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| ID | PMID | YEAR | Sequence | Name | Length | Linear/Cyclic | Chirality | Chem-MOD | C-ter MOD | N-ter MOD | Nature | Origin | Cell Line | Cancer Type | Assay | Activity | Testing Time | Tissue Affected | Patents |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 38319435 | 2024 | Temporin-SHf | 8 | Linear | L | None | Amidation | Free | Antimicrobial | Pelophylax saharica | HepG-2 | Liver Cancer | MTT assay | IC50 = 32.64 ± 1.350 µM | 24-h | Liver | None | ||
| None | 2022 | ATRA1-R3W2 - HYD | 21 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | H-358 | Lung Cancer | Cytotoxicity assay | LD50 ~24.5 μM | 6-h | Lung | US011447533B2 | ||
| 38319435 | 2024 | Temporin-SHf | 8 | Linear | L | None | Amidation | Free | Antimicrobial | Pelophylax saharica | PC-3 | Prostate Cancer | MTT assay | IC50 = 36.67 ± 0.729 µM | 24-h | Prostate | None | ||
| 38319435 | 2024 | Temporin-SHf | 8 | Linear | L | None | Amidation | Free | Antimicrobial | Pelophylax saharica | MCF-7 | Breast Cancer | MTT assay | IC50 = 32.76 ± 1.528 µM | 24-h | Breast | None | ||
| 38319435 | 2024 | Temporin-SHf | 8 | Linear | L | None | Amidation | Free | Antimicrobial | Pelophylax saharica | A-549 | Lung Cancer | MTT assay | IC50 = 24.03 ± 0.945 µM | 24-h | Lung | None | ||
| 37853814 | 2024 | NRC-07 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | 52.5 ± 5.0% cell viability at 150 µM | 24-h | Breast | None | ||
| 37853814 | 2024 | NRC-07 | 25 | Linear | L | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | 14.0 ± 3.0% cell viability at 150 µM | 24-h | Breast | None | ||
| 38491556 | 2024 | HMM-ID | 34 | Linear | L | None | Free | Free | Anticancer | Red Sea Brine | U2OS | Osteosarcoma | MTT assay | IC50 = 100.5 µg/ml | 24-h | Bone | None | ||
| 38272230 | 2024 | RP7 SCR | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | PC-3 | Prostate Cancer | MTT assay | IC50 = 128 ± 11.65 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | RP7 SCR | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | DU-145 | Prostate Cancer | MTT assay | IC50 = 137 ± 5.98 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | RP7 SCR | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MCF-7 | Breast Cancer | MTT assay | IC50 = 150 ± 10.32 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | RP7 SCR | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 156 ± 8.15 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | D-RP-7 | 7 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | DU-145 | Prostate Cancer | MTT assay | IC50 = 121.59 ± 6.56 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | D-RP-7 | 7 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | PC-3 | Prostate Cancer | MTT assay | IC50 = 101 ± 5.73 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | D-RP-7 | 7 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 95 ± 7.71 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | D-RP-7 | 7 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MCF-7 | Breast Cancer | MTT assay | IC50 = 90 ± 10.31 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | RP-7 | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | PC-3 | Prostate Cancer | MTT assay | IC50 = 113 ± 8.02 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | RP-7 | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | DU-145 | Prostate Cancer | MTT assay | IC50 = 120.72 ± 7.08 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | RP-7 | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MCF-7 | Breast Cancer | MTT assay | IC50 = 110.12 ± 4.23 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | LA3IK-SCR | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | DU-145 | Prostate Cancer | MTT assay | IC50 = 351.76 ± 7.18 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | RP-7 | 7 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 139.03 ± 8.41 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | LA3IK-SCR | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | PC-3 | Prostate Cancer | MTT assay | IC50 = 319 ± 13.64 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | LA3IK-SCR | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MCF-7 | Breast Cancer | MTT assay | IC50 = 133 ± 9.52 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | LA3IK-SCR | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 243 ± 8.16 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | D-LA3IK | 6 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | PC-3 | Prostate Cancer | MTT assay | IC50 = 98.71 ± 6.17 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | D-LA3IK | 6 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | DU-145 | Prostate Cancer | MTT assay | IC50 = 89.11 ± 8.12 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | D-LA3IK | 6 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MCF-7 | Breast Cancer | MTT assay | IC50 = 91.2 ± 8.21 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | LA3IK | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | DU-145 | Prostate Cancer | MTT assay | IC50 = 335.7 ± 3.09 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | D-LA3IK | 6 | Linear | D | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 197.72 ± 5.42 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | LA3IK | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MCF-7 | Breast Cancer | MTT assay | IC50 = 90.23 ± 7.32 µM | 24-h | Breast | None | ||
| 38272230 | 2024 | LA3IK | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | PC-3 | Prostate Cancer | MTT assay | IC50 = 321.4 ± 11.79 µM | 24-h | Prostate | None | ||
| 38272230 | 2024 | LA3IK | 6 | Linear | L | None | Amidation | Acetylation | Anticancer | Migration and invasion enhancer 1 (MIEN1) | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 223.6 ± 5.62 µM | 24-h | Breast | None | ||
| 38464729 | 2024 | U7 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | HepG-2 | Liver Cancer | MTT assay | IC50 = 523 µM | 48-h | Liver | None | ||
| 38464729 | 2024 | U7 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | MCF-7 | Breast Cancer | MTT assay | IC50 = 554 µM | 48-h | Breast | None | ||
| 38464729 | 2024 | U7 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | T-47D | Breast Cancer | MTT assay | IC50 = 584 ± 29.99 µM | 48-h | Breast | None | ||
| 38464729 | 2024 | U3 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | HepG-2 | Liver Cancer | MTT assay | IC50 = 561 µM | 48-h | Liver | None | ||
| 38464729 | 2024 | U3 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | T-47D | Breast Cancer | MTT assay | IC50 = 517.6 ± 34.86 µM | 48-h | Breast | None | ||
| 38464729 | 2024 | U3 | 11 | Linear | L | None | Free | Free | Anticancer | Phoenix dactylifera | MCF-7 | Breast Cancer | MTT assay | IC50 = 555 µM | 48-h | Breast | None | ||
| 37298595 | 2023 | NT-12 | 9 | Linear | L | Tle = L-tert-leucine | Free | Free | Anticancer | Synthetic analogue of Neurotensin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | NT-12 | 9 | Linear | L | Tle = L-tert-leucine | Free | Free | Anticancer | Synthetic analogue of Neurotensin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | NT-11 | 6 | Linear | L | None | Free | Free | Anticancer | Synthetic analogue of Neurotensin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | NT-12 | 9 | Linear | L | Tle = L-tert-leucine | Free | Free | Anticancer | Synthetic analogue of Neurotensin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | NT-9 | 6 | Linear | L | None | Free | Free | Anticancer | Synthetic analogue of Neurotensin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | NT-10 | 6 | Linear | L | None | Free | Free | Anticancer | Synthetic analogue of Neurotensin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-7 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (D)Pip—(D)-piperidine-2-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-8 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (D)Pip—(D)-piperidine-2-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-5 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (L)Pip—(L)-piperidine-2-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-6 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; (L)Pip—(L)-piperidine-2-carboxylic acid;(D)Pip—(D)-piperidine-2-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-3 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Acc = 1-aminocyclohexane-1-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-4 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Acc = 1-aminocyclohexane-1-carboxylic acid | Free | Aaa = [(3S,5S,7S)-adamantan-1-yl]acetic acid | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-1 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Apc =1-aminocyclopentyl-1-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37298595 | 2023 | BK-2 | 10 | Linear | Mix | Hyp = hydroxyproline; Thi = thienylalanine; Apc =1-aminocyclopentyl-1-carboxylic acid | Free | Free | Anticancer | Synthetic analogue of Bradykinin | HCT-116 | Colorectal Cancer | MTS assay | Not Available | 24-h | Colon | None | ||
| 37344820 | 2023 | Moricin | 43 | Linear | L | None | Free | Free | Antimicrobial | Bombyx mori | MDA-MB-231 | Triple-negative Breast Cancer | Trypan blue assay | 70% cell viability at 6.25 µg/ml | 24-h | Breast | None | ||
| 37344820 | 2023 | Moricin | 43 | Linear | L | None | Free | Free | Antimicrobial | Bombyx mori | MDA-MB-231 | Triple-negative Breast Cancer | LDH release assay | Significant decrease in cell viability at 6.25 μg/ml | 24-h | Breast | None | ||
| 37880286 | 2023 | MC–FA | 27 | Linear | L | None | Folic Acid | Free | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 12.63 µg/mL | 24-h | Breast | None | ||
| 37344820 | 2023 | Moricin | 43 | Linear | L | None | Free | Free | Antimicrobial | Bombyx mori | MDA-MB-231 | Triple-negative Breast Cancer | MTT assay | 70% cell viability at 6.25 µg/ml | 24-h | Breast | None | ||
| 37880286 | 2023 | MC–FA | 27 | Linear | L | None | Folic Acid | Free | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 66.43 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | MC–FA | 27 | Linear | L | None | Folic Acid | Free | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 35.22 µg/ mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | CM–FA | 27 | Linear | L | None | Amidation | Folic Acid | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 35.75 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | CM–FA | 27 | Linear | L | None | Amidation | Folic Acid | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 10.38 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | CM–FA | 27 | Linear | L | None | Amidation | Folic Acid | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 67.34 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | Mel-C | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 160.62 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | Mel-C | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 58.63 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | Mel-C | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 50.72 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | C-Mel | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | MCF-7 | Breast Cancer | MTT assay | IC50 = 110.59 µg/mL | 24-h | Breast | None | ||
| 37880286 | 2023 | C-Mel | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | C-33A | Cervical Cancer | MTT assay | IC50 = 44.76 µg/mL | 24-h | Cervix | None | ||
| 37880286 | 2023 | C-Mel | 27 | Linear | L | None | Amidation | Free | Anticancer; Antibacterial | Synthetic analogue | HeLa | Cervical Cancer | MTT assay | IC50 = 64.15 µg/mL | 24-h | Cervix | None | ||
| 37251837 | 2023 | CPSA-CPSC-L-ACAN | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | Anticancer | Recombinant Fusion Peptide | HeLa | Cervical Cancer | MTT assay | IC50 = 63.15 μg/ml | 24-h | Cervix | None | ||
| 36873017 | 2023 | LK-LE3 | 30 | Cyclic | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 10.2 µM at pH 6 | 24-h | Cervix | None | ||
| 36873017 | 2023 | LK-LE2 | 30 | Cyclic | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 12.9 µM at pH 6 | 24-h | Cervix | None | ||
| 36873017 | 2023 | LK-LE1 | 30 | Cyclic(C1-C16) | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 11.3 µM at pH 6 | 24-h | Cervix | None | ||
| 37104235 | 2023 | LHRH-BinBC | 195 | Linear | L | None | Free | Fused a luteinizing hormone-releasing hormone (LHRH) peptide | Mosquitocidal, Anticancer | Synthetic | MCF-7 | Breast Cancer | LDH leakage assay | 40% LDH efflux at 16 µM | 48-h | Breast | None | ||
| 37104235 | 2023 | LHRH-BinBC | 195 | Linear | L | None | Free | Fused a luteinizing hormone-releasing hormone (LHRH) peptide | Mosquitocidal, Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 10.96 μM | 48-h | Breast | None | ||
| 37001908 | 2023 | A11 | 11 | Linear | L | None | Free | Free | Anticancer | Annexin A1 | A-375 | Skin Cancer | Biotin Pull Down assay | Not Available | 24-h | Skin | None | ||
| 37001908 | 2023 | A11 | 11 | Linear | L | None | Free | Free | Anticancer | Annexin A1 | MDA-MB-231 | Breast Cancer | Biotin Pull Down assay | Not Available | 24-h | Breast | None | ||
| 37001908 | 2023 | A11 | 11 | Linear | L | None | Free | Free | Anticancer | Annexin A1 | H-460 | Lung Cancer | Biotin Pull Down assay | Not Available | 24-h | Lung | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HepG-2 | Liver Cancer | Cell Viability assay | IC50 = 34.05 ± 0.53 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HT-29 | Colon Cancer | Cell Viability assay | IC50 = 42.6 ± 4.0 μM | 48-h | Colon | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HeLa | Cervical Cancer | HDAC inhibition assay | IC50 = 0.446±0.095 µM | Not Available | Cervix | None | ||
| 36934526 | 2023 | WP2 | 14 | Linear | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | Huh-7 | Liver Cancer | Cell Viability assay | IC50 = 28.12 ± 1.5 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | Huh-7 | Liver Cancer | Cell Viability assay | IC50 = 43.74 ± 5.4 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HepG-2 | Liver Cancer | Cell Viability assay | IC50 = 52.23 ± 0.9 μM | 48-h | Liver | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HT-29 | Colon Cancer | Cell Viability assay | IC50 = 54.6 ± 2.1 μM | 48-h | Colon | None | ||
| 36934526 | 2023 | WP1 | 14 | Cyclic(M6-M10) | L | None | Hydroxamic acid | Acetylation | Anticancer | Derived from RLL peptide | HeLa | Cervical Cancer | HDAC inhibition assay | IC50 = 0.310±0.064 µM | Not Available | Cervix | None | ||
| 37734650 | 2023 | NKL-MUT | 27 | Linear | L | None | Free | Free | Antimicrobial | Trematomus bernacchii | B16-F10 | Skin Cancer | luciferase-based ATPlite assay | ATP level = 0.023 ± 0.007 at 40 μM | 12-h | Skin | None | ||
| 34986732 | 2023 | trans-Phakellistatin 18 | 7 | Cyclic | L | Proline residues in trans-configuration | Free | Free | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 67.5 ± 2.938 µM | Not Available | Liver | None | ||
| 37734650 | 2023 | NKL-WT | 27 | Linear | L | None | Free | Free | Antimicrobial | Trematomus bernacchii | B16-F10 | Skin Cancer | luciferase-based ATPlite assay | ATP level = 0.753 ± 0.254 at 40 μM | 12-h | Skin | None | ||
| 36840453 | 2023 | AMP-WF3 | 25 | Linear | L | None | Free | Free | Anticancer | Poecilia Mexicana fish | Jurkat | Blood Cancer | MTT assay | IC50 = 50 µM | 24-h | Blood | None | ||
| 31234333 | 2023 | LFB | 33 | Linear | L | None | Free | Free | Antimicrobial | Limnonectes fujianensis | HCT-116 | Colon Cancer | LDH leakage assay | LDH release above 80% | 24-h | Colon | None | ||
| 31234333 | 2023 | LFB | 33 | Linear | L | None | Free | Free | Antimicrobial | Limnonectes fujianensis | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.02 μM | 24-h | Colon | None | ||
| 31234333 | 2023 | LFB | 33 | Linear | L | None | Free | Free | Antimicrobial | Limnonectes fujianensis | U-251-MG | Brain Tumor | MTT assay | IC50 = 2.32 μM | 24-h | Brain | None | ||
| 31234333 | 2023 | LFB | 33 | Linear | L | None | Free | Free | Antimicrobial | Limnonectes fujianensis | MDA-MB-435 | Breast Cancer | MTT assay | IC50 = 18.99 μM | 24-h | Breast | None | ||
| 31234333 | 2023 | LFB | 33 | Linear | L | None | Free | Free | Antimicrobial | Limnonectes fujianensis | H-460 | Lung Cancer | MTT assay | IC50 = 3.47 μM | 24-h | Lung | None | ||
| 37764521 | 2023 | GE18 | 18 | Linear | L | None | Free | Free | Antimicrobial | Aphanomyces invadans | MCF-7 | Breast Cancer | MTT assay | IC50 = 35.34 µM | 24-h | Breast | None | ||
| 36626098 | 2023 | LFchimera | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic - Lectoferrin chimera | Jurkat | Blood Cancer | MTT assay | cell viability ~ 8% at 20 µM | 6-h | Blood | None | ||
| 36626098 | 2023 | LFchimera | 35 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic - Lectoferrin chimera | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 44% at 10 µM | 12-h | Liver | None | ||
| 36626098 | 2023 | LFampin265–284 | 20 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | Jurkat | Blood Cancer | MTT assay | cell viability ~ 47% at 10 µM | 6-h | Blood | None | ||
| 36626098 | 2023 | LFampin265–284 | 20 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 50% at 1 µM | 12-h | Liver | None | ||
| 36626098 | 2023 | LFcin17–30 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | Jurkat | Blood Cancer | MTT assay | cell viability ~ 70% at 20 µM | 6-h | Blood | None | ||
| 36626098 | 2023 | LFcin17–30 | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Lectoferrin Peptide | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 50% at 1 µM | 12-h | Liver | None | ||
| 36626098 | 2023 | bLF | 25 | Linear | L | None | Free | Free | Antimicrobial | Bos Taurus | Jurkat | Blood Cancer | MTT assay | cell viability ~ 17.5% at 20 µM | 4-h | Blood | None | ||
| 36509220 | 2023 | KM8-Aib | 18 | Linear | L | Aib = 2-Aminoisobutyric acid | Amidation | Free | Antimicrobial | Synthetic derivative of KM8 | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 36626098 | 2023 | bLF | 25 | Linear | L | None | Free | Free | Antimicrobial | Bos Taurus | HepG-2 | Liver Cancer | MTT assay | cell viability ~ 21% at 10 µM | 24-h | Liver | None | ||
| 36509220 | 2023 | KM8 | 18 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic derivative of Mastoparan | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 36509220 | 2023 | Mastoparan | 14 | Linear | L | None | Amidation | Free | Antimicrobial | Wasp venom | Not Available | Not Available | Not Available | Not Available | Not Available | Not Available | None | ||
| 37380046 | 2023 | RP7 | 7 | Linear | L | None | Free | Free | Anticancer | RAGE(receptor for advanced glycation end product) inhibitor | BT-549 | Breast Cancer | MTT assay | IC50 = 29.9 µM | 48-h | Breast | None | ||
