL-1 | Tumor | MTT/MTS assay | LC50<3.125 µM | Not Available | Pancreatic | AU_2004_246909_A1 | ||
| None | 2004 | DDA-DL6K6-22 | 12 | Linear | Mix | None | Amidation | CH3(CH2)10CO | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | 22RV1 | Prostate Cancer | MTT/MTS assay | LC50<3.125 µM | Not Available | Prostate | AU_2004_246909_A1 | ||
| None | 2004 | DDA-DL6K6-22 | 12 | Linear | Mix | None | Amidation | CH3(CH2)10CO | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | CL-1 | Tumor | MTT/MTS assay | LC50<3.125 µM | Not Available | Pancreatic | AU_2004_246909_A1 | ||
| None | 2004 | DL6K6 | 12 | Linear | Mix | None | Amidation | Free | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | CL-1 | Tumor | MTT/MTS assay | LC50>100 µM | Not Available | Pancreatic | AU_2004_246909_A1 | ||
| None | 2004 | DL6K6 | 12 | Linear | Mix | None | Amidation | Free | Antimicrobial, Antifungal and Anticancer | Synthetic Peptide | 22RV1 | Prostate Cancer | MTT/MTS assay | LC50>100 µM | Not Available | Prostate | AU_2004_246909_A1 | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-VM1 | Leukemia Cancer | Cell Viability assay | 40% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-VLB | Leukemia Cancer | Cell Viability assay | 40% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-VLB | Leukemia Cancer | Cell Viability assay | 44% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-WT | Leukemia Cancer | Cell Viability assay | 40% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-WT | Leukemia Cancer | Cell Viability assay | 44% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-VM1 | Leukemia Cancer | Cell Viability assay | 44% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin A | 12 | Cyclic | L | Aoc = 3-aminooctanoic acid ,Hyp = 4- hydroxyproline, Dhb = didehydrobutyrine, Hse = Homoserine | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-VM1 | Leukemia Cancer | Cell Viability assay | No inhibition at 4 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin B | 13 | Cyclic | L | Ade = 3-aminodecanoyl, Hleu =hydroxyleucyl, Hasn = hydoxyasparaginyl | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-WT | Leukemia Cancer | Cell Viability assay | 50% inhibition at 1 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin A | 12 | Cyclic | L | Aoc = 3-aminooctanoic acid ,Hyp = 4- hydroxyproline, Dhb = didehydrobutyrine, Hse = Homoserine | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-WT | Leukemia Cancer | Cell Viability assay | No inhibition at 4 µM | 96-h | Blood | None | ||
| 15875779, 1429232 | 2005 | Laxaphycin A | 12 | Cyclic | L | Aoc = 3-aminooctanoic acid ,Hyp = 4- hydroxyproline, Dhb = didehydrobutyrine, Hse = Homoserine | Free | Free | Antifungal | Terrestrial blue-green alga Anabaena laxa or the marine cyanobacterium Lyngbya Majuscula | CEM-VLB | Leukemia Cancer | Cell Viability assay | No inhibition at 4 µM | 96-h | Blood | None | ||
| 15467750 | 2004 | HIV-TAT48-57 | 10 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 65% apoptosis at 50 µM | 16 to 24-h | Cervix | None | ||
| 15467750 | 2004 | HIV-TAT48-57 | 10 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 15% apoptosis at 20 µM | 16 to 24-h | Cervix | None | ||
| 15467750 | 2004 | HIV-TAT48-57 | 10 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 35% apoptosis at 30 µM | 16 to 24-h | Cervix | None | ||
| 15467750 | 2004 | HIV-TAT48-57 | 10 | Linear | L | None | Free | Free | Anticancer | Not Available | HeLa | Cervical Cancer | LDH leakage assay | 7% apoptosis at 10 µM | 16 to 24-h | Cervix | None | ||
| 15313924 | 2004 | (HHPHG)4 | 20 | Linear | L | None | Amidation | Acetylation | Antiangiogenesis and Antitumor | Synthetic Peptide | Not Available | Tumor | Tropomyosin binding assay | IC50=0.245 µM | Not Available | Not Available | None | ||
| 15313924 | 2004 | (HHPHG)4 | 20 | Linear | L | None | Free | Free | Antiangiogenesis and Antitumor | Synthetic Peptide | Not Available | Tumor | Tropomyosin binding assay | IC50=0.256 µM | Not Available | Not Available | None | ||
| 15313924 | 2004 | (HHPHG)3 | 15 | Linear | L | None | Free | Free | Antiangiogenesis and Antitumor | Synthetic Peptide | Not Available | Tumor | Tropomyosin binding assay | IC50=1.25 µM | Not Available | Not Available | None | ||
| 15313924 | 2004 | (HHPHG)3 | 15 | Linear | L | None | Amidation | Acetylation | Antiangiogenesis and Antitumor | Synthetic Peptide | Not Available | Tumor | Tropomyosin binding assay | IC50=1.56 µM | Not Available | Not Available | None | ||
| 15313924 | 2004 | (HHPHG)2 | 10 | Linear | L | None | Free | Free | Antiangiogenesis and Antitumor | Synthetic Peptide | Not Available | Tumor | Tropomyosin binding assay | IC50=11.6 µM | Not Available | Not Available | None | ||
| 15313924 | 2004 | (HHPHG)2 | 10 | Linear | L | None | Amidation | Acetylation | Antiangiogenesis and Antitumor | Synthetic Peptide | Not Available | Tumor | Tropomyosin binding assay | IC50=26.9 µM | Not Available | Not Available | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | retro | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 23 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 22 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 19 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= >10 µM | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 18 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 17 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 16 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 15 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 14 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 13 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 11 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 7 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= >100 µM | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= >100 µM | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | 5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= > 1 µM | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 6 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | 3 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 6 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Breast tumor cellline | Breast Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Breast | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1D | 16 | Linear | D | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Prostate tumor cellline | Prostate Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Prostate | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Liver tumor celline | Liver Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Liver | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Ovary tumor cellline | Ovarian Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Ovary | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Brain tumor cellline | Brain Tumor | Sulforhodamine B assay | IC50= 5 M | Not Available | Brain | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Skin tumor cellline | Skin Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Skin | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Colon tumor cellline | Colon Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Colon | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Lung tumor cellline | Lung Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Lung | None | ||
| 12631273, 9266696 | 2003 | Citropin 1.1 | 16 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Amphibian skin secretions | Leukemia tumor cellline | Leukemia Cancer | Sulforhodamine B assay | IC50= 5 M | Not Available | Blood | None | ||
| 20515045 | 2010 | ES-2 | 11 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 60% inhibition at 10µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | ES-2 | 11 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 60% inhibition at 5µg/ml | NA | Not Available | None | ||
| 20515045 | 2010 | ES-2 | 11 | Linear | L | None | Free | Free | Antitumor | Endostatin derived synthetic peptide | BAE | Tumor | MTT/MTS assay | 60% inhibition at 2.5µg/ml | NA | Not Available | None | ||
| 23893605 | 2013 | NK-11 | 11 | Linear | L | None | Amidation | Free | Anticancer | NK2 derived inactive control peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 >> 100 µM | 24-h | Skin | None | ||
| 23893605 | 2013 | NK-11 | 11 | Linear | L | None | Amidation | Free | Anticancer | NK2 derived inactive control peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC-50 >> 100 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | NK-11 | 11 | Linear | L | None | Amidation | Free | Anticancer | NK2 derived inactive control peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC-50 >> 100 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | NK-11 | 11 | Linear | L | None | Amidation | Free | Anticancer | NK2 derived inactive control peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC-50>> 100 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | NK-11 | 11 | Linear | L | None | Amidation | Free | Anticancer | NK2 derived inactive control peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC-50 >> 100 µM | 4-h | Skin | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50= 22.25 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50= 12.55 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50= 22.51 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50= 29.10 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50= 14.8 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50= 21.48 µM | 72-h | Renal | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50= 14.53 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50= 27.39 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50= 24.76 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50= 47.69 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50= 27.00 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50= 26.70 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50= 41.21 µM | 72-h | Renal | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50= 25.20 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50= 14.58 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50= 24.32 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50= 13.16 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50= 14.80 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50= 13.77 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50= 15.88 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50= 22.06 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50= 22.59 µM | 72-h | Renal | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50= 13.97 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50= 24.31 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50= 46.51 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50= 20.36 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50= 24.63 µM | 72-h | Colon | None | ||
| 22481251 | 2012 | P7 | 11 | Linear | L | None | Free | Free | Antiproliferative and Antiangiogenic | NA | B16-F10 | Skin Cancer | WST-1 assay | IC50= 1 µM | 48-h | Skin | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50= 22.88 µM | 72-h | Renal | None | ||
| 22100226 | 2012 | HAL-2/11 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/13 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/24 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/6 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/20 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/18 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/19 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/8 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/2 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/22 | 12 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/15 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 34 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/29 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/19 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/21 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/20 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/17 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/10 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/5 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/12 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/18 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 30±10 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/6 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-1/22 | 12 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/11 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 49±9 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | HAL-2/13 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 60 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/6 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/24 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/20 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/19 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/18 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/8 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/2 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 35±5 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 38±6 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/22 | 12 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 35±3 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/15 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/29 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/21 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/19 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/20 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/10 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 60 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 50 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/18 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 18±2 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/5 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 44±5 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/12 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/17 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/11 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 14±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 44±8 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/22 | 12 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/6 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-1/4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | HAL-2/19 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 16±4 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/20 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 30±5 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/24 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 34 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/6 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 23±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/13 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 13±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/2 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 6±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 14±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/8 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 15±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/18 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 14±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/29 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/15 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 14±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 12±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/22 | 12 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 12 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-2/4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/19 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/21 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 30±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/20 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 22±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/10 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 13±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/17 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 35±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/5 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 9±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/12 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 43±14 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/18 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 4±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/9 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 9±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/4 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/6 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 15±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1 | 12 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 11±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | HAL-1/22 | 12 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Halictines and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 15±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/26 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 9±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/24 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 11 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/25 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 12±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/21 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 22±4 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/20 | 13 | Linear | L | O = Ornithine | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 25±3 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/19 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 43±11 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/10 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 16 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/16 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 70 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/9 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 14±4 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/6 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 15 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/3 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 22 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/4 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 29 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 17 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/1 | 13 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 11 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 32 