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IDPMIDYEARSequenceNameLengthLinear/CyclicChiralityChem-MODC-ter MODN-ter MODNatureOriginCell LineCancer TypeAssayActivityTesting TimeTissue AffectedPatents
7713
383194352024
FFFLSRIF
Temporin-SHf8LinearLNoneAmidationFreeAntimicrobialPelophylax saharicaHepG-2Liver CancerMTT assayIC50 = 32.64 ± 1.350 µM24-hLiverNone
7714
None2022
RRWKRFFKRWKGGVIGVTFPF
ATRA1-R3W2 - HYD21LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticH-358Lung CancerCytotoxicity assayLD50 ~24.5 μM6-hLungUS011447533B2
7712
383194352024
FFFLSRIF
Temporin-SHf8LinearLNoneAmidationFreeAntimicrobialPelophylax saharicaPC-3Prostate CancerMTT assayIC50 = 36.67 ± 0.729 µM24-hProstateNone
7711
383194352024
FFFLSRIF
Temporin-SHf8LinearLNoneAmidationFreeAntimicrobialPelophylax saharicaMCF-7Breast CancerMTT assayIC50 = 32.76 ± 1.528 µM24-hBreastNone
7710
383194352024
FFFLSRIF
Temporin-SHf8LinearLNoneAmidationFreeAntimicrobialPelophylax saharicaA-549Lung CancerMTT assayIC50 = 24.03 ± 0.945 µM24-hLungNone
7709
378538142024
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerMTT assay52.5 ± 5.0% cell viability at 150 µM24-hBreastNone
7708
378538142024
RWGKWFKKATHVGKHVGKAALTAYL
NRC-0725LinearLNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerMTT assay14.0 ± 3.0% cell viability at 150 µM24-hBreastNone
7704
384915562024
AAEKEFIKYPYPTPLQYQQLATRLKVEKKLVRRW
HMM-ID34LinearLNoneFreeFreeAnticancerRed Sea BrineU2OSOsteosarcomaMTT assayIC50 = 100.5 µg/ml24-hBoneNone
7702
382722302024
RPPLVIC
RP7 SCR7LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)PC-3Prostate CancerMTT assayIC50 = 128 ± 11.65 µM24-hProstateNone
7703
382722302024
RPPLVIC
RP7 SCR7LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)DU-145Prostate CancerMTT assayIC50 = 137 ± 5.98 µM24-hProstateNone
7701
382722302024
RPPLVIC
RP7 SCR7LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MCF-7Breast CancerMTT assayIC50 = 150 ± 10.32 µM24-hBreastNone
7700
382722302024
RPPLVIC
RP7 SCR7LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MDA-MB-231Breast CancerMTT assayIC50 = 156 ± 8.15 µM24-hBreastNone
7699
382722302024
rppcvil
D-RP-77LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)DU-145Prostate CancerMTT assayIC50 = 121.59 ± 6.56 µM24-hProstateNone
7698
382722302024
rppcvil
D-RP-77LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)PC-3Prostate CancerMTT assayIC50 = 101 ± 5.73 µM24-hProstateNone
7696
382722302024
rppcvil
D-RP-77LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MDA-MB-231Breast CancerMTT assayIC50 = 95 ± 7.71 µM24-hBreastNone
7697
382722302024
rppcvil
D-RP-77LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MCF-7Breast CancerMTT assayIC50 = 90 ± 10.31 µM24-hBreastNone
7694
382722302024
RPPCVIL
RP-77LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)PC-3Prostate CancerMTT assayIC50 = 113 ± 8.02 µM24-hProstateNone
7695
382722302024
RPPCVIL
RP-77LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)DU-145Prostate CancerMTT assayIC50 = 120.72 ± 7.08 µM24-hProstateNone
7693
382722302024
RPPCVIL
RP-77LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MCF-7Breast CancerMTT assayIC50 = 110.12 ± 4.23 µM24-hBreastNone
7691
382722302024
LAKAVI
LA3IK-SCR6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)DU-145Prostate CancerMTT assayIC50 = 351.76 ± 7.18 µM24-hProstateNone
7692
382722302024
RPPCVIL
RP-77LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MDA-MB-231Breast CancerMTT assayIC50 = 139.03 ± 8.41 µM24-hBreastNone
7690
382722302024
LAKAVI
LA3IK-SCR6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)PC-3Prostate CancerMTT assayIC50 = 319 ± 13.64 µM24-hProstateNone
7689
382722302024
LAKAVI
LA3IK-SCR6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MCF-7Breast CancerMTT assayIC50 = 133 ± 9.52 µM24-hBreastNone
7688
382722302024
LAKAVI
LA3IK-SCR6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MDA-MB-231Breast CancerMTT assayIC50 = 243 ± 8.16 µM24-hBreastNone
7686
382722302024
laiavk
D-LA3IK6LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)PC-3Prostate CancerMTT assayIC50 = 98.71 ± 6.17 µM24-hProstateNone
7687
382722302024
laiavk
D-LA3IK6LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)DU-145Prostate CancerMTT assayIC50 = 89.11 ± 8.12 µM24-hProstateNone
7685
382722302024
laiavk
D-LA3IK6LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MCF-7Breast CancerMTT assayIC50 = 91.2 ± 8.21 µM24-hBreastNone
7683
382722302024
LAIAVK
LA3IK6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)DU-145Prostate CancerMTT assayIC50 = 335.7 ± 3.09 µM24-hProstateNone
7684
382722302024
laiavk
D-LA3IK6LinearDNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MDA-MB-231Breast CancerMTT assayIC50 = 197.72 ± 5.42 µM24-hBreastNone
7681
382722302024
LAIAVK
LA3IK6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MCF-7Breast CancerMTT assayIC50 = 90.23 ± 7.32 µM24-hBreastNone
7682
382722302024
LAIAVK
LA3IK6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)PC-3Prostate CancerMTT assayIC50 = 321.4 ± 11.79 µM24-hProstateNone
7680
382722302024
LAIAVK
LA3IK6LinearLNoneAmidationAcetylationAnticancerMigration and invasion enhancer 1 (MIEN1)MDA-MB-231Breast CancerMTT assayIC50 = 223.6 ± 5.62 µM24-hBreastNone
7675
384647292024
NCSIHGDIPAY
U711LinearLNoneFreeFreeAnticancerPhoenix dactyliferaHepG-2Liver CancerMTT assayIC50 = 523 µM48-hLiverNone
7673
384647292024
NCSIHGDIPAY
U711LinearLNoneFreeFreeAnticancerPhoenix dactyliferaMCF-7Breast CancerMTT assayIC50 = 554 µM48-hBreastNone
7674
384647292024
NCSIHGDIPAY
U711LinearLNoneFreeFreeAnticancerPhoenix dactyliferaT-47DBreast CancerMTT assayIC50 = 584 ± 29.99 µM48-hBreastNone
7666
384647292024
NGSIPATWASL
U311LinearLNoneFreeFreeAnticancerPhoenix dactyliferaHepG-2Liver CancerMTT assayIC50 = 561 µM48-hLiverNone
7665
384647292024
NGSIPATWASL
U311LinearLNoneFreeFreeAnticancerPhoenix dactyliferaT-47DBreast CancerMTT assayIC50 = 517.6 ± 34.86 µM48-hBreastNone
7664
384647292024
NGSIPATWASL
U311LinearLNoneFreeFreeAnticancerPhoenix dactyliferaMCF-7Breast CancerMTT assayIC50 = 555 µM48-hBreastNone
7658
372985952023
PEGKRPY-Tle-L
NT-129LinearLTle = L-tert-leucineFreeFreeAnticancerSynthetic analogue of NeurotensinHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7659
372985952023
PEGKKPY-Tle-L
NT-129LinearLTle = L-tert-leucineFreeFreeAnticancerSynthetic analogue of NeurotensinHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7656
372985952023
RRPYAL
NT-116LinearLNoneFreeFreeAnticancerSynthetic analogue of NeurotensinHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7657
372985952023
PEGRKPY-Tle-L
NT-129LinearLTle = L-tert-leucineFreeFreeAnticancerSynthetic analogue of NeurotensinHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7654
372985952023
RRPYIL
NT-96LinearLNoneFreeFreeAnticancerSynthetic analogue of NeurotensinHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7655
372985952023
RRPAIL
NT-106LinearLNoneFreeFreeAnticancerSynthetic analogue of NeurotensinHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7652
372985952023
rRP-Hyp-G-Thi-S-(D)Pip-Thi-R
BK-710LinearMixHyp = hydroxyproline; Thi = thienylalanine; (D)Pip—(D)-piperidine-2-carboxylic acidFreeFreeAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7653
372985952023
Aaa-rRP-Hyp-G-Thi-S-(D)Pip-Thi-R
BK-810LinearMixHyp = hydroxyproline; Thi = thienylalanine; (D)Pip—(D)-piperidine-2-carboxylic acidFreeAaa = [(3S,5S,7S)-adamantan-1-yl]acetic acidAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7650
372985952023
rRP-Hyp-G-Thi-S-f-(L)Pip-R
BK-510LinearMixHyp = hydroxyproline; Thi = thienylalanine; (L)Pip—(L)-piperidine-2-carboxylic acidFreeFreeAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7651
372985952023
Aaa-rRP-Hyp-G-Thi-S-(D)Pip-(L)Pip-R
BK-610LinearMixHyp = hydroxyproline; Thi = thienylalanine; (L)Pip—(L)-piperidine-2-carboxylic acid;(D)Pip—(D)-piperidine-2-carboxylic acidFreeAaa = [(3S,5S,7S)-adamantan-1-yl]acetic acidAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7648
372985952023
Aaa-rRP-Hyp-G-Thi-S-Acc-Thi-R
BK-310LinearMixHyp = hydroxyproline; Thi = thienylalanine; Acc = 1-aminocyclohexane-1-carboxylic acidFreeAaa = [(3S,5S,7S)-adamantan-1-yl]acetic acidAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7649
372985952023
Aaa-rRP-Hyp-G-Thi-S-f-Acc-R
BK-410LinearMixHyp = hydroxyproline; Thi = thienylalanine; Acc = 1-aminocyclohexane-1-carboxylic acidFreeAaa = [(3S,5S,7S)-adamantan-1-yl]acetic acidAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7646
372985952023
rRP-Hyp-G-Thi-S-Apc-Thi-R
BK-110LinearMixHyp = hydroxyproline; Thi = thienylalanine; Apc =1-aminocyclopentyl-1-carboxylic acidFreeFreeAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7647
372985952023
rRP-Hyp-G-Thi-S-f-Apc-R
BK-210LinearMixHyp = hydroxyproline; Thi = thienylalanine; Apc =1-aminocyclopentyl-1-carboxylic acidFreeFreeAnticancerSynthetic analogue of BradykininHCT-116Colorectal CancerMTS assayNot Available24-hColonNone
7645
373448202023
AKIPIKAAIKTVGKAVGKGLRAINIASTANDVFNFLKPKKRKA
Moricin43LinearLNoneFreeFreeAntimicrobialBombyx moriMDA-MB-231Triple-negative Breast CancerTrypan blue assay70% cell viability at 6.25 µg/ml24-hBreastNone
7644
373448202023
AKIPIKAAIKTVGKAVGKGLRAINIASTANDVFNFLKPKKRKA
Moricin43LinearLNoneFreeFreeAntimicrobialBombyx moriMDA-MB-231Triple-negative Breast CancerLDH release assaySignificant decrease in cell viability at 6.25 μg/ml24-hBreastNone
7642
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
MC–FA27LinearLNoneFolic AcidFreeAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 12.63 µg/mL24-hBreastNone
7643
373448202023
AKIPIKAAIKTVGKAVGKGLRAINIASTANDVFNFLKPKKRKA
Moricin43LinearLNoneFreeFreeAntimicrobialBombyx moriMDA-MB-231Triple-negative Breast CancerMTT assay70% cell viability at 6.25 µg/ml24-hBreastNone
7640
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
MC–FA27LinearLNoneFolic AcidFreeAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 66.43 µg/mL24-hCervixNone
7641
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
MC–FA27LinearLNoneFolic AcidFreeAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 35.22 µg/ mL24-hCervixNone
7638
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
CM–FA27LinearLNoneAmidationFolic AcidAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 35.75 µg/mL24-hCervixNone
7639
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
CM–FA27LinearLNoneAmidationFolic AcidAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 10.38 µg/mL24-hBreastNone
7637
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
CM–FA27LinearLNoneAmidationFolic AcidAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 67.34 µg/mL24-hCervixNone
7636
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
Mel-C27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 160.62 µg/mL24-hBreastNone
7635
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