| 37380046 | 2023 | RP7 | 7 | Linear | L | None | Free | Free | Anticancer | RAGE(receptor for advanced glycation end product) inhibitor | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 24.5 µM | 48-h | Breast | None | ||
| 36567478 | 2023 | mtp1 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTS assay | 17.4% decrease in cell viability at 10 μM | 24-h | Lung | None | ||
| 36567478 | 2023 | mtp1 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTS assay | 33.6% decrease in cell viability at 10 μM | 24-h | Breast | None | ||
| 36567478 | 2023 | mtp1 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTS assay | 30.2 % decrease in cell viability at 10 μM | 24-h | Cervix | None | ||
| 37273629 | 2023 | PS9 | 9 | Linear | L | None | Free | Free | Anticancer | Aphanomyces invadans | MCF-7 | Breast Cancer | LDH leakage assay | 71.25 ± 1.3% LDH release at 40 μM | 24-h | Breast | None | ||
| 37273629 | 2023 | PS9 | 9 | Linear | L | None | Free | Free | Anticancer | Aphanomyces invadans | MCF-7 | Breast Cancer | Neutral Red Uptake assay | IC50 value range between 25.27 - 43.28 μM | 24-h | Breast | None | ||
| 37098530 | 2023 | Mellitin | 26 | Linear | L | None | Amidation | Free | Anticancer | Main component of honey bee venom | K-562 | Leukemia Cancer | Sulforhodamine B assay | IC50 = 1.84 ± 0.75 μg/ml | 96-h | Blood | None | ||
| 37068520 | 2023 | Test peptide | 5 | Linear | L | None | Amidation | Free | Anti cancer | Neuropep Peptide | A-549 | Lung Cancer | MTT assay | IC50 = 26.417±0.660 µM | 48 h | Lung | None | ||
| 37068520 | 2023 | Test peptide | 5 | Linear | L | None | Amidation | Free | Anti cancer | Neuropep Peptide | MDA-MB-231 | Lung Cancer | MTT assay | IC50 = 39.047±0.770 µM | 48 h | Lung | None | ||
| 36830725 | 2023 | Pep-1-Phor21 | 30 | Linear | L | None | Free | Free | Anticancer | Hybrid peptide PEP1 and Phor 21 | PC-3 | Prostrate Cancer | AlamarBlue assay | IC50 ≤ 0.6 μM | 24-h | Prostate | None | ||
| 36830725 | 2023 | Pep-1-Phor21 | 30 | Linear | L | None | Free | Free | Anticancer | Hybrid peptide PEP1 and Phor 21 | DU-145 | Prostrate Cancer | AlamarBlue assay | IC50 = 2.57 ± 2.02 µM | 24-h | Prostate | None | ||
| 36168817 | 2023 | Rapeseed peptide | 7 | Linear | L | None | Free | Free | Anticancer | extracted from rapeseed protein | HepG-2 | Liver Cancer | Apoptosis assay | 28.39 ± 0.80% apoptosis rate at 0.5 mmol/L | NA | Liver | None | ||
| 36830725 | 2023 | Pep-1-Phor21 | 30 | Linear | L | None | Free | Free | Anticancer | Hybrid peptide PEP1 and Phor 21 | LNCaP | Liver Cancer | AlamarBlue assay | IC50 = 55.13 ± 13.56 µM | 24-h | Liver | None | ||
| 36168817 | 2023 | Rapeseed peptide | 7 | Linear | L | None | Free | Free | Anticancer | extracted from rapeseed protein | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.56 mmol/L | 24-h | Liver | None | ||
| 37514049 | 2023 | Salamandrin - I | 12 | Linear | L | None | Amidation | Free | Antioxidant | Salamandra salamandra | HL-60 | Leukemia Cancer | LDH leakage assay | Absorbance ~ 2 at 490 nm at 27 27 µM | 48-h | Blood | None | ||
| 37514049 | 2023 | Salamandrin - I | 12 | Linear | L | None | Amidation | Free | Antioxidant | Salamandra salamandra | HL-60 | Leukemia Cancer | MTT assay | IC50 = 27 µM | 48-h | Blood | None | ||
| 37580909 | 2023 | mPNC-NLS | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | Cytotoxicity assay | IC50 = 45 μM | 24-h | Lung | None | ||
| 37580909 | 2023 | mPNC-NLS | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | U-87 | Brain Tumor | MTT assay | IC50 = 56.9 μM | 24-h | Brain | None | ||
| 37580909 | 2023 | mPNC-NLS | 21 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 44.9 μM | 24-h | Lung | None | ||
| 36730301 | 2023 | Lasioglossin - III | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Lasioglossum laticeps | HepG-2 | Liver Cancer | Not Available | IC50 = 7.75 μM | Not Available | Liver | None | ||
| 36730301 | 2023 | Lasioglossin - III | 15 | Linear | L | None | Amidation | Free | Antimicrobial | Lasioglossum laticeps | A-549 | Lung Cancer | Not Available | IC50 = 26.36 μM | Not Available | Lung | None | ||
| 37483971 | 2023 | ATMP1 | 24 | Linear | L | None | Free | Free | Antimicrobial | Anabas testudineus | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 8.25 ± 0.14 μg/ml | 48-h | Breast | None | ||
| 37483971 | 2023 | ATMP5 | 24 | Linear | L | None | Free | Free | Anticancer; Antimicrobial | Synthetic Analog of ATMP1 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 64.04 ± 0.021 μg /ml | 24-h | Breast | None | ||
| None | 2023 | Raniseptin-3 | 28 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Boana raniceps | B16-F10 | Skin Cancer | MTT assay | IC50 = 6.56 uM | 3-h | Skin | None | ||
| 36910465 | 2023 | ALA-A2 | 13 | Linear | L | None | Free | Free | Anticancer | Alpha-Lactalbumin | HT-29 | Colon Cancer | MTT assay | ~50% cell viability | 24-h | Colon | None | ||
| None | 2023 | Raniseptin-6 | 29 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Boana raniceps | B16-F10 | Skin Cancer | MTT assay | IC50 = 8.69 uM | 3-h | Skin | None | ||
| 36910465 | 2023 | ALA-A2 | 13 | Linear | L | None | Free | Free | Anticancer | Alpha-Lactalbumin | A-549 | Lung Cancer | MTT assay | ~50% cell viability | 24-h | Lung | None | ||
| 37310533 | 2023 | PMAP-NC | 23 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analgog of PMAP-24 | A-549 | Lung Cancer | MTT assay | IC50 = 7.1 μM | 4-h | Lung | None | ||
| 37310533 | 2023 | PMAP-NC | 23 | Linear | L | None | Free | Free | Antimicrobial | Synthetic Analgog of PMAP-23 | MDA-MB-361 | Breast Cancer | MTT assay | IC50 = 6.4 μM | 4-h | Breast | None | ||
| 37183466 | 2023 | CM11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Cecropin-Melittin Hybrid Peptide | Raji | Blood Cancer | MTT assay | Survival rate = 51% at 32 μg/ml | 24-h | Blood | None | ||
| 37183466 | 2023 | CM11 | 11 | Linear | L | None | Amidation | Free | Antimicrobial | Cecropin-Melittin Hybrid Peptide | Jurkat | Blood Cancer | MTT assay | Survival rate = 47% at 32 μg/ml | 24-h | Blood | None | ||
| 37764334 | 2023 | 14VL23 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 16.4 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14VL23 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 5.7 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V5K | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 6.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V5K | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 8.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L2V | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 0.6 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L2V | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 2.2 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14G | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 31.7 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14G | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 48.7 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 4.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | 14V | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 7.0 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L14 | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-460 | Lung Cancer | MTT assay | IC50 = 20.1 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | L14 | 22 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Dermaseptin-SS1- Analog | H-838 | Lung Cancer | MTT assay | IC50 = 64.4 µM | 24-h | Lung | None | ||
| 37764334 | 2023 | Dermaseptin-SS1 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Brown-belly leaf frog, Phyllomedusa Tarsius | H-460 | Lung Cancer | MTT assay | IC50 = 1.3 µM | 24-h | Lung | None | ||
| 36982610 | 2023 | K2-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 9 µM | 24-h | Breast | None | ||
| 37764334 | 2023 | Dermaseptin-SS1 | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Brown-belly leaf frog, Phyllomedusa Tarsius | H-838 | Lung Cancer | MTT assay | IC50 = 7.7 µM | 24-h | Lung | None | ||
| 36982610 | 2023 | K56-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =12 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K6-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =8 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K259-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =10 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K25-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =9 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K259-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 =13 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | Leu4-NH2 | 10 | Linear | L | U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 > 20 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | K2569-Lol | 10 | Linear | L | U = 2-Aminoisobutyric acid | Lol = leucinol | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 12 µM | 24-h | Breast | None | ||
| 36982610 | 2023 | Api8-NH2 | 10 | Linear | L | Z =4-aminopiperidine-4-carboxylic acid , U = 2-Aminoisobutyric acid | Amidation | Oct = 1-octanoyl | Antimicrobial and Antifungal | Trichogin GA | MDA-MB-231 | Breast Cancer | MTS assay | IC50 > 20 µM | 24-h | Breast | None | ||
| 36678914 | 2023 | trichoderin A analogue 18 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | decanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.2 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 19 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | dodecanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.2 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 17 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Octanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.6 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 16 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Hexanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.5 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 14 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Propanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 1.8 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 15 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Butanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.9 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 13 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Ethanoyl | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 6.0 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 12 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 > 9 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 4 | 10 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderin A | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.5 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 19 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | dodecanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.1 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A | 10 | Linear | L | MDA = 2-methyl decanoic acid; AHMOD = 2-amino-6-hydroxy-4-methyl-8-oxodecanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderma sp. fungus, strain 05FI48 | PANC-1 | Pancreatic Cancer | CyQUANT Direct assay | IC50 = 0.3 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 18 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | decanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.2 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 17 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid; AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Octanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.4 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 16 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Hexanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.4 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 15 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Butanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.5 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 13 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Ethanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 > 1 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 14 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Propanoyl | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.6 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 12 | 9 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 > 1 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A | 10 | Linear | L | MDA = 2-methyl decanoic acid; AHMOD = 2-amino-6-hydroxy-4-methyl-8-oxodecanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderma sp. fungus, strain 05FI48 | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.4 μM | 24-h | Pancreas | None | ||
| 36678914 | 2023 | trichoderin A analogue 4 | 10 | Linear | L | AHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanol | Free | Free | Antitubercular | Trichoderin A | BxPC-3 | Pancreatic Cancer | PrestoBlue assay | IC50 = 0.4 μM | 24-h | Pancreas | None | ||
| 37228702 | 2023 | B1AW-K | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | analogue of B1AW | U251-MG | Brain Tumor | MTT assay | IC50 = 3.860 µM | 24-h | Brain | None | ||
| 37228702 | 2023 | B1AW-K | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | analogue of B1AW | H-838 | Lung Cancer | MTT assay | IC50 = 5.15 µM | 24-h | Lung | None | ||
| 37228702 | 2023 | B1AW-K | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | analogue of B1AW | PC-3 | Prostate Cancer | MTT assay | IC50 = 4.283 µM | 24-h | Prostate | None | ||
| 37228702 | 2023 | B1AW | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Wuyi torrent frog, Amolops wuyiensis | U251-MG | Brain Tumor | MTT assay | IC50 = 33.56 µM | 24-h | Brain | None | ||
| 37228702 | 2023 | B1AW | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Wuyi torrent frog, Amolops wuyiensis | H-838 | Lung Cancer | MTT assay | IC50 = 32.15 µM | 24-h | Lung | None | ||
| 37228702 | 2023 | B1AW | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Wuyi torrent frog, Amolops wuyiensis | PC-3 | Prostate Cancer | MTT assay | IC50 = 33.46 µM | 24-h | Prostate | None | ||
| 37508198 | 2023 | Figanin 2BN | 27 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | HT-29 | Colon Cancer | MTT assay | LC50 = 14.1 uM | 24-h | Colon | None | ||
| 37508198 | 2023 | Figanin 2BN | 27 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | MDA-MB-231 | Breast Cancer | MTT assay | LC50 = 8.1 uM | 24-h | Breast | None | ||
| 37508198 | 2023 | Figanin 2BN | 27 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | A-549 | Lung Cancer | MTT assay | LC50 = 6.7 uM | 24-h | Lung | None | ||
| 37508198 | 2023 | Picturin 1BN | 25 | Linaer | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | HT-29 | Colon Cancer | MTT assay | LC50 = 84.9 uM | 24-h | Colon | None | ||
| 37508198 | 2023 | Picturin 1BN | 25 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | MDA-MB-231 | Breast Cancer | MTT assay | LC50 = 64.2 uM | 24-h | Breast | None | ||
| 37508198 | 2023 | Picturin 1BN | 25 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | A-549 | Lung Cancer | MTT assay | LC50 = 30.7 µM | 24-h | Lung | None | ||
| 37508198 | 2023 | Picturin 2BN | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | HT-29 | Colon Cancer | MTT assay | LC50 52.2 uM | 24-h | Colon | None | ||
| 37508198 | 2023 | Picturin 2BN | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | MDA-MB-231 | Breast Cancer | MTT assay | LC50 26.3 uM | 24-h | Breast | None | ||
| 37508198 | 2023 | Picturin 2BN | 23 | Linear | L | None | Amidation | Free | Antimicrobial and Antitumor | Giant Gladiator Treefrog (Boana boans) | A-549 | Lung Cancer | MTT assay | LC50 = 23 µM | 24-h | Lung | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 32.47 µM | 36-h | Lung | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | CCK-8 assay | IC50 = 25.65 µM | 36-h | Bone | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | CCK-8 assay | IC50 = 42.95 µM | 36-h | Cervix | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | ZR-75-30 | Breast Cancer | CCK-8 assay | IC50 = 23.57 µM | 36-h | Breast | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | CCK-8 assay | IC50 = 31.05 µM | 36-h | Breast | None | ||
| 37598210 | 2023 | M1-20 | 30 | Linear | D | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | CCK-8 assay | IC50 = 18.15 µM | 36-h | Breast | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | ZR-75-30 | Breast Cancer | Cell Viability assay | IC50 = 12.92 µM | 72-h | Breast | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | U-251 | BrainTumor | Cell Viability assay | IC50 = 18.17 µM | 72-h | Brain | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | Cell Viability assay | IC50 = 22.00 µM | 72-h | Lung | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | HCT-116 | Colon Cancer | Cell Viability assay | IC50 = 9.08 µM | 72-h | Colon | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | 786-0 | Renal Cancer | Cell Viability assay | IC50 = 13.5 µM | 72-h | Renal | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Cell Viability assay | IC50 = 31.83 µM | 72-h | Cervix | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | 5637 | Bladder cancer | Cell Viability assay | IC50 = 9.33 µM | 72-h | Bladder | None | ||
| 37344857 | 2023 | M1-21 | 31 | Linear | Mix | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | Cell Viability assay | IC50 = 24.25 µM | 72-h | Breast | None | ||
| 37396945 | 2023 | p28 | 28 | Linear | L | None | Free | Free | Antitumor | Pseudomonas aeruginosa | CT-26 | Colorectal Cancer | MTT assay | IC50 ~ 150 μg/ml | 24-h | Colon | None | ||
| 37396945 | 2023 | p28 | 28 | Linear | L | None | Free | Free | Antitumor | Pseudomonas aeruginosa | HT-29 | Colon Cancer | MTT assay | IC50 ~ 200 μg/ml | 24-h | Colon | None | ||
| 36687035 | 2023 | 1-R | 8 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 130 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | 1-R | 8 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 > 150 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | R-1 | 8 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 > 150 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | R-1 | 8 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 58 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | 1 | 7 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 105 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | 1 | 7 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 > 170 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-R | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 68 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-R | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 73 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | R-1-RR | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 95 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-RR | 11 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 67 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | R-1-RR | 10 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 122 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | LfcinB(21-25)Pal | 9 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | LfcinB | MCF-7 | Breast Cancer | MTT assay | IC50 = 81 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | RR-1-RR | 11 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | Synthetic analogue of LfcinB(21-25)Pal | MCF-7 | Breast Cancer | MTT assay | IC50 = 58 µM | 24-h | Breast | None | ||