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/25 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 14±1 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/26 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 18±1 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 12±6 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | MAC1/24 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 16±1 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/20 | 13 | Linear | L | O = Ornithine | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 35±4 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/21 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 17±2 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/19 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 68±2 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/16 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/10 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/9 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 13±3 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/4 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 49±9 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/6 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 29±3 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/3 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 11±1 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/1 | 13 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 19±2 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 16 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/26 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 8±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 23±4 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | MAC1/24 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 8±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/25 | 13 | Linear | L | AC6C = cyclohexyl-1-carboxylic acid | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 7±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/20 | 13 | Linear | L | O = Ornithine | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 10±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/21 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 9±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/16 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 32±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/19 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 21±4 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/10 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 15±6 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/6 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 8±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/9 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 8±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/4 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 15±5 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 16±3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/3 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 9±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1/1 | 13 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 12±4 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | MAC1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Macropins and their analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 10±4 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/37 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50= 4±1 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/34 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 5±3 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/36 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/27 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 18 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/26 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 6 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/24 | 15 | Linear | L | O = Ornithine | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 5±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/25 | 15 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 4 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/23 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 6 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/22 | 15 | Linear | L | Aib = 1-amino-isobutyric acid | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 25±4 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/19 | 15 | Linear | L | Aib = 1-amino-isobutyric acid | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 8±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/18 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 7±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/17 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/16 | 15 | Linear | L | Nal = 3-(1-naphthyl)alanine | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 9±3 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/12 | 15 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 5±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/11 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 4±1 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/9 | 15 | Linear | L | None | Methoxylation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/10 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 9 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/8 | 15 | Linear | L | None | Free | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 9 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/4 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 18 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/6 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 6±3 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/3 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | Not tested | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/2 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 7±2 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 5±3 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | CCRF-CEM | Leukemia Cancer | MTT/MTS assay | IC50 = 3±1 µM | 48-h | Blood | None | ||
| 22100226 | 2012 | LL-III/37 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 13 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/34 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 37 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/36 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/27 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/25 | 15 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 20 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/26 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 30 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/24 | 15 | Linear | L | O = Ornithine | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 20 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/23 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 15 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/19 | 15 | Linear | L | Aib = 1-amino-isobutyric acid | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 28 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/22 | 15 | Linear | L | Aib = 1-amino-isobutyric acid | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 100 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/18 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/17 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/16 | 15 | Linear | L | Nal = 3-(1-naphthyl)alanine | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 42 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/12 | 15 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 20 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/10 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/11 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 48 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/9 | 15 | Linear | L | None | Methoxylation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 25± 5 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/6 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/8 | 15 | Linear | L | None | Free | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | Not tested | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/4 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/2 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 11 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/3 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 12± 3 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/37 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 5±1 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | SW | Colon Cancer | MTT/MTS assay | IC50 = 18±4 µM | 48-h | Colon | None | ||
| 22100226 | 2012 | LL-III/36 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 8 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/27 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 13±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/34 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 5±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/26 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 5±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/24 | 15 | Linear | L | O = Ornithine | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 3±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/25 | 15 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 4±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/23 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 4 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/22 | 15 | Linear | L | Aib = 1-amino-isobutyric acid | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 11±7 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/18 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 3 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/19 | 15 | Linear | L | Aib = 1-amino-isobutyric acid | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 3±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/17 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50= 9 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/12 | 15 | Linear | D | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 6±2 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/15 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 7±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/16 | 15 | Linear | L | Nal = 3-(1-naphthyl)alanine | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 6±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/9 | 15 | Linear | L | None | Methoxylation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 3±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/10 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 9±4 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/11 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 8±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/4 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 7±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/6 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 > 40 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/8 | 15 | Linear | L | None | Free | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 12±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/2 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | Not tested | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/3 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | Not tested | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 4±1 µM | 48-h | Cervix | None | ||
| 22100226 | 2012 | LL-III/1 | 15 | Linear | L | None | Amidation | Free | Antimicrobial and Antifungal | Lasioglossin III and its analogs | HeLa | Cervical Cancer | MTT/MTS assay | IC50 = 3±1 µM | 48-h | Cervix | None | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | ~15% cytotoxicity at 10 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | <3% cytotoxicity at 10 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | 20% cytotoxicity at 1 µM | 24-h | Bladder | WO2012042540A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HTB-9 | Bladder Cancer | MTT/MTS assay | ~10% cytotoxicity at 10 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | 20% cytotoxicity at 10 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | <10% cytotoxicity at 10 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | ~5% cytotoxicity at 10 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | ~10% cytotoxicity at 1 µM | 48-h | Cervix | WO2012042540A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | CaSki | Cervical Cancer | MTT/MTS assay | ~15% cytotoxicity at 1 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | 20% cytotoxicity at 10 µM | 72-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 72-h | Cervix | WO2012042540A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | <10% cytotoxicity at 10 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | 10% cytotoxicity at 1 µM | 48-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | 5% cytotoxicity at 10 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | SiHa | Cervical Cancer | MTT/MTS assay | ~15% cytotoxicity at 1 µM | 24-h | Cervix | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | 15% cytotoxicity at 10 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <20% cytotoxicity at 1 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | 10% cytotoxicity at 10 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | <3% cytotoxicity at 10 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | HCT-116 | Colon Cancer | MTT/MTS assay | 20% cytotoxicity at 1 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | <45% cytotoxicity at 10 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~45% cytotoxicity at 1 µM | 72-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | <25% cytotoxicity at 10 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | ~25% cytotoxicity at 1 µM | 48-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | <10% cytotoxicity at 10 µM | 24-h | Bladder | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | UM-UC-3 | Bladder Cancer | MTT/MTS assay | 10% cytotoxicity at 1 µM | 24-h | Bladder | WO2012042540A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 10 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 72-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | >20% cytotoxicity at 10 µM | 48-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | <5% cytotoxicity at 1 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | <20% cytotoxicity at 10 µM | 24-h | Colon | WO_2012042540_A2 | ||
| None | 2012 | TG20 | 20 | Linear | L | None | Free | Free | Anticancer | Derived from the SAG1 surface protein from the parasite Toxoplasma gondii | COLO-205 | Colon Cancer | MTT/MTS assay | ~15% cytotoxicity at 1 µM | 48-h | Colon | WO2012042540A2 | ||
| None | 2004 | Synthetic peptide | 20 | Linear | L | None | Free | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Synthetic peptide | SNU-601 | Gastric Cancer | MTT/MTS assay | 0% survival rate at 100 µM | NA | Stomach | US_6800727_B2 | ||
| None | 2004 | Synthetic peptide | 20 | Linear | L | None | Free | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Synthetic peptide | SNU-601 | Gastric Cancer | MTT/MTS assay | ~20% survival rate at 10 µM | NA | Stomach | US_6800727_B2 | ||
| None | 2004 | Synthetic peptide | 20 | Linear | L | None | Free | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Synthetic peptide | Jurkat | Blood Cancer | MTT/MTS assay | 0% survival rate at 100 µM | NA | Blood | US_6800727_B2 | ||
| None | 2004 | Synthetic peptide | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Synthetic peptide | Jurkat | Blood Cancer | MTT/MTS assay | ~60% survival rate at 10 µM | NA | Blood | US_6800727_B2 | ||
| None | 2004 | Synthetic peptide | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Synthetic peptide | Calu-6 | Lung Cancer | MTT/MTS assay | 0% survival rate at 100 µM | NA | Lung | US_6800727_B2 | ||
| None | 2004 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Ceropin-Melittin hybrid | Calu-6 | Lung Cancer | MTT/MTS assay | ~90% survival rate at 10 µM | NA | Lung | US_6800727_B2 | ||
| None | 2004 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Ceropin-Melittin hybrid | Calu-6 | Lung Cancer | MTT/MTS assay | <20% survival rate at 100 µM | NA | Lung | US_6800727_B2 | ||
| None | 2004 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Ceropin-Melittin hybrid | Jurkat | Blood Cancer | MTT/MTS assay | 100% survival rate at 10 µM | NA | Blood | US_6800727_B2 | ||
| None | 2004 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Ceropin-Melittin hybrid | Jurkat | Blood Cancer | MTT/MTS assay | 0% survival rate at 100 µM | NA | Blood | US_6800727_B2 | ||
| None | 2004 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Ceropin-Melittin hybrid | SNU-601 | Gastric Cancer | MTT/MTS assay | ~80% survival rate at 10 µM | NA | Stomach | US_6800727_B2 | ||
| None | 2004 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Ceropin-Melittin hybrid | SNU-601 | Gastric Cancer | MTT/MTS assay | 10% survival rate at 100 µM | NA | Stomach | US_6800727_B2 | ||
| None | 2004 | Synthetic peptide | 20 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer, antibacterial, antifungal | Synthetic peptide | Calu-6 | Lung Cancer | MTT/MTS assay | 35% survival rate at 10 µM | NA | Lung | US_6800727_B2 | ||
| 23533710 | 2013 | LfcinB | 12 | Linear | L | None | Amidation | Free | Antihypertensive and Antimicrobial and Antiviral and Antioxidant | Bovine milk | AZ-97 | Colon Cancer | MTT/MTS assay | Inhibition at 0.1g/l | NA | Colon | None | ||
| 23893605 | 2013 | NK11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 >>100 µM | 30-Min | Skin | None | ||
| 23893605 | 2013 | NK11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 >>100 µM | 2-h | Skin | None | ||
| 23893605 | 2013 | NK11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 >>100 µM | 4-h | Skin | None | ||
| 23893605 | 2013 | NK11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | E42/02 | Skin Cancer | MTT/MTS assay | IC50 >>100 µM | 24-h | Skin | None | ||
| 21453492, 23533710 | 2011 | LfcinB | 12 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Bovine lactoferrin (Lf-B) | Kelly | Brain Tumor | MTT/MTS assay | IC50 =141 ± 3 µM | 30-Min | Brain | None | ||
| 21453492, 23533710 | 2011 | LfcinB | 12 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Bovine lactoferrin (Lf-B) | MT-1 | Breast Cancer | MTT/MTS assay | IC50 > 160 µM | 30-Min | Breast | None | ||