Mel-C27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 58.63 µg/mL24-hCervixNone
7634
378802862023
GIGAVLKVLTTGLPALISWIKRKRQQC
Mel-C27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 50.72 µg/mL24-hCervixNone
7633
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
C-Mel27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueMCF-7Breast CancerMTT assayIC50 = 110.59 µg/mL24-hBreastNone
7632
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
C-Mel27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueC-33ACervical CancerMTT assayIC50 = 44.76 µg/mL24-hCervixNone
7631
378802862023
CGIGAVLKVLTTGLPALISWIKRKRQQ
C-Mel27LinearLNoneAmidationFreeAnticancer; AntibacterialSynthetic analogueHeLaCervical CancerMTT assayIC50 = 64.15 µg/mL24-hCervixNone
7629
372518372023
Not Available
CPSA-CPSC-L-ACANNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableAnticancerRecombinant Fusion PeptideHeLaCervical CancerMTT assayIC50 = 63.15 μg/ml24-hCervixNone
7628
368730172023
CLKKLLKLLKKLLKLCLEELLHHLEELLHH
LK-LE330CyclicLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 10.2 µM at pH 624-hCervixNone
7627
368730172023
CLKKLLKLLKKLLKLCLEHLLEHLEHLLEH
LK-LE230CyclicLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 12.9 µM at pH 624-hCervixNone
7626
368730172023
CLKKLLKLLKKLLKLCLHELLEHLHELLEH
LK-LE130Cyclic(C1-C16)LNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 11.3 µM at pH 624-hCervixNone
7624
371042352023
QHWSYGLRPGGRGPKDAVRAVKGSALLPCIIVHDPNLNNSDKMKFNTYYLLEYKEYWHQLWSQIIPAHQTVKIQERTGISEVVQNSMIEDLNMYIGADFGMYFYLRSSGFKEQITRGLNRPLSQTTTQLGERVEEMEYYNSNDLDVRYVKYALAREFTLKRVNGEIVKNWVAVDYRMAGIQSYPNAPITNPLTLT
LHRH-BinBC195LinearLNoneFreeFused a luteinizing hormone-releasing hormone (LHRH) peptideMosquitocidal, AnticancerSyntheticMCF-7Breast CancerLDH leakage assay40% LDH efflux at 16 µM48-hBreastNone
7623
371042352023
QHWSYGLRPGGRGPKDAVRAVKGSALLPCIIVHDPNLNNSDKMKFNTYYLLEYKEYWHQLWSQIIPAHQTVKIQERTGISEVVQNSMIEDLNMYIGADFGMYFYLRSSGFKEQITRGLNRPLSQTTTQLGERVEEMEYYNSNDLDVRYVKYALAREFTLKRVNGEIVKNWVAVDYRMAGIQSYPNAPITNPLTLT
LHRH-BinBC195LinearLNoneFreeFused a luteinizing hormone-releasing hormone (LHRH) peptideMosquitocidal, AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 10.96 μM48-hBreastNone
7622
370019082023
EYVQTVKSSKG
A1111LinearLNoneFreeFreeAnticancerAnnexin A1A-375Skin CancerBiotin Pull Down assayNot Available24-hSkinNone
7620
370019082023
EYVQTVKSSKG
A1111LinearLNoneFreeFreeAnticancerAnnexin A1MDA-MB-231Breast CancerBiotin Pull Down assayNot Available24-hBreastNone
7621
370019082023
EYVQTVKSSKG
A1111LinearLNoneFreeFreeAnticancerAnnexin A1H-460Lung CancerBiotin Pull Down assayNot Available24-hLungNone
7618
369345262023
RLLRLLRLRRLLRL
WP214LinearLNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHepG-2Liver CancerCell Viability assayIC50 = 34.05 ± 0.53 μM48-hLiverNone
7619
369345262023
RLLRLLRLRRLLRL
WP214LinearLNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHT-29Colon CancerCell Viability assayIC50 = 42.6 ± 4.0 μM48-hColonNone
7616
369345262023
RLLRLLRLRRLLRL
WP214LinearLNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHeLaCervical CancerHDAC inhibition assayIC50 = 0.446±0.095 µMNot AvailableCervixNone
7617
369345262023
RLLRLLRLRRLLRL
WP214LinearLNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHuh-7Liver CancerCell Viability assayIC50 = 28.12 ± 1.5 μM48-hLiverNone
7613
369345262023
RLLRLMRLRMLLRM
WP114Cyclic(M6-M10)LNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHuh-7Liver CancerCell Viability assayIC50 = 43.74 ± 5.4 μM48-hLiverNone
7614
369345262023
RLLRLMRLRMLLRM
WP114Cyclic(M6-M10)LNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHepG-2Liver CancerCell Viability assayIC50 = 52.23 ± 0.9 μM48-hLiverNone
7615
369345262023
RLLRLMRLRMLLRM
WP114Cyclic(M6-M10)LNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHT-29Colon CancerCell Viability assayIC50 = 54.6 ± 2.1 μM48-hColonNone
7612
369345262023
RLLRLMRLRMLLRM
WP114Cyclic(M6-M10)LNoneHydroxamic acidAcetylationAnticancerDerived from RLL peptideHeLaCervical CancerHDAC inhibition assayIC50 = 0.310±0.064 µMNot AvailableCervixNone
7611
377346502023
KLKSKLMVVANKIGLLKSLARKFVKSH
NKL-MUT27LinearLNoneFreeFreeAntimicrobialTrematomus bernacchiiB16-F10Skin Cancerluciferase-based ATPlite assayATP level = 0.023 ± 0.007 at 40 μM12-hSkinNone
7609
349867322023
trans(P)PIPYPIF
trans-Phakellistatin 187CyclicLProline residues in trans-configurationFreeFreeAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 67.5 ± 2.938 µMNot AvailableLiverNone
7610
377346502023
KLKSKLMVVCNKIGLLKSLCRKFVKSH
NKL-WT27LinearLNoneFreeFreeAntimicrobialTrematomus bernacchiiB16-F10Skin Cancerluciferase-based ATPlite assayATP level = 0.753 ± 0.254 at 40 μM12-hSkinNone
7608
368404532023
FLKSLWRGVKAIFNGARQGYKEHKN
AMP-WF325LinearLNoneFreeFreeAnticancerPoecilia Mexicana fishJurkatBlood CancerMTT assayIC50 = 50 µM24-hBloodNone
7607
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisHCT-116Colon CancerLDH leakage assayLDH release above 80%24-hColonNone
7606
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisHCT-116Colon CancerMTT assayIC50 = 2.02 μM24-hColonNone
7605
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisU-251-MGBrain TumorMTT assayIC50 = 2.32 μM24-hBrainNone
7604
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisMDA-MB-435Breast CancerMTT assayIC50 = 18.99 μM24-hBreastNone
7603
312343332023
GLFSVVKGVLKGVGKNVSGSLLDQLKCKISGGC
LFB33LinearLNoneFreeFreeAntimicrobialLimnonectes fujianensisH-460Lung CancerMTT assayIC50 = 3.47 μM24-hLungNone
7602
377645212023
GAGIVVASIDTGVRVSHE
GE1818LinearLNoneFreeFreeAntimicrobialAphanomyces invadansMCF-7Breast CancerMTT assayIC50 = 35.34 µM24-hBreastNone
7601
366260982023
FKCRRWQWRMKKLG-K-RSKNKGFKEQAKSLLKWILD
LFchimera35LinearLNoneAmidationFreeAntimicrobialSynthetic - Lectoferrin chimeraJurkatBlood CancerMTT assaycell viability ~ 8% at 20 µM6-hBloodNone
7600
366260982023
FKCRRWQWRMKKLG-K-RSKNKGFKEQAKSLLKWILD
LFchimera35LinearLNoneAmidationFreeAntimicrobialSynthetic - Lectoferrin chimeraHepG-2Liver CancerMTT assaycell viability ~ 44% at 10 µM12-hLiverNone
7599
366260982023
DLIWKLLSKAQEKFGKNKSR
LFampin265–28420LinearLNoneAmidationFreeAntimicrobialLectoferrin PeptideJurkatBlood CancerMTT assaycell viability ~ 47% at 10 µM6-hBloodNone
7598
366260982023
DLIWKLLSKAQEKFGKNKSR
LFampin265–28420LinearLNoneAmidationFreeAntimicrobialLectoferrin PeptideHepG-2Liver CancerMTT assaycell viability ~ 50% at 1 µM12-hLiverNone
7597
366260982023
FKCRRWQWRMKKLG
LFcin17–3014LinearLNoneAmidationFreeAntimicrobialLectoferrin PeptideJurkatBlood CancerMTT assaycell viability ~ 70% at 20 µM6-hBloodNone
7596
366260982023
FKCRRWQWRMKKLG
LFcin17–3014LinearLNoneAmidationFreeAntimicrobialLectoferrin PeptideHepG-2Liver CancerMTT assaycell viability ~ 50% at 1 µM12-hLiverNone
7595
366260982023
FKCRRWQWRMKKLGAPSITCVRRAF
bLF25LinearLNoneFreeFreeAntimicrobialBos TaurusJurkatBlood CancerMTT assaycell viability ~ 17.5% at 20 µM4-hBloodNone
7593
365092202023
KLLKINLK(Aib)LAALAKKIL
KM8-Aib18LinearLAib = 2-Aminoisobutyric acidAmidationFreeAntimicrobialSynthetic derivative of KM8Not AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
7594
366260982023
FKCRRWQWRMKKLGAPSITCVRRAF
bLF25LinearLNoneFreeFreeAntimicrobialBos TaurusHepG-2Liver CancerMTT assaycell viability ~ 21% at 10 µM24-hLiverNone
7592
365092202023
KLLKINLKALAALAKKIL
KM818LinearLNoneAmidationFreeAntimicrobialSynthetic derivative of MastoparanNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
7591
365092202023
INLKALAALAKKIL
Mastoparan14LinearLNoneAmidationFreeAntimicrobialWasp venomNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNot AvailableNone
7590
373800462023
ATRQPNH
RP77LinearLNoneFreeFreeAnticancerRAGE(receptor for advanced glycation end product) inhibitorBT-549Breast CancerMTT assayIC50 = 29.9 µM48-hBreastNone
7589
373800462023
ATRQPNH
RP77LinearLNoneFreeFreeAnticancerRAGE(receptor for advanced glycation end product) inhibitorMDA-MB-231Breast CancerMTT assayIC50 = 24.5 µM48-hBreastNone
7588
365674782023
DGDWDAWTRETS
mtp112LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerMTS assay17.4% decrease in cell viability at 10 μM24-hLungNone
7586
365674782023
DGDWDAWTRETS
mtp112LinearLNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerMTS assay33.6% decrease in cell viability at 10 μM24-hBreastNone
7587
365674782023
DGDWDAWTRETS
mtp112LinearLNoneFreeFreeAnticancerSyntheticHeLaCervical CancerMTS assay30.2 % decrease in cell viability at 10 μM24-hCervixNone
7585
372736292023
PSRKVMLWS
PS99LinearLNoneFreeFreeAnticancerAphanomyces invadansMCF-7Breast CancerLDH leakage assay71.25 ± 1.3% LDH release at 40 μM24-hBreastNone
7584
372736292023
PSRKVMLWS
PS99LinearLNoneFreeFreeAnticancerAphanomyces invadansMCF-7Breast CancerNeutral Red Uptake assayIC50 value range between 25.27 - 43.28 μM24-hBreastNone
7583
370985302023
GIGAVLKVLTTGLPALISWIKRKRQQ
Mellitin26LinearLNoneAmidationFreeAnticancerMain component of honey bee venomK-562Leukemia CancerSulforhodamine B assayIC50 = 1.84 ± 0.75 μg/ml96-hBloodNone
7581
370685202023
YSFGL
Test peptide5LinearLNoneAmidationFreeAnti cancerNeuropep PeptideA-549Lung CancerMTT assayIC50 = 26.417±0.660 µM48 hLungNone
7582
370685202023
YSFGL
Test peptide5LinearLNoneAmidationFreeAnti cancerNeuropep PeptideMDA-MB-231Lung CancerMTT assayIC50 = 39.047±0.770 µM48 hLungNone
7580
368307252023
CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK
Pep-1-Phor2130LinearLNoneFreeFreeAnticancerHybrid peptide PEP1 and Phor 21PC-3Prostrate CancerAlamarBlue assayIC50 ≤ 0.6 μM24-hProstateNone
7579
368307252023
CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK
Pep-1-Phor2130LinearLNoneFreeFreeAnticancerHybrid peptide PEP1 and Phor 21DU-145Prostrate CancerAlamarBlue assayIC50 = 2.57 ± 2.02 µM24-hProstateNone
7577
361688172023
NDGNQPL
Rapeseed peptide7LinearLNoneFreeFreeAnticancerextracted from rapeseed proteinHepG-2Liver CancerApoptosis assay28.39 ± 0.80% apoptosis rate at 0.5 mmol/LNALiverNone
7578
368307252023
CGEMGWVRCKFAKFAKKFAKFAKKFAKFAK
Pep-1-Phor2130LinearLNoneFreeFreeAnticancerHybrid peptide PEP1 and Phor 21LNCaPLiver CancerAlamarBlue assayIC50 = 55.13 ± 13.56 µM24-hLiverNone
7576
361688172023
NDGNQPL
Rapeseed peptide7LinearLNoneFreeFreeAnticancerextracted from rapeseed proteinHepG-2Liver CancerMTT assayIC50 = 1.56 mmol/L24-hLiverNone
7575
375140492023
FAVWGCADYRGY
Salamandrin - I12LinearLNoneAmidationFreeAntioxidantSalamandra salamandraHL-60Leukemia CancerLDH leakage assayAbsorbance ~ 2 at 490 nm at 27 27 µM48-hBloodNone
7574
375140492023
FAVWGCADYRGY
Salamandrin - I12LinearLNoneAmidationFreeAntioxidantSalamandra salamandraHL-60Leukemia CancerMTT assayIC50 = 27 µM48-hBloodNone
7573
375809092023
QETFSDLWKLLVQRKRQKLMP
mPNC-NLS21LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerCytotoxicity assayIC50 = 45 μM24-hLungNone
7572
375809092023
QETFSDLWKLLVQRKRQKLMP
mPNC-NLS21LinearLNoneFreeFreeAnticancerSyntheticU-87Brain TumorMTT assayIC50 = 56.9 μM24-hBrainNone