| 36687035 | 2023 | LfcinB(21-25)Pal | 9 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | LfcinB | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 103 µM | 24-h | Breast | None | ||
| 37818062 | 2023 | P10 | 13 | Linear | L | None | Free | Free | Anticancer | 40S ribosomal protein fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.01 at 50 μg/ml | 48-h | Bone | None | ||
| 36687035 | 2023 | LfcinB(21-25)Pal | 9 | Linear | L | None | Amidation | Free | Antibacterial and Anticancer | LfcinB | MDA-MB-468 | Breast Cancer | MTT assay | IC50 = 72 µM | 24-h | Breast | None | ||
| 37818062 | 2023 | P09 | 13 | Linear | L | None | Free | Free | Anticancer | Eukaryotic Translation Elongation Factor 1 Gamma (Eef1G) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.07 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P10 | 13 | Linear | L | None | Free | Free | Anticancer | 40S ribosomal protein fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 1.08 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P09 | 13 | Linear | L | None | Free | Free | Anticancer | Eukaryotic Translation Elongation Factor 1 Gamma (Eef1G) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.85 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P08 | 16 | Linear | L | None | Free | Free | Anticancer | Lamin A/C (LMNA) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.92 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P08 | 16 | Linear | L | None | Free | Free | Anticancer | Lamin A/C (LMNA) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.06 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P07 | 13 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.96 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P07 | 13 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.96 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P06 | 18 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.92 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P06 | 18 | Linear | L | None | Free | Free | Anticancer | FLNA (Filamin A) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.17 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P03 | 13 | Linear | L | None | Free | Free | Anticancer | Triosephosphate Isomerase (TPI) fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.98 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P01 | 16 | Linear | L | None | Free | Free | Anticancer | Histone H1.4 (H1-4) Fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 1.13 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P03 | 13 | Linear | L | None | Free | Free | Anticancer | Triosephosphate Isomerase (TPI) fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 1.04 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P04 | 20 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.83 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P01 | 16 | Linear | L | None | Free | Free | Anticancer | Histone H1.4 (H1-4) Fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.84 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P04 | 20 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.86 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P02 | 15 | Linear | L | None | Free | Free | Anticancer | Rho GDP Dissociation Inhibitor Alpha fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.88 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P02 | 15 | Linear | L | None | Free | Free | Anticancer | Rho GDP Dissociation Inhibitor Alpha fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.93 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P05 | 12 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | U-2 OS | Bone Cancer | MTT assay | Relative viability = 0.98 at 50 μg/ml | 48-h | Bone | None | ||
| 37818062 | 2023 | P05 | 12 | Linear | L | None | Free | Free | Anticancer | Aldolase A fragment | MG-63 | Bone Cancer | MTT assay | Relative viability = 0.85 at 50 μg/ml | 48-h | Bone | None | ||
| 37495988 | 2023 | 37-mer peptide | 37 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | SK-OV-3 | Ovarian cancer | MTT assay | IC50 = 27.45 ± 1.5085 μM | 24-h | Ovary | None | ||
| 37495988 | 2023 | 37-mer peptide | 37 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 33.65 ± 1.09 μM | 24-h | Liver | None | ||
| 37495988 | 2023 | 37-mer peptide | 37 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | SNU-449 | Liver Cancer | MTT assay | IC50 = 76.4 ± 0.6015 μM | 24-h | Liver | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant_R5 (R5-Aurm) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | HT-29 | Colon Cancer | MTT assay | 54.22% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant_R5 (R5-Aurm) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | SW-480 | Colon Cancer | MTT assay | 40.62% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_R5 (R5-Aur) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | HT-29 | Colon Cancer | MTT assay | 61.56% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant (Aurm) | 13 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | HT-29 | Colon Cancer | MTT assay | 66.10% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_R5 (R5-Aur) | 18 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | SW-480 | Colon Cancer | MTT assay | 43.89% cell viability | 24-h | Colon | None | ||
| 37646048 | 2023 | Aurein 1.2_mutant (Aurm) | 13 | Linear | L | None | Free | Acetylation | Antimicrobial | Synthetic | SW-480 | Colon Cancer | MTT assay | 51.63% cell viability | 24-h | Colon | None | ||
| 37867694 | 2023 | 1[dR] 5[Orn] [Pal] | 9 | Linear | Mix | O=Ornithine | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 109 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | 5[Orn] [Pal] | 9 | Linear | L | O=Ornithine | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 64 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | 1[Orn] [Pal] | 9 | Linear | L | O=Ornithine | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 91 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | CH3CO-Ahx-[Pal] | 10 | Linear | L | Ahx = Amino Hexanoic Acid | Amidation | Acetylation | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 31 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | 1[dR][Pal] | 9 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 105 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | 9[Orn] [Pal] | 9 | Linear | L | O=Ornithine | Amidation | Free | Anticancer | Synthetic | DU-145 | Prostrate Cancer | MTT assay | IC50 = 62 μM | 24-h | Prostate | None | ||
| 37867694 | 2023 | 9[Orn] [Pal] | 9 | Linear | L | O=Ornithine | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT assay | IC50 = 109 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | 9[Orn] [Pal] | 9 | Linear | L | O=Ornithine | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 40 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | Ahx-[Pal] | 10 | Linear | L | Ahx = Amino Hexanoic Acid | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT assay | IC50 = 119 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | Ahx-[Pal] | 10 | Linear | L | Ahx = Amino Hexanoic Acid | Amidation | Free | Anticancer | Synthetic | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 40 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | LfcinB (21-25)Pal | 9 | Linear | L | None | Amidation | Free | Anticancer | LfcinB | DU-145 | Prostrate Cancer | MTT assay | IC50 = 40 μM | 24-h | Prostate | None | ||
| 37867694 | 2023 | LfcinB (21-25)Pal | 9 | Linear | L | None | Amidation | Free | Anticancer | LfcinB | HT-29 | Colon Cancer | MTT assay | IC50 = 100 μM | 24-h | Colon | None | ||
| 37867694 | 2023 | LfcinB (21-25)Pal | 9 | Linear | L | None | Amidation | Free | Anticancer | LfcinB | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 86 μM | 24-h | Colon | None | ||
| 36410436 | 2023 | FHV-2D5 | 23 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-G | 48-h | Liver | None | ||
| 36410436 | 2023 | HTLV-II-Rex-2D5 | 21 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-G | 48-h | Liver | None | ||
| 36410436 | 2023 | TAT-2D5 | 21 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-G | 48-h | Liver | None | ||
| 36410436 | 2023 | 6F (I113-P122) | 20 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-D | 48-h | Liver | None | ||
| 36410436 | 2023 | 6E(V116-M135) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-D | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D5(G45-Y51) | 17 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | IC50 = 19.4 μM | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D3(G45-N52) | 18 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D2(Q44-Y51) | 18 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2D(Q44-R55) | 22 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2C(Q44-Q58) | 25 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | 2A(F39-Q58) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-C | 48-h | Liver | None | ||
| 36410436 | 2023 | #6(M108-L127) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | MCF-7 | Breast Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Breast | None | ||
| 36410436 | 2023 | #6(M108-L127) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Liver | None | ||
| 36410436 | 2023 | #5(D93-F112) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Liver | None | ||
| 36410436 | 2023 | #2(D33-N52) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | MCF-7 | Breast Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Breast | None | ||
| 36410436 | 2023 | #2(D33-N52) | 30 | Linear | L | None | Free | Free | Anticancer | STAP-2 PH domain–derived peptide | DU-145 | Liver Cancer | CellTiter-Glo assay | Graph figure 1-B | 48-h | Liver | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 12.29 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 16.29 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 17.70 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 22.37 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-PR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 32.32 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 29.90 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 32.51 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 52.01 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 28.78 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-AR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 41.31 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 33.85 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 30.29 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 15.87 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 62.17 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-FR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 31.51 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.459 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.810 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 12.40 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.944 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 23.18 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-TR | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 4.637 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 42.88 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 23.51 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 20.58 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | MCF-7 | Breast Cancer | MTT assay | IC50 = 20.26 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-4K | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 22.55 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | HCT-116 | Colon Cancer | MTT assay | IC50 = 47.02 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | U-251-MG | Brain Tumor | MTT assay | IC50 = 25.09 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | PC-3 | Prostate Cancer | MTT assay | IC50 = 17.98 μM | 24-h | Prostate | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | MCF-7 | Breast Cancer | MTT assay | IC50 = 26.49 μM | 24-h | Breast | None | ||
| 37833918 | 2023 | Crabrolin-4R | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic Analog of Crabrolin | H-838 | Lung Cancer | MTT assay | IC50 = 11.40 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | HCT-116 | Colon Cancer | MTT assay | IC50 = 8.539 μM | 24-h | Colon | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | U-251-MG | Brain Tumor | MTT assay | IC50 = 20.13 μM | 24-h | Brain | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | H-838 | Lung Cancer | MTT assay | IC50 = 27.71 μM | 24-h | Lung | None | ||
| 37833918 | 2023 | Crabrolin | 13 | Linear | L | None | Amidation | Free | Antimicrobial | European hornet (Vespa crabro) | PC-3 | Prostate Cancer | MTT assay | IC50 = 32.13 μM | 24-h | Prostate | None | ||
| 35889301 | 2022 | Sansalvimide A | 5 | Cyclic | L | X = OLeu | Cyclized | Cyclized | Anticancer | Fusarium sp. | HCT-116 | Colon Cancer | Not Available | IC50 = 9.8 µg/ml | Not Available | Colon | None | ||
| 35889301 | 2022 | Sansalvimide A | 5 | Cyclic | L | X = OLeu | Cyclized | Cyclized | Anticancer | Fusarium sp. | Colo-205 | Colon Cancer | Not Available | IC50 = 3.5 µg/ml | Not Available | Colon | None | ||
| 35889301 | 2022 | Sansalvimide A | 5 | Cyclic | L | X = OLeu | Cyclized | Cyclized | Anticancer | Fusarium sp. | SK-MEL-2 | Skin Cancer | Not Available | IC50 = 5.9 µg/ml | Not Available | Skin | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | EJ | Bladder Cancer | MTS assay | 89.6% apoptotic cells at 50 μg/mL | 24-h | Bladder | None | ||
| None | 2022 | MP12 | 12 | Linear | L | None | Free | Free | Antiproliferative | Aphanomyces invadans | Hep-2 | Larynx Cancer | MTT assay | IC50 = 24.7 ± 0.34 μM | Not Available | Larynx | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | EC-109 | Esophageal Cancer | MTS assay | 57.1% apoptotic cells at 50 μg/mL | 24-h | Esophagus | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | HepG-2 | Liver Cancer | MTS assay | 44.2% apoptotic cells at 50 μg/mL | 24-h | Liver | None | ||
| 33630204 | 2022 | LvHemB1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | hemocyanin of Litopenaeus vannamei | HeLa | Cervical cancer | MTS assay | 65.1% apoptotic cells at 50 μg/mL | 24-h | Cervix | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | SW-620 | Colon Cancer | MTT assay | IC50 >27 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | L02 | Colorectal Cancer | MTT assay | IC50 >150 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 10.88 ± 0.72 μg/mL | 48-h | Colon | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | DLD-1 | Colorectal Cancer | MTT assay | IC50 = 2.14 ± 0.28 μg/mL | 48-h | Colon | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | MCF-7 | Breast Cancer | MTT assay | IC50 = 24.60 μM | 24-h | Breast | None | ||
| 35200639 | 2022 | P6 | 20 | Linear | L | None | Free | Free | Antitumor | Arca inflata | HT-29 | Colorectal Cancer | MTT assay | IC50 = 4.43 ± 0.15 μg/mL | 48-h | Colon | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | U-251-MG | Brain Tumor | MTT assay | IC50 = 25.06 μM | 24-h | Brain | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | H-157 | Non-small cell lung cancer | MTT assay | IC50 = 24 μM | 24-h | Lung | None | ||
| 35606468 | 2022 | Nigrocin-M1 | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Analogue of Nigrocin M1 | PC-3 | Prostate cancer | MTT assay | IC50 = 31.27 μM | 24-h | Prostate | None | ||
| 35606468 | 2022 | Nigrocin-PN | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Pelophylax nigromaculatus | PC-3 | Prostate cancer | MTT assay | IC50 = 53.03 μM | 24-h | Prostate | None | ||
| 35606468 | 2022 | Nigrocin-PN | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Pelophylax nigromaculatus | U-251-MG | Brain Tumor | MTT assay | IC50 = 73.65 μM | 24-h | Brain | None | ||
| 35606468 | 2022 | Nigrocin-PN | 21 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Pelophylax nigromaculatus | H-157 | Non-small cell lung cancer | MTT assay | IC50 = 18.04 μM | 24-h | Lung | None | ||
| 36212827 | 2022 | Lt-MAP2 | 13 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Derivative of Lataracin-3a | C1498 | Blood Cancer | Cytotoxicity assay | EC50 = 43.9 ± 0.5 µg/mL | 24-h | Blood | None | ||
| 36212827 | 2022 | Lt-MAP2 | 13 | Linear | L | None | Free | Free | Antimicrobial and Antitumor | Synthetic; Derivative of Lataracin-3a | K-562 | Blood Cancer | Cytotoxicity assay | EC50 = 44 ± 3 µg/mL | 24-h | Blood | None | ||
| 36426386 | 2022 | [D4K,A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 46 ± 12 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | [D4K,A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 25 ± 1 μM | 24-h | Lung | None | ||
| 36426386 | 2022 | [D4K,A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 31 ± 1 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | [D4K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 20 ± 1 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | [D4K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 12 ± 1 μM | 24-h | Lung | None | ||
| 36426386 | 2022 | [D4K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 15 ± 1 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | Ocellatin-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Leptodactylus nesiotus | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 69 ± 10 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | Ocellatin-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Leptodactylus nesiotus | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 35 ± 1 μM | 24-h | Lung | None | ||
| 36426386 | 2022 | Ocellatin-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Leptodactylus nesiotus | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 51 ± 16 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | [A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | MDA-MB-231 | Breast Cancer | CellTiter-Glo assay | LC50 = 69 ± 18 μM | 24-h | Breast | None | ||