| 21453492, 23533710 | 2011 | LfcinB | 12 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Bovine lactoferrin (Lf-B) | HT-29 | Colon Cancer | MTT/MTS assay | IC50 > 160 µM | 30-Min | Colon | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 6.5 ± 1.07% cell viability at 80 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 26.9 ± 0.5% cell viability at 60 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 47.5 ± 1.66% cell viability at 40 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 63.8 ± 0.8% cell viability at 20 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | A-375 | Skin Cancer | MTT/MTS assay | 86 ± 0.57% cell viability at 10 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 13.8 ± 1.44% cell viability at 80 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 31.5 ± 1.49% cell viability at 60 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 50 ± 3.09% cell viability at 40 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Synthetic peptide | M14 | Skin Cancer | MTT/MTS assay | 71.1 ± 2.84% cell viability at 20 µM | NA | Skin | None | ||
| 19957017 | 2010 | P18 | 18 | Linear | L | None | Free | Free | Antibacterial | Bovine lactoferrin (Lf-B) | M14 | Skin Cancer | MTT/MTS assay | 92.2 ± 1.02% cell viability at 10 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | Ramos | Lymphoma Cancer | MTT/MTS assay | IC50 = 10 µM | NA | Blood | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | Raji | Lymphoma Cancer | MTT/MTS assay | IC50 = 13 µM | NA | Blood | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | Sudhl-4 | Skin Cancer | MTT/MTS assay | IC50 = 16 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | KMM-1 | Skin Cancer | MTT/MTS assay | IC50 = 57 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | U-266 | Lymphoma Cancer | MTT/MTS assay | IC50 = 55 µM | NA | Blood | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | KMS-5 | Skin Cancer | MTT/MTS assay | IC50 = 38 µM | NA | Skin | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | HT-29 | Colon Cancer | MTT/MTS assay | IC50 =148±8 µM | NA | Colon | None | ||
| 19527490, 23533710 | 2009 | LfcinB | 12 | Linear | L | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | FEMX | Skin Cancer | MTT/MTS assay | IC50 =40±7 µM | NA | Skin | None | ||
| 18815734 | 2008 | PST13-RK | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =80 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | PST13-RK | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 =90 µg/ml | NA | Lung | None | ||
| 18815734 | 2008 | Tritrpticin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50 =142 µg/ml | NA | Breast | None | ||
| 18815734 | 2008 | Tritrpticin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of tritrpticin | A-549 | Lung Cancer | MTT/MTS assay | IC50 >200 µg/ml | NA | Lung | None | ||
| 22934601 | 2012 | PTP-7b | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic peptide | A-549 | Lung Cancer | MTT/MTS assay | IC50 =32 µM | NA | Lung | None | ||
| 22934601 | 2012 | PTP-7a | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic peptide | A-549 | Lung Cancer | MTT/MTS assay | IC50 =28 µM | NA | Lung | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 =12.55 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 =22.25 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 =29.10 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 =22.51 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50 =14.80 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50 =14.53 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-K4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50 =21.48 µM | 72-h | Renal | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 =27.39 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 =47.69 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50 =27.00 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 =26.70 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50 =41.21 µM | 72-h | Renal | None | ||
| 22644847 | 2012 | GA-K3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50 =25.20 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 =13.16 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 =14.58 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50 =14.80 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 =13.77 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 =24.32 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50 =22.59 µM | 72-h | Renal | None | ||
| 22644847 | 2012 | GA-W4 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50 =15.88 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 =22.06 µM | 72-h | Ovary | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 =46.51 µM | 72-h | Prostate | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 =13.97 µM | 72-h | Skin | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 =24.31 µM | 72-h | Stomach | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | HCT-116 | Colon Cancer | MTT/MTS assay | IC50 =24.63 µM | 72-h | Colon | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-549 | Lung Cancer | MTT/MTS assay | IC50 =20.36 µM | 72-h | Lung | None | ||
| 22644847 | 2012 | GA-W3 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Undecapeptide analogues derived from Brevinin-1EMa | A-498 | Renal Cancer | MTT/MTS assay | IC50 =22.88 µM | 72-h | Renal | None | ||
| 22413859 | 2012 | SVS-2 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | MDA-MB-436 | Breast Cancer | MTT/MTS assay | IC50 >100 µM | 24-h | Breast | None | ||
| 22413859 | 2012 | SVS-2 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 >100 µM | 24-h | Breast | None | ||
| 22413859 | 2012 | SVS-2 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | KB | Oral Cancer | MTT/MTS assay | IC50 >100 µM | 24-h | Oral mucosa | None | ||
| 22413859 | 2012 | SVS-2 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic peptide | A-549 | Lung Cancer | MTT/MTS assay | IC50 >100 µM | 24-h | Lung | None | ||
| 22413859 | 2012 | D-SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | MDA-MB-436 | Breast Cancer | MTT/MTS assay | IC50 =3.2±0.4 µM | 24-h | Breast | None | ||
| 22413859 | 2012 | D-SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 =4.7±0.4 µM | 24-h | Breast | None | ||
| 22413859 | 2012 | D-SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | KB | Oral Cancer | MTT/MTS assay | IC50 =4.5±0.5 µM | 24-h | Oral mucosa | None | ||
| 22413859 | 2012 | D-SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | A-549 | Lung Cancer | MTT/MTS assay | IC50 =3.2±0.6 µM | 24-h | Lung | None | ||
| 22413859 | 2012 | SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | MDA-MB-436 | Breast Cancer | MTT/MTS assay | IC50 =5.6±0.5 µM | 24-h | Breast | None | ||
| 22413859 | 2012 | SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 =8.1±0.8 µM | 24-h | Breast | None | ||
| 22413859 | 2012 | SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Bovine lactoferrin (Lf-B) | KB | Oral Cancer | MTT/MTS assay | NA | 24-h | Oral mucosa | None | ||
| 22413859 | 2012 | SVS-1 | 18 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic peptide | A-549 | Lung Cancer | MTT/MTS assay | NA | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-S2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 = 1.8 µM | 24-h | Breast | None | ||
| 23770440 | 2013 | TsAP-S2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 1.6 µM | 24-h | Prostate | None | ||
| 23770440 | 2013 | TsAP-S2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | U251-MG | Brain Tumor | MTT/MTS assay | IC50 = 2.0 µM | 24-h | Brain | None | ||
| 23770440 | 2013 | TsAP-S2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | HI-57 | Lung Cancer | MTT/MTS assay | IC50 = 0.83 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-S2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | H-838 | Lung Cancer | MTT/MTS assay | IC50 = 1.6 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-S1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 = 1.8 µM | 24-h | Breast | None | ||
| 23770440 | 2013 | TsAP-S1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 2.1 µM | 24-h | Prostate | None | ||
| 23770440 | 2013 | TsAP-S1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | U251-MG | Brain Tumor | MTT/MTS assay | IC50 = 2.9 µM | 24-h | Brain | None | ||
| 23770440 | 2013 | TsAP-2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | U251-MG | Brain Tumor | MTT/MTS assay | IC50 = 15.4 µM | 24-h | Brain | None | ||
| 23770440 | 2013 | TsAP-S1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | HI-57 | Lung Cancer | MTT/MTS assay | IC50 = 1.5 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-S1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Derivative of TsAP-1, Brazilian yellow scorpion venom peptide | H-838 | Lung Cancer | MTT/MTS assay | IC50 = 1.6 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | H-838 | Lung Cancer | MTT/MTS assay | IC50 = 11.0 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | MCF-7 | Breast Cancer | MTT/MTS assay | IC50 = 6.4 µM | 24-h | Breast | None | ||
| 23770440 | 2013 | TsAP-2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 13.3 µM | 24-h | Prostate | None | ||
| 23770440 | 2013 | TsAP-1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | HI-57 | Lung Cancer | MTT/MTS assay | IC50 =55.9 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | H-838 | Lung Cancer | MTT/MTS assay | IC50 =52.5 µM | 24-h | Lung | None | ||
| 23770440 | 2013 | TsAP-2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Venom-derived cDNot Available library of the Brazilian yellow scorpion, Tityus serrulatus | HI-57 | Lung Cancer | MTT/MTS assay | IC50 = 4.1 µM | 24-h | Lung | None | ||
| 23993331 | 2013 | MAP-04-04 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability >80% at 75 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-04 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability >80% at 100 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-03 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=61.5 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-03 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability <40% at 75 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-03 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability >20% at 100 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-03 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability ~100% at 25 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-04 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability >80% at 50 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-03 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability >80% at 25 µM | 48-h | Breast | None | ||
| 23993331 | 2013 | MAP-04-03 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Analogs of Ixosin-B amide | MCF-7 | Breast Cancer | MTT/MTS assay | Cell viability ~50% at 50 µM | 48-h | Breast | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 3 % Cytotoxicity at 6.25 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 3 % Cytotoxicity at 3.125 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 8 % Cytotoxicity at 12.5 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 75 % Cytotoxicity at 25 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 4 % Cytotoxicity at 3.125 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 90 % Cytotoxicity at 50 mg/L | 24-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 4 % Cytotoxicity at 6.25 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 12 % Cytotoxicity at 12.5 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 76 % Cytotoxicity at 50 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 70 % Cytotoxicity at 25 mg/L | 12-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 10 % Cytotoxicity at 3.125 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 5 %Cytotoxicity at 12.5 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 7 % Cytotoxicity at 6.25 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 70 % Cytotoxicity at 25 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 5 % Cytotoxicity at 3.125 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 75 % Cytotoxicity at 50 mg/L | 6-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 10 % Cytotoxicity at 6.25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 8 % Cytotoxicity at 12.5 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 60 % Cytotoxicity at 50 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HT-1080 | Fibrosarcoma | MTT/MTS assay | 50 % Cytotoxicity at 25 mg/L | 3-h | Fibrous connective tissue | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 8 % Cytotoxicity at 12.5 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 3 % Cytotoxicity at 6.25 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 3 % Cytotoxicity at 3.125 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 75 % Cytotoxicity at 25 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 4 % Cytotoxicity at 3.125 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 90 % Cytotoxicity at 50 mg/L | 24-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 4 % Cytotoxicity at 6.25 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 70 % Cytotoxicity at 25 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 12 % Cytotoxicity at 12.5 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 10 % Cytotoxicity at 3.125 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 76 % Cytotoxicity at 50 mg/L | 12-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 5 % Cytotoxicity at 12.5 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 7 % Cytotoxicity at 6.25 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 70 % Cytotoxicity at 25 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 75 % Cytotoxicity at 50 mg/L | 6-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 10 % Cytotoxicity at 6.25 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 5 % Cytotoxicity at 3.125 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 8 % Cytotoxicity at 12.5 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 50 % Cytotoxicity at 25 mg/L | 3-h | Cervix | None | ||
| 23598079 | 2013 | Epinecidin-8 | 16 | Linear | L | None | Free | Free | Antimicrobial | Epinephelus nebulosus | HeLa | Cervical Cancer | MTT/MTS assay | 60 % Cytotoxicity at 50 mg/L | 3-h | Cervix | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | LNCaP | Prostate Cancer | WST-1 assay | IC50= 15.8 µM | 72-h | Prostate | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | COLO-587 | Human epithelial Cancer | WST-1 assay | IC50= 13.5 µM | 72-h | Pancreatic | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | HuCCT-1 | Human epithelial Cancer | WST-1 assay | IC50= 17.1 µM | 72-h | Bileduct | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | U-251 | Brain Tumor | WST-1 assay | IC50= 17.0 µM | 72-h | Brain | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | SF-295 | Brain Tumor | WST-1 assay | IC50= 19.1 µM | 72-h | Brain | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | SN-19 | Brain Tumor | WST-1 assay | IC50= 21.9 µM | 72-h | Brain | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | ZR75-1 | Breast Cancer | WST-1 assay | IC50= 19.4 µM | 72-h | Breast | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | BT-20 | Breast Cancer | WST-1 assay | IC50= 20.0 µM | 72-h | Breast | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | MDA-MB-231 | Breast Cancer | WST-1 assay | IC50= 27.0 µM | 72-h | Breast | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | SK-BR-3 | Breast Cancer | WST-1 assay | IC50= 25.7 µM | 72-h | Breast | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | T-47D | Breast Cancer | WST-1 assay | IC50= 14.1 µM | 72-h | Breast | None | ||
| 21849092 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Transferrin receptor (TfR) | BT-474 | Breast Cancer | WST-1 assay | IC50= 34.5 µM | 72-h | Breast | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | WM1158 | Skin Cancer | MTT/MTS assay | LC50 = 4.1 µM | 24-h | Skin | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | 4T1 | Breast Cancer | MTT/MTS assay | LC50 = 6.2 µM | 24-h | Breast | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | RENCA | Renal Cancer | MTT/MTS assay | LC50 = 1.3 µM | 24-h | Renal | None | ||
| 23583573 | 2013 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | Bcap-37 | Breast Cancer | MTT/MTS assay | 30 % Cell viability at 40 µM | 1-h | Breast | None | ||
| 20212453 | 2010 | Camel | 15 | Linear | L | None | Free | Free | Antimicrobial | Ceropin-Melittin hybrid | B16-F10 | Skin Cancer | MTT/MTS assay | LC50 = 1.75 µM | 24-h | Skin | None | ||
| 23583573 | 2013 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | Bcap-37 | Breast Cancer | MTT/MTS assay | 45% Cell viability at 30 µM | 1-h | Breast | None | ||
| 23583573 | 2013 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | Bcap-37 | Breast Cancer | MTT/MTS assay | 70% Cell viability at 20 µM | 1-h | Breast | None | ||
| 16707464 | 2006 | D-K6L9 | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Host Defense lytic Peptide | MB-231 | Prostate Cancer | Enzyme Immunoassay (EIA) | LC50=3 µMol/L | 960-h | Prostate | None | ||
| 16707464 | 2006 | D-K6L9 | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Host DefenseÐLike Lytic Peptide | CL-1 | Lung Cancer | Enzyme Immunoassay (EIA) | LC50=3 µMol/L | Not Available | Lung | None | ||
| 16707464 | 2006 | D-K6L9 | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Host Defense lytic Peptide | 22RV1 | Prostate Cancer | Enzyme Immunoassay (EIA) | LC50=6 µMol/L | Not Available | Prostate | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Interleukin-4 receptor a (IL-4Ra) chain | MDA-MB-231 | Breast Cancer | WST-1 assay | IC50=18.5 µMol/L | 24-h | Breast | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Interleukin-4 receptor a (IL-4Ra) chain | H-322 | Lung Cancer | WST-1 assay | IC50=27.1 µMol/L | 24-h | Lung | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Interleukin-4 receptor a (IL-4Ra) chain | A-172 | Brain Tumor | WST-1 assay | IC50=30.5 µMol/L | 24-h | Brain | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Interleukin-4 receptor a (IL-4Ra) chain | T98G | Brain Tumor | WST-1 assay | IC50=77.3 µMol/L | 24-h | Brain | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Bovine lactoferrin (Lf-B) | KB | Oral Cancer | WST-1 assay | IC50=37.4 µMol/L | 24-h | Oral mucosa | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Interleukin-4 receptor a (IL-4Ra) chain | SU.86.86 | Pancreatic Cancer | WST-1 assay | IC50=28.0 µMol/L | 24-h | Pancreatic | None | ||
| 22084165 | 2011 | Lytik | 17 | Linear | Mix | None | Free | Free | Anticancer | Interleukin-4 receptor a (IL-4Ra) chain | BXPC-3 | Pancreatic Cancer | WST-1 assay | IC50=37.1 µMol/L | 24-h | Pancreatic | None | ||
| 23577112, 21871946 | 2012 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | MCF-7 | Breast Cancer | LDH leakage assay | 32% Cytotoxicity at 40 µM | 1-h | Breast | None | ||
| 23577112, 21871946 | 2012 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | MCF-7 | Breast Cancer | MTT/MTS assay | 61% Cell viability at 40 µM | 1-h | Breast | None | ||
| 23577112, 21871946 | 2012 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | MDA-MB-231 | Breast Cancer | MTT/MTS assay | 22% Cell viability at 40 µM | 1-h | Breast | None | ||