7571
375809092023
QETFSDLWKLLVQRKRQKLMP
mPNC-NLS21LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 44.9 μM24-hLungNone
7570
367303012023
VNWKKILGKIIKVVK
Lasioglossin - III15LinearLNoneAmidationFreeAntimicrobialLasioglossum laticepsHepG-2Liver CancerNot AvailableIC50 = 7.75 μMNot AvailableLiverNone
7569
367303012023
VNWKKILGKIIKVVK
Lasioglossin - III15LinearLNoneAmidationFreeAntimicrobialLasioglossum laticepsA-549Lung CancerNot AvailableIC50 = 26.36 μMNot AvailableLungNone
7568
374839712023
THPPTTTTTTTTTTTYTAAPATTT
ATMP124LinearLNoneFreeFreeAntimicrobialAnabas testudineusMDA-MB-231Breast CancerMTT assayIC50 = 8.25 ± 0.14 μg/ml48-hBreastNone
7567
374839712023
THPPTTTTTTTTTTTYTAAPATTT
ATMP524LinearLNoneFreeFreeAnticancer; AntimicrobialSynthetic Analog of ATMP1MDA-MB-231Breast CancerMTT assayIC50 = 64.04 ± 0.021 μg /ml24-hBreastNone
7566
None2023
AWLDKLKSIGKVVGKVAIGVAKNLLNPQ
Raniseptin-328LinearLNoneFreeFreeAntimicrobial and AntitumorBoana ranicepsB16-F10Skin CancerMTT assayIC50 = 6.56 uM3-hSkinNone
7564
369104652023
KLWCKSSQVPQSR
ALA-A213LinearLNoneFreeFreeAnticancerAlpha-LactalbuminHT-29Colon CancerMTT assay~50% cell viability24-hColonNone
7565
None2023
ALLDKLKSLGKVVGKVALGVVQNYLNPRQ
Raniseptin-629LinearLNoneFreeFreeAntimicrobial and AntitumorBoana ranicepsB16-F10Skin CancerMTT assayIC50 = 8.69 uM3-hSkinNone
7563
369104652023
KLWCKSSQVPQSR
ALA-A213LinearLNoneFreeFreeAnticancerAlpha-LactalbuminA-549Lung CancerMTT assay~50% cell viability24-hLungNone
7562
373105332023
RIIDRLWLVRRPQKPKFVLVWVL
PMAP-NC23LinearLNoneFreeFreeAntimicrobialSynthetic Analgog of PMAP-24A-549Lung CancerMTT assayIC50 = 7.1 μM4-hLungNone
7561
373105332023
RIIDRLWLVRRPQKPKFVLVWVL
PMAP-NC23LinearLNoneFreeFreeAntimicrobialSynthetic Analgog of PMAP-23MDA-MB-361Breast CancerMTT assayIC50 = 6.4 μM4-hBreastNone
7560
371834662023
WKLFKKILKVL
CM1111LinearLNoneAmidationFreeAntimicrobialCecropin-Melittin Hybrid PeptideRajiBlood CancerMTT assaySurvival rate = 51% at 32 μg/ml24-hBloodNone
7559
371834662023
WKLFKKILKVL
CM1111LinearLNoneAmidationFreeAntimicrobialCecropin-Melittin Hybrid PeptideJurkatBlood CancerMTT assaySurvival rate = 47% at 32 μg/ml24-hBloodNone
7558
377643342023
ALWKSILKNAGKAVLNEINQIV
14VL2323LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 16.4 µM24-hLungNone
7557
377643342023
ALWKSILKNAGKAVLNEINQIV
14VL2323LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 5.7 µM24-hLungNone
7556
377643342023
ALWKKILKNAGKAVLNEINQIVQ
14V5K23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 6.1 µM24-hLungNone
7555
377643342023
ALWKKILKNAGKAVLNEINQIVQ
14V5K23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 8.1 µM24-hLungNone
7554
377643342023
ALWKSILKNVGKVLNEINQIVQ
L2V22LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 0.6 µM24-hLungNone
7553
377643342023
ALWKSILKNVGKVLNEINQIVQ
L2V22LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 2.2 µM24-hLungNone
7552
377643342023
ALWKSILKNAGKAGLNEINQIVQ
14G23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 31.7 µM24-hLungNone
7551
377643342023
ALWKSILKNAGKAGLNEINQIVQ
14G23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 48.7 µM24-hLungNone
7550
377643342023
ALWKSILKNAGKAVLNEINQIVQ
14V23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 4.1 µM24-hLungNone
7549
377643342023
ALWKSILKNAGKAVLNEINQIVQ
14V23LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 7.0 µM24-hLungNone
7548
377643342023
ALWKSILKNAGKALNEINQIVQ
L1422LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-460Lung CancerMTT assayIC50 = 20.1 µM24-hLungNone
7547
377643342023
ALWKSILKNAGKALNEINQIVQ
L1422LinearLNoneAmidationFreeAntimicrobial and AnticancerDermaseptin-SS1- AnalogH-838Lung CancerMTT assayIC50 = 64.4 µM24-hLungNone
7546
377643342023
ALWKSILKNAGKAALNEINQIV
Dermaseptin-SS123LinearLNoneAmidationFreeAntimicrobial and AnticancerBrown-belly leaf frog, Phyllomedusa TarsiusH-460Lung CancerMTT assayIC50 = 1.3 µM24-hLungNone
7544
369826102023
UKLUGGLUGI
K2-NH210LinearLU = 2-Aminoisobutyric acidAmidationOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 = 9 µM24-hBreastNone
7545
377643342023
ALWKSILKNAGKAALNEINQIV
Dermaseptin-SS123LinearLNoneAmidationFreeAntimicrobial and AnticancerBrown-belly leaf frog, Phyllomedusa TarsiusH-838Lung CancerMTT assayIC50 = 7.7 µM24-hLungNone
7542
369826102023
UGLUKKLUGI
K56-Lol10LinearLU = 2-Aminoisobutyric acidLol = leucinolOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 =12 µM24-hBreastNone
7543
369826102023
UGLUGKLUGI
K6-NH210LinearLU = 2-Aminoisobutyric acidAmidationOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 =8 µM24-hBreastNone
7540
369826102023
UKLUKGLUKI
K259-Lol10LinearLU = 2-Aminoisobutyric acidLol = leucinolOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 =10 µM24-hBreastNone
7541
369826102023
UKLUKGLUGI
K25-Lol10LinearLU = 2-Aminoisobutyric acidLol = leucinolOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 =9 µM24-hBreastNone
7539
369826102023
UKLUKGLUKI
K259-NH210LinearLU = 2-Aminoisobutyric acidAmidationOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 =13 µM24-hBreastNone
7537
369826102023
UGLLGGLUGI
Leu4-NH210LinearLU = 2-Aminoisobutyric acidAmidationOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 > 20 µM24-hBreastNone
7538
369826102023
UKLUKKLUKI
K2569-Lol10LinearLU = 2-Aminoisobutyric acidLol = leucinolOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 = 12 µM24-hBreastNone
7536
369826102023
UGLUGGLZGI
Api8-NH210LinearLZ =4-aminopiperidine-4-carboxylic acid , U = 2-Aminoisobutyric acidAmidationOct = 1-octanoylAntimicrobial and AntifungalTrichogin GAMDA-MB-231Breast CancerMTS assayIC50 > 20 µM24-hBreastNone
7534
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 189LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreedecanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.2 μM24-hPancreasNone
7535
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 199LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreedodecanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.2 μM24-hPancreasNone
7533
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 179LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeOctanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.6 μM24-hPancreasNone
7532
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 169LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeHexanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.5 μM24-hPancreasNone
7530
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 149LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreePropanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 1.8 μM24-hPancreasNone
7531
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 159LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeButanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.9 μM24-hPancreasNone
7529
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 139LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeEthanoylAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 6.0 μM24-hPancreasNone
7528
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 129LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeFreeAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 > 9 μM24-hPancreasNone
7527
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 410LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeFreeAntitubercularTrichoderin APANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.5 μM24-hPancreasNone
7525
366789142023
MDA-P-AHMOD-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 199LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreedodecanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.1 μM24-hPancreasNone
7526
366789142023
MDA-P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A10LinearLMDA = 2-methyl decanoic acid; AHMOD = 2-amino-6-hydroxy-4-methyl-8-oxodecanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeFreeAntitubercularTrichoderma sp. fungus, strain 05FI48PANC-1Pancreatic CancerCyQUANT Direct assayIC50 = 0.3 μM24-hPancreasNone
7524
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 189LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreedecanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.2 μM24-hPancreasNone
7523
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 179LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid; AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeOctanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.4 μM24-hPancreasNone
7522
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 169LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeHexanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.4 μM24-hPancreasNone
7521
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 159LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeButanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.5 μM24-hPancreasNone
7519
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 139LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeEthanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 > 1 μM24-hPancreasNone
7520
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 149LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreePropanoylAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.6 μM24-hPancreasNone
7518
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 129LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeFreeAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 > 1 μM24-hPancreasNone
7516
366789142023
MDA-P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A10LinearLMDA = 2-methyl decanoic acid; AHMOD = 2-amino-6-hydroxy-4-methyl-8-oxodecanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeFreeAntitubercularTrichoderma sp. fungus, strain 05FI48BxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.4 μM24-hPancreasNone
7517
366789142023
P-Cha-Aib-Aib-IV-Aib-Aib-AMAE
trichoderin A analogue 410LinearLAHMOD replaced by Cha(L-cyclohexylalanine); MDA = 2-methyl decanoic acid; Aib = a-aminoisobutyric acid;AMAE = 2-[(20-aminopropyl) methylamino] ethanolFreeFreeAntitubercularTrichoderin ABxPC-3Pancreatic CancerPrestoBlue assayIC50 = 0.4 μM24-hPancreasNone
7515
372287022023
FLPLLAGLAANFLPKIICKIARKC
B1AW-K24LinearLNoneAmidationFreeAntimicrobial and Antitumoranalogue of B1AWU251-MGBrain TumorMTT assayIC50 = 3.860 µM24-hBrainNone
7514
372287022023
FLPLLAGLAANFLPKIICKIARKC
B1AW-K24LinearLNoneAmidationFreeAntimicrobial and Antitumoranalogue of B1AWH-838Lung CancerMTT assayIC50 = 5.15 µM24-hLungNone
7513
372287022023
FLPLLAGLAANFLPKIICKIARKC
B1AW-K24LinearLNoneAmidationFreeAntimicrobial and Antitumoranalogue of B1AWPC-3Prostate CancerMTT assayIC50 = 4.283 µM24-hProstateNone
7512
372287022023
FLPLLAGLAANFLPQIICKIARKC
B1AW24LinearLNoneAmidationFreeAntimicrobial and AntitumorWuyi torrent frog, Amolops wuyiensisU251-MGBrain TumorMTT assayIC50 = 33.56 µM24-hBrainNone