| 36426386 | 2022 | [A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | HT-29 | Colorectal Cancer | CellTiter-Glo assay | LC50 = 59 ± 4 μM | 24-h | Colon | None | ||
| 36426386 | 2022 | [A18K]OCN-3N | 19 | Linear | L | None | Amidation | Free | Host Defense | Synthetic; Derivative of ocellatin-3N | A-549 | Lung Cancer | CellTiter-Glo assay | LC50 = 30 ± 1 μM | 24-h | Lung | None | ||
| 35209215 | 2022 | RT2 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Crocodylus siamensis | CaCo-2 | Colon Cancer | MTT assay | IC50 = 29.74 μM | 24-h | Colon | None | ||
| 35628312 | 2022 | rScyreprocin | 90 | Linear | L | None | His-Tag | Free | Antimicrobial | Recombinant product of Scyreprocin | HeLa | Cervical cancer | MTS assay | IC50 = 3.34 x 104 µM | 24-h | Cervix | None | ||
| 35628312 | 2022 | rScyreprocin | 90 | Linear | L | None | His-Tag | Free | Antimicrobial | Recombinant product of Scyreprocin | DU-145 | Prostate cancer | MTS assay | IC50 = 1158.30 µM | 24-h | Prostate | None | ||
| 35628312 | 2022 | rScyreprocin | 90 | Linear | L | None | His-Tag | Free | Antimicrobial | Recombinant product of Scyreprocin | T-24 | Urinary Bladder Cancer | MTS assay | IC50 = 1.94 x 105 µM | 24-h | Bladder | None | ||
| 35628312 | 2022 | rScyreprocin | 90 | Linear | L | None | His-Tag | Free | Antimicrobial | Recombinant product of Scyreprocin | HepG-2 | Liver Cancer | MTS assay | IC50 = 441.01 µM | 24-h | Liver | None | ||
| 35628312 | 2022 | rScyreprocin | 90 | Linear | L | None | His-Tag | Free | Antimicrobial | Recombinant product of Scyreprocin | H-460 | Lung Cancer | MTS assay | IC50 = 6.27 µM | 72-h | Lung | None | ||
| 34999227 | 2022 | LA-C1b | 18 | Linear | L | Lauric acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | LA-C1b | 18 | Linear | L | Lauric acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | OA-C1b | 18 | Linear | L | Octanoic acid acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | OA-C1b | 18 | Linear | L | Octanoic acid acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | LA-C1b | 18 | Linear | L | Lauric acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 34999227 | 2022 | PA-C1b | 18 | Linear | L | Palmitic acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | OA-C1b | 18 | Linear | L | Octanoic acid acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 34999227 | 2022 | PA-C1b | 18 | Linear | L | Palmitic acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 34999227 | 2022 | PA-C1b | 18 | Linear | L | Palmitic acid conjugated to the 17th Lys-residue | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | Chensinin-1b | 18 | Linear | L | None | Amidation | Free | Antmicrobial and Anticancer | Synthetic | A-375 | Skin Cancer | Not Available | Not Available | Not Available | Skin | None | ||
| 34999227 | 2022 | Chensinin-1b | 18 | Linear | L | None | Amidation | Free | Antmicrobial and Anticancer | Synthetic | HeLa | Cervical Cancer | Not Available | Not Available | Not Available | Cervix | None | ||
| 34999227 | 2022 | Chensinin-1b | 18 | Linear | L | None | Amidation | Free | Antmicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | Not Available | Not Available | Not Available | Breast | None | ||
| 36555235 | 2022 | AC-P19 | 19 | Linear | L | None | Free | Free | Anticancer | Synthetic | H-460 | Lung Cancer | WST-8 assay | IC50 = 49.08 µM | 24-h | Lung | None | ||
| 36483599 | 2022 | Q7 | 15 | Linear | L | None | Free | Free | Anticancer | Pisum sativum | HEC-1-A | Endometrial Cancer | MTT assay | IC50 = 129.82 ± 7.53 μM | 48-h | Endometrium | None | ||
| 36555235 | 2022 | AC-P19 | 19 | Linear | L | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | WST-8 assay | IC50 = 52.14 µM | 24-h | Lung | None | ||
| None | 2022 | RF13 | 13 | Linear | L | None | Free | Free | Anticancer | VSP26B of C. striatus | HEp-2 | Larynx Cancer | MTT assay | IC50 = 49.65 µM | 24-h | Larynx | None | ||
| 35246758 | 2022 | Nisin ZP | 34 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Lactococcus lactis | H-1299 | Lung Cancer | MTT assay | IC50 = 137.3 ± 9.1 μM | 48-h | Lung | None | ||
| 35246758 | 2022 | Nisin ZP | 34 | Cyclic | L | None | Cyclized | Cyclized | Antimicrobial | Lactococcus lactis | A-549 | Lung Cancer | MTT assay | IC50 = 132.4 ± 6.4 μM | 48-h | Lung | None | ||
| 36555235 | 2022 | AC-P19M | 19 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Synthetic analogue of AC-P19 | H-460 | Lung Cancer | WST-8 assay | IC50 = 6.29 µM | 24-h | Lung | None | ||
| 36555235 | 2022 | AC-P19M | 19 | Linear | L | None | Free | Free | Anticancer and Antimicrobial | Synthetic analogue of AC-P19 | A-549 | Lung Cancer | WST-8 assay | IC50 = 9.84 µM | 24-h | Lung | None | ||
| 36183673 | 2022 | GV1001 | 16 | Linear | L | None | Free | Free | Anticancer | Human telomerase reverse transcriptase (hTERT) | A-549 | Lung Cancer | Cell Viability assay | Graph Fig 2A | 24-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | HCC-827 | Lung Adenocarcinoma | MTT assay | IC50 between 4.0 and 5.5 μM | 72-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | H-1975 | Non Small Cell Lung Cancer (NSCLC) | MTT assay | IC50 between 4.0 and 5.5 μM | 72-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | H-358 | Non Small Cell Lung Cancer (NSCLC) | MTT assay | IC50 = 4.00 ± 0.20 μM | 72-h | Lung | None | ||
| 35764196 | 2022 | D-LAK-120-A | 25 | Linear | D | None | Amidation | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 5.55 ± 0.13 μM | 72-h | Lung | None | ||
| 36287985 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | HepG-2 | Liver Cancer | MTT assay | IC50 = 5.524 µM | 24-h | Liver | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | H-460 | Lung Cancer | MTT assay | IC50 = 7.07 ± 0.81 µM | 24-h | Lung | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | PC-9 | Lung Cancer | MTT assay | IC50 = 6.34 ± 0.53 µM | 24-h | Lung | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | H-3122 | Lung Cancer | MTT assay | IC50 = 4.64 ± 0.18 µM | 24-h | Lung | None | ||
| 35878176 | 2022 | SMP24 | 24 | Linear | L | None | Free | Free | Antimicrobial | Egyptian scorpion Scorpio maurus palmatus | A-549 | Lung Cancer | MTT assay | IC50 = 4.06 ± 0.60 µM | 24-h | Lung | None | ||
| 36713538 | 2022 | NTP-217 | 9 | Linear | L | Dip = β-diphenylalanine | Amidation | rhodamine B - GABA | Anticancer | Synthetic | Huh-7 | Liver Cancer | MTT assay | IC50 = 40.1 ± 1.3 µM | 4-h | Liver | None | ||
| 36713538 | 2022 | NTP-217 | 9 | Linear | L | Dip = β-diphenylalanine | Amidation | rhodamine B - GABA | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 48.8 ± 0.7 µM | 4-h | Liver | None | ||
| 36713538 | 2022 | NTP-217 | 9 | Linear | L | Dip = β-diphenylalanine | Amidation | rhodamine B - GABA | Anticancer | Synthetic | Hep3B | Liver Cancer | MTT assay | IC50 = 45.7 ± 1.7 µM | 4-h | Liver | None | ||
| 36713538 | 2022 | NTP-217 | 9 | Linear | L | Dip = β-diphenylalanine | Amidation | rhodamine B - GABA | Anticancer | Synthetic | Hepa 1-6 | Liver Cancer | MTT assay | IC50 = 21.6 ± 1.0 µM | 4-h | Liver | None | ||
| 36713538 | 2022 | NTP-217 | 9 | Linear | L | Dip = β-diphenylalanine | Amidation | rhodamine B - GABA | Anticancer | Synthetic | PLC/PRF/5 | Liver Cancer | MTT assay | IC50 = 14.6 ± 1.1 µM | 4-h | Liver | None | ||
| 36713538 | 2022 | NTP-217 | 9 | Linear | L | Dip = β-diphenylalanine | Amidation | rhodamine B - GABA | Anticancer | Synthetic | HCCLM-3 | Liver Cancer | MTT assay | IC50 = 22.4 ± 5.1 µM | 4-h | Liver | None | ||
| 36121385 | 2022 | ST101 | 38 | Linear | D | None | Free | Free | Anticancer | Synthetic | T98G | Brain Tumor | Annexin V/ PI staining assay | mean EC50 value of 2.1 ± 0.4 μmol/L | 48-h | Brain | None | ||
| 36121385 | 2022 | ST101 | 38 | Linear | D | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | Annexin V/ PI staining assay | mean EC50 value of 2.1 ± 0.4 μmol/L | 48-h | Lung | None | ||
| 36121385 | 2022 | ST101 | 38 | Linear | D | None | Free | Free | Anticancer | Synthetic | DU-145 | Prostate Cancer | Annexin V/ PI staining assay | mean EC50 value of 2.1 ± 0.4 μmol/L | 48-h | Prostate | None | ||
| 36121385 | 2022 | ST101 | 38 | Linear | D | None | Free | Free | Anticancer | Synthetic | A-375 | Skin Cancer | Annexin V/ PI staining assay | mean EC50 value of 2.1 ± 0.4 μmol/L | 48-h | Skin | None | ||
| 36121385 | 2022 | ST101 | 38 | Linear | D | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | Annexin V/ PI staining assay | mean EC50 value of 2.1 ± 0.4 μmol/L | 48-h | Breast | None | ||
| 36121385 | 2022 | ST101 | 38 | Linear | D | None | Free | Free | Anticancer | Synthetic | U-251 | Brain Tumor | Annexin V/ PI staining assay | mean EC50 value of 2.1 ± 0.4 μmol/L | 48-h | Brain | None | ||
| 35601827 | 2022 | LyeTx-I-b | 24 | Linear | L | None | Amidated | Acetylation | Antimicrobial | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 2.47 µM | 48-h | Breast | None | ||
| 35013881 | 2022 | Brevinin-2R | 25 | Linear | L | None | Free | Free | Antimicrobial | Rana ridibunda | HeLa | Cervical Cancer | MTT assay | IC50 = 131.5 μg/ml | 24-h | Cervix | None | ||
| 36186562 | 2022 | C16-E4Y | 5 | Linear | L | None | Free | Palmitoyl | Anticancer | Synthetic | MCF-7 | Breast Cancer | WST-8 assay | 50 % cell viability at 0.05 wt % | 24-h | Breast | None | ||
| 36465844 | 2022 | HAZ | 21 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 5.44 μM | 4-h | Lung | None | ||
| 36186562 | 2022 | C16-E4Y | 5 | Linear | L | None | Free | Palmitoyl | Anticancer | Synthetic | A-431 | Skin Cancer | WST-8 assay | 10 % cell viability at 0.05 wt % | 24-h | Skin | None | ||
| 36186562 | 2022 | C16-E4Y | 5 | Linear | L | None | Free | Palmitoyl | Anticancer | Synthetic | HeLa | Cervical Cancer | WST-8 assay | 60% cell viability at 0.05 wt % | 24-h | Cervix | None | ||
| 36186562 | 2022 | C16-E4Y | 5 | Linear | L | None | Free | Palmitoyl | Anticancer | Synthetic | HepG-2 | Liver Cancer | WST-8 assay | 50 % cell viability at 0.05 wt % | 24-h | Liver | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | AlamarBlue assay | 75% cell viability at 20 μM | Not Available | Breast | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | AlamarBlue assay | IC50 = 9 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-480 | Colon Cancer | AlamarBlue assay | IC50 = 8 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut3 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-620 | Colon Cancer | AlamarBlue assay | IC50 = 9 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | AlamarBlue assay | 80% cell viability at 20 μM | Not Available | Breast | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-620 | Colon Cancer | AlamarBlue assay | IC50 = 40 ± 3 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | AlamarBlue assay | IC50 = 50 ± 3 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43-mut2 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-480 | Colon Cancer | AlamarBlue assay | IC50 = 34 ± 2 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | AlamarBlue assay | 50% cell viability at 20 μM | Not Available | Breast | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-620 | Colon Cancer | AlamarBlue assay | IC50 = 10 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HT-29 | Colon Cancer | AlamarBlue assay | IC50 = 11 ± 1 μM | 24-h | Colon | None | ||
| 35631675 | 2022 | HB43 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | SW-480 | Colon Cancer | AlamarBlue assay | IC50 = 12 ± 4 μM | 24-h | Colon | None | ||
| 36360120 | 2022 | HTDT-6-2-3-2 | 7 | Linear | L | None | Free | Free | Anticancer | Enteromorpha prolifera | HepG-2 | Liver Cancer | CCK-8 assay | IC50 = 1.2564 ± 0.0548 mg/mL | 48-h | Liver | None | ||
| 36360120 | 2022 | HTDT-6-2-3-2 | 7 | Linear | L | None | Free | Free | Anticancer | Enteromorpha prolifera | A-549 | Lung Cancer | CCK-8 assay | IC50 = 0.9867 ± 0.0857 mg/mL | 48-h | Lung | None | ||
| 36360120 | 2022 | HTDT-6-2-3-2 | 7 | Linear | L | None | Free | Free | Anticancer | Enteromorpha prolifera | NCI-H-460 | Lung Cancer | CCK-8 assay | IC50 = 0.3686 ± 0.0935 mg/mL | 48-h | Lung | None | ||
| 35774163 | 2022 | D-NAF-1 | 24 | Linear | D | None | Free | Free | Anticancer | NAF-1/CISD2 | MDA-MB-231 | Breast Cancer | Not Available | IC50 = 12.8 ± 0.2 μM | NA | Breast | None | ||
| 35774163 | 2022 | NAF-1 | 24 | Linear | L | None | Free | Free | Anticancer | NAF-1/CISD2 | MDA-MB-231 | Breast Cancer | Not Available | IC50 = 18.3 ± 0.4 μM | NA | Breast | None | ||
| 35094208 | 2022 | CIGB-552 | 20 | Linear | Mix | None | Free | Acetylation | Antitumor | Synthetic | A-549 | Lung Cancer | Sulforhodamine B assay | IC50 = 44.6 μM | 48-h | Lung | None | ||
| 35094208 | 2022 | CIGB-552 | 20 | Linear | Mix | None | Free | Acetylation | Antitumor | Synthetic | NCI-H-460 | Lung Cancer | Sulforhodamine B assay | IC50 = 287.9 μM | 48-h | Lung | None | ||
| 36672551 | 2022 | CIGB-300 | 25 | Cyclic | L | X = Beta- Alanine | Free | Biotinylated | Anticancer | Synthetic | NCI-H-460 | Lung Cancer | Crystal Violet assay | IC50 = 30 ± 5.3 µM | 48-h | Lung | None | ||
| 35745643 | 2022 | BmPLA2 | 24 | Linear | L | None | Free | Free | Anticancer | phospholipase A2 isoform from B. moojeni venom | RD | Rhabdomyosarcoma | MTT assay | 60% reduction in cell viability | 24-h | Muscle | None | ||
| 35745643 | 2022 | BmPLA2 | 24 | Linear | L | None | Free | Free | Anticancer | phospholipase A2 isoform from B. moojeni venom | CaCo-2 | Colorectal Cancer | MTT assay | IC50 = 0.6 µM | 24-h | Colon | None | ||
| 36174494 | 2022 | At12 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 14.0 µM | NA | Lung | None | ||
| 36174494 | 2022 | At12 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 13.4 µM | NA | Liver | None | ||
| 36174494 | 2022 | At11 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 7.6 µM | NA | Liver | None | ||
| 36174494 | 2022 | At11 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 7.9 µM | NA | Lung | None | ||
| 36174494 | 2022 | At10 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.2 µM | NA | Liver | None | ||
| 36174494 | 2022 | At10 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4.4 µM | NA | Lung | None | ||
| 36174494 | 2022 | At9 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 51.7 µM | NA | Liver | None | ||
| 36174494 | 2022 | At9 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 100 µM | NA | Lung | None | ||
| 36174494 | 2022 | At8 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 8.9 µM | NA | Liver | None | ||
| 36174494 | 2022 | At8 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 13.4 µM | NA | Lung | None | ||
| 36174494 | 2022 | At7 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 8.8 µM | NA | Liver | None | ||
| 36174494 | 2022 | At7 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 10.3 µM | NA | Lung | None | ||
| 36174494 | 2022 | At6 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 70.8 µM | NA | Liver | None | ||
| 36174494 | 2022 | At6 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 > 100 µM | NA | Lung | None | ||
| 36174494 | 2022 | At5 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 3.6 µM | NA | Lung | None | ||
| 36174494 | 2022 | At5 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.5 µM | NA | Liver | None | ||
| 36174494 | 2022 | At4 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.5 µM | NA | Liver | None | ||
| 36174494 | 2022 | At4 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 7.2 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; K13L; Q15K], At3 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4.3 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; K13L; Q15K], At3 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.2 µM | NA | Liver | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; Q15K], At2 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 >100 µM | NA | Liver | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25) [P4K; S5K; G8K; Q15K], At2 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 >100 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25), At1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 > 100 µM | NA | Lung | None | ||
| 36174494 | 2022 | Ponericin-W1 (11-25), At1 | 15 | Linear | L | None | Amidation | Acetylation | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 >100 µM | NA | Liver | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | MCF-7 | Breast Cancer | MTT assay | EC50 = 0.724 ± 0.340 mol/L × 10-3 | 24-h | Breast | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | A-2058 | Skin Cancer | MTT assay | EC50 = 0.744 ± 0.208 mol/L × 10-3 | 24-h | Skin | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | U-87 | Brain Tumor | MTT assay | EC50 = 0.427 ± 0.053 mol/L × 10-3 | 24-h | Brain | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | HeLa | Cervical Cancer | MTT assay | EC50 = 0.525 ± 0.160 mol/L × 10-3 | 24-h | Cervix | None | ||
| 35190586 | 2022 | RB4 | 24 | Linear | L | None | Amidation | Free | Anticancer | Derived from protein PLP2 | B16-F10-Nex 2 | Skin Cancer | MTT assay | EC50 = 0.263 ± 0.585 mol/L × 10-3 | 24-h | Skin | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | WiDr | Colon Cancer | MTT assay | IC50 = 197.3 μM | 24-h | Colon | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | AGS | Stomach Cancer | MTT assay | IC50 = 29.8 μM | 24-h | Stomach | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | A-549 | Lung Cancer | MTT assay | IC50 = 42.1 μM | 24-h | Lung | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | Hep3B | Liver Cancer | MTT assay | IC50 = 77.5 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | Huh-7 | Liver Cancer | MTT assay | IC50 = 60 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple-a | 25 | Linear | L | None | Amidation | Free | Antimicrobial | C-terminal-amidated derivative of Pleurocidin | J5 | Liver Cancer | MTT assay | IC50 = 11 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | AGS | Stomach Cancer | MTT assay | IC50 = 186.5 μM | 24-h | Stomach | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | A-549 | Lung Cancer | MTT assay | IC50 = 300.8 μM | 24-h | Lung | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | Hep3B | Liver Cancer | MTT assay | IC50 = 340.9 μM | 24-h | Liver | None | ||