| 23577112, 21871946 | 2012 | Tempoprin-1CEa | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Chinese brown frog Rana chensinensis. | MDA-MB-231 | Breast Cancer | LDH leakage assay | 61% Cytotoxicity at 40 µM | 1-h | Breast | None | ||
| 24246647 | 2014 | Short α-helical peptides | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha-helical proteins | HL-60 | Leukemia Cancer | MTT/MTS assay | 70% Cytotoxicity at 5 µM Approx | 24-h | Blood | None | ||
| 24246647 | 2014 | Short α-helical peptides | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha-helical proteins | HL-60 | Leukemia Cancer | MTT/MTS assay | 90% Cytotoxicity at 5 µM Approx | 24-h | Blood | None | ||
| 24246647 | 2014 | Short α-helical peptides | 10 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha-helical proteins | HL-60 | Leukemia Cancer | MTT/MTS assay | 100% Cytotoxicity at 5 µM Approx | 24-h | Blood | None | ||
| 24246647 | 2014 | Short α-helical peptides | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha-helical proteins | HeLa | Cervical Cancer | MTT/MTS assay | 95% Cytotoxicity at 4 µM Approx | 24-h | Cervix | None | ||
| 24246647 | 2014 | Short α-helical peptides | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha-helical proteins | HeLa | Cervical Cancer | MTT/MTS assay | 80% Cytotoxicity at 4 µM Approx | 24-h | Cervix | None | ||
| 24246647 | 2014 | Short α-helical peptides | 10 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha-helical proteins | HeLa | Cervical Cancer | MTT/MTS assay | 99% Cytotoxicity at 4 µM Approx | 24-h | Cervix | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | J774A.1 | Tumor | MTT/MTS assay | IC50=12 µM | 96-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | J774A.1 | Tumor | MTT/MTS assay | IC50=17 µM | 96-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | J774A.1 | Tumor | MTT/MTS assay | IC50=26 µM | 24-h | Blood | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | J774A.1 | Tumor | MTT/MTS assay | IC50=47 µM | 24-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=36 µM | 96-h | Blood | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=25 µM | 96-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=45 µM | 72-h | Blood | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=36 µM | 72-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=43 µM | 48-h | Blood | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=37 µM | 48-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=43 µM | 24-h | Blood | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=39 µM | 24-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=38 µM | 2-h | Blood | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | HUT-102 | Lymphoma Cancer | MTT/MTS assay | IC50=93 µM | 2-h | Blood | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=10 µM | 48-h | Breast | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=16 µM | 48-h | Breast | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=12 µM | 24-h | Breast | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=29 µM | 24-h | Breast | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=18 µM | 2-h | Breast | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | MDA-MB-231 | Breast Cancer | MTT/MTS assay | IC50=39 µM | 2-h | Breast | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | LNCaP | Prostate Cancer | MTT/MTS assay | IC50=8 µM | 48-h | Prostate | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | LNCaP | Prostate Cancer | MTT/MTS assay | IC50=28 µM | 48-h | Prostate | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | LNCaP | Prostate Cancer | MTT/MTS assay | IC50=23 µM | 24-h | Prostate | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | LNCaP | Prostate Cancer | MTT/MTS assay | IC50=9 µM | 24-h | Prostate | None | ||
| 23000474 | 2012 | 9R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | LNCaP | Prostate Cancer | MTT/MTS assay | IC50=44 µM | 2-h | Prostate | None | ||
| 23000474 | 2012 | 9S1R | 10 | Linear | L | None | Free | Free | Anticancer | Nullomer derived anticancer peptides (NulloPs): | LNCaP | Prostate Cancer | MTT/MTS assay | IC50=26 µM | 2-h | Prostate | None | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =760 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =380 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =325 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =820 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =275 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =550 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =320 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =285 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =55 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =275 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =640 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =220 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =610 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =940 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =14 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =780 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =810 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =87 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =660 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =540 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =130 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =70 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =43 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 = >1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =670 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =20 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =380 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =74 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =260 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =570 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =210 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =345 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | Not Available | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =300 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =15 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =33 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | Not Available | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =280 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =22 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =15 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =185 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =620 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | Not Available | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =27 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =62 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK06 R-AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =260 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =25 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | HeLa | Cervical Cancer | MTT/MTS assay | LD50 =80 µg/ml | 24-h | Cervix | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =120 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =320 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =450 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =145 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =260 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =640 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =97 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =74 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =340 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =440 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =350 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =900 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =145 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =10 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =800 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =240 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =640 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =11 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =18 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =66 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =730 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =83 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =690 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =31 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =675 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =660 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =270 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =470 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =290 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =66 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =81 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =47 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =435 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =90 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =40 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =77 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =32 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =280 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =45 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =12 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =435 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =310 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =10 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =19 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =5 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK06 R-AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =280 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =16 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | PC-3 | Prostate Cancer | MTT/MTS assay | LD50 =8 µg/ml | 24-h | Prostate | US_06875744_B2 | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =345 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =720 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =240 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =540 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =640 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =300 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =74 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =470 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | Not Available | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =410 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =50 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =185 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =660 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =93 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =93 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =225 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =850 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =450 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =770 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =76 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =460 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =620 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =33 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =74 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =50 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =470 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =8 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =95 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =920 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =52 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =27 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =340 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | Not Available | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =320 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =25 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =860 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =80 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =670 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =320 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =130 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =450 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =270 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =127 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =370 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =80 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =65 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =17 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =290 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =72 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =6 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =245 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =420 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =33 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =57 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =16 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =24 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | H-1299 | Lung Cancer | MTT/MTS assay | LD50 =16 µg/ml | 24-h | Lung | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50D V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM V | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM V | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 17 CV | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =770 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =920 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =640 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =310 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =240 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =220 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =520 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =165 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =110 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =185 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =250 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =525 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =38 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =135 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =36 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =660 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =670 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =635 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =10 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =220 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =535 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =75 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =100 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =690 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =26 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =445 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =820 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =11 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =125 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =750 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =24 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =460 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =445 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =200 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =250 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =200 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =155 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =740 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =205 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =16 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =90 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =40 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =40 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =43 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =47 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =290 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =510 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =21 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =56 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =53 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =93 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK06 R-AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =300 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50D V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM V | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM V | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 17 CV | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | Not Available | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =920 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =770 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =640 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =310 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =240 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =220 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =520 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =165 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =330 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =185 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =110 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =250 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =38 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =525 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =535 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =220 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =635 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =10 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =670 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =660 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =36 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =135 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =26 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =445 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =690 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =75 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =100 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =820 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =11 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =830 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =125 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =750 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =24 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =460 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =445 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =200 