7511
372287022023
FLPLLAGLAANFLPQIICKIARKC
B1AW24LinearLNoneAmidationFreeAntimicrobial and AntitumorWuyi torrent frog, Amolops wuyiensisH-838Lung CancerMTT assayIC50 = 32.15 µM24-hLungNone
7510
372287022023
FLPLLAGLAANFLPQIICKIARKC
B1AW24LinearLNoneAmidationFreeAntimicrobial and AntitumorWuyi torrent frog, Amolops wuyiensisPC-3Prostate CancerMTT assayIC50 = 33.46 µM24-hProstateNone
7509
375081982023
FLGVALKLGKVLGKALLPLASSLLHSQ
Figanin 2BN27LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)HT-29Colon CancerMTT assayLC50 = 14.1 uM24-hColonNone
7508
375081982023
FLGVALKLGKVLGKALLPLASSLLHSQ
Figanin 2BN27LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)MDA-MB-231Breast CancerMTT assayLC50 = 8.1 uM24-hBreastNone
7507
375081982023
FLGVALKLGKVLGKALLPLASSLLHSQ
Figanin 2BN27LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)A-549Lung CancerMTT assayLC50 = 6.7 uM24-hLungNone
7506
375081982023
GIFKDTLKKVVAAVLTTVADNIHPK
Picturin 1BN25LinaerLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)HT-29Colon CancerMTT assayLC50 = 84.9 uM24-hColonNone
7505
375081982023
GIFKDTLKKVVAAVLTTVADNIHPK
Picturin 1BN25LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)MDA-MB-231Breast CancerMTT assayLC50 = 64.2 uM24-hBreastNone
7504
375081982023
GIFKDTLKKVVAAVLTTVADNIHPK
Picturin 1BN25LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)A-549Lung CancerMTT assayLC50 = 30.7 µM24-hLungNone
7503
375081982023
GLMDMLKKVGKVALTVAKSALLP
Picturin 2BN23LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)HT-29Colon CancerMTT assayLC50 52.2 uM24-hColonNone
7502
375081982023
GLMDMLKKVGKVALTVAKSALLP
Picturin 2BN23LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)MDA-MB-231Breast CancerMTT assayLC50 26.3 uM24-hBreastNone
7501
375081982023
GLMDMLKKVGKVALTVAKSALLP
Picturin 2BN23LinearLNoneAmidationFreeAntimicrobial and AntitumorGiant Gladiator Treefrog (Boana boans)A-549Lung CancerMTT assayLC50 = 23 µM24-hLungNone
7500
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticA-549Lung CancerCCK-8 assayIC50 = 32.47 µM36-hLungNone
7499
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticU-2 OSBone CancerCCK-8 assayIC50 = 25.65 µM36-hBoneNone
7498
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticHeLaCervical CancerCCK-8 assayIC50 = 42.95 µM36-hCervixNone
7497
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticZR-75-30Breast CancerCCK-8 assayIC50 = 23.57 µM36-hBreastNone
7496
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerCCK-8 assayIC50 = 31.05 µM36-hBreastNone
7495
375982102023
grrrqrrkkrlgpfsidllikslsdnmtdl
M1-2030LinearDNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerCCK-8 assayIC50 = 18.15 µM36-hBreastNone
7494
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticZR-75-30Breast CancerCell Viability assayIC50 = 12.92 µM72-hBreastNone
7493
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticU-251BrainTumorCell Viability assayIC50 = 18.17 µM72-hBrainNone
7492
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticA-549Lung CancerCell Viability assayIC50 = 22.00 µM72-hLungNone
7491
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticHCT-116Colon CancerCell Viability assayIC50 = 9.08 µM72-hColonNone
7490
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSynthetic786-0Renal CancerCell Viability assayIC50 = 13.5 µM72-hRenalNone
7489
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticHeLaCervical CancerCell Viability assayIC50 = 31.83 µM72-hCervixNone
7488
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSynthetic5637Bladder cancerCell Viability assayIC50 = 9.33 µM72-hBladderNone
7487
373448572023
rrrqrrkkrg-QTQPRLGPPQTPAGGCSILIF
M1-2131LinearMixNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerCell Viability assayIC50 = 24.25 µM72-hBreastNone
7480
373969452023
LSTAADMQGVVTDGMASGLDKDYLKPDD
p2828LinearLNoneFreeFreeAntitumorPseudomonas aeruginosaCT-26Colorectal CancerMTT assayIC50 ~ 150 μg/ml24-hColonNone
7479
373969452023
LSTAADMQGVVTDGMASGLDKDYLKPDD
p2828LinearLNoneFreeFreeAntitumorPseudomonas aeruginosaHT-29Colon CancerMTT assayIC50 ~ 200 μg/ml24-hColonNone
7477
366870352023
WQWRWQWR
1-R8LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMCF-7Breast CancerMTT assayIC50 = 130 µM24-hBreastNone
7478
366870352023
WQWRWQWR
1-R8LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMDA-MB-231Breast CancerMTT assayIC50 > 150 µM24-hBreastNone
7476
366870352023
RWQWRWQW
R-18LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMDA-MB-231Breast CancerMTT assayIC50 > 150 µM24-hBreastNone
7475
366870352023
RWQWRWQW
R-18LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMCF-7Breast CancerMTT assayIC50 = 58 µM24-hBreastNone
7473
366870352023
WQWRWQW
17LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMCF-7Breast CancerMTT assayIC50 = 105 µM24-hBreastNone
7474
366870352023
WQWRWQW
17LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMDA-MB-231Breast CancerMTT assayIC50 > 170 µM24-hBreastNone
7471
366870352023
RRWQWRWQWR
RR-1-R10LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMCF-7Breast CancerMTT assayIC50 = 68 µM24-hBreastNone
7472
366870352023
RRWQWRWQWR
RR-1-R10LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMDA-MB-231Breast CancerMTT assayIC50 = 73 µM24-hBreastNone
7470
366870352023
RWQWRWQWRR
R-1-RR10LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMDA-MB-231Breast CancerMTT assayIC50 = 95 µM24-hBreastNone
7468
366870352023
RRWQWRWQWRR
RR-1-RR11LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMDA-MB-231Breast CancerMTT assayIC50 = 67 µM24-hBreastNone
7469
366870352023
RWQWRWQWRR
R-1-RR10LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMCF-7Breast CancerMTT assayIC50 = 122 µM24-hBreastNone
7466
366870352023
RWQWRWQWR
LfcinB(21-25)Pal9LinearLNoneAmidationFreeAntibacterial and AnticancerLfcinBMCF-7Breast CancerMTT assayIC50 = 81 µM24-hBreastNone
7467
366870352023
RRWQWRWQWRR
RR-1-RR11LinearLNoneAmidationFreeAntibacterial and AnticancerSynthetic analogue of LfcinB(21-25)PalMCF-7Breast CancerMTT assayIC50 = 58 µM24-hBreastNone
7465
366870352023
RWQWRWQWR
LfcinB(21-25)Pal9LinearLNoneAmidationFreeAntibacterial and AnticancerLfcinBMDA-MB-231Breast CancerMTT assayIC50 = 103 µM24-hBreastNone
7463
378180622023
FAAATGATPIAGR
P1013LinearLNoneFreeFreeAnticancer40S ribosomal protein fragmentU-2 OSBone CancerMTT assayRelative viability = 1.01 at 50 μg/ml48-hBoneNone
7464
366870352023
RWQWRWQWR
LfcinB(21-25)Pal9LinearLNoneAmidationFreeAntibacterial and AnticancerLfcinBMDA-MB-468Breast CancerMTT assayIC50 = 72 µM24-hBreastNone
7461
378180622023
AAGTLYTYPENWR
P0913LinearLNoneFreeFreeAnticancerEukaryotic Translation Elongation Factor 1 Gamma (Eef1G) fragmentU-2 OSBone CancerMTT assayRelative viability = 1.07 at 50 μg/ml48-hBoneNone
7462
378180622023
FAAATGATPIAGR
P1013LinearLNoneFreeFreeAnticancer40S ribosomal protein fragmentMG-63Bone CancerMTT assayRelative viability = 1.08 at 50 μg/ml48-hBoneNone
7460
378180622023
AAGTLYTYPENWR
P0913LinearLNoneFreeFreeAnticancerEukaryotic Translation Elongation Factor 1 Gamma (Eef1G) fragmentMG-63Bone CancerMTT assayRelative viability = 0.85 at 50 μg/ml48-hBoneNone
7458
378180622023
NSNLVGAAHEELQQSR
P0816LinearLNoneFreeFreeAnticancerLamin A/C (LMNA) fragmentMG-63Bone CancerMTT assayRelative viability = 0.92 at 50 μg/ml48-hBoneNone
7459
378180622023
NSNLVGAAHEELQQSR
P0816LinearLNoneFreeFreeAnticancerLamin A/C (LMNA) fragmentU-2 OSBone CancerMTT assayRelative viability = 1.06 at 50 μg/ml48-hBoneNone
7456
378180622023
VEPGLGADNSVVR
P0713LinearLNoneFreeFreeAnticancerFLNA (Filamin A) fragmentMG-63Bone CancerMTT assayRelative viability = 0.96 at 50 μg/ml48-hBoneNone
7457
378180622023
VEPGLGADNSVVR
P0713LinearLNoneFreeFreeAnticancerFLNA (Filamin A) fragmentU-2 OSBone CancerMTT assayRelative viability = 0.96 at 50 μg/ml48-hBoneNone
7454
378180622023
GAGTGGLGLAVEGPSEAK
P0618LinearLNoneFreeFreeAnticancerFLNA (Filamin A) fragmentMG-63Bone CancerMTT assayRelative viability = 0.92 at 50 μg/ml48-hBoneNone
7455
378180622023
GAGTGGLGLAVEGPSEAK
P0618LinearLNoneFreeFreeAnticancerFLNA (Filamin A) fragmentU-2 OSBone CancerMTT assayRelative viability = 1.17 at 50 μg/ml48-hBoneNone
7453
378180622023
HVFGESDELIGQK
P0313LinearLNoneFreeFreeAnticancerTriosephosphate Isomerase (TPI) fragmentU-2 OSBone CancerMTT assayRelative viability = 0.98 at 50 μg/ml48-hBoneNone
7451
378180622023
SETAPAAPAAPAPAEK
P0116LinearLNoneFreeFreeAnticancerHistone H1.4 (H1-4) FragmentU-2 OSBone CancerMTT assayRelative viability = 1.13 at 50 μg/ml48-hBoneNone
7452
378180622023
HVFGESDELIGQK
P0313LinearLNoneFreeFreeAnticancerTriosephosphate Isomerase (TPI) fragmentMG-63Bone CancerMTT assayRelative viability = 1.04 at 50 μg/ml48-hBoneNone
7449
378180622023
IGEHTPSALAIMENANVLAR
P0420LinearLNoneFreeFreeAnticancerAldolase A fragmentU-2 OSBone CancerMTT assayRelative viability = 0.83 at 50 μg/ml48-hBoneNone
7450
378180622023
SETAPAAPAAPAPAEK
P0116LinearLNoneFreeFreeAnticancerHistone H1.4 (H1-4) FragmentMG-63Bone CancerMTT assayRelative viability = 0.84 at 50 μg/ml48-hBoneNone
7448
378180622023
IGEHTPSALAIMENANVLAR
P0420LinearLNoneFreeFreeAnticancerAldolase A fragmentMG-63Bone CancerMTT assayRelative viability = 0.86 at 50 μg/ml48-hBoneNone
7446
378180622023
AEEYEFLTPMEEAPK
P0215LinearLNoneFreeFreeAnticancerRho GDP Dissociation Inhibitor Alpha fragmentMG-63Bone CancerMTT assayRelative viability = 0.88 at 50 μg/ml48-hBoneNone
7447
378180622023
AEEYEFLTPMEEAPK
P0215LinearLNoneFreeFreeAnticancerRho GDP Dissociation Inhibitor Alpha fragmentU-2 OSBone CancerMTT assayRelative viability = 0.93 at 50 μg/ml48-hBoneNone
7445
378180622023
ADDGRPFPQVIK
P0512LinearLNoneFreeFreeAnticancerAldolase A fragmentU-2 OSBone CancerMTT assayRelative viability = 0.98 at 50 μg/ml48-hBoneNone
7444
378180622023
ADDGRPFPQVIK
P0512LinearLNoneFreeFreeAnticancerAldolase A fragmentMG-63Bone CancerMTT assayRelative viability = 0.85 at 50 μg/ml48-hBoneNone
7443
374959882023
TKEQKEQIAKATGLTTKQVRNWYVQLNASIKVCMCSC
37-mer peptide37LinearLNoneFreeFreeAntimicrobialSyntheticSK-OV-3Ovarian cancerMTT assayIC50 = 27.45 ± 1.5085 μM24-hOvaryNone
7442
374959882023
TKEQKEQIAKATGLTTKQVRNWYVQLNASIKVCMCSC
37-mer peptide37LinearLNoneFreeFreeAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 33.65 ± 1.09 μM24-hLiverNone
7441
374959882023
TKEQKEQIAKATGLTTKQVRNWYVQLNASIKVCMCSC
37-mer peptide37LinearLNoneFreeFreeAntimicrobialSyntheticSNU-449Liver CancerMTT assayIC50 = 76.4 ± 0.6015 μM24-hLiverNone
7440
376460482023
RRRRRGLFDIIKKIIKSF
Aurein 1.2_mutant_R5 (R5-Aurm)18LinearLNoneFreeAcetylationAntimicrobialSyntheticHT-29Colon CancerMTT assay54.22% cell viability24-hColonNone
7439
376460482023
RRRRRGLFDIIKKIIKSF
Aurein 1.2_mutant_R5 (R5-Aurm)18LinearLNoneFreeAcetylationAntimicrobialSyntheticSW-480Colon CancerMTT assay40.62% cell viability24-hColonNone
7438
376460482023
RRRRRGLFDIIKKIAESF
Aurein 1.2_R5 (R5-Aur)18LinearLNoneFreeAcetylationAntimicrobialSyntheticHT-29Colon CancerMTT assay61.56% cell viability24-hColonNone