| 36005521 | 2022 | Ple | 25 | Linear | L | None | Free | Free | Antimicrobial | Pleuronectes americanus | J5 | Liver Cancer | MTT assay | IC50 = 54.9 μM | 24-h | Liver | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 14.0 ± 1.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-474 | Breast Cancer | MTT assay | IC50 = 15.7 ± 1.5 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 4.2 ± 2.2 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP2319 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 4.5 ± 0.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 21.1 ± 2.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-474 | Breast Cancer | MTT assay | IC50 = 37.5 ± 1.7 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 3.5 ± 1.5 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0769 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 9.0 ± 0.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0667 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 71.2 ± 1.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0667 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-474 | Breast Cancer | MTT assay | IC50 = 92.8 ± 1.1 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0667 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 88.8 ± 1.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0275 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | SK-BR-3 | Breast Cancer | MTT assay | IC50 = 34.0 ± 1.0 μM | 24-h | Breast | None | ||
| 34679257 | 2022 | vCPP0275 | 20 | Linear | L | None | Amidation | Free | Anticancer and Cell Penetrating | Capsid protein of the Torque teno douroucouli virus | BT-20 | Breast Cancer | MTT assay | IC50 = 44.8 ± 1.1 μM | 24-h | Breast | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | SNB-19 | Brain Tumor | CCK-8 assay | IC50 = 12.0 ± 0.6 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | SF-268 | Brain Tumor | CCK-8 assay | IC50 = 4.8 ± 0.1 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-138 | Brain Tumor | CCK-8 assay | IC50 = 7.5 ± 0.3 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | LN229 | Brain Tumor | CCK-8 assay | IC50 = 4.7 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | SW-1783 | Brain Tumor | CCK-8 assay | IC50 = 4.8 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | D54 | Brain Tumor | CCK-8 assay | IC50 = 8.4 ± 0.1 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-118 | Brain Tumor | CCK-8 assay | IC50 = 6.8 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-373 | Brain Tumor | CCK-8 assay | IC50 = 5.0 ± 0.2 μM | 72-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | T98G | Brain Tumor | CCK-8 assay | IC50 = 7.1 ± 0.2 μM | 96-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | A-172 | Brain Tumor | CCK-8 assay | IC50 = 6.4 ± 0.4 μM | 96-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U-251 | Brain Tumor | CCK-8 assay | IC50 = 4.9 ± 0.3 μM | 96-h | Brain | None | ||
| 35053455 | 2022 | ATX-101 | 25 | Linear | L | None | Free | Acetylation | Antitumor and Cell Penetrating | Synthetic | U87-MG | Brain Tumor | CCK-8 assay | IC50 = 4.3 ± 0.3 μM | 96-h | Brain | None | ||
| 35660629 | 2022 | NRC-03 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | skin mucous secretions of winter flounder | SCC-9 | Oral Cancer | CCK-8 assay | IC50 = 45 μg/ml | 24-h | Tongue | None | ||
| 34509120 | 2022 | GI-15 | 17 | Linear | L | None | Amidation | LC-Propargylglycine | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 16.6 ± 0.8 µM | 72-h | Cervix | None | ||
| 35660629 | 2022 | NRC-03 | 26 | Linear | L | None | Amidation | Free | Antimicrobial | skin mucous secretions of winter flounder | CAL-27 | Oral Cancer | CCK-8 assay | IC50 = 45 μg/ml | 24-h | Tongue | None | ||
| 34509120 | 2022 | GI-15 | 17 | Linear | L | None | Amidation | LC-Propargylglycine | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 13.6 ± 0.2 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | CI-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 7.7 ± 0.2 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | CI-15 | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 2.7 ± 0.5 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 26.7 ± 1.3 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 15.6 ± 1.0 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | IR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 > 100 µM | 72-h | Colon | None | ||
| 34509120 | 2022 | IR13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 > 100 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 83 ± 9 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | IK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 47±5 µM | 72-h | Cervix | None | ||
| 34509120 | 2022 | LK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 23 ± 2 µM | 72-h | Colon | None | ||
| 35323457 | 2022 | Z-8 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 15.88 ± 1.42 µg/ml | NA | Lung | None | ||
| 34509120 | 2022 | IK13 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 29 ± 6 µM | 72-h | Colon | None | ||
| 35323457 | 2022 | Z-8 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 20.16 ± 2.24 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-8 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 7.97 ± 0.61 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-7 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 9.97 ± 1.00 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-8 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.82 ± 1.18 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-8 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 9.00 ± 0.83 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-7 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 16.52 ± 1.7 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-7 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 18.21 ± 1.35 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-7 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 13.28 ± 3.28 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-7 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 13.85 ± 1.99 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-6 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 4.59 ± 0.27 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-6 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 5.69 ± 0.37 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-6 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 5.96 ± 0.41 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-6 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 1.65 ± 0.3 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-6 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.91 ± 0.17 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-5 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 12.12 ± 0.95 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-5 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 9.5 ± 1.13 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-4 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 13.43 ± 1.96 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-5 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 14.98 ± 0.93 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-5 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 8.48 ± 1.12 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-4 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 7.38 ± 0.83 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-4 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 9.85 ± 0.95 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-3 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 4.88 ± 0.58 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-4 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 15.23 ± 1.14 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-4 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 22.09 ± 1.12 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-3 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 5.57 ± 0.45 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-3 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 6.43 ± 0.43 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-3 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 5.05 ± 0.45 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-3 | 5 | Cyclic | Mix | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 6.34 ± 0.6 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-2 | 5 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 14.5 ± 0.36 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-2 | 5 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 7.97 ± 2.06 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-2 | 5 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 2.25 ± 0.42 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-2 | 5 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 11.95 ± 0.64 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Z-2 | 5 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 14.45 ± 1.1 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-1 | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4.92 ± 0.84 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Z-2 | 5 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 4.68 ± 1.22 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-1 | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 17.81 ± 0.6 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-1 | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 11.56 ± 0.65 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Z-1 | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.85 ± 1.28 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Z-1 | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Synthetic | HepG-2 | Liver Cancer | MTT assay | IC50 = 7.57 ± 0.17 µg/ml | NA | Liver | None | ||
| 35323457 | 2022 | Galaxamide | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Galaxaura filamentosa | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 8.73 ± 0.29 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Galaxamide | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Galaxaura filamentosa | A-549 | Lung Cancer | MTT assay | IC50 = 6.99 ± 0.63 µg/ml | NA | Lung | None | ||
| 35323457 | 2022 | Galaxamide | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Galaxaura filamentosa | MCF-7 | Breast Cancer | MTT assay | IC50 = 11.33 ± 2.95 µg/ml | NA | Breast | None | ||
| 35323457 | 2022 | Galaxamide | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Galaxaura filamentosa | HeLa | Cervical Cancer | MTT assay | IC50 = 8.53 ± 0.73 µg/ml | NA | Cervix | None | ||
| 35323457 | 2022 | Galaxamide | 5 | Cyclic | L | N-Me-L = N-methyl-Lysine | Cyclized | Cyclized | Anticancer | Galaxaura filamentosa | HepG-2 | Liver Cancer | MTT assay | IC50 = 5.20 ± 0.52 µg/ml | NA | Liver | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 72.06 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 71.18 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 193.4 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 167 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-3i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 120.6 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 2.94 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 5.28 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 3.07 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.35 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-i | 17 | Linear | Mix | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 4.46 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 27.76 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 99.36 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 49.50 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 35.28 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-4K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 85.52 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 3.29 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 0.38 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 3.01 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 0.51 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-3K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 2.83 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 22.09 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 24.03 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 22.67 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 27.32 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-K12 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 25.75 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-157 | Lung Cancer | MTT assay | IC50 = 2.78 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 2.84 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | H-838 | Lung Cancer | MTT assay | IC50 = 3.07 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | PC-3 | Prostate Cancer | MTT assay | IC50 = 2.64 μM | 24-h | Prostate | None | ||
| 35740884 | 2022 | Temporin-PKE-2K | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | U251-MG | Brain Tumor | MTT assay | IC50 = 2.49 μM | 24-h | Brain | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | H-157 | Lung Cancer | MTT assay | IC50 = 17.40 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | HCT-116 | Colorectal Cancer | MTT assay | IC50 = 21.31 μM | 24-h | Colon | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | H-838 | Lung Cancer | MTT assay | IC50 = 16.38 μM | 24-h | Lung | None | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | PC-3 | Prostate Cancer | MTT assay | IC50 = 7.29 μM | 24-h | Prostate | None | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 57.03 ± 6.09 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740884 | 2022 | Temporin-PKE | 17 | Linear | L | None | Amidation | Free | Antimicrobial | skin secretion of Pelophylax kl. esculentus | U251-MG | Brain Tumor | MTT assay | IC50 = 23.24 μM | 24-h | Brain | None | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 57.99 ± 5.04 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 33.92 ± 5.90 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 57.45 ± 6.03 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 35.71 ± 8.50 µM | 48-h | Breast | US_10550155_B2 | ||
| 35740895 | 2022 | Jeff-[G10a]2-SHa | 26 | Linear | Mix | Jeffamine linker | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 70.71 ± 5.39 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 1.84 ± 0.17 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 2.24 ± 0.05 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 2.31 ± 0.08 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 6.94 ± 0.27 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 3.74 ± 3.46 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 3.77 ± 0.12 µM | 48-h | Breast | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]3-SHa | 41 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | HepG-2 | Liver Cancer | Resazurin dye assay | IC50 = 5.49 ± 0.37 µM | 48-h | Liver | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 4.72 ± 0.36 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 6.31 ± 0.66 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 8.71 ± 0.35 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 4.42 ± 0.06 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 3.79 ± 1.61 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | HepG-2 | Liver Cancer | Resazurin dye assay | IC50 = 14.31 ± 1.37 µM | 48-h | Liver | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]2-SHa | 27 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 5.69 ± 1.46 µM | 48-h | Breast | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MNT-1 | Skin Cancer | Resazurin dye assay | IC50 = 15.25 ± 0.80 µM | 48-h | Skin | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | PC-3 | Prostate Cancer | Resazurin dye assay | IC50 = 13.04 ± 1.99 µM | 48-h | Prostate | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MiaPaCa.2 | Pancreatic Cancer | Resazurin dye assay | IC50 = 22.36 ± 6.07 µM | 48-h | Pancreas | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-2780 | Ovarian Cancer | Resazurin dye assay | IC50 = 14.75 ± 7.35 µM | 48-h | Ovary | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | A-549 | Lung Cancer | Resazurin dye assay | IC50 = 14.52 ± 1.44 µM | 48-h | Lung | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | HepG-2 | Liver Cancer | Resazurin dye assay | IC50 = 31.63 ± 1.56 µM | 48-h | Liver | US_10550155_B2 | ||
| 35740895 | 2022 | [G10a]-SHa | 13 | Linear | Mix | None | Amidation | Free | Antimicrobial and Anticancer | Analog of temporin SHa | MCF-7 | Breast Cancer | Resazurin dye assay | IC50 = 15.05 ± 8.51 µM | 48-h | Breast | US_10550155_B2 | ||
| 35631515 | 2022 | K4F6K4 | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | AnnexinV-FITC/PI double staining assay | apoptotic cells (early and late) increased from 9.59 ± 1.00% to 43.03 ± 2.13% | 12-h | Lung | None | ||
| 35631515 | 2022 | K4F8K4 | 16 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 571.87 ± 66.23 μg/mL | 48-h | Lung | None | ||
| 35631515 | 2022 | K4F6K4 | 14 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 62.64 ± 9.55 μg/mL | 48-h | Lung | None | ||
| 35631515 | 2022 | K2F6K2 | 10 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 1146.23 ± 346.83 μg/mL | 48-h | Lung | None | ||
| 35631515 | 2022 | K3F6K3 | 12 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 123.10 ± 35.19 μg/mL | 48-h | Lung | None | ||
| 36364156 | 2022 | PS14 | 14 | Linear | L | None | Free | Free | Anticancer and Anti-inflammatory | Aphanomyces invadans | Hep-2 | Larynx Cancer | LDH leakage assay | 45.56 ± 2% LDH release at 20 µM | 24-h | Larynx | None | ||
| 36364155 | 2022 | PS14 | 14 | Linear | L | None | Free | Free | Anticancer and Anti-inflammatory | Aphanomyces invadans | Hep-2 | Larynx Cancer | MTT assay | IC50 = 21 µM | 24-h | Larynx | None | ||