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =250 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =200 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =155 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =740 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =205 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =16 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =90 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =40 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =40 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =43 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =700 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =47 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =290 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =510 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =21 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =56 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =7 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =53 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =300 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =93 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | BMKC | Skin Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Skin | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50D V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM V | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM V | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 17 CV | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =530 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =870 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =310 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =770 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =360 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =370 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =345 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =750 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =61 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =740 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =235 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =380 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =185 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =285 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =38 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =600 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =125 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =570 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =800 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =630 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =115 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =27 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =800 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =325 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =570 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =57 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =90 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =170 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =51 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =340 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =17 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =250 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =145 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =345 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =345 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 = µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =100 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =42 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =215 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =740 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =14 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =100 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =47 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =32 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =120 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =435 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =13 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =30 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =14 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK06 R-AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =210 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =59 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | SW-480 | Colon Cancer | MTT/MTS assay | LD50 =26 µg/ml | 24-h | Colon | US_06875744_B2 | ||
| None | 2005 | FLAK50J | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | Not Available | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50D V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =45 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM V | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =130 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM V | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =86 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =92 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 17 CV | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =23 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | KSL-7 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =315 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | KSL-1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =340 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK-120C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK-120D | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =550 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK-120G | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =950 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Flak 96L | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =555 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Flak 96I | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Flak 96J | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =770 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Flak 96H | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK96D | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =305 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK96F | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =510 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK96C | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =940 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK96B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =230 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK121 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Modelin-5-CO2H | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =320 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Modelin-5 | 16 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =61 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50T9 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK100-CO2H | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =135 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50T8 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =315 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK95 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50T6 | 11 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50T7 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =430 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK92B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK99 | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =160 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK91B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =315 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FKRLA | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =106 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK98 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =110 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK96 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK93B | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =44 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z10 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z9 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z7 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z8 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =625 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z5 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =500 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z2 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Z1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 T5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =440 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 T3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =90 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 T4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 T1 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =615 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 T2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =18 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q10 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =360 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q8 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =730 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q9 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =400 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q7 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =54 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q6 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =70 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q5 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q4 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =730 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q3 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =150 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q2 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =500 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 Q1 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =35 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAG26-D3 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =180 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK26-D2 | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | VISHNU3 | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAG26-D1 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =620 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | CA(1-& HECATE(11/23) | 20 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =11 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 50P | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =46 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 50O | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 50N | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =250 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50K | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50L | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50I | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =65 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50B | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =23 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Indolocidin-ac | 13 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =12 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 75 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =540 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 72 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 56 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =42 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 58 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =970 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 54 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =465 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Shiva 10(1-18 AC) | 18 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =190 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 50G | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =90 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 50H | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =475 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 17 C | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =80 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | Indolicidin | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =64 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 26 Ac | 17 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =105 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK82 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =31 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK81 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK80 | 10 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =>1000 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 50E | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =500 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50D | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =16 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50C | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =60 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | CAME-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =45 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK26V AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =32 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50F | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =40 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50V | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =23 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK77 | 12 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =575 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK71 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =300 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK57 | 14 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =260 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK51 | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK50 | 13 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 06R-AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =98 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK62 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =760 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK44 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =130 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK43 AM | 15 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =17 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 25 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 26 AM | 17 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =9 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK 17 AM | 16 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =21 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK06 R-AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =140 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK06 AC | 19 | Linear | L | None | Free | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =65 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2005 | FLAK06 AM | 19 | Linear | L | None | Amidation | Free | Anticancer | FLAK peptides | MCF-7 | Breast Cancer | MTT/MTS assay | LD50 =14 µg/ml | 24-h | Breast | US_06875744_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 14.58 mM | 24-h | Ovary | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 13.16 mM | 24-h | Skin | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 24.32 mM | 24-h | Prostate | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | IC50 = 57 mM | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 13.77 mM | 24-h | Stomach | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 14.8 mM | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 15.88 mM | 24-h | Lung | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | Not Available | 24-h | Renal | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 22.06 mM | 24-h | Ovary | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 13.97 mM | 24-h | Skin | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 46.51 mM | 24-h | Prostate | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | IC50 = 48 mM | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 22.31 mM | 24-h | Stomach | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 24.63 mM | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 20.36 mM | 24-h | Lung | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | Not Available | 24-h | Renal | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 12.55 mM | 24-h | Ovary | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 22.25 mM | 24-h | Skin | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 29.1 mM | 24-h | Prostate | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 22.51 mM | 24-h | Stomach | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 14.8 mM | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 14.53 mM | 24-h | Lung | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | IC50 = 21.48 mM | 24-h | Renal | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 24.76 mM | 24-h | Ovary | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 27.39 mM | 24-h | Skin | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 47.69 mM | 24-h | Prostate | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 26.7 mM | 24-h | Stomach | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 25.2 mM | 24-h | Lung | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | IC50 = 41.21 mM | 24-h | Renal | WO_2007133033_A1 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | IC50 = 57 mM | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | IC50 = 48 mM | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | NCI-H630 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 14.8 mM | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 24.63 mM | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 14.8 mM | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | HCTl-16 | Colon Cancer | MTT/MTS assay | IC50 = 27 mM | 24-h | Colon | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | Not Available | 24-h | Renal | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 24.32 mM | 24-h | Prostate | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 13.77 mM | 24-h | Stomach | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 14.58 mM | 24-h | Ovary | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 14.8 mM | 24-h | Lung | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 4 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 13.16 mM | 24-h | Skin | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | Not Available | 24-h | Renal | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 46.51 mM | 24-h | Prostate | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 24.31 mM | 24-h | Stomach | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 22.06 mM | 24-h | Ovary | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 20.36 mM | 24-h | Lung | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 3 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 13.97 mM | 24-h | Skin | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | IC50 = 21.48 mM | 24-h | Renal | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 29.1 mM | 24-h | Prostate | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 22.51 mM | 24-h | Stomach | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 12.55 mM | 24-h | Ovary | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 14.53 mM | 24-h | Lung | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 2 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 22.25 mM | 24-h | Skin | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-498 | Renal Cancer | MTT/MTS assay | IC50 = 41.21 mM | 24-h | Renal | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | PC-3 | Prostate Cancer | MTT/MTS assay | IC50 = 47.69 mM | 24-h | Prostate | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | MKN-45 | Gastric Cancer | MTT/MTS assay | IC50 = 26.7 mM | 24-h | Stomach | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-OV-3 | Ovarian Cancer | MTT/MTS assay | IC50 = 24.76 mM | 24-h | Ovary | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | SK-MEL-2 | Skin Cancer | MTT/MTS assay | IC50 = 27.39 mM | 24-h | Skin | US_008076284_B2 | ||