7436
376460482023
GLFDIIKKIIKSF
Aurein 1.2_mutant (Aurm)13LinearLNoneFreeAcetylationAntimicrobialSyntheticHT-29Colon CancerMTT assay66.10% cell viability24-hColonNone
7437
376460482023
RRRRRGLFDIIKKIAESF
Aurein 1.2_R5 (R5-Aur)18LinearLNoneFreeAcetylationAntimicrobialSyntheticSW-480Colon CancerMTT assay43.89% cell viability24-hColonNone
7435
376460482023
GLFDIIKKIIKSF
Aurein 1.2_mutant (Aurm)13LinearLNoneFreeAcetylationAntimicrobialSyntheticSW-480Colon CancerMTT assay51.63% cell viability24-hColonNone
7434
378676942023
rWQWOWQWR
1[dR] 5[Orn] [Pal]9LinearMixO=OrnithineAmidationFreeAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 109 μM24-hColonNone
7433
378676942023
RWQWOWQWR
5[Orn] [Pal]9LinearLO=OrnithineAmidationFreeAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 64 μM24-hColonNone
7432
378676942023
OWQWRWQWR
1[Orn] [Pal]9LinearLO=OrnithineAmidationFreeAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 91 μM24-hColonNone
7430
378676942023
CH3-CO-Ahx-RWQWRWQWR
CH3CO-Ahx-[Pal]10LinearLAhx = Amino Hexanoic AcidAmidationAcetylationAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 31 μM24-hColonNone
7431
378676942023
rWQWRWQWR
1[dR][Pal]9LinearMixNoneAmidationFreeAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 105 μM24-hColonNone
7429
378676942023
RWQWRWQWO
9[Orn] [Pal]9LinearLO=OrnithineAmidationFreeAnticancerSyntheticDU-145Prostrate CancerMTT assayIC50 = 62 μM24-hProstateNone
7427
378676942023
RWQWRWQWO
9[Orn] [Pal]9LinearLO=OrnithineAmidationFreeAnticancerSyntheticHT-29Colon CancerMTT assayIC50 = 109 μM24-hColonNone
7428
378676942023
RWQWRWQWO
9[Orn] [Pal]9LinearLO=OrnithineAmidationFreeAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 40 μM24-hColonNone
7425
378676942023
Ahx-RWQWRWQWR
Ahx-[Pal]10LinearLAhx = Amino Hexanoic AcidAmidationFreeAnticancerSyntheticHT-29Colon CancerMTT assayIC50 = 119 μM24-hColonNone
7426
378676942023
Ahx-RWQWRWQWR
Ahx-[Pal]10LinearLAhx = Amino Hexanoic AcidAmidationFreeAnticancerSyntheticCaCo-2Colorectal CancerMTT assayIC50 = 40 μM24-hColonNone
7424
378676942023
RWQWRWQWR
LfcinB (21-25)Pal9LinearLNoneAmidationFreeAnticancerLfcinBDU-145Prostrate CancerMTT assayIC50 = 40 μM24-hProstateNone
7423
378676942023
RWQWRWQWR
LfcinB (21-25)Pal9LinearLNoneAmidationFreeAnticancerLfcinBHT-29Colon CancerMTT assayIC50 = 100 μM24-hColonNone
7422
378676942023
RWQWRWQWR
LfcinB (21-25)Pal9LinearLNoneAmidationFreeAnticancerLfcinBCaCo-2Colorectal CancerMTT assayIC50 = 86 μM24-hColonNone
7421
364104362023
RRRRNRTRRNRRRVRGGLTIYFY
FHV-2D523LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-G48-hLiverNone
7420
364104362023
TRRQRTRRARRNRGGLTIYFY
HTLV-II-Rex-2D521LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-G48-hLiverNone
7419
364104362023
GRKKRRQRRRPPQGGLTIYFY
TAT-2D521LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-G48-hLiverNone
7418
364104362023
RRRRRRRRGGILTVVELRVP
6F (I113-P122)20LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-D48-hLiverNone
7417
364104362023
RRRRRRRRGGVVELRVPTDLTLLPGHLYMM
6E(V116-M135)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-D48-hLiverNone
7416
364104362023
RRRRRRRRGGGLTIYFY
2D5(G45-Y51)17LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayIC50 = 19.4 μM48-hLiverNone
7415
364104362023
RRRRRRRRGGGLTIYFYN
2D3(G45-N52)18LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7414
364104362023
RRRRRRRRGGQGLTIYFY
2D2(Q44-Y51)18LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7413
364104362023
RRRRRRRRGGQGLTIYFYNSNR
2D(Q44-R55)22LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7412
364104362023
RRRRRRRRGGQGLTIYFYNSNRDFQ
2C(Q44-Q58)25LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7411
364104362023
RRRRRRRRGGFWAGLQGLTIYFYNSNRDFQ
2A(F39-Q58)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-C48-hLiverNone
7410
364104362023
RRRRRRRRGGMWKGFILTVVELRVPTDLTL
#6(M108-L127)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideMCF-7Breast CancerCellTiter-Glo assayGraph figure 1-B48-hBreastNone
7409
364104362023
RRRRRRRRGGMWKGFILTVVELRVPTDLTL
#6(M108-L127)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-B48-hLiverNone
7408
364104362023
RRRRRRRRGGDQEIKFKVETLECREMWKGF
#5(D93-F112)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-B48-hLiverNone
7407
364104362023
RRRRRRRRGGDRDYKKFWAGLQGLTIYFYN
#2(D33-N52)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideMCF-7Breast CancerCellTiter-Glo assayGraph figure 1-B48-hBreastNone
7406
364104362023
RRRRRRRRGGDRDYKKFWAGLQGLTIYFYN
#2(D33-N52)30LinearLNoneFreeFreeAnticancerSTAP-2 PH domain–derived peptideDU-145Liver CancerCellTiter-Glo assayGraph figure 1-B48-hLiverNone
7405
378339182023
RLRRILRKIVRRL
Crabrolin-PR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinMCF-7Breast CancerMTT assayIC50 = 12.29 μM24-hBreastNone
7404
378339182023
RLRRILRKIVRRL
Crabrolin-PR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinHCT-116Colon CancerMTT assayIC50 = 16.29 μM24-hColonNone
7403
378339182023
RLRRILRKIVRRL
Crabrolin-PR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinU-251-MGBrain TumorMTT assayIC50 = 17.70 μM24-hBrainNone
7402
378339182023
RLRRILRKIVRRL
Crabrolin-PR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinPC-3Prostate CancerMTT assayIC50 = 22.37 μM24-hProstateNone
7401
378339182023
RLRRILRKIVRRL
Crabrolin-PR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinH-838Lung CancerMTT assayIC50 = 32.32 μM24-hLungNone
7399
378339182023
RLPRILRKIVRRL
Crabrolin-AR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinHCT-116Colon CancerMTT assayIC50 = 29.90 μM24-hColonNone
7400
378339182023
RLPRILRKIVRRL
Crabrolin-AR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinMCF-7Breast CancerMTT assayIC50 = 32.51 μM24-hBreastNone
7398
378339182023
RLPRILRKIVRRL
Crabrolin-AR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinU-251-MGBrain TumorMTT assayIC50 = 52.01 μM24-hBrainNone
7397
378339182023
RLPRILRKIVRRL
Crabrolin-AR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinPC-3Prostate CancerMTT assayIC50 = 28.78 μM24-hProstateNone
7396
378339182023
RLPRILRKIVRRL
Crabrolin-AR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinH-838Lung CancerMTT assayIC50 = 41.31 μM24-hLungNone
7395
378339182023
RLPRILRKIVRAL
Crabrolin-FR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinMCF-7Breast CancerMTT assayIC50 = 33.85 μM24-hBreastNone
7394
378339182023
RLPRILRKIVRAL
Crabrolin-FR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinHCT-116Colon CancerMTT assayIC50 = 30.29 μM24-hColonNone
7392
378339182023
RLPRILRKIVRAL
Crabrolin-FR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinPC-3Prostate CancerMTT assayIC50 = 15.87 μM24-hProstateNone
7393
378339182023
RLPRILRKIVRAL
Crabrolin-FR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinU-251-MGBrain TumorMTT assayIC50 = 62.17 μM24-hBrainNone
7391
378339182023
RLPRILRKIVRAL
Crabrolin-FR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinH-838Lung CancerMTT assayIC50 = 31.51 μM24-hLungNone
7390
378339182023
FLPRILRKIVRAL
Crabrolin-TR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinMCF-7Breast CancerMTT assayIC50 = 3.459 μM24-hBreastNone
7389
378339182023
FLPRILRKIVRAL
Crabrolin-TR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinHCT-116Colon CancerMTT assayIC50 = 2.810 μM24-hColonNone
7388
378339182023
FLPRILRKIVRAL
Crabrolin-TR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinU-251-MGBrain TumorMTT assayIC50 = 12.40 μM24-hBrainNone
7387
378339182023
FLPRILRKIVRAL
Crabrolin-TR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinPC-3Prostate CancerMTT assayIC50 = 3.944 μM24-hProstateNone
7385
378339182023
FLPKILRKIVTAL
Crabrolin-4K13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinMCF-7Breast CancerMTT assayIC50 = 23.18 μM24-hBreastNone
7386
378339182023
FLPRILRKIVRAL
Crabrolin-TR13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinH-838Lung CancerMTT assayIC50 = 4.637 μM24-hLungNone
7384
378339182023
FLPKILRKIVTAL
Crabrolin-4K13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinHCT-116Colon CancerMTT assayIC50 = 42.88 μM24-hColonNone
7383
378339182023
FLPKILRKIVTAL
Crabrolin-4K13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinU-251-MGBrain TumorMTT assayIC50 = 23.51 μM24-hBrainNone
7382
378339182023
FLPKILRKIVTAL
Crabrolin-4K13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinPC-3Prostate CancerMTT assayIC50 = 20.58 μM24-hProstateNone
7380
378339182023
FLPRILRKIVTAL
Crabrolin-4R13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinMCF-7Breast CancerMTT assayIC50 = 20.26 μM24-hBreastNone
7381
378339182023
FLPKILRKIVTAL
Crabrolin-4K13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinH-838Lung CancerMTT assayIC50 = 22.55 μM24-hLungNone
7379
378339182023
FLPRILRKIVTAL
Crabrolin-4R13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinHCT-116Colon CancerMTT assayIC50 = 47.02 μM24-hColonNone
7378
378339182023
FLPRILRKIVTAL
Crabrolin-4R13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinU-251-MGBrain TumorMTT assayIC50 = 25.09 μM24-hBrainNone
7377
378339182023
FLPRILRKIVTAL
Crabrolin-4R13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinPC-3Prostate CancerMTT assayIC50 = 17.98 μM24-hProstateNone
7375
378339182023
FLPLILRKIVTAL
Crabrolin13LinearLNoneAmidationFreeAntimicrobialEuropean hornet (Vespa crabro)MCF-7Breast CancerMTT assayIC50 = 26.49 μM24-hBreastNone
7376
378339182023
FLPRILRKIVTAL
Crabrolin-4R13LinearLNoneAmidationFreeAntimicrobialSynthetic Analog of CrabrolinH-838Lung CancerMTT assayIC50 = 11.40 μM24-hLungNone
7374
378339182023
FLPLILRKIVTAL
Crabrolin13LinearLNoneAmidationFreeAntimicrobialEuropean hornet (Vespa crabro)HCT-116Colon CancerMTT assayIC50 = 8.539 μM24-hColonNone
7373
378339182023
FLPLILRKIVTAL
Crabrolin13LinearLNoneAmidationFreeAntimicrobialEuropean hornet (Vespa crabro)U-251-MGBrain TumorMTT assayIC50 = 20.13 μM24-hBrainNone
7371
378339182023
FLPLILRKIVTAL
Crabrolin13LinearLNoneAmidationFreeAntimicrobialEuropean hornet (Vespa crabro)H-838Lung CancerMTT assayIC50 = 27.71 μM24-hLungNone
7372
378339182023
FLPLILRKIVTAL
Crabrolin13LinearLNoneAmidationFreeAntimicrobialEuropean hornet (Vespa crabro)PC-3Prostate CancerMTT assayIC50 = 32.13 μM24-hProstateNone
7368
358893012022
LXVLF
Sansalvimide A5CyclicLX = OLeuCyclizedCyclizedAnticancerFusarium sp.HCT-116Colon CancerNot AvailableIC50 = 9.8 µg/mlNot AvailableColonNone
7369
358893012022
LXVLF
Sansalvimide A5CyclicLX = OLeuCyclizedCyclizedAnticancerFusarium sp.Colo-205Colon CancerNot AvailableIC50 = 3.5 µg/mlNot AvailableColonNone
7370
358893012022
LXVLF
Sansalvimide A5CyclicLX = OLeuCyclizedCyclizedAnticancerFusarium sp.SK-MEL-2Skin CancerNot AvailableIC50 = 5.9 µg/mlNot AvailableSkinNone
7365
336302042022
DVNFLLHKIYGNIRY
LvHemB115LinearLNoneAmidationAcetylationAntimicrobialhemocyanin of Litopenaeus vannameiEJBladder CancerMTS assay89.6% apoptotic cells at 50 μg/mL24-hBladderNone