| 35246961 | 2022 | d-EEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 4.78 ± 0.02 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | d-EEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.29 ± 0.01 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-EEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 0.29 ± 0.01 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 5.84 ± 0.04 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | d-DEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.36 ± 0 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DEK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 0.44 ± 0.10 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DHK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 1.24 ± 0.03 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | d-DHK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 0.32 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | d-DHK | 15 | Linear | Mix | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.23 ± 0.04 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 9.65 ± 1.20 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.35 ± 0.40 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.23 ± 0.11 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.57 ± 0.24 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.60 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.20 ± 1.84 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.40 ± 0.71 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.19 ± 0.40 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.72 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.20 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 10.40 ± 1.70 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DKK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.95 ± 0.35 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.88 ± 1.24 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.59 ± 0.92 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.40 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.65 ± 1.91 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.15 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.75 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 25.00 ± 0 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.35 ± 0.35 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.71 ± 0.13 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 20.45 ± 2.05 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.75 ±0.49 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.02 ± 0.12 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 8.15 ± 0.49 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.60 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.35 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 143.20 ± 80.33 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.45 ± 2.19 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.35 ± 1.06 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 32.88 ± 4.07 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.08 ± 0.18 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.10 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 19.88 ± 2.65 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 0.70 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEK | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.14 ± 0.52 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 13.30 ± 0.99 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.20 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.40 ± 0.85 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 18.88 ± 1.24 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.10 ± 0.57 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.45 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 23.83 ± 0.81 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.18 ± 0.31 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.75 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 21.13 ± 3.01 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.80 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.45 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 39.75 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 4.45 ± 0.49 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 5.20 ± 0.71 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 185 ± 7 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 9.50 ± 0.99 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 117 ± 7 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 21.10 ± 6.93 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 16.05 ± 3.18 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 25.35 ± 2.76 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 11.90 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 55.85 ± 18.88 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DHH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 21.45 ± 2.47 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 49.25 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.35 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.30 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 106 ± 14 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 10.95 ± 1.06 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 19.60 ± 3.96 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 28.60 ± 10.75 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.30 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.60 ± 0.85 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 36.48 ± 3.92 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 3.60 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEH | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 5.35 ± 1.91 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 12.75 ± 1.20 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.70 ± 0 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.05 ± 0.64 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 15.95 ± 0.78 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.90 ± 0.42 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.70 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 8.00 ± 0.71 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.30 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 1.80 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 9.93 ± 0.25 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 1.57 ± 0.33 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DKE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 2.10 ± 0 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 53 ± 2.83 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.92 ± 0.17 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.70 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 53.25 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 10.75 ± 0.78 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 16.70 ± 2.26 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 18.25 ± 1.06 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.55 ± 0.07 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.90 ± 0.28 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 17.25 ± 1.06 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.80 ± 0.14 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DHE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.75 ± 0.92 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 49.38 ± 13.26 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | KEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 2.05 ± 0.21 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | KEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 3.75 ± 0.78 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 47.50 ± 11 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | HEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 4.95 ± 0.49 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | HEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 6.50 ± 0.71 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 78.75 ± 5.30 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | EEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 10.55 ± 3.46 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | EEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 6.25 ± 1.77 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | U-2 OS | Bone Cancer | MTT assay | IC50 = 61.00 ± 1.41 µM | 72-h | Bone | None | ||
| 35246961 | 2022 | DEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER-shEcad | Breast Cancer | MTT assay | IC50 = 6.05 ± 2.76 µM | 72-h | Breast | None | ||
| 35246961 | 2022 | DEE | 15 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HMLER | Breast Cancer | MTT assay | IC50 = 5.55 ± 0.35 µM | 72-h | Breast | None | ||
| 36355026 | 2022 | LJP-12 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.72 ± 0.05 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-12 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 0.41 ± 0.04 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-12 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 0.60 ± 0.08 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-11 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.70 ± 0.07 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-11 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 0.61 ± 0.07 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-10 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 3.53 ± 0.34 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-11 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 0.49 ± 0.05 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-10 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.69 ± 0.22 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-9 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.51 ± 0.07 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-10 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 3.52 ± 0.35 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-9 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 0.69 ± 0.08 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-8 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.76 ± 0.08 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-9 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 0.53 ± 0.05 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-8 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 0.63 ± 0.05 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-8 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 0.44 ± 0.04 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-7 | 7 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.66 ± 0.11 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-7 | 7 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 1.44 ± 0.12 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-7 | 7 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 2.53 ± 0.24 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-5 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 1.49 ± 0.13 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-6 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.06 ± 0.31 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-5 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 2.78 ± 0.26 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-4 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.68 ± 0.07 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-5 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 2.44 ± 0.22 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-4 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 0.65 ± 0.07 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-3 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 1.70 ± 0.15 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-4 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 0.62 ± 0.07 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-3 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 1.42 ± 0.12 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-2 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 1.71 ± 0.13 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-2 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.62 ± 0.05 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-2 | 6 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 2.25 ± 0.22 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-1 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | HepG-2 | Liver Cancer | MTT assay | IC50 = 0.45 ± 0.05 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-1 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | H-22 | Liver Cancer | MTT assay | IC50 = 0.36 ± 0.03 mM | 48-h | Liver | None | ||
| 36355026 | 2022 | LJP-1 | 5 | Linear | L | None | Free | Free | Anticancer | Laminaria japonica | Huh-7 | Liver Cancer | MTT assay | IC50 = 0.48 ± 0.05 mM | 48-h | Liver | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | B16-F10 | Skin Cancer | MTS assay | IC50 = 6.65 ± 0.33 μM | 48-h | Skin | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | SMMC-7721 | Liver Cancer | MTS assay | IC50 = 6.87 ± 0.51 μM | 48-h | Liver | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | A-549 | Lung Cancer | MTS assay | IC50 = 5.81 ± 0.23 μM | 48-h | Lung | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | SW-480 | Blood Cancer | MTS assay | IC50 = 10.37 ± 0.40 μM | 48-h | Blood | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | MDA-MB-231 | Breast Cancer | MTS assay | IC50 = 5.44 ± 0.33 μM | 48-h | Breast | None | ||
| 34361728 | 2021 | GA - 8 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 60.70 ± 0.6 µg/mL | 24-h | Colon | None | ||
| 33916789 | 2021 | Brevinin-1RL1 | 24 | Cyclic(C18-C24) | L | None | Free | Free | Antimicrobial | Rana limnocharis | HCT-116 | Colon Cancer | MTS assay | IC50 = 5.87 ± 0.15 μM | 48-h | Colon | None | ||
| 34361728 | 2021 | GA - 7 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HepG-2 | Liver Cancer | MTT assay | IC50 = 3.30 ± 0.1 µg/mL | 24-h | Liver | None | ||
| 34361728 | 2021 | GA - 8 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 6.90 ± 1.1 µg/mL | 24-h | Breast | None | ||
| 34361728 | 2021 | GA - 7 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.70 ± 0.2 µg/mL | 24-h | Breast | None | ||
| 34361728 | 2021 | GA - 7 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.0 ± 1.1 µg/mL | 24-h | Colon | None | ||
| 34361728 | 2021 | GA - 5 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.0 ± 0.3 µg/mL | 24-h | Breast | None | ||
| 34361728 | 2021 | GA - 5 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 5.2 ± 0.8 µg/mL | 24-h | Colon | None | ||
| 34361728 | 2021 | GA - 4 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 73.0 ± 1.4 µg/mL | 24-h | Colon | None | ||
| 34361728 | 2021 | GA - 3 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 7.40 ± 0.4 µg/mL | 24-h | Colon | None | ||
| 34361728 | 2021 | GA - 4 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 6.10 ± 0.4 µg/mL | 24-h | Breast | None | ||
| 34361728 | 2021 | GA - 2 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | HCT-116 | Colon Cancer | MTT assay | IC50 = 70.30 ± 0.9 µg/mL | 24-h | Colon | None | ||
| 34361728 | 2021 | GA - 3 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.1 ± 0.7 µg/mL | 24-h | Breast | None | ||
| 34361728 | 2021 | GA - 2 | Not Available | Linear | L | None | Free | 18beta-glycyrrhetinic-acid | Antimicrobial and Anticancer | Synthetic (glycyrrhetinic acid (GA)-based peptides) | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.70 ± 1.3 µg/mL | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 1.97 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 18.1 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 2.99 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 21.6 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 5.25 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 17.5 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 5.52 µM | 24-h | Not Available | None | ||
| 34135370 | 2021 | Piscidin 3 | 22 | Linear | L | None | Free | Free | Anticancer | Morone chrysops x Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 26.01 µM | 24-h | Not Available | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 2.17 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | HeLa | Cervical Cancer | MTT assay | IC50 = 2.22 µM | 24-h | Cervix | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 2.15 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | A-549 | Lung Cancer | MTT assay | IC50 = 4.2 µM | 24-h | Lung | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 3.92 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 5.83 µM | 24-h | Breast | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | Cu2+ bound | Free | Free | Anticancer | Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 5.31 µM | 24-h | Not Available | None | ||
| 34135370 | 2021 | Piscidin 1, Moronecidin | 22 | Linear | L | None | Free | Free | Anticancer | Morone saxatilis | HT-1080 | Fibrosarcoma | MTT assay | IC50 = 5.58 µM | 24-h | Not Available | None | ||
| 33603033 | 2021 | L. squarrosulus purifed fraction | 19 | Linear | L | None | Free | Free | Anticancer | Lentinus squarrosulus (Mont.) | H-460 | Lung Cancer | MTT assay | Graph Figure 2 | 24-h | Lung | None | ||
| 34789753 | 2021 | Palustrin - Ca | 31 | Linear | L | None | Free | Free | Host Defence Peptide | Lithobates catesbeianus | SGC-7901 | Gastric Cancer | Not Available | IC50 = 0.951 μg/ml | Not Available | Stomach | None | ||
| 33677023 | 2021 | Pep | 21 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 2 µM | 24-h | Breast | None | ||
| 33677023 | 2021 | Pep | 21 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 4 µM | 24-h | Lung | None | ||
| 34531430 | 2021 | PCC-1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Poecilocoris lewisi | G361 | Skin Cancer | MTS assay | IC50 = 57.8 µM | 48-h | Skin | None | ||
| 34531430 | 2021 | PCC-1 | 17 | Linear | L | None | Amidation | Free | Antimicrobial | Poecilocoris lewisi | SK-Mel-28 | Skin Cancer | MTS assay | IC50 = 50.8 µM | 48-h | Skin | None | ||
| 33981363 | 2021 | 17BIPHE2 | 17 | Linear | L | None | Free | Free | Antimicrobial | Derivative of LL-37 | NCI-H-1975 | Lung Cancer | MTT assay | IC50 = 71.42 µmol/L | 24-h | Lung | None | ||
| 33690977 | 2021 | NMTP-5 | 24 | Linear | D | Z = C10H7CH2C(O), M, 4-(Trifluoromethyl)-D-phenylalanine | Free | Free | Anticancer | Not Available | SK-HEP-1 | Liver Cancer | MTT assay | IC50 = 53.84 ± 4.35 µM | 48-h | Liver | None | ||
| 33567789 | 2021 | Si15 | 7 | Linear | L | nL = nor-Leu | Amidation | Caffeic acid (Caf) | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 140.3 ± 7.12 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si15 | 7 | Linear | L | nL = nor-Leu | Amidation | Caffeic acid (Caf) | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 346.3 ± 7.91 µM | 72-h | Breast | None | ||
| 33981363 | 2021 | 17BIPHE2 | 17 | Linear | L | None | Free | Free | Antimicrobial | Derivative of LL-37 | A-549 | Lung Cancer | MTT assay | IC50 = 34.33 µmol | 24-h | Lung | None | ||