| None | 2011 | Gaegurin peptides SEQID NO: 1 | 11 | Linear | L | None | Free | Free | Antimicrobial | Korean frog Rana rugosa | A-549 | Lung Cancer | MTT/MTS assay | IC50 = 25.2 mM | 24-h | Lung | US_008076284_B2 | ||
| 11691780 | 2001 | DP1 | 14 | Linear | L | None | Free | Free | Antimicrobial | Protein transduction domain | MCA205 | Renal Cancer | MTT/MTS assay | LC50 =< 50 µM | 168-h | Renal | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | MEC | Breast Cancer | MTT/MTS assay | 29.33 Inhibition ratio at 50 µg/ml | 24-h | Breast | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | MEC | Breast Cancer | MTT/MTS assay | 19.76 Inhibition ratio at 50 µg/ml | 24-h | Breast | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | MEC | Breast Cancer | MTT/MTS assay | 27.99 Inhibition ratio at 50 µg/ml | 24-h | Breast | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | MEC | Breast Cancer | MTT/MTS assay | 24.15Inhibition ratio at 50 µg/ml | 24-h | Breast | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | HEK-293T | Renal Cancer | MTT/MTS assay | 32.52 Inhibition ratio at 50 µg/ml | 24-h | Renal | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | HEK-293T | Renal Cancer | MTT/MTS assay | 27.86 Inhibition ratio at 50 µg/ml | 24-h | Renal | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HEK-293T | Renal Cancer | MTT/MTS assay | 30.90 Inhibition ratio at 50 µg/ml | 24-h | Renal | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HEK-293T | Renal Cancer | MTT/MTS assay | 30.82 Inhibition ratio at 50 µg/ml | 24-h | Renal | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | HL7702 | Liver Cancer | MTT/MTS assay | 38.13 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | HL7702 | Liver Cancer | MTT/MTS assay | 36.25 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HL7702 | Liver Cancer | MTT/MTS assay | 37.00 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HL7702 | Liver Cancer | MTT/MTS assay | 37.22 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | A-549 | Lung Cancer | MTT/MTS assay | 52.50 Inhibition ratio at 50 µg/ml | 24-h | Lung | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | A-549 | Lung Cancer | MTT/MTS assay | 47.26Inhibition ratio at 50 µg/ml | 24-h | Lung | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | A-549 | Lung Cancer | MTT/MTS assay | 50.64 Inhibition ratio at 50 µg/ml | 24-h | Lung | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | A-549 | Lung Cancer | MTT/MTS assay | 45.62 Inhibition ratio at 50 µg/ml | 24-h | Lung | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | BGC-823 | Gastric Cancer | MTT/MTS assay | 73.705 Inhibition ratio at 50 µg/ml | 24-h | Stomach | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | BGC-823 | Gastric Cancer | MTT/MTS assay | 62.49 Inhibition ratio at 50 µg/ml | 24-h | Stomach | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | BGC-823 | Gastric Cancer | MTT/MTS assay | 50.85 Inhibition ratio at 50 µg/ml | 24-h | Stomach | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | BGC-823 | Gastric Cancer | MTT/MTS assay | 48.19 Inhibition ratio at 50 µg/ml | 24-h | Stomach | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide aNot Available temporins | HepG-2 | Liver Cancer | MTT/MTS assay | 73.07 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide aNot Available temporins | HepG-2 | Liver Cancer | MTT/MTS assay | 60.22 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HepG-2 | Liver Cancer | MTT/MTS assay | 55.98 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HepG-2 | Liver Cancer | MTT/MTS assay | 50.90 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | HeLa | Cervical Cancer | MTT/MTS assay | 78.045 Inhibition ratio at 50 µg/ml | 24-h | Cervix | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | HeLa | Cervical Cancer | MTT/MTS assay | 73.09 Inhibition ratio at 50 µg/ml | 24-h | Cervix | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HeLa | Cervical Cancer | MTT/MTS assay | 56.81 Inhibition ratio at 50 µg/ml | 24-h | Cervix | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | HeLa | Cervical Cancer | MTT/MTS assay | 52.32 Inhibition ratio at 50 µg/ml | 24-h | Cervix | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | SMMC-7721 | Liver Cancer | MTT/MTS assay | 86.175 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | SMMC-7721 | Liver Cancer | MTT/MTS assay | 70.39 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | SMMC-7721 | Liver Cancer | MTT/MTS assay | 59.37 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | SMMC-7721 | Liver Cancer | MTT/MTS assay | 52.77 Inhibition ratio at 50 µg/ml | 24-h | Liver | None | ||
| 22641352 | 2012 | RGD-Las | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | SW-1116 | Colorectal Cancer | MTT/MTS assay | 81.465 Inhibition ratio at 50 µg/ml | 24-h | Colon | None | ||
| 22641352 | 2012 | RGD-La | 16 | Linear | L | None | Free | Free | Anticancer | Arg-Gly-Asp(RGD) tripeptide ana temporins | SW-1116 | Colorectal Cancer | MTT/MTS assay | 72.69 Inhibition ratio at 50 µg/ml | 24-h | Colon | None | ||
| 22641352 | 2012 | Temporin-Las | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | SW-1116 | Colorectal Cancer | MTT/MTS assay | 62.73 Inhibition ratio at 50 µg/ml | 24-h | Colon | None | ||
| 22641352 | 2012 | Temporin-La | 13 | Linear | L | None | Free | Free | Anticancer | Temporins family | SW-1116 | Colorectal Cancer | MTT/MTS assay | 57.62 Inhibition ratio at 50 µg/ml | 24-h | Colon | None | ||
| 12366526 | 2002 | L15 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=178 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L14 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=423 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L13 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=29 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L12 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=25 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L11 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=248 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L10 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=35 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L9 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=52 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L8 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=180 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L7 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=16 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L6 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=15 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L5 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=14 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L4 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=57 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L3 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=141 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L2 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=>440 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L1 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | HT-29 | Colon Cancer | MTT/MTS assay | IC50=>404 µM | 4-h | Colon | None | ||
| 12366526 | 2002 | L14 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=141 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L15 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=92 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L13 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=12 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L12 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=10 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L10 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=20 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L11 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=75 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L9 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=32 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L7 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=11 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L8 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=87 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L6 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=12 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L4 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=16 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L5 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=8 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L3 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=18 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L2 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=>254 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L1 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | MT-1 | Breast Cancer | MTT/MTS assay | IC50=>404 µM | 4-h | Breast | None | ||
| 12366526 | 2002 | L14 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=125 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L15 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=87 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L13 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=14 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L12 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=7.9 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L11 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=116 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L10 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=24 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L8 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=110 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L9 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=35 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L7 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=16 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L6 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=11 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L5 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=6.6 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L4 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=31 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L3 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=32 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L1 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=>404 µM | 4-h | Skin | None | ||
| 12366526 | 2002 | L2 | 18 | Cyclic | L | None | Free | Free | Antimicrobial | Lactoferrin | Meth A | Skin Cancer | MTT/MTS assay | IC50=144 µM | 4-h | Skin | None | ||
| 18656352 | 2008 | A5 | 12 | Linear | L | None | Free | Free | Anticancer | Cyclin B (285-296) | HCT-116 | Colon Cancer | MTT/MTS assay | Not Available | 24-h | Colon | None | ||
| 16637646 | 2006 | dLL-37(17-32)c | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-4,17-27) | 15 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-32)b | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | LC50=25 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-29) | 13 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | LC50=55 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-12) | 12 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | HBMEC | Prostate Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | dLL-37(17-32)c | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-29) | 13 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | LC50=57 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-4,17-27) | 15 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-32)b | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | LC50=30 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-12) | 12 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KB | Oral Cancer | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | dLL-37(17-32)c | 16 | Linear | Mix | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-4,17-27) | 15 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-29) | 13 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | LC50=60 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(17-32)b | 16 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | LC50=30 µM | 24-h | Not Available | None | ||
| 16637646 | 2006 | LL-37(1-12) | 12 | Linear | L | None | Free | Free | Antibacterial | LL-37,a series of peptide fragments | KBv | Tumor | MTT/MTS assay | Not Available | 24-h | Not Available | None | ||
| 12646578 | 2003 | l3,4,8,10K5L7 | 12 | Linear | Mix | None | Free | Free | Antibacterial | Diastereomeric peptide | D-122 | Lung Cancer | XTT assay | LC50 = >50 µM | 24-h | Lung | None | ||
| 12646578 | 2003 | l3,10,13K7,8K4R2L9 | 15 | Linear | Mix | None | Free | Free | Antibacterial | Diastereomeric peptide | D-122 | Lung Cancer | XTT assay | LC50= 4.5 µM | 24-h | Lung | None | ||
| 12646578 | 2003 | l3,4,8,10K5L7 | 12 | Linear | Mix | None | Free | Free | Antibacterial | Diastereomeric peptide | B16-F10 | Skin Cancer | XTT assay | LC50 = 100 µM | 24-h | Skin | None | ||
| 12646578 | 2003 | l3,10,13K7,8K4R2L9 | 15 | Linear | Mix | None | Free | Free | Antibacterial | Diastereomeric peptide | B16-F10 | Skin Cancer | XTT assay | LC50 = 2.5 µM | 24-h | Skin | None | ||
| 21955251 | 2011 | Cationic Amphiphilic | 16 | Cyclic | L | None | Free | Free | Antimicrobial | AMP | HL-60 | Pancreatic Cancer | WST-1 assay | IC50 = 25 µM | Not Available | Pancreatic | None | ||
| 21955251 | 2011 | Cationic Amphiphilic | 11 | Cyclic | L | None | Free | Free | Antimicrobial | AMP | HL-60 | Pancreatic Cancer | WST-1 assay | IC50 = >500 µM | Not Available | Pancreatic | None | ||
| 21955251 | 2011 | Cationic Amphiphilic | 16 | Cyclic | L | None | Free | Free | Antimicrobial | AMP | HeLa | Cervical Cancer | WST-1 assay | IC50 = 15 µM | Not Available | Cervix | None | ||
| 21955251 | 2011 | Cationic Amphiphilic | 11 | Cyclic | L | None | Free | Free | Antimicrobial | AMP | HeLa | Cervical Cancer | WST-1 assay | IC50 = 160 µM | Not Available | Cervix | None | ||
| 9022710 | 1996 | Temporin A | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Frog Rana temporaria | U-937 | Lymphoma Cancer | MTT/MTS assay | 15% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 8335113, 21403917 | 1993 | Protegrin 1 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Alpha helical peptide without cysteines | U-937 | Lymphoma Cancer | MTT/MTS assay | 61% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 14508884, 21403917 | 2003 | OmigaNAn MBI-226 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Helical peptide with a predominance of one or more amino acids tryptophane-rich | U-937 | Lymphoma Cancer | MTT/MTS assay | 27% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 16512752, 21403917 | 2006 | Demegen P-113 | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Amphibian skin peptide | U-937 | Lymphoma Cancer | MTT/MTS assay | 15% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 10504394, 21403917 | 2009 | Citropin1.1 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Australian blue mountains tree frog, Litoria citropa | U-937 | Lymphoma Cancer | MTT/MTS assay | 60% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 10455241, 21403917 | 2009 | Citropin1.1 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Australian blue mountains tree frog, Litoria citropa | U-937 | Lymphoma Cancer | MTT/MTS assay | 60% Cytotoxicity at 0.5 µg/ml | 6-h | Blood | None | ||
| 18931881 | 2008 | PNC-28 | 10 | Linear | L | None | Free | Free | Anticancer | Antennapedia | MiaPaCa.2 | Pancreatic Cancer | MTT/MTS assay | Cytotoxicity=80% µMo/ml | 48-h | Pancreatic | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Prostate tumor cellline | Prostate Cancer | Not Available | LC50 = 10 µM | Not Available | Prostate | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Renal tumor cellline | Renal Cancer | Not Available | LC50 = 10 µM | Not Available | Renal | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Ovary tumor cellline | Ovarian Cancer | Not Available | LC50 = 10 µM | Not Available | Ovary | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Brain tumor cellline | Brain Tumor | Not Available | LC50 = 10 µM | Not Available | Brain | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Skin tumor cellline | Skin Cancer | Not Available | LC50 = 10 µM | Not Available | Skin | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Colon tumor cellline | Colon Cancer | Not Available | LC50 = 10 µM | Not Available | Colon | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Lung tumor cellline | Lung Cancer | Not Available | LC50 = 10 µM | Not Available | Lung | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Leukemia tumor cellline | Leukemia Cancer | Not Available | LC50=10-100 µM | Not Available | Blood | None | ||