7367
None2022
MDNHVCIPLCPP
MP1212LinearLNoneFreeFreeAntiproliferativeAphanomyces invadansHep-2Larynx CancerMTT assayIC50 = 24.7 ± 0.34 μMNot AvailableLarynxNone
7363
336302042022
DVNFLLHKIYGNIRY
LvHemB115LinearLNoneAmidationAcetylationAntimicrobialhemocyanin of Litopenaeus vannameiEC-109Esophageal CancerMTS assay57.1% apoptotic cells at 50 μg/mL24-hEsophagusNone
7364
336302042022
DVNFLLHKIYGNIRY
LvHemB115LinearLNoneAmidationAcetylationAntimicrobialhemocyanin of Litopenaeus vannameiHepG-2Liver CancerMTS assay44.2% apoptotic cells at 50 μg/mL24-hLiverNone
7362
336302042022
DVNFLLHKIYGNIRY
LvHemB115LinearLNoneAmidationAcetylationAntimicrobialhemocyanin of Litopenaeus vannameiHeLaCervical cancerMTS assay65.1% apoptotic cells at 50 μg/mL24-hCervixNone
7360
352006392022
WYIRKIRRFFKWLKKKLKKK
P620LinearLNoneFreeFreeAntitumorArca inflataSW-620Colon CancerMTT assayIC50 >27 μg/mL48-hColonNone
7361
352006392022
WYIRKIRRFFKWLKKKLKKK
P620LinearLNoneFreeFreeAntitumorArca inflataL02Colorectal CancerMTT assayIC50 >150 μg/mL48-hColonNone
7359
352006392022
WYIRKIRRFFKWLKKKLKKK
P620LinearLNoneFreeFreeAntitumorArca inflataHCT-116Colorectal CancerMTT assayIC50 = 10.88 ± 0.72 μg/mL48-hColonNone
7358
352006392022
WYIRKIRRFFKWLKKKLKKK
P620LinearLNoneFreeFreeAntitumorArca inflataDLD-1Colorectal CancerMTT assayIC50 = 2.14 ± 0.28 μg/mL48-hColonNone
7355
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1MCF-7Breast CancerMTT assayIC50 = 24.60 μM24-hBreastNone
7357
352006392022
WYIRKIRRFFKWLKKKLKKK
P620LinearLNoneFreeFreeAntitumorArca inflataHT-29Colorectal CancerMTT assayIC50 = 4.43 ± 0.15 μg/mL48-hColonNone
7354
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1U-251-MGBrain TumorMTT assayIC50 = 25.06 μM24-hBrainNone
7352
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1H-157Non-small cell lung cancerMTT assayIC50 = 24 μM24-hLungNone
7353
356064682022
GLLGKILGAGKKVLLGVSGLL
Nigrocin-M121LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Analogue of Nigrocin M1PC-3Prostate cancerMTT assayIC50 = 31.27 μM24-hProstateNone
7350
356064682022
GLLGKILGAGKKVLCGVSGLC
Nigrocin-PN21LinearLNoneFreeFreeAntimicrobial and AntitumorPelophylax nigromaculatusPC-3Prostate cancerMTT assayIC50 = 53.03 μM24-hProstateNone
7351
356064682022
GLLGKILGAGKKVLCGVSGLC
Nigrocin-PN21LinearLNoneFreeFreeAntimicrobial and AntitumorPelophylax nigromaculatusU-251-MGBrain TumorMTT assayIC50 = 73.65 μM24-hBrainNone
7349
356064682022
GLLGKILGAGKKVLCGVSGLC
Nigrocin-PN21LinearLNoneFreeFreeAntimicrobial and AntitumorPelophylax nigromaculatusH-157Non-small cell lung cancerMTT assayIC50 = 18.04 μM24-hLungNone
7347
362128272022
LIKKLKEYLKKLI
Lt-MAP213LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Derivative of Lataracin-3aC1498Blood CancerCytotoxicity assayEC50 = 43.9 ± 0.5 µg/mL24-hBloodNone
7348
362128272022
LIKKLKEYLKKLI
Lt-MAP213LinearLNoneFreeFreeAntimicrobial and AntitumorSynthetic; Derivative of Lataracin-3aK-562Blood CancerCytotoxicity assayEC50 = 44 ± 3 µg/mL24-hBloodNone
7346
364263862022
GIFKVLKNLAKGVITSLKS
[D4K,A18K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NHT-29Colorectal CancerCellTiter-Glo assayLC50 = 46 ± 12 μM24-hColonNone
7344
364263862022
GIFKVLKNLAKGVITSLKS
[D4K,A18K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NA-549Lung CancerCellTiter-Glo assayLC50 = 25 ± 1 μM24-hLungNone
7345
364263862022
GIFKVLKNLAKGVITSLKS
[D4K,A18K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NMDA-MB-231Breast CancerCellTiter-Glo assayLC50 = 31 ± 1 μM24-hBreastNone
7343
364263862022
GIFKVLKNLAKGVITSLKS
[D4K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NHT-29Colorectal CancerCellTiter-Glo assayLC50 = 20 ± 1 μM24-hColonNone
7341
364263862022
GIFKVLKNLAKGVITSLKS
[D4K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NA-549Lung CancerCellTiter-Glo assayLC50 = 12 ± 1 μM24-hLungNone
7342
364263862022
GIFKVLKNLAKGVITSLKS
[D4K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NMDA-MB-231Breast CancerCellTiter-Glo assayLC50 = 15 ± 1 μM24-hBreastNone
7340
364263862022
GIFDVLKNLAKGVITSLAS
Ocellatin-3N19LinearLNoneAmidationFreeHost DefenseLeptodactylus nesiotusHT-29Colorectal CancerCellTiter-Glo assayLC50 = 69 ± 10 μM24-hColonNone
7338
364263862022
GIFDVLKNLAKGVITSLAS
Ocellatin-3N19LinearLNoneAmidationFreeHost DefenseLeptodactylus nesiotusA-549Lung CancerCellTiter-Glo assayLC50 = 35 ± 1 μM24-hLungNone
7339
364263862022
GIFDVLKNLAKGVITSLAS
Ocellatin-3N19LinearLNoneAmidationFreeHost DefenseLeptodactylus nesiotusMDA-MB-231Breast CancerCellTiter-Glo assayLC50 = 51 ± 16 μM24-hBreastNone
7336
364263862022
GIFDVLKNLAKGVITSLKS
[A18K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NMDA-MB-231Breast CancerCellTiter-Glo assayLC50 = 69 ± 18 μM24-hBreastNone
7337
364263862022
GIFDVLKNLAKGVITSLKS
[A18K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NHT-29Colorectal CancerCellTiter-Glo assayLC50 = 59 ± 4 μM24-hColonNone
7335
364263862022
GIFDVLKNLAKGVITSLKS
[A18K]OCN-3N19LinearLNoneAmidationFreeHost DefenseSynthetic; Derivative of ocellatin-3NA-549Lung CancerCellTiter-Glo assayLC50 = 30 ± 1 μM24-hLungNone
7334
352092152022
NGVQPKYRWWRWWRRWW
RT217LinearLNoneAmidationFreeAntimicrobialCrocodylus siamensisCaCo-2Colon CancerMTT assayIC50 = 29.74 μM24-hColonNone
7333
356283122022
MKEDSNILDKTAKMTKQNKALLFTAGGAAAFMAGYYYYHCNYRNPAPKKSGSTTSQDKTDAQAVQSIPSPSGNKGKESKDPKVKHHHHHH
rScyreprocin90LinearLNoneHis-TagFreeAntimicrobialRecombinant product of ScyreprocinHeLaCervical cancerMTS assayIC50 = 3.34 x 104 µM24-hCervixNone
7332
356283122022
MKEDSNILDKTAKMTKQNKALLFTAGGAAAFMAGYYYYHCNYRNPAPKKSGSTTSQDKTDAQAVQSIPSPSGNKGKESKDPKVKHHHHHH
rScyreprocin90LinearLNoneHis-TagFreeAntimicrobialRecombinant product of ScyreprocinDU-145Prostate cancerMTS assayIC50 = 1158.30 µM24-hProstateNone
7331
356283122022
MKEDSNILDKTAKMTKQNKALLFTAGGAAAFMAGYYYYHCNYRNPAPKKSGSTTSQDKTDAQAVQSIPSPSGNKGKESKDPKVKHHHHHH
rScyreprocin90LinearLNoneHis-TagFreeAntimicrobialRecombinant product of ScyreprocinT-24Urinary Bladder CancerMTS assayIC50 = 1.94 x 105 µM24-hBladderNone
7330
356283122022
MKEDSNILDKTAKMTKQNKALLFTAGGAAAFMAGYYYYHCNYRNPAPKKSGSTTSQDKTDAQAVQSIPSPSGNKGKESKDPKVKHHHHHH
rScyreprocin90LinearLNoneHis-TagFreeAntimicrobialRecombinant product of ScyreprocinHepG-2Liver CancerMTS assayIC50 = 441.01 µM24-hLiverNone
7329
356283122022
MKEDSNILDKTAKMTKQNKALLFTAGGAAAFMAGYYYYHCNYRNPAPKKSGSTTSQDKTDAQAVQSIPSPSGNKGKESKDPKVKHHHHHH
rScyreprocin90LinearLNoneHis-TagFreeAntimicrobialRecombinant product of ScyreprocinH-460Lung CancerMTS assayIC50 = 6.27 µM72-hLungNone
7327
349992272022
SKVWRHWRRFWHRAHRLH
LA-C1b18LinearLLauric acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticHeLaCervical CancerNot AvailableNot AvailableNot AvailableCervixNone
7328
349992272022
SKVWRHWRRFWHRAHRLH
LA-C1b18LinearLLauric acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticA-375Skin CancerNot AvailableNot AvailableNot AvailableSkinNone
7324
349992272022
SKVWRHWRRFWHRAHRLH
OA-C1b18LinearLOctanoic acid acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticHeLaCervical CancerNot AvailableNot AvailableNot AvailableCervixNone
7325
349992272022
SKVWRHWRRFWHRAHRLH
OA-C1b18LinearLOctanoic acid acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticA-375Skin CancerNot AvailableNot AvailableNot AvailableSkinNone
7326
349992272022
SKVWRHWRRFWHRAHRLH
LA-C1b18LinearLLauric acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticMCF-7Breast CancerNot AvailableNot AvailableNot AvailableBreastNone
7322
349992272022
SKVWRHWRRFWHRAHRLH
PA-C1b18LinearLPalmitic acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticA-375Skin CancerNot AvailableNot AvailableNot AvailableSkinNone
7323
349992272022
SKVWRHWRRFWHRAHRLH
OA-C1b18LinearLOctanoic acid acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticMCF-7Breast CancerNot AvailableNot AvailableNot AvailableBreastNone
7320
349992272022
SKVWRHWRRFWHRAHRLH
PA-C1b18LinearLPalmitic acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticMCF-7Breast CancerNot AvailableNot AvailableNot AvailableBreastNone
7321
349992272022
SKVWRHWRRFWHRAHRLH
PA-C1b18LinearLPalmitic acid conjugated to the 17th Lys-residueAmidationFreeAnticancerSyntheticHeLaCervical CancerNot AvailableNot AvailableNot AvailableCervixNone
7319
349992272022
SKVWRHWRRFWHRAHRLH
Chensinin-1b18LinearLNoneAmidationFreeAntmicrobial and AnticancerSyntheticA-375Skin CancerNot AvailableNot AvailableNot AvailableSkinNone
7318
349992272022
SKVWRHWRRFWHRAHRLH
Chensinin-1b18LinearLNoneAmidationFreeAntmicrobial and AnticancerSyntheticHeLaCervical CancerNot AvailableNot AvailableNot AvailableCervixNone
7317
349992272022
SKVWRHWRRFWHRAHRLH
Chensinin-1b18LinearLNoneAmidationFreeAntmicrobial and AnticancerSyntheticMCF-7Breast CancerNot AvailableNot AvailableNot AvailableBreastNone
7316
365552352022
FAKKLAKLKKKLAKLALAL
AC-P1919LinearLNoneFreeFreeAnticancerSyntheticH-460Lung CancerWST-8 assayIC50 = 49.08 µM24-hLungNone
7314
364835992022
EQQQQQQPQNRRFRE
Q715LinearLNoneFreeFreeAnticancerPisum sativumHEC-1-AEndometrial CancerMTT assayIC50 = 129.82 ± 7.53 μM48-hEndometriumNone
7315
365552352022
FAKKLAKLKKKLAKLALAL
AC-P1919LinearLNoneFreeFreeAnticancerSyntheticA-549Lung CancerWST-8 assayIC50 = 52.14 µM24-hLungNone
7313
None2022
RRGKGGRRVTMSF
RF1313LinearLNoneFreeFreeAnticancerVSP26B of C. striatusHEp-2Larynx CancerMTT assayIC50 = 49.65 µM24-hLarynxNone
7312
352467582022
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin ZP34CyclicLNoneCyclizedCyclizedAntimicrobialLactococcus lactisH-1299Lung CancerMTT assayIC50 = 137.3 ± 9.1 μM48-hLungNone
7311
352467582022
ITSISLCTPGCKTGALMGCNMKTATCNCSIHVSK
Nisin ZP34CyclicLNoneCyclizedCyclizedAntimicrobialLactococcus lactisA-549Lung CancerMTT assayIC50 = 132.4 ± 6.4 μM48-hLungNone
7310
365552352022
FAKKLAKLKKKLAKLAKKR
AC-P19M19LinearLNoneFreeFreeAnticancer and AntimicrobialSynthetic analogue of AC-P19H-460Lung CancerWST-8 assayIC50 = 6.29 µM24-hLungNone
7309
365552352022
FAKKLAKLKKKLAKLAKKR
AC-P19M19LinearLNoneFreeFreeAnticancer and AntimicrobialSynthetic analogue of AC-P19A-549Lung CancerWST-8 assayIC50 = 9.84 µM24-hLungNone
7308
361836732022
EARPALLTSRLRFIPK
GV100116LinearLNoneFreeFreeAnticancerHuman telomerase reverse transcriptase (hTERT)A-549Lung CancerCell Viability assayGraph Fig 2A24-hLungNone
7307
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticHCC-827Lung AdenocarcinomaMTT assayIC50 between 4.0 and 5.5 μM72-hLungNone
7306
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticH-1975Non Small Cell Lung Cancer (NSCLC)MTT assayIC50 between 4.0 and 5.5 μM72-hLungNone
7305
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticH-358Non Small Cell Lung Cancer (NSCLC)MTT assayIC50 = 4.00 ± 0.20 μM72-hLungNone
7304
357641962022
kklalalakkwlalakklalalakk
D-LAK-120-A25LinearDNoneAmidationFreeAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 5.55 ± 0.13 μM72-hLungNone
7303