| 33567789 | 2021 | Si14 | 7 | Linear | L | nL = nor-Leu | Amidation | 1,8-naphthalimide-Gly | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 593.3 ± 60.3 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si14 | 7 | Linear | L | nL = nor-Leu | Amidation | 1,8-naphthalimide-Gly | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 1049 ± 49.77 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si11 | 7 | Linear | L | β-Ala | Amidation | Caffeic acid (Caf) | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 1087 ± 70.71 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si13 | 7 | Linear | L | nL = nor-Leu | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 1704 ± 112 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si2 | 7 | Linear | L | β-Ala | Amidation | 1,8-naphthalimide-Gly | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 840 ± 21.18 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si11 | 7 | Linear | L | β-Ala | Amidation | Caffeic acid (Caf) | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 228.8 ± 7.18 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si2 | 7 | Linear | L | β-Ala | Amidation | 1,8-naphthalimide-Gly | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 662.9 ± 20.02 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si8 | 7 | Linear | L | None | Amidation | Caffeic acid (Caf) | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 514.3 ± 26.82 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si3 | 8 | Linear | L | β-Ala | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 176.3 ± 4.66 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si7 | 7 | Linear | L | None | Amidation | 1,8-naphthalimide-Gly | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 1195 ± 131.5 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si8 | 7 | Linear | L | None | Amidation | Caffeic acid (Caf) | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 128.6 ± 8.03 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si1 | 14 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 746.5 ± 7.6 µM | 72-h | Breast | None | ||
| 33567789 | 2021 | Si1 | 14 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 124.1 ± 8.12 µM | 72-h | Breast | None | ||
| 33428507 | 2021 | L8H6 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 16.4 µM | 24-h | Cervix | None | ||
| 33428507 | 2021 | L9H5-1 | 14 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HeLa | Cervical Cancer | MTT assay | IC50 = 5.4 µM | 24-h | Cervix | None | ||
| None | 2021 | SKACP003 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-453 | Breast Cancer | MTT assay | IC50 = 156 ± 0.5 µM | 24-h | Breast | None | ||
| None | 2021 | SKACP003 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 212 ± 0.5 µM | 24-h | Breast | None | ||
| None | 2021 | SKACP003 | 12 | Linear | L | None | Free | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 193 ± 0.5 µM | 24-h | Breast | None | ||
| 32381104 | 2021 | Sur-X | 35 | Linear | L | None | Free | TAT Peptide | Anticancer | Synthetic | HT-29 | Colon Cancer | MTT assay | Not Available | Not Available | Colon | None | ||
| 32381104 | 2021 | Sur-X | 35 | Linear | L | None | Free | TAT Peptide | Anticancer | Synthetic | RKO | Colon Cancer | MTT assay | 25% cell viability at at 20 μM | 24-h | Colon | None | ||
| 32381104 | 2021 | Sur-X | 35 | Linear | L | None | Free | TAT Peptide | Anticancer | Synthetic | HCT-15 | Colon Cancer | MTT assay | Not Available | Not Available | Colon | None | ||
| 32381104 | 2021 | Sur-X | 35 | Linear | L | None | Free | TAT Peptide | Anticancer | Synthetic | HCT-116 | Colon Cancer | MTT assay | 20% cell viability at at 20 μM | 24-h | Colon | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | Sup-B15 | Blood Cancer | Trypan blue assay | IC50 = 90 ± 14 µM | 24-h | Blood | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | RS4;11 | Blood Cancer | Trypan blue assay | IC50 = 184 ± 23 µM | 24-h | Blood | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | Raji | Lymphoma Cancer | Trypan blue assay | IC50 = 89 ± 24 µM | 24-h | Blood | None | ||
| 34440185 | 2021 | HMP-S7 | 17 | Linear | L | None | Free | Free | Anticancer | Human Milk | Jurkat | Blood Cancer | Trypan blue assay | IC50 = 186 ± 37 µM | 24-h | Blood | None | ||
| 33442881 | 2021 | [Arg]11-VmCT1 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 25.8 ± 5.2 μmol/L | 24-h | Breast | None | ||
| 33442881 | 2021 | [Arg]7-VmCT1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 18.0 ± 2.7 μmol/L | 24-h | Breast | None | ||
| 33442881 | 2021 | [Arg]3-VmCT1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 20.6 ± 3.1 μmol/L | 24-h | Breast | None | ||
| 33442881 | 2021 | VmCT1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Vaejovis mexicanus smithi | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.3 ± 1.4 μmol/L | 24-h | Breast | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | HepG-2 | Liver Cancer | CCK-8 assay | IC50 = 7.0 ± 1.0 µM | 24-h | Liver | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | HeLa | Cervical Cancer | CCK-8 assay | IC50 = 4.7 ± 1.4 µM | 24-h | Cervix | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | IC50 = 6.2 ± 1.4 µM | 24-h | Lung | None | ||
| 34941705 | 2021 | LVTX-9-C18 | 19 | Linear | L | None | Amidation | CH3-(CH2)16-CO | Anticancer | Synthetic | 4T1 | Breast Cancer | CCK-8 assay | IC50 = 7.6 ± 1.3 µM | 24-h | Breast | None | ||
| 34941705 | 2021 | LVTX-9 | 19 | Linear | L | None | Amidation | Free | Anticancer | Lycosa vittata | A-549 | Lung Cancer | CCK-8 assay | IC50 = 51.7 ± 4.3 µM | 24-h | Lung | None | ||
| 33244888 | 2021 | Protonectin-F | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Protonoectin | HCT-116 | Colon Cancer | Resazurin dye assay | CC50 = 9.8 ± 1.2 µM | 24-h | Colon | None | ||
| 33244888 | 2021 | Protonectin-F | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Protonoectin | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 16.0 ± 1.2 µM | 24-h | Skin | None | ||
| 33244888 | 2021 | Protonectin | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Parachartergus fraternus | HCT-116 | Colon Cancer | Resazurin dye assay | CC50 = 8.0 ± 0.5 µM | 24-h | Colon | None | ||
| 33244888 | 2021 | Protonectin | 12 | Linear | L | None | Amidation | Free | Antimicrobial | Parachartergus fraternus | MM96L | Skin Cancer | Resazurin dye assay | CC50 = 14.8 ± 0.9 µM | 24-h | Skin | None | ||
| 34309373 | 2021 | Pal-pFL-N-Ter-TAT | 32 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W) | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | MCF-7 | Breast Cancer | MTT assay | IC50 = 11.85 μM | 24-h | Breast | None | ||
| 34309373 | 2021 | Pal-pFL-N-Ter-TAT | 32 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W) | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-549 | Lung Cancer | MTT assay | IC50 = 31.17 μM | 24-h | Lung | None | ||
| 34309373 | 2021 | Pal-pFL-N-Ter-TAT | 32 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W) | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-375 | Skin Cancer | MTT assay | IC50 = 5.5 ± 1.1 μM | 24-h | Skin | None | ||
| 34309373 | 2021 | pFL-N-Ter-TAT | 32 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | pFL = hydrophobic peptide fragment (FPWWWPFL) | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-375 | Skin Cancer | MTT assay | IC50 = 11.1 ± 0.1 μM | 24-h | Skin | None | ||
| 34309373 | 2021 | Pal-N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | MCF-7 | Breast Cancer | MTT assay | IC50 = 27.26 μM | 24-h | Breast | None | ||
| 34309373 | 2021 | Pal-N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-549 | Lung Cancer | MTT assay | IC50 = 44.98 μM | 24-h | Lung | None | ||
| 34309373 | 2021 | Pal-N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Palmitic acid | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-375 | Skin Cancer | MTT assay | IC50 = 36.67(Supplementary material)/15.2 ± 0.7 μM(Published paper) | 24-h | Skin | None | ||
| 34309373 | 2021 | N-Ter | 12 | Linear | L | None | Free | Free | Anticancer | Analogue of N-terminal fragment of the VDAC1 protein | A-375 | Skin Cancer | MTT assay | IC50(A-375)> 50.0 μM | 24-h | Skin | None | ||
| 34117917 | 2021 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | N-terminal region of Helicobacter pylori ribosomal protein L1 | HT-29 | Colon Cancer | MTT assay | IC50 ~ 0.5 µg/mL | 24-h | Colon | None | ||
| 34117917 | 2021 | HPRP-A1 | 15 | Linear | L | None | Amidation | Acetylation | Anticancer | N-terminal region of Helicobacter pylori ribosomal protein L1 | CT-26 | Colorectal Cancer | MTT assay | IC50 between 0.5 and 1 µg/mL | 24-h | Colon | None | ||
| 34848729 | 2021 | AtMP2 | 22 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 6.97 ± 0.24 μg/ml | 48-h | Breast | None | ||
| 34848729 | 2021 | AtMP2 | 22 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MCF-7 | Breast Cancer | MTT assay | IC50 = 5.89 ± 0.14 μg/ml | 48-h | Breast | None | ||
| 34848729 | 2021 | AtMP1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 9.35 ± 0.25 μg/ml | 48-h | Breast | None | ||
| 34848729 | 2021 | AtMP1 | 24 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Anabastestudineus skin mucus fraction 2 | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.25 ± 0.14 μg/ml | 48-h | Breast | None | ||
| 33517264 | 2021 | Hepcidin | 20 | Linear | L | None | Free | Free | Antimicrobial and Anticancer | Homo sapiens | U-266 | Lymphoma Cancer | MTT assay | NA | NA | Blood | None | ||
| 34796903 | 2021 | A4W-GGN5 | 11 | Linear | L | None | Amidation | Free | Anticancer | Gaegurin 5 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 22.07 ± 1.63 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | A4W-GGN5 | 11 | Linear | L | None | Amidation | Free | Anticancer | Gaegurin 5 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 98.63 ± 1.17 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop2-PS2Aa | 12 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 15.95 ± 0.69 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop1-HCoV-229E | 11 | Linear | L | None | Amidation | Free | Anticancer | Alphacoronavirus (HCoV-229E) | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 125.0 ± 1.32 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop2-PS2Aa | 12 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 92.99 ± 0.98 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop1-PS2Aa | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 106.2 ± 1.67 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | Loop1-PS2Aa | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 23.76 ± 1.25 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | P264-G274 | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-620 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 11.28 ± 0.52 µM | 48-h | Colon | None | ||
| 34796903 | 2021 | P264-G274 | 11 | Linear | L | None | Amidation | Free | Anticancer | Parasporin-2Aa1 | SW-480 | Colorectal Cancer | Sulforhodamine B assay | EC50 = 90.98 ± 0.75 µM | 48-h | Colon | None | ||
| 33245189 | 2021 | Tachyplesin | 17 | Linear | L | None | Amidation | Free | Antibacterial | Horseshoe crab | H-460 | Lung Cancer | MTT assay | IC50 = 25 µg/ml | 24-h | Lung | None | ||
| 33245189 | 2021 | Tachyplesin | 17 | Linear | L | None | Amidation | Free | Antibacterial | Horseshoe crab | A-549 | Lung Cancer | MTT assay | IC50 = 35 µg/ml | 24-h | Lung | None | ||
| 33562681 | 2021 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | Aska-SS | Synovial Sarcoma | MTS assay | IC50 = 32.41 μg/mL | NA | Muscle | None | ||
| 33562681 | 2021 | TP4 | 25 | Linear | L | None | Free | Free | Antimicrobial | Oreochromis niloticus | SW982 | Synovial Sarcoma | MTS assay | IC50 = 29.20 μg/mL | NA | Muscle | None | ||
| 34449322 | 2021 | rhCGA-N46 | 46 | Linear | L | None | Free | Free | Antimicrobial | Found in neurons and endocrine cells in Humans | HCT-116 | Colon Cancer | MTT assay | IC50 = 1.997 µg/ml | 24-h | Colon | None | ||
| 34073203 | 2021 | Ranatuerin-2 | 31 | Linear | L | None | Free | Free | Anticancer | Rana catesbeiana | LoVo | Colon Cancer | MTT assay | IC50 = 128 µM | 24-h | Colon | None | ||
| 34073203 | 2021 | Ranatuerin-2 | 31 | Linear | L | None | Free | Free | Anticancer | Rana catesbeiana | HeLa | Cervical Cancer | MTT assay | IC50 > 128 µM | 24-h | Cervix | None | ||
| 34073203 | 2021 | Ranatuerin-2 | 31 | Linear | L | None | Free | Free | Anticancer | Rana catesbeiana | MCF-7 | Breast Cancer | MTT assay | IC50 > 128 µM | 24-h | Breast | None | ||
| 34073203 | 2021 | Ranatuerin-2 | 31 | Linear | L | None | Free | Free | Anticancer | Rana catesbeiana | A-549 | Lung Cancer | MTT assay | IC50 > 128 µM | 24-h | Lung | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | MDA-MB-435 DOX-R | Breast Cancer | MTS assay | IC50 = 3.4 µM | 24-h | Breast | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | MDA-MB-435 WT | Breast Cancer | MTS assay | IC50 = 3.5 µM | 24-h | Breast | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | CT-26 | Colorectal Cancer | MTS assay | IC50 = 2.2 µM | 24-h | Colon | None | ||
| 34461456 | 2021 | D-melittin | 27 | Linear | D | None | Free | Free | Anticancer | Synthetic | A-549 | Lung Cancer | MTS assay | IC50 = 4.5 µM | 24-h | Lung | None | ||
| 33462944 | 2021 | GP-3 | 6 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | Colo-320 | Colon Cancer | MTT assay | IC50 = 149 ± 15.2 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-3 | 6 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | CT-26 | Colorectal Cancer | MTT assay | IC50 = 133 ± 12.5 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-3 | 6 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | CaCo-2 | Colon Cancer | MTT assay | IC50 = 162 ± 17.1 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-2 | 5 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | CaCo-2 | Colon Cancer | MTT assay | IC50 = 154 ± 15.8 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-2 | 5 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | Colo-320 | Colon Cancer | MTT assay | IC50 = 142 ± 14.9 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-1 | 6 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | Colo-320 | Colon Cancer | MTT assay | IC50 = 111 ± 12.0 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-2 | 5 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | CT-26 | Colorectal Cancer | MTT assay | IC50 = 114 ± 12.1 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-1 | 6 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | CaCo-2 | Colon Cancer | MTT assay | IC50 = 104 ± 11.3 µM | 48-h | Colon | None | ||
| 33462944 | 2021 | GP-1 | 6 | Linear | L | None | Amidation | Free | Anticancer | Ginseng Leaf Peptide | CT-26 | Colorectal Cancer | MTT assay | IC50 = 86.4 ± 9.46 µM | 48-h | Colon | None | ||
| 34073203 | 2021 | Brevinin-2DYb | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | LoVo | Colon Cancer | MTT assay | IC50 = 35.05 µM | 24-h | Colon | None | ||
| 34073203 | 2021 | Brevinin-2DYb | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | HeLa | Cervical Cancer | MTT assay | IC50 = 23.26 µM | 24-h | Cervix | None | ||
| 34073203 | 2021 | Brevinin-2DYb | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | MCF-7 | Breast Cancer | MTT assay | IC50 = 37.84 µM | 24-h | Breast | None | ||
| 34073203 | 2021 | Brevinin-2DYb | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | A-549 | Lung Cancer | MTT assay | IC50 = 24.01 µM | 24-h | Lung | None | ||
| 34073203 | 2021 | Odorranain-C1 | 33 | Linear | L | None | Free | Free | Anticancer | Odorrana grahami | LoVo | Colon Cancer | MTT assay | IC50 = 55.22 µM | 24-h | Colon | None | ||
| 34073203 | 2021 | Odorranain-C1 | 33 | Linear | L | None | Free | Free | Anticancer | Odorrana grahami | HeLa | Cervical Cancer | MTT assay | IC50 = 52.83 µM | 24-h | Cervix | None | ||
| 34073203 | 2021 | Odorranain-C1 | 33 | Linear | L | None | Free | Free | Anticancer | Odorrana grahami | MCF-7 | Breast Cancer | MTT assay | IC50 = 41.21 µM | 24-h | Breast | None | ||
| 34073203 | 2021 | Odorranain-C1 | 33 | Linear | L | None | Free | Free | Anticancer | Odorrana grahami | A-549 | Lung Cancer | MTT assay | IC50 = 27.31 µM | 24-h | Lung | None | ||
| 34073203 | 2021 | Ranatuerin-2Lb | 32 | Linear | L | None | Free | Free | Anticancer | Rana luteiventris | LoVo | Colon Cancer | MTT assay | IC50 = 59.78 µM | 24-h | Colon | None | ||
| 34073203 | 2021 | Ranatuerin-2Lb | 32 | Linear | L | None | Free | Free | Anticancer | Rana luteiventris | MCF-7 | Breast Cancer | MTT assay | IC50 = 45.25 µM | 24-h | Breast | None | ||
| 34073203 | 2021 | Ranatuerin-2Lb | 32 | Linear | L | None | Free | Free | Anticancer | Rana luteiventris | HeLa | Cervical Cancer | MTT assay | IC50 = 37.23 µM | 24-h | Cervix | None | ||
| 34073203 | 2021 | Ranatuerin-2Lb | 32 | Linear | L | None | Free | Free | Anticancer | Rana luteiventris | A-549 | Lung Cancer | MTT assay | IC50 = 15.32 µM | 24-h | Lung | None | ||
| 34073203 | 2021 | Brevinin-2DYd | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | LoVo | Colon Cancer | MTT assay | IC50 = 8.05 µg/ml | 24-h | Colon | None | ||
| 34073203 | 2021 | Brevinin-2DYd | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | HeLa | Cervical Cancer | MTT assay | IC50 = 19.69 µg/ml | 24-h | Cervix | None | ||
| 34073203 | 2021 | Brevinin-2DYd | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | MCF-7 | Breast Cancer | MTT assay | IC50 = 25.74 µg/ml | 24-h | Breast | None | ||
| 34073203 | 2021 | Brevinin-2DYd | 33 | Linear | L | None | Free | Free | Anticancer | Rana dybowskii | A-549 | Lung Cancer | MTT assay | IC50 = 2.975 µg/ml | 24-h | Lung | None | ||
| 33919639 | 2021 | Pugnin B | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | PC-3 | Prostate Cancer | MTT assay | 90% Cytotoxicity at 100 µM | 24-h | Prostate | None | ||
| 33919639 | 2021 | Pugnin B | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | MCF-7 | Breast Cancer | MTT assay | 5% Cytotoxicity at 100 µM | 24-h | Breast | None | ||
| 33919639 | 2021 | Pugnin A | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | PC-3 | Prostate Cancer | MTT assay | 74% Cytotoxicity at 100 µM | 24-h | Prostate | None | ||
| 34935253 | 2021 | LCP-3 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | CaCo-2 | Colon Cancer | MTT assay | IC50 = 68.2 ± 7.11 μM | 48-h | Colon | None | ||
| 33919639 | 2021 | Pugnin A | 13 | Linear | L | None | Free | Free | Antibacterial and Anticancer | Synthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax) | MCF-7 | Breast Cancer | MTT assay | 12% Cytotoxicity at 100 µM | 24-h | Breast | None | ||
| 34935253 | 2021 | LCP-3 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | MKN-45 | Gastric Cancer | MTT assay | IC50 = 86.9 ± 9.11 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-3 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | HepG-2 | Gastric Cancer | MTT assay | IC50 = 85.2 ± 9.27 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-2 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | HepG-2 | Gastric Cancer | MTT assay | IC50 = 96.9 ± 9.91 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-2 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | CaCo-2 | Colon Cancer | MTT assay | IC50 = 100 ± 11.6 μM | 48-h | Colon | None | ||