| 10951191 | 2000 | Aurein 3.3 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Breast tumor cellline | Breast Cancer | Not Available | LC50 = 10 µM | Not Available | Breast | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Prostate tumor cellline | Prostate Cancer | Not Available | LC50 = 10 µM | Not Available | Prostate | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Renal tumor cellline | Renal Cancer | Not Available | LC50 = 10 µM | Not Available | Renal | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Ovary tumor cellline | Ovarian Cancer | Not Available | LC50 = 10 µM | Not Available | Ovary | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Skin tumor cellline | Skin Cancer | Not Available | LC50 = 10 µM | Not Available | Skin | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Brain tumor cellline | Brain Tumor | Not Available | LC50 = 10 µM | Not Available | Brain | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Lung tumor cellline | Lung Cancer | Not Available | LC50 = 10 µM | Not Available | Lung | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Colon tumor cellline | Colon Cancer | Not Available | LC50=10-100 µM | Not Available | Colon | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Leukemia tumor cellline | Leukemia Cancer | Not Available | LC50 = 10 µM | Not Available | Blood | None | ||
| 10951191 | 2000 | Aurein 3.2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Breast tumor cellline | Breast Cancer | Not Available | LC50 = 10 µM | Not Available | Breast | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Prostate tumor cellline | Prostate Cancer | Not Available | LC50 = 10 µM | Not Available | Prostate | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Renal tumor cellline | Renal Cancer | Not Available | LC50=10-100 µM | Not Available | Renal | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Ovary tumor cellline | Ovarian Cancer | Not Available | LC50=10-100 µM | Not Available | Ovary | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Skin tumor cellline | Skin Cancer | Not Available | LC50=10-100 µM | Not Available | Skin | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Brain tumor cellline | Brain Tumor | Not Available | LC50=10-100 µM | Not Available | Brain | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Colon tumor cellline | Colon Cancer | Not Available | LC50 = 10 µM | Not Available | Colon | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Lung tumor cellline | Lung Cancer | Not Available | LC50 = 10 µM | Not Available | Lung | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Leukemia tumor cellline | Leukemia Cancer | Not Available | LC50 = 10 µM | Not Available | Blood | None | ||
| 10951191 | 2000 | Aurein 3.1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Breast tumor cellline | Breast Cancer | Not Available | LC50=10-100 µM | Not Available | Breast | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Prostate tumor cellline | Prostate Cancer | Not Available | LC50 = 10 µM | Not Available | Prostate | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Renal tumor cellline | Renal Cancer | Not Available | LC50 = 10 µM | Not Available | Renal | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Ovary tumor cellline | Ovarian Cancer | Not Available | LC50 = 10 µM | Not Available | Ovary | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Skin tumor cellline | Skin Cancer | Not Available | LC50 = 10 µM | Not Available | Skin | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Brain tumor cellline | Brain Tumor | Not Available | LC50 = 10 µM | Not Available | Brain | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Colon tumor cellline | Colon Cancer | Not Available | LC50=10-100 µM | Not Available | Colon | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Lung tumor cellline | Lung Cancer | Not Available | LC50 = 10 µM | Not Available | Lung | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Leukemia tumor cellline | Leukemia Cancer | Not Available | LC50=10-100 µM | Not Available | Blood | None | ||
| 10951191 | 2000 | Aurein2.6 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Breast tumor cellline | Breast Cancer | Not Available | LC50 = 10 µM | Not Available | Breast | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Prostate tumor cellline | Prostate Cancer | Not Available | LC50 = 10 µM | Not Available | Prostate | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Renal tumor cellline | Renal Cancer | Not Available | LC50 = 10 µM | Not Available | Renal | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Ovary tumor cellline | Ovarian Cancer | Not Available | LC50 = 10 µM | Not Available | Ovary | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Skin tumor cellline | Skin Cancer | Not Available | LC50 = 10 µM | Not Available | Skin | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Brain tumor cellline | Brain Tumor | Not Available | LC50 = 10 µM | Not Available | Brain | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Colon tumor cellline | Colon Cancer | Not Available | LC50=10-100 µM | Not Available | Colon | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Lung tumor cellline | Lung Cancer | Not Available | LC50 = 10 µM | Not Available | Lung | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Leukemia tumor cellline | Leukemia Cancer | Not Available | LC50=10-100 µM | Not Available | Blood | None | ||
| 10951191 | 2000 | Aurein2.5 | 16 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Breast tumor cellline | Breast Cancer | Not Available | LC50 = 10 µM | Not Available | Breast | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Prostate tumor cellline | Prostate Cancer | Not Available | LC50 = 10 µM | Not Available | Prostate | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Ovary tumor cellline | Ovarian Cancer | Not Available | LC50 = 10 µM | Not Available | Ovary | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Renal tumor cellline | Renal Cancer | Not Available | LC50 = 10 µM | Not Available | Renal | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Skin tumor cellline | Skin Cancer | Not Available | LC50 = 10 µM | Not Available | Skin | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Brain tumor cellline | Brain Tumor | Not Available | LC50 = 10 µM | Not Available | Brain | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Colon tumor cellline | Colon Cancer | Not Available | LC50 = 10 µM | Not Available | Colon | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Lung tumor cellline | Lung Cancer | Not Available | LC50 = 10 µM | Not Available | Lung | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Leukemia tumor cellline | Leukemia Cancer | Not Available | LC50=10-100 µM | Not Available | Blood | None | ||
| 10951191 | 2000 | Aurein1.2 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Southern bell frog | Breast tumor cellline | Breast Cancer | Not Available | LC50 = 10 µM | Not Available | Breast | None | ||
| 9352466 | 1997 | P8 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=1.8 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P7 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=2.4 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P5 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=3.2 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P6 | 19 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=3.1 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P4 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=2.8 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=10.9 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P2 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=47.7 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P1 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=4.5 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=15.8 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | CA-ME | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H146 | Lung Cancer | MTT/MTS assay | IC50=28.6 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P8 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=2.3 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P7 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=2.4 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P5 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=2.9 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P6 | 19 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=2 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P4 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=1.3 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=9.3 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P2 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=37.9 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P1 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=3.5 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | CA-ME | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=28.6 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H128 | Lung Cancer | MTT/MTS assay | IC50=16.1 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P8 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=2.6 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P7 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=3.1 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P6 | 19 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=1.7 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P5 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=2.9 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P4 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=1.9 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=9.3 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P2 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=36.2 µM | 72-h | Lung | None | ||
| 10675500 | 2000 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=44 µM | 72-h | Breast | None | ||
| 10675500 | 2000 | CA-MA1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=100 µM | 72-h | Breast | None | ||
| 10675500 | 2000 | CA-MA2 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=28 µM | 72-h | Breast | None | ||
| 10675500 | 2000 | CA-MA3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=>100 µM | 72-h | Breast | None | ||
| 9352466 | 1997 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=15.8 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | CA-ME | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=32.2 µM | 72-h | Lung | None | ||
| 9352466 | 1997 | P1 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A-Magainin 2 | NCI-H69 | Lung Cancer | MTT/MTS assay | IC50=3.4 µM | 72-h | Lung | None | ||
| 10675500 | 2000 | CA-MA1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | A-549 | Lung Cancer | MTT/MTS assay | IC50=100 µM | 72-h | Lung | None | ||
| 10675500 | 2000 | CA-MA2 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | A-549 | Lung Cancer | MTT/MTS assay | IC50=25 µM | 72-h | Lung | None | ||
| 10675500 | 2000 | CA-MA3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | A-549 | Lung Cancer | MTT/MTS assay | IC50=>100 µM | 72-h | Lung | None | ||
| 10675500 | 2000 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | Jurkat | Blood Cancer | MTT/MTS assay | IC50=30 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | Jurkat | Blood Cancer | MTT/MTS assay | IC50=65 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA2 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | Jurkat | Blood Cancer | MTT/MTS assay | IC50=20 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | Jurkat | Blood Cancer | MTT/MTS assay | IC50=75 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | A-549 | Lung Cancer | MTT/MTS assay | IC50=60 µM | 72-h | Lung | None | ||
| 10675500 | 2000 | CA-MA3 | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=>100 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA2 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=35.1 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA | 20 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=65 µM | 72-h | Blood | None | ||
| 10675500 | 2000 | CA-MA1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin-Magainin hybrid peptides | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=85.3 µM | 72-h | Blood | None | ||
| 12005420 | 2001 | C-9 | 13 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-10 | 13 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-8 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=30 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-6 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=27 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-7 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-5 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=67 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-3 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=62 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-4 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=25 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-2 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=23 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=31 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-5L | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=10 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-4L | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=3 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-3L | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=4.2 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-4 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=24 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-5 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-2 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=7 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-3 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=11 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | [S9]-P18 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=3 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=6 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | [L9]-P18 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=3 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | P18 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=3.5 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | CA-MA-P | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | K-562 | Leukemia Cancer | MTT/MTS assay | IC50=25 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-10 | 13 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-9 | 13 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-8 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=54 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-7 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-6 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=21 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-5 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=81 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-4 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=31 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-3 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=74 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-2 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=26 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=32 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-5L | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=14 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-4L | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=6 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-3L | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=4 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-5 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=100.0 <µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-4 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=23 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-3 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=17 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-2 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=11 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | N-1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=12 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | [S9]-P18 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=7 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | [L9]-P18 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=9 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | P18 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=4 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | CA-MA-P | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | Jurkat | Blood Cancer | MTT/MTS assay | IC50=20 µM | 48-h | Blood | None | ||
| 12005420 | 2001 | C-10 | 13 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=100. <µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-9 | 13 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=100. <µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-8 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=83 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-7 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=100. <µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-6 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=47 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-5 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=100 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-4 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=54 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-3 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=79 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-2 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=38 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | C-1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=26 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-5L | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=17 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-4L | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=5 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-3L | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=5 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-5 | 14 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=100. <µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-4 | 15 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=32 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-3 | 16 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=17 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-2 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=11 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | N-1 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=9.5 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | [S9]-P18 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=4 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | [L9]-P18 | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=3 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | P18 | 17 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=8 µM | 48-h | Breast | None | ||