362879852022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusHepG-2Liver CancerMTT assayIC50 = 5.524 µM24-hLiverNone
7302
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusH-460Lung CancerMTT assayIC50 = 7.07 ± 0.81 µM24-hLungNone
7301
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusPC-9Lung CancerMTT assayIC50 = 6.34 ± 0.53 µM24-hLungNone
7300
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusH-3122Lung CancerMTT assayIC50 = 4.64 ± 0.18 µM24-hLungNone
7299
358781762022
IWSFLIKAATKLLPSLFGGGKKDS
SMP2424LinearLNoneFreeFreeAntimicrobialEgyptian scorpion Scorpio maurus palmatusA-549Lung CancerMTT assayIC50 = 4.06 ± 0.60 µM24-hLungNone
7296
367135382022
KKWWKKW-Dip-K
NTP-2179LinearLDip = β-diphenylalanineAmidationrhodamine B - GABAAnticancerSyntheticHuh-7Liver CancerMTT assayIC50 = 40.1 ± 1.3 µM4-hLiverNone
7297
367135382022
KKWWKKW-Dip-K
NTP-2179LinearLDip = β-diphenylalanineAmidationrhodamine B - GABAAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 48.8 ± 0.7 µM4-hLiverNone
7298
367135382022
KKWWKKW-Dip-K
NTP-2179LinearLDip = β-diphenylalanineAmidationrhodamine B - GABAAnticancerSyntheticHep3BLiver CancerMTT assayIC50 = 45.7 ± 1.7 µM4-hLiverNone
7293
367135382022
KKWWKKW-Dip-K
NTP-2179LinearLDip = β-diphenylalanineAmidationrhodamine B - GABAAnticancerSyntheticHepa 1-6Liver CancerMTT assayIC50 = 21.6 ± 1.0 µM4-hLiverNone
7294
367135382022
KKWWKKW-Dip-K
NTP-2179LinearLDip = β-diphenylalanineAmidationrhodamine B - GABAAnticancerSyntheticPLC/PRF/5Liver CancerMTT assayIC50 = 14.6 ± 1.1 µM4-hLiverNone
7295
367135382022
KKWWKKW-Dip-K
NTP-2179LinearLDip = β-diphenylalanineAmidationrhodamine B - GABAAnticancerSyntheticHCCLM-3Liver CancerMTT assayIC50 = 22.4 ± 5.1 µM4-hLiverNone
7292
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticT98GBrain TumorAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hBrainNone
7291
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticA-549Lung CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hLungNone
7290
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticDU-145Prostate CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hProstateNone
7289
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticA-375Skin CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hSkinNone
7288
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hBreastNone
7287
361213852022
vaeareelerlearlgqargelkkwkmrrnqfwlklqr
ST10138LinearDNoneFreeFreeAnticancerSyntheticU-251Brain TumorAnnexin V/ PI staining assaymean EC50 value of 2.1 ± 0.4 μmol/L48-hBrainNone
7276
356018272022
IWLTALKFLGKNLGKLAKQQLAKL
LyeTx-I-b24LinearLNoneAmidatedAcetylationAntimicrobialSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 2.47 µM48-hBreastNone
7275
350138812022
KLKNFAKGVAQSLLNKASCKLSGQC
Brevinin-2R25LinearLNoneFreeFreeAntimicrobialRana ridibundaHeLaCervical CancerMTT assayIC50 = 131.5 μg/ml24-hCervixNone
7273
361865622022
EEEEY
C16-E4Y5LinearLNoneFreePalmitoylAnticancerSyntheticMCF-7Breast CancerWST-8 assay50 % cell viability at 0.05 wt %24-hBreastNone
7274
364658442022
GVKFAKRFWRFAKKAFKRFEK
HAZ21LinearLNoneFreeFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 5.44 μM4-hLungNone
7270
361865622022
EEEEY
C16-E4Y5LinearLNoneFreePalmitoylAnticancerSyntheticA-431Skin CancerWST-8 assay10 % cell viability at 0.05 wt %24-hSkinNone
7271
361865622022
EEEEY
C16-E4Y5LinearLNoneFreePalmitoylAnticancerSyntheticHeLaCervical CancerWST-8 assay60% cell viability at 0.05 wt %24-hCervixNone
7272
361865622022
EEEEY
C16-E4Y5LinearLNoneFreePalmitoylAnticancerSyntheticHepG-2Liver CancerWST-8 assay50 % cell viability at 0.05 wt %24-hLiverNone
7269
356316752022
FAKLLAKLARRLL
HB43-mut313LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerAlamarBlue assay75% cell viability at 20 μMNot AvailableBreastNone
7268
356316752022
FAKLLAKLARRLL
HB43-mut313LinearLNoneAmidationFreeAnticancerSyntheticHT-29Colon CancerAlamarBlue assayIC50 = 9 ± 1 μM24-hColonNone
7266
356316752022
FAKLLAKLARRLL
HB43-mut313LinearLNoneAmidationFreeAnticancerSyntheticSW-480Colon CancerAlamarBlue assayIC50 = 8 ± 1 μM24-hColonNone
7267
356316752022
FAKLLAKLARRLL
HB43-mut313LinearLNoneAmidationFreeAnticancerSyntheticSW-620Colon CancerAlamarBlue assayIC50 = 9 ± 1 μM24-hColonNone
7265
356316752022
FAKLLAKLAKLLK
HB43-mut213LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerAlamarBlue assay80% cell viability at 20 μMNot AvailableBreastNone
7263
356316752022
FAKLLAKLAKLLK
HB43-mut213LinearLNoneAmidationFreeAnticancerSyntheticSW-620Colon CancerAlamarBlue assayIC50 = 40 ± 3 μM24-hColonNone
7264
356316752022
FAKLLAKLAKLLK
HB43-mut213LinearLNoneAmidationFreeAnticancerSyntheticHT-29Colon CancerAlamarBlue assayIC50 = 50 ± 3 μM24-hColonNone
7262
356316752022
FAKLLAKLAKLLK
HB43-mut213LinearLNoneAmidationFreeAnticancerSyntheticSW-480Colon CancerAlamarBlue assayIC50 = 34 ± 2 μM24-hColonNone
7261
356316752022
FAKLLAKLAKKLL
HB4313LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerAlamarBlue assay50% cell viability at 20 μMNot AvailableBreastNone
7259
356316752022
FAKLLAKLAKKLL
HB4313LinearLNoneAmidationFreeAnticancerSyntheticSW-620Colon CancerAlamarBlue assayIC50 = 10 ± 1 μM24-hColonNone
7260
356316752022
FAKLLAKLAKKLL
HB4313LinearLNoneAmidationFreeAnticancerSyntheticHT-29Colon CancerAlamarBlue assayIC50 = 11 ± 1 μM24-hColonNone
7258
356316752022
FAKLLAKLAKKLL
HB4313LinearLNoneAmidationFreeAnticancerSyntheticSW-480Colon CancerAlamarBlue assayIC50 = 12 ± 4 μM24-hColonNone
7256
363601202022
GPLGAGP
HTDT-6-2-3-27LinearLNoneFreeFreeAnticancerEnteromorpha proliferaHepG-2Liver CancerCCK-8 assayIC50 = 1.2564 ± 0.0548 mg/mL48-hLiverNone
7257
363601202022
GPLGAGP
HTDT-6-2-3-27LinearLNoneFreeFreeAnticancerEnteromorpha proliferaA-549Lung CancerCCK-8 assayIC50 = 0.9867 ± 0.0857 mg/mL48-hLungNone
7255
363601202022
GPLGAGP
HTDT-6-2-3-27LinearLNoneFreeFreeAnticancerEnteromorpha proliferaNCI-H-460Lung CancerCCK-8 assayIC50 = 0.3686 ± 0.0935 mg/mL48-hLungNone
7254
357741632022
flgvlallgylavrpflpkkkqqk
D-NAF-124LinearDNoneFreeFreeAnticancerNAF-1/CISD2MDA-MB-231Breast CancerNot AvailableIC50 = 12.8 ± 0.2 μMNABreastNone
7253
357741632022
FLGVLALLGYLAVRPFLPKKKQQK
NAF-124LinearLNoneFreeFreeAnticancerNAF-1/CISD2MDA-MB-231Breast CancerNot AvailableIC50 = 18.3 ± 0.4 μMNABreastNone
7252
350942082022
HARIKpTFRRlKWKYKGKFW
CIGB-55220LinearMixNoneFreeAcetylationAntitumorSyntheticA-549Lung CancerSulforhodamine B assayIC50 = 44.6 μM48-hLungNone
7251
350942082022
HARIKpTFRRlKWKYKGKFW
CIGB-55220LinearMixNoneFreeAcetylationAntitumorSyntheticNCI-H-460Lung CancerSulforhodamine B assayIC50 = 287.9 μM48-hLungNone
7250
366725512022
GRKKRRQRRRPPQ-X-CWMSPRHLGTC
CIGB-30025CyclicLX = Beta- AlanineFreeBiotinylatedAnticancerSyntheticNCI-H-460Lung CancerCrystal Violet assayIC50 = 30 ± 5.3 µM48-hLungNone
7249
357456432022
FKWQFEMLIMKIAKTSGFMFYSSY
BmPLA224LinearLNoneFreeFreeAnticancerphospholipase A2 isoform from B. moojeni venomRDRhabdomyosarcomaMTT assay60% reduction in cell viability24-hMuscleNone
7248
357456432022
FKWQFEMLIMKIAKTSGFMFYSSY
BmPLA224LinearLNoneFreeFreeAnticancerphospholipase A2 isoform from B. moojeni venomCaCo-2Colorectal CancerMTT assayIC50 = 0.6 µM24-hColonNone
7246
361744942022
KIIIKIKKKIKIIIK
At1215LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 14.0 µMNALungNone
7247
361744942022
KIIIKIKKKIKIIIK
At1215LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 13.4 µMNALiverNone
7245
361744942022
IIIKKIKKKIKKIII
At1115LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 7.6 µMNALiverNone
7244
361744942022
IIIKKIKKKIKKIII
At1115LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 7.9 µMNALungNone
7243
361744942022
IKKIIKIIKKIIKKI
At1015LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 3.2 µMNALiverNone
7242
361744942022
IKKIIKIIKKIIKKI
At1015LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 4.4 µMNALungNone
7241
361744942022
KVVKKVKKKVKKVVK
At915LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 51.7 µMNALiverNone
7240
361744942022
KVVKKVKKKVKKVVK
At915LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 100 µMNALungNone
7239
361744942022
KLLKKLKKKLKKLLK
At815LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 8.9 µMNALiverNone
7238
361744942022
KLLKKLKKKLKKLLK
At815LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 13.4 µMNALungNone
7237
361744942022
KIIKKIKKKIKKIIK
At715LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 8.8 µMNALiverNone
7236
361744942022
KIIKKIKKKIKKIIK
At715LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 10.3 µMNALungNone
7235
361744942022
KVVKKVVKVVKKVVK
At615LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 70.8 µMNALiverNone
7234
361744942022
KVVKKVVKVVKKVVK
At615LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 > 100 µMNALungNone
7232
361744942022
KIIKKIIKIIKKIIK
At515LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 3.6 µMNALungNone
7233
361744942022
KIIKKIIKIIKKIIK
At515LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 1.5 µMNALiverNone
7231
361744942022
KLLKKLLKLLKKLLK
At415LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 2.5 µMNALiverNone
7230
361744942022
KLLKKLLKLLKKLLK
At415LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 7.2 µMNALungNone
7228
361744942022
KLLKKVVKLFKKLLK
Ponericin-W1 (11-25) [P4K; S5K; G8K; K13L; Q15K], At315LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 4.3 µMNALungNone
7229
361744942022
KLLKKVVKLFKKLLK
Ponericin-W1 (11-25) [P4K; S5K; G8K; K13L; Q15K], At315LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 = 2.2 µMNALiverNone
7227
361744942022
KLLKKVVKLFKKKKK
Ponericin-W1 (11-25) [P4K; S5K; G8K; Q15K], At215LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 >100 µMNALiverNone
7226
361744942022
KLLKKVVKLFKKKKK
Ponericin-W1 (11-25) [P4K; S5K; G8K; Q15K], At215LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 >100 µMNALungNone
7224
361744942022
KLLPSVVGLFKKKKQ
Ponericin-W1 (11-25), At115LinearLNoneAmidationAcetylationAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 > 100 µMNALungNone
7225
361744942022
KLLPSVVGLFKKKKQ
Ponericin-W1 (11-25), At115LinearLNoneAmidationAcetylationAntimicrobialSyntheticHepG-2Liver CancerMTT assayIC50 >100 µMNALiverNone
7223
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2MCF-7Breast CancerMTT assayEC50 = 0.724 ± 0.340 mol/L × 10-324-hBreastNone
7222
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2A-2058Skin CancerMTT assayEC50 = 0.744 ± 0.208 mol/L × 10-324-hSkinNone
7221
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2U-87Brain TumorMTT assayEC50 = 0.427 ± 0.053 mol/L × 10-324-hBrainNone
7220
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2HeLaCervical CancerMTT assayEC50 = 0.525 ± 0.160 mol/L × 10-324-hCervixNone
7219
351905862022
MADSERLSAPGCWAACTNFSRTRK
RB424LinearLNoneAmidationFreeAnticancerDerived from protein PLP2B16-F10-Nex 2Skin CancerMTT assayEC50 = 0.263 ± 0.585 mol/L × 10-324-hSkinNone
7218
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinWiDrColon CancerMTT assayIC50 = 197.3 μM24-hColonNone