| 34935253 | 2021 | LCP-3 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | SGC-7901 | Gastric Cancer | MTT assay | IC50 = 101 ± 10.6 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-2 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | SGC-7901 | Gastric Cancer | MTT assay | IC50 = 116 ± 12.4 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-2 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | MKN-45 | Gastric Cancer | MTT assay | IC50 = 107 ± 11.8 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-1 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | MKN-45 | Gastric Cancer | MTT assay | IC50 = 128 ± 13.5 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-1 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | HepG-2 | Gastric Cancer | MTT assay | IC50 = 123 ± 12.9 μM | 48-h | Stomach | None | ||
| 34935253 | 2021 | LCP-1 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | CaCo-2 | Colon Cancer | MTT assay | IC50 = 131 ± 13.4 μM | 48-h | Colon | None | ||
| 33757145 | 2021 | P2 | 8 | Linear | L | None | Free | Free | Anticancer | Zingiber officinale | Raji | Lymphoma Cancer | MTT assay | IC50 = 700 μg/mL | 24-h | Blood | None | ||
| 34935253 | 2021 | LCP-1 | 4 | Cyclic | L | None | Cyclized | Cyclized | Anticancer | Laminaria japonica | SGC-7901 | Gastric Cancer | MTT assay | IC50 = 111 ± 10.6 μM | 48-h | Stomach | None | ||
| 33757145 | 2021 | P2 | 8 | Linear | L | None | Free | Free | Anticancer | Zingiber officinale | MOLT-4 | Luekemia Cancer | MTT assay | IC50 = 700 μg/mL | 24-h | Blood | None | ||
| 34309373 | 2021 | N-Ter-TAT | 24 | Linear | L | Dansylglycine = fluorescent amino acid residue located in the side chain of lysine | TAT | Free | Anticancer | Synthetic | A-375 | Skin Cancer | MTT assay | IC50 > 50.0 μM | 24-h | Skin | None | ||
| 33757145 | 2021 | P2 | 8 | Linear | L | None | Free | Free | Anticancer | Zingiber officinale | NB-4 | Luekemia Cancer | MTT assay | IC50 = 600 μg/mL | 24-h | Blood | None | ||
| 34394384 | 2021 | MIPP | 8 | Linear | L | None | Free | Free | Anticancer | Morchella importuna | HeLa | Cervical Cancer | MTT assay | Inhibitory rate = 59.36 ± 3.67% at 400 μg/mL | 24-h | Cervix | None | ||
| 33582221 | 2021 | Dermaseptin-TO | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tomopterna | PC-3 | Prostate Cancer | MTT assay | Graph Figure-7 | 24-h | Prostate | None | ||
| 33582221 | 2021 | Dermaseptin-TO | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tomopterna | H-157 | Lung Cancer | MTT assay | Graph Figure-7 | 24-h | Lung | None | ||
| 33582221 | 2021 | Dermaseptin-TO | 28 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa tomopterna | U251-MG | Brain Tumor | MTT assay | Graph Figure-7 | 24-h | Brain | None | ||
| 34572719 | 2021 | LyeTxI-b | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 5.77 ± 0.83 µM | 48-h | Breast | None | ||
| 34572719 | 2021 | LyeTxI-b | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | MCF-7 | Breast Cancer | MTT assay | IC50 = 7.34 ± 3.09 µM | 48-h | Breast | None | ||
| 34572719 | 2021 | LyeTxI-b | 24 | Linear | L | None | Amidation | Free | Antimicrobial and Anticancer | Synthetic | 4T1 | Breast Cancer | MTT assay | IC50 = 6.5 ± 5.30 µM | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | MDA-MB-231 | Breast Cancer | Annexin V-FITC assay | ~80% cell death at 200 µg/ml | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | MCF-7 | Breast Cancer | Annexin V-FITC assay | ~50% cell death at 300 µg/ml | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | SK-BR-3 | Breast Cancer | Annexin V-FITC assay | ~80% cell death at 100 µg/ml | 48-h | Breast | None | ||
| 34236134 | 2021 | Bovine Lactoferricin (LfcinB) | 25 | Linear | L | None | Free | Free | Antimicrobial | Bovine Milk | MDA-MB-468 | Breast Cancer | Annexin V-FITC assay | ~60% cell death at 300 µg/ml | 48-h | Breast | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.721 µM | 24-h | Colon | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | MCF-7 | Breast Cancer | MTT assay | IC50 = 3.17 µM | 24-h | Breast | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | U251-MG | Brain Tumor | MTT assay | IC50 = 3.492 µM | 24-h | Brain | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | PC-3 | Prostate Cancer | MTT assay | IC50 = 2.629 µM | 24-h | Prostate | None | ||
| 34564615 | 2021 | B1OS-D-L | 24 | Linear | Mix | None | Free | Free | Antimicrobial | B-1OS | H-838 | Lung Cancer | MTT assay | IC50 = 2.553 µM | 24-h | Lung | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | HCT-116 | Colon Cancer | MTT assay | IC50 = 11.03 µM | 24-h | Colon | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | MCF-7 | Breast Cancer | MTT assay | IC50 = 8.883 µM | 24-h | Breast | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | U251-MG | Brain Tumor | MTT assay | IC50 = 8.629 µM | 24-h | Brain | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.473 µM | 24-h | Prostate | None | ||
| 34564615 | 2021 | B1OS-L | 24 | Linear | L | None | Free | Free | Antimicrobial | B-1OS | H-838 | Lung Cancer | MTT assay | IC50 = 3.976 µM | 24-h | Lung | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | HCT-116 | Colon Cancer | MTT assay | IC50 = 33.69 µM | 24-h | Colon | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | MCF-7 | Breast Cancer | MTT assay | IC50 = 112 µM | 24-h | Breast | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | U251-MG | Brain Tumor | MTT assay | IC50 = 233.0 µM | 24-h | Brain | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | PC-3 | Prostate Cancer | MTT assay | IC50 = 95.94 µM | 24-h | Prostate | None | ||
| 34564615 | 2021 | B1OS | 23 | Linear | L | None | Free | Free | Antimicrobial | Odorrana schmackeri | H-838 | Lung Cancer | MTT assay | IC50 = 36.84 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | HCT-116 | Colon Cancer | MTT assay | IC50 = 3.583 µM | 24-h | Colon | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | H-157 | Lung Cancer | MTT assay | IC50 = 2.811 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 2.243 µM | 24-h | Breast | None | ||
| 32812694 | 2021 | Brevinin-1HY | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.425 µM | 24-h | Prostate | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | HCT-116 | Colon Cancer | MTT assay | IC50 = 342.8 µM | 24-h | Colon | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | H-157 | Lung Cancer | MTT assay | IC50 = 278.9 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 214.7 µM | 24-h | Breast | None | ||
| 32812694 | 2021 | Brevinin-1Ha | 21 | Linear | L | None | Free | Free | Antimicrobial | Analogue of Brevinin-1H | PC-3 | Prostate Cancer | MTT assay | IC50 = 186.9 µM | 24-h | Prostate | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | HCT-116 | Colon Cancer | MTT assay | IC50 = 2.599 µM | 24-h | Colon | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | H-157 | Lung Cancer | MTT assay | IC50 = 3.37 µM | 24-h | Lung | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | MDA-MB-435S | Breast Cancer | MTT assay | IC50 = 3.47 µM | 24-h | Breast | None | ||
| 32812694 | 2021 | Brevinin-1H | 21 | Linear | L | None | Free | Free | Antimicrobial | Amolops hainanensis | PC-3 | Prostate Cancer | MTT assay | IC50 = 5.87 µM | 24-h | Prostate | None | ||
| 33489681 | 2021 | Chickpea | 7 | Linear | L | None | Free | Free | Anticancer | Cicer arietinum L. | MCF-7 | Breast Cancer | Sulforhodamine B assay | IC50 = 110.3 ± 2.97µM | NA | Breast | None | ||
| 33489681 | 2021 | Chickpea | 7 | Linear | L | None | Free | Free | Anticancer | Cicer arietinum L. | MDA-MB-231 | Breast Cancer | Sulforhodamine B assay | IC50 = 107.2 ± 1.62µM | NA | Breast | None | ||
| 33489681 | 2021 | Chickpea | 7 | Linear | L | None | Free | Free | Anticancer | Cicer arietinum L. | A-549 | Lung Cancer | Sulforhodamine B assay | IC50 = 126.4 ± 1.98 µM | NA | Lung | None | ||
| 33489681 | 2021 | Chickpea | 7 | Linear | L | None | Free | Free | Anticancer | Cicer arietinum L. | HepG-2 | Liver Cancer | Sulforhodamine B assay | IC50 = 113.7 ± 0.99 µM | NA | Liver | None | ||
| 33489681 | 2021 | Chickpea | 7 | Linear | L | None | Free | Free | Anticancer | Cicer arietinum L. | Ishikawa | Endometrial Cancer | Sulforhodamine B assay | IC50 = 101.5 ± 1.83 µM | NA | Endometrium | None | ||
| 33489681 | 2021 | Chickpea | 7 | Linear | L | None | Free | Free | Anticancer | Cicer arietinum L. | PA-1 | Ovarian Cancer | Sulforhodamine B assay | IC50 = 133.4 ± 0.70µM | NA | Ovary | None | ||
| 33595876 | 2021 | VS-9 | 9 | Linear | L | None | Free | Free | Anticancer | Allium sativum | K-562 | Blood Cancer | MTT assay | IC50 = 1.57 mM | 48-h | Blood | None | ||
| 33595876 | 2021 | VS-9 | 9 | Linear | L | None | Free | Free | Anticancer | Allium sativum | MOLT-4 | Blood Cancer | MTT assay | IC50 = 0.84 mM | 48-h | Blood | None | ||
| 34867962 | 2021 | SSTP1 | 18 | Linear | L | None | Free | Free | Host Defense Peptide | Indosylvirana aurantiaca | HSC-4 | Tongue Squamous Cell Carcinoma | MTT assay | IC50 = 10.22 μM | 48-h | Tongue | None | ||
| 34867962 | 2021 | SSTP1 | 18 | Linear | L | None | Free | Free | Host Defense Peptide | Indosylvirana aurantiaca | MDA-MB-231 | Breast Cancer | MTT assay | IC50 = 4.5 μM | 48-h | Breast | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 1499 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 427.3 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 180.8 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6KW | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 118.4 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 593.7 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 88.28 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 186.1 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-6K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 55.65 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 2.679 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 1.546 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 1.796 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-5K | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 2.605 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | U251-MG | Brain Tumor | MTT assay | IC50 = 32.18 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-157 | Lung Cancer | MTT assay | IC50 = 6.143 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | H-838 | Lung Cancer | MTT assay | IC50 = 10.11 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1-K4 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Analogue of t-DPH1 | PC-3 | Prostate Cancer | MTT assay | IC50 = 18.99 μM | 24-h | Prostate | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | U251-MG | Brain Tumor | MTT assay | IC50 = 34.25 μM | 24-h | Brain | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | H-157 | Lung Cancer | MTT assay | IC50 = 10.20 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | H-838 | Lung Cancer | MTT assay | IC50 = 23.51 μM | 24-h | Lung | None | ||
| 34943741 | 2021 | t-DPH1 | 21 | Linear | L | None | Amidation | Free | Antimicrobial | Phyllomedusa hypochondrialis | PC-3 | Prostate Cancer | MTT assay | IC50 = 14.67 μM | 24-h | Prostate | None | ||
| None | 2021 | DN4 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | 191.67 ± 12.02 μM | 24-h | Liver | None | ||
| None | 2021 | DN1 | 13 | Linear | L | None | Free | Free | Antimicrobial | Synthetic | HepG-2 | Liver Cancer | MTT assay | 152.17 ± 7.73 μM | 24-h | Liver | None | ||
| None | 2023 | MAD1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | OVCAR-3 | Ovarian Cancer | MTT assay | IC50 = 14.2 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | MAD1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 36.2 μM | 48-h | Lung | US11571454 B2 | ||
| None | 2023 | MAD1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | NCI/ADR-RES | Ovarian Cancer | MTT assay | IC50 = 85.6 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | A-549 | Lung Cancer | MTT assay | IC50 = 11.9 μM | 48-h | Lung | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | OVCAR-3 | Ovarian Cancer | MTT assay | IC50 = 8.6 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | NCI/ADR-RES | Ovarian Cancer | MTT assay | IC50 = 14.0 μM | 48-h | Lung | US11571454 B2 | ||
| None | 2023 | DAP1 | 13 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | T-24 | Bladder Cancer | MTT assay | IC50 = 15.3 μM | 48-h | Bladder | US11571454 B2 | ||
| None | 2023 | AMP1 | 9 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | OVCAR-3 | Ovarian Cancer | MTT assay | IC50 = 51.1 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2023 | AMP2 | 9 | Linear | L | None | Amidation | Free | Antimicrobial | Synthetic | OVCAR-3 | Ovarian Cancer | MTT assay | IC50 = 53.5 μM | 48-h | Ovary | US11571454 B2 | ||
| None | 2022 | P1C | 7 | Linear | L | None | Acetylation | Free | Anticancer | Synthetic | BXPC-3 | Pancreatic Cancer | Cell Proliferation assay | ~40% reduction in cell growth at 20 μM | 72-h | Pancreas | US011214593B2 | ||
| None | 2022 | P1A | 7 | Linear | L | None | Free | Free | Anticancer | Synthetic | BXPC-4 | Pancreatic Cancer | Cell Proliferation assay | ~50% reduction in cell growth at 20 μM | 72-h | Pancreas | US011214593B2 | ||
| None | 2022 | P1B | 7 | Linear | L | None | Acetylation | Free | Anticancer | Synthetic | BXPC-5 | Pancreatic Cancer | Cell Proliferation assay | ~50% reduction in cell growth at 20 μM | 72-h | Pancreas | US011214593B2 | ||
| None | 2022 | Sample Peptide 1 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 48% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 2 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 0.4% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 3 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 45.8% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 4 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 85.6% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 5 from US011339203B2 | 41 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 77.6% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 6 from US011339203B2 | 34 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 59.7% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 7 from US011339203B2 | 34 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | CAKI-2 | Renal Cancer | CCK-8 assay | Cell Viability = 66.3% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 2 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | PC-3 | Prostate Cancer | CCK-8 assay | Cell Viability = 2.5% at 25 μM | 48-h | Kidney | US011339203B2 | ||
| None | 2022 | Sample Peptide 2 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-2058 | Skin Cancer | CCK-8 assay | Cell Viability = 0.2% at 25 μM | 48-h | Skin | US011339203B2 | ||
| None | 2022 | Sample Peptide 2 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H2444 | Lung Cancer | CCK-8 assay | Cell Viability = 0.6% at 25 μM | 48-h | Lung | US011339203B2 | ||
| None | 2022 | Sample Peptide 2 from US011339203B2 | 35 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 assay | Cell Viability = 1.4% at 25 μM | 48-h | Lung | US011339203B2 | ||
| None | 2023 | Sample Peptide 1 from EP3604345B1 | 33 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H2444 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 6.8% at 25 μM | 48-h | Lung | EP3604345B1;US11352408B2 | ||
| None | 2023 | Sample Peptide 2 from EP3604345B1 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H2444 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 3.6% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 3 from EP3604345B1 | 31 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H2444 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 87.7% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 1 from EP3604345B1 | 33 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 11.8% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 2 from EP3604345B1 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 4.9% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 3 from EP3604345B1 | 31 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 120.6% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 4 from EP3604345B1 | 33 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 102.6% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 5 from EP3604345B1 | 13 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | HCC-827 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 106.5% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 2 from EP3604345B1 | 29 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-549 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 9.1% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 1 from EP3604345B1 | 33 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H446 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 0.5% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 3 from EP3604345B1 | 31 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | NCI-H446 | Lung Cancer | CCK-8 / WST-8 | Cell Viability = 56.7% at 25 μM | 48-h | Lung | EP3604345B1 | ||
| None | 2023 | Sample Peptide 1 from EP3604345B1 | 33 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-2058 | Skin Cancer | CCK-8 / WST-8 | Cell Viability = 6.7% at 25 μM | 48-h | Skin | EP3604345B1 | ||
| None | 2023 | Sample Peptide 3 from EP3604345B1 | 31 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | A-2058 | Skin Cancer | CCK-8 / WST-8 | Cell Viability = 87.5% at 25 μM | 48-h | Skin | EP3604345B1 | ||
| None | 2023 | Sample Peptide 1 from EP3604345B1 | 33 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | CCK-8 / WST-8 | Cell Viability = 62.3% at 25 μM | 48-h | Breast | EP3604345B1 | ||
| None | 2023 | Sample Peptide 3 from EP3604345B1 | 31 | Linear | L | None | Amidation | Free | Anticancer | Synthetic | MDA-MB-231 | Breast Cancer | CCK-8 / WST-8 | Cell Viability = 81.7% at 25 μM | 48-h | Breast | EP3604345B1 | ||
| 37874670 | 2023 | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | NCI-H2122 | NSCLC | CellTiter-Glo Cell Viability assay | IC50 = 1.4 ± 0.3 nmol/L | Not available | Lung | None | ||
| 37874670 | 2023 | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | MiaPaCa.2 | Pancreatic Cancer | CellTiter-Glo Cell Viability assay | IC50 = 1.4 ± 0.2 nmol/L | Not available | Pancreas | None | ||
| 37874670 | 2023 | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | NCI-H441 | NSCLC | CellTiter-Glo Cell Viability assay | IC50 = 2.9 ± 0.7 nmol/L | Not available | Lung | None | ||
| 37874670 | 2023 | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | LS 180 | Colon Cancer | CellTiter-Glo Cell Viability assay | IC50 = 2.7 ± 0.4 nmol/L | Not available | Colon | None | ||
| 37874670 | 2023 | LUNA18 | Not Available | Cyclic | L | None | Free | Alkylation | Anticancer and Antitumor | Synthetic | GSU | Stomach Cancer | CellTiter-Glo Cell Viability assay | IC50 = 0.17 ± 0.02 nmol/L | Not available | Stomach | None |