| 12005420 | 2001 | CA-MA-P | 18 | Linear | L | None | Amidation | Free | Antibacterial | Ceropin A | MDA-MB-361 | Breast Cancer | MTT/MTS assay | IC50=20 µM | 48-h | Breast | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | SH-SY-5Y2 | Brain Tumor | MTT/MTS assay | IC50=60 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | SK-N-DZ | Brain Tumor | MTT/MTS assay | IC50=37 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | SHEP-12 | Brain Tumor | MTT/MTS assay | IC50=45 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Temporins family | IMR-32 | Brain Tumor | MTT/MTS assay | IC50=29 µM | 48-h | Brain | None | ||
| 16572423 | 2008 | Lactoferricin B | 15 | Linear | L | None | Amidation | Free | Antibacterial | Temporins family | Kelly | Brain Tumor | MTT/MTS assay | IC50=15.5 µM | 48-h | Brain | None | ||
| 14499271 | 2003 | PTP7 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=5.25 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP8 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=32.23 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP5 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=5.43 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP6 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=17.56 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP2 | 20 | Cyclic(C14-C20) | L | None | Free | Free | Antibacterial | Gaegurin | MCF-7 | Breast Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Breast | None | ||
| 14499271 | 2003 | PTP7 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=5.4 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP8 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=30.79 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP5 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | Not Available | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP6 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=15.07 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP2 | 20 | Cyclic(C14-C20) | L | None | Free | Free | Antibacterial | Gaegurin | Hep3B | Liver Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Liver | None | ||
| 14499271 | 2003 | PTP7 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | PC-3 | Prostate Cancer | MTT/MTS assay | IC50=5.01 µg/ml | 96-h | Prostate | None | ||
| 14499271 | 2003 | PTP8 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | PC-3 | Prostate Cancer | MTT/MTS assay | IC50=28.9 µg/ml | 96-h | Prostate | None | ||
| 14499271 | 2003 | PTP5 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | PC-3 | Prostate Cancer | MTT/MTS assay | Not Available | 96-h | Prostate | None | ||
| 14499271 | 2003 | PTP6 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | PC-3 | Prostate Cancer | MTT/MTS assay | IC50=13.27 µg/ml | 96-h | Prostate | None | ||
| 14499271 | 2003 | PTP2 | 20 | Cyclic(C14-C20) | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP7 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=6.71 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP8 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=26.8 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP5 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=15.11 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP6 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=14 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP2 | 20 | Cyclic(C14-C20) | L | None | Free | Free | Antibacterial | Gaegurin | 293 | Renal Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Renal | None | ||
| 14499271 | 2003 | PTP8 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=24.58 µg/ml | 96-h | Lung | None | ||
| 14499271 | 2003 | PTP6 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=13.94 µg/ml | 96-h | Lung | None | ||
| 14499271 | 2003 | PTP7 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=8.01 µg/ml | 96-h | Lung | None | ||
| 14499271 | 2003 | PTP5 | 13 | Linear | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=9.09 µg/ml | 96-h | Lung | None | ||
| 14499271 | 2003 | PTP2 | 20 | Cyclic(C14-C20) | L | None | Free | Free | Antibacterial | Gaegurin | A-549 | Lung Cancer | MTT/MTS assay | IC50=>100 µg/ml | 96-h | Lung | None | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | RG1 | Glioblastoma | AlamarBlue assay | EC50 ~ 7 μM | 72-96 h | Brain | WO 2019/025432 A1;US011352395B2 | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | GMB-27 | Glioblastoma | AlamarBlue assay | EC50 ~ 7.5 μM | 72-96 h | Brain | WO 2019/025432 Al;US20200157150A1 | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | 12015 | Glioblastoma | AlamarBlue assay | EC50 ~ 10 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | 12089 | Glioblastoma | AlamarBlue assay | EC50 ~ 4 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | RG6 | Glioblastoma | AlamarBlue assay | EC50 ~ 5 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | RG4 | Glioblastoma | AlamarBlue assay | EC50 ~ 5 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | RG5 | Glioblastoma | AlamarBlue assay | EC50 ~ 7 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS10 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links L(3) and A(10) | Free | Free | Anticancer | Synthetic | 12053 | Glioblastoma | AlamarBlue assay | EC50 ~ 50 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS02 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links D(5) and S(10) | Free | Free | Anticancer | Synthetic | NCI-H524 | Lung Cancer | AlamarBlue assay | EC50 ~ 5 μM | 72-96 h | Lung | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS16 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and R(15) | Free | Free | Anticancer | Synthetic | RG1 | Glioblastoma | AlamarBlue assay | EC50 ~ 15 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-NS16 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and R(15) | Free | Free | Anticancer | Synthetic | 12053 | Glioblastoma | AlamarBlue assay | EC50 ~ 10 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2019 | IDP-Na05 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links S(8) and H(15) | Free | Free | Anticancer | Synthetic | RG1 | Glioblastoma | AlamarBlue assay | EC50 ~ 10 μM | 72-96 h | Brain | WO 2019/025432 Al | ||
| None | 2020 | IDP-wtL05 | 17 | Linear | L | None | Free | Free | Anticancer | Synthetic | RPMI | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS05 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(4) and F(11) | Free | Free | Anticancer | Synthetic | HL-60 | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 5 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS05 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(4) and F(11) | Free | Free | Anticancer | Synthetic | RPMI | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 6 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS13 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and R(15) | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Breast | US20200239547A1 | ||
| None | 2020 | IDP-LS13 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and R(15) | Free | Free | Anticancer | Synthetic | HL-60 | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 7 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS13 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and R(15) | Free | Free | Anticancer | Synthetic | RPMI | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 9 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS13 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and R(15) | Free | Free | Anticancer | Synthetic | U266 | Lymphoma Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS15 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(15) and Q(17) | Free | Free | Anticancer | Synthetic | RPMI | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 7 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS15 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(15) and Q(17) | Free | Free | Anticancer | Synthetic | U266 | Lymphoma Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 8 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS16 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links I(6) and Y(13) | Free | Free | Anticancer | Synthetic | RPMI | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 15 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS16 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links I(6) and Y(13) | Free | Free | Anticancer | Synthetic | U266 | Lymphoma Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS17 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links S(8) and Q(15) | Free | Free | Anticancer | Synthetic | RPMI | Leukemia Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-LS17 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links S(8) and Q(15) | Free | Free | Anticancer | Synthetic | U266 | Lymphoma Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 16 μM | 48-72 h | Blood | US20200239547A1 | ||
| None | 2020 | IDP-Lb01 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links S(1) and I(8) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 22.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb01 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links S(1) and I(8) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 12.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb01 | 16 | Linear | L | -(CH2)2-CH=CH-(CH2)3; a biradical linker links S(1) and I(8) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 22.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb02 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links K(2) and L(9) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 22.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb02 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)2; a biradical linker links K(2) and L(9) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 7.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb02 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links K(2) and L(9) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 15 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb03 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links A(3) and S(10) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 22.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb03 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links A(3) and S(10) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb03 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links A(3) and S(10) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 15 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb04 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links P(4) and K(11) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 > 30 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb04 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links P(4) and K(11) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 12.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb04 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links P(4) and K(11) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 > 30 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb05 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links K(5) and A(12) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb05 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links K(5) and A(12) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 7.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb05 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links K(5) and A(12) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 12.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb06 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links V(6) and L(13) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 12.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb06 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links V(6) and L(13) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 7.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-Lb06 | 16 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links V(6) and L(13) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 12.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-La05 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and Q(15) | Free | Free | Anticancer | Synthetic | NCl-H187 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 22.5 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-La05 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and Q(15) | Free | Free | Anticancer | Synthetic | NCl-H82 | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 15 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2020 | IDP-La05 | 17 | Linear | L | -(CH2)6-CH=CH-(CH2)3; a biradical linker links R(8) and Q(15) | Free | Free | Anticancer | Synthetic | NCl-H510A | Lung Cancer | MTT/Alamamar-Blue/Hexosaminidase activity test | EC50 ~ 10 μM | 48-72 h | Lung | US20200239547A1 | ||
| None | 2023 | MAD1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | OVCAR-3 | Ovarian Cancer | MTT assay | IC50 = 14.2 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | MAD1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 36.2 μM | 48-h | Lung | US11571454 B2 | ||
| None | 2023 | MAD1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | NCI/ADR-RES | Ovarian Cancer | MTT assay | IC50 = 85.6 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 11.9 μM | 48-h | Lung | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | OVCAR-3 | Ovarian Cancer | MTT assay | IC50 = 8.6 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | NCI/ADR-RES | Ovarian Cancer | MTT assay | IC50 = 14.0 μM | 48-h | Lung | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | T-24 | Bladder Cancer | MTT assay | IC50 = 15.3 μM | 48-h | Bladder | US11571454 B2 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | U343 | Glioblastoma | MTT assay | IC50 = 0.781 μM | 48-h | Brain | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | U373MG | Glioblastoma | MTT assay | IC50 = 0.8717 μM | 48-h | Brain | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | U251 | Glioblastoma | MTT assay | IC50 = 0.7607 μM | 48-h | Brain | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | U87-MG | Glioblastoma | MTT assay | IC50 = 0.9164 μM | 48-h | Brain | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.064 μM | 48-h | Liver | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | Hep3B | Liver Cancer | MTT assay | IC50 = 0.7847 μM | 48-h | Liver | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | 293T | Renal Cancer | MTT assay | IC50 = 1.107 μM | 48-h | Renal | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 9.74 μM | 48-h | Breast | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 0.8061 μM | 48-h | Breast | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HL-60 | Blood Cancer | MTT assay | IC50 = 1.111 μM | 48-h | Blood | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | K-562 | Blood Cancer | MTT assay | IC50 = 1.103 μM | 48-h | Blood | EP3279210 B1 | ||
| None | 2016 | 5-2C | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | Hel | Blood Cancer | MTT assay | IC50 = 1.055 μM | 48-h | Blood | EP3279210 B1 | ||
| None | 2018 | hBD3-3 | 15 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Cell Proliferation assay | Concentration dependent reduction in colony formation between 100 μM and 200 μM. | 48-h | Breast | US009993519B2 | ||
| None | 2018 | hBD3-3 M1 | 15 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Cell Proliferation assay | Concentration dependent reduction in colony formation between 100 μM and 200 μM. | 48-h | Breast | US009993519B2 | ||
| None | 2018 | hBD3-3 M2 | 15 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Cell Proliferation assay | Concentration dependent reduction in colony formation between 100 μM and 200 μM. | 48-h | Breast | US009993519B2 | ||
| None | 2018 | hBD3-3 | 15 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Annexin V/ PI staining assay | Inhibition in growth by apoptosis as cells positive for annexin V formed 50% of test group | 8-h | Breast | US009993519B2 | ||
| None | 2018 | hBD3-3 M1 | 15 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Annexin V/ PI staining assay | Inhibition in growth by apoptosis as cells positive for annexin V formed 50% of test group | 8-h | Breast | US009993519B2 | ||
| None | 2018 | hBD3-3 M2 | 15 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Annexin V/ PI staining assay | Inhibition in growth by apoptosis as cells positive for annexin V formed 50% of test group | 8-h | Breast | US009993519B2 | ||
| None | 2017 | Alpha-gliadin peptide p31-43 | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | 9.4% growth inhibition at 70 μg/mL | 72-h | Lung | US009669068B2 | ||
| None | 2017 | Alpha-gliadin peptide p31-43 | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic | NCI-H1975 | Lung Cancer | MTT assay | 36.3% growth inhibition at 70 μg/mL | 72-h | Lung | US009669068B2 | ||
| None | 2017 | Alpha-gliadin peptide p31-43 | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic | PANC-1 | Pancreatic Cancer | MTT assay | 26.2% growth inhibition at 70 μg/mL | 72-h | Pancreas | US009669068B2 | ||
| None | 2017 | Alpha-gliadin peptide p31-43 | 13 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | TUNEL assay | Mean apoptotic rate = 36% at 200 μg/mL | 72-h | Lung | US009669068B2 | ||
| None | 2023 | Sample Peptide 5 from EP3604345B1 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 106.5% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2016 | ALRN-6924 | 17 | Linear | Mix | staple between Ala4 and d-Ala11 | Free | Free | Antitumor | Synthetic | TP53-WT subcutaneous mouse xenograft models | Breast Cancer | Not Available | Tumor suppression at doses 2.5 mg/kg to 5mg/kg | 28 days | Breast | WO2016049359A1 | ||
| None | 2018 | Balixafortide | 16 | Cyclic ; Disulfide bridge: Cys2-Cys9 | Mix | Dab = 2,4-diaminobutyric acid | Free | Free | Anticancer and Antitumor | Synthetic | Namalwa | Lymphoma | HUVEC sprouting | IC50< 10 nM | Not available | Blood | None | ||
| None | 2018 | Balixafortide | 16 | Cyclic ; Disulfide bridge: Cys2-Cys9 | Mix | Dab = 2,4-diaminobutyric acid | Free | Free | Anticancer and Antitumor | Synthetic | Jurkat | Blood Cancer | HUVEC sprouting | IC50< 10 nM | Not available | Blood | None | ||
| None | 2018 | Balixafortide | 16 | Cyclic ; Disulfide bridge: Cys2-Cys9 | Mix | Dab = 2,4-diaminobutyric acid | Free | Free | Anticancer and Antitumor | Synthetic | MDA-MB-231 | Breast Cancer | HUVEC sprouting | IC50< 20 nM | Not available | Breast | None | ||
| 15289344 | 2004 | PCK3145 | 15 | Linear | L | None | Free | Free | Anticancer and Antitumor | Derived from prostate secretory protein PSP-94 | Mat Ly Lu | Prostate Cancer | TUNEL assay | Not available | 15 days | Prostate | None | ||
| 30210643 | 2018 | SOR-C13 | 13 | Linear | L | None | Free | Free | Anticancer and Antitumor | Synthetic | SKOV-3 | Ovarian Cancer | IP; daily; on days 1 to 12 | Effectively inhibited the growth of tumor | 12 days | Ovary | None |