7217
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinAGSStomach CancerMTT assayIC50 = 29.8 μM24-hStomachNone
7216
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinA-549Lung CancerMTT assayIC50 = 42.1 μM24-hLungNone
7215
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinHep3BLiver CancerMTT assayIC50 = 77.5 μM24-hLiverNone
7214
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinHuh-7Liver CancerMTT assayIC50 = 60 μM24-hLiverNone
7213
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple-a25LinearLNoneAmidationFreeAntimicrobialC-terminal-amidated derivative of PleurocidinJ5Liver CancerMTT assayIC50 = 11 μM24-hLiverNone
7212
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusAGSStomach CancerMTT assayIC50 = 186.5 μM24-hStomachNone
7211
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusA-549Lung CancerMTT assayIC50 = 300.8 μM24-hLungNone
7210
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusHep3BLiver CancerMTT assayIC50 = 340.9 μM24-hLiverNone
7209
360055212022
GWGSFFKKAAHVGKHVGKAALTHYL
Ple25LinearLNoneFreeFreeAntimicrobialPleuronectes americanusJ5Liver CancerMTT assayIC50 = 54.9 μM24-hLiverNone
7208
346792572022
WRRRYRRWRRRRRWRRRPRR
vCPP231920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusSK-BR-3Breast CancerMTT assayIC50 = 14.0 ± 1.0 μM24-hBreastNone
7207
346792572022
WRRRYRRWRRRRRWRRRPRR
vCPP231920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-474Breast CancerMTT assayIC50 = 15.7 ± 1.5 μM24-hBreastNone
7206
346792572022
WRRRYRRWRRRRRWRRRPRR
vCPP231920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-20Breast CancerMTT assayIC50 = 4.2 ± 2.2 μM24-hBreastNone
7205
346792572022
WRRRYRRWRRRRRWRRRPRR
vCPP231920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusMDA-MB-231Breast CancerMTT assayIC50 = 4.5 ± 0.1 μM24-hBreastNone
7204
346792572022
RRLTLRQLLGLGSRRRRRSR
vCPP076920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusSK-BR-3Breast CancerMTT assayIC50 = 21.1 ± 2.0 μM24-hBreastNone
7203
346792572022
RRLTLRQLLGLGSRRRRRSR
vCPP076920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-474Breast CancerMTT assayIC50 = 37.5 ± 1.7 μM24-hBreastNone
7202
346792572022
RRLTLRQLLGLGSRRRRRSR
vCPP076920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-20Breast CancerMTT assayIC50 = 3.5 ± 1.5 μM24-hBreastNone
7201
346792572022
RRLTLRQLLGLGSRRRRRSR
vCPP076920LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusMDA-MB-231Breast CancerMTT assayIC50 = 9.0 ± 0.1 μM24-hBreastNone
7200
346792572022
RPRRRATTRRRITTGTRRRR
vCPP066720LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusSK-BR-3Breast CancerMTT assayIC50 = 71.2 ± 1.1 μM24-hBreastNone
7199
346792572022
RPRRRATTRRRITTGTRRRR
vCPP066720LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-474Breast CancerMTT assayIC50 = 92.8 ± 1.1 μM24-hBreastNone
7198
346792572022
RPRRRATTRRRITTGTRRRR
vCPP066720LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-20Breast CancerMTT assayIC50 = 88.8 ± 1.0 μM24-hBreastNone
7197
346792572022
KKRYKKKYKAYKPYKKKKKF
vCPP027520LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusSK-BR-3Breast CancerMTT assayIC50 = 34.0 ± 1.0 μM24-hBreastNone
7196
346792572022
KKRYKKKYKAYKPYKKKKKF
vCPP027520LinearLNoneAmidationFreeAnticancer and Cell PenetratingCapsid protein of the Torque teno douroucouli virusBT-20Breast CancerMTT assayIC50 = 44.8 ± 1.1 μM24-hBreastNone
7195
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticSNB-19Brain TumorCCK-8 assayIC50 = 12.0 ± 0.6 μM72-hBrainNone
7194
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticSF-268Brain TumorCCK-8 assayIC50 = 4.8 ± 0.1 μM72-hBrainNone
7193
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-138Brain TumorCCK-8 assayIC50 = 7.5 ± 0.3 μM72-hBrainNone
7192
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticLN229Brain TumorCCK-8 assayIC50 = 4.7 ± 0.2 μM72-hBrainNone
7191
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticSW-1783Brain TumorCCK-8 assayIC50 = 4.8 ± 0.2 μM72-hBrainNone
7190
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticD54Brain TumorCCK-8 assayIC50 = 8.4 ± 0.1 μM72-hBrainNone
7189
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-118Brain TumorCCK-8 assayIC50 = 6.8 ± 0.2 μM72-hBrainNone
7188
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-373Brain TumorCCK-8 assayIC50 = 5.0 ± 0.2 μM72-hBrainNone
7187
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticT98GBrain TumorCCK-8 assayIC50 = 7.1 ± 0.2 μM96-hBrainNone
7186
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticA-172Brain TumorCCK-8 assayIC50 = 6.4 ± 0.4 μM96-hBrainNone
7185
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU-251Brain TumorCCK-8 assayIC50 = 4.9 ± 0.3 μM96-hBrainNone
7184
350534552022
MDRWLVKWKKKRKIRRRRRRRRRRR
ATX-10125LinearLNoneFreeAcetylationAntitumor and Cell PenetratingSyntheticU87-MGBrain TumorCCK-8 assayIC50 = 4.3 ± 0.3 μM96-hBrainNone
7183
356606292022
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationFreeAntimicrobialskin mucous secretions of winter flounderSCC-9Oral CancerCCK-8 assayIC50 = 45 μg/ml24-hTongueNone
7181
345091202022
LC-Propargyl-GIIKKIIKKIIKKII
GI-1517LinearLNoneAmidationLC-PropargylglycineAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 16.6 ± 0.8 µM72-hCervixNone
7182
356606292022
GRRKRKWLRRIGKGVKIIGGAALDHL
NRC-0326LinearLNoneAmidationFreeAntimicrobialskin mucous secretions of winter flounderCAL-27Oral CancerCCK-8 assayIC50 = 45 μg/ml24-hTongueNone
7180
345091202022
LC-Propargyl-GIIKKIIKKIIKKII
GI-1517LinearLNoneAmidationLC-PropargylglycineAnticancerSyntheticHCT-116Colorectal CancerMTT assayIC50 = 13.6 ± 0.2 µM72-hColonNone
7178
345091202022
CIIKKIIKKIIKKII
CI-1515LinearLNoneAmidationFreeAnticancerSyntheticHCT-116Colorectal CancerMTT assayIC50 = 7.7 ± 0.2 µM72-hColonNone
7179
345091202022
CIIKKIIKKIIKKII
CI-1515LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 2.7 ± 0.5 µM72-hCervixNone
7177
345091202022
CLLRRLLRRLLRR
LR1313LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 26.7 ± 1.3 µM72-hCervixNone
7176
345091202022
CLLRRLLRRLLRR
LR1313LinearLNoneAmidationFreeAnticancerSyntheticHCT-116Colorectal CancerMTT assayIC50 = 15.6 ± 1.0 µM72-hColonNone
7174
345091202022
CIIRRIIRRIIRR
IR1313LinearLNoneAmidationFreeAnticancerSyntheticHCT-116Colorectal CancerMTT assayIC50 > 100 µM72-hColonNone
7175
345091202022
CIIRRIIRRIIRR
IR1313LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 > 100 µM72-hCervixNone
7173
345091202022
CLLKKLLKKLLKK
LK1313LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 83 ± 9 µM72-hCervixNone
7171
345091202022
CIIKKIIKKIIKK
IK1313LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 47±5 µM72-hCervixNone
7172
345091202022
CLLKKLLKKLLKK
LK1313LinearLNoneAmidationFreeAnticancerSyntheticHCT-116Colorectal CancerMTT assayIC50 = 23 ± 2 µM72-hColonNone
7169
353234572022
lPlPl
Z-85CyclicMixNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 15.88 ± 1.42 µg/mlNALungNone
7170
345091202022
CIIKKIIKKIIKK
IK1313LinearLNoneAmidationFreeAnticancerSyntheticHCT-116Colorectal CancerMTT assayIC50 = 29 ± 6 µM72-hColonNone
7167
353234572022
lPlPl
Z-85CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 20.16 ± 2.24 µg/mlNABreastNone
7168
353234572022
lPlPl
Z-85CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 7.97 ± 0.61 µg/mlNACervixNone
7164
353234572022
LPlPl
Z-75CyclicMixNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 9.97 ± 1.00 µg/mlNALungNone
7165
353234572022
lPlPl
Z-85CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 7.82 ± 1.18 µg/mlNABreastNone
7166
353234572022
lPlPl
Z-85CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 9.00 ± 0.83 µg/mlNALiverNone
7162
353234572022
LPlPl
Z-75CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 16.52 ± 1.7 µg/mlNABreastNone
7163
353234572022
LPlPl
Z-75CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 18.21 ± 1.35 µg/mlNACervixNone
7160
353234572022
LPlPl
Z-75CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 13.28 ± 3.28 µg/mlNABreastNone
7161
353234572022
LPlPl
Z-75CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 13.85 ± 1.99 µg/mlNALiverNone
7157
353234572022
lPLPl
Z-65CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 4.59 ± 0.27 µg/mlNABreastNone
7158
353234572022
lPLPl
Z-65CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 5.69 ± 0.37 µg/mlNACervixNone
7159
353234572022
lPLPl
Z-65CyclicMixNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 5.96 ± 0.41 µg/mlNALungNone
7155
353234572022
lPLPl
Z-65CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 1.65 ± 0.3 µg/mlNABreastNone
7156
353234572022
lPLPl
Z-65CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 2.91 ± 0.17 µg/mlNALiverNone
7153
353234572022
LPLPl
Z-55CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 12.12 ± 0.95 µg/mlNACervixNone
7154
353234572022
LPLPl
Z-55CyclicMixNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 9.5 ± 1.13 µg/mlNALungNone
7150
353234572022
LPlPL
Z-45CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 13.43 ± 1.96 µg/mlNABreastNone
7151
353234572022
LPLPl
Z-55CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 14.98 ± 0.93 µg/mlNALiverNone
7152
353234572022
LPLPl
Z-55CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 8.48 ± 1.12 µg/mlNABreastNone
7148
353234572022
LPlPL
Z-45CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 7.38 ± 0.83 µg/mlNACervixNone
7149
353234572022
LPlPL
Z-45CyclicMixNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 9.85 ± 0.95 µg/mlNALungNone
7145
353234572022
lPLPL
Z-35CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 4.88 ± 0.58 µg/mlNABreastNone
7146
353234572022
LPlPL
Z-45CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 15.23 ± 1.14 µg/mlNALiverNone
7147
353234572022
LPlPL
Z-45CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 22.09 ± 1.12 µg/mlNABreastNone
7143
353234572022
lPLPL
Z-35CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 5.57 ± 0.45 µg/mlNACervixNone
7144
353234572022
lPLPL
Z-35CyclicMixNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 6.43 ± 0.43 µg/mlNALungNone
7141
353234572022
lPLPL
Z-35CyclicMixNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 5.05 ± 0.45 µg/mlNALiverNone
7142
353234572022
lPLPL
Z-35CyclicMixNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 6.34 ± 0.6 µg/mlNABreastNone
7138
353234572022
LPLPL
Z-25CyclicLNoneCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 14.5 ± 0.36 µg/mlNACervixNone
7139
353234572022
LPLPL
Z-25CyclicLNoneCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 7.97 ± 2.06 µg/mlNALungNone
7140
353234572022
LPLPL
Z-25CyclicLNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 2.25 ± 0.42 µg/mlNABreastNone
7136
353234572022
LPLPL
Z-25CyclicLNoneCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 11.95 ± 0.64 µg/mlNALiverNone
7137
353234572022
LPLPL
Z-25CyclicLNoneCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 14.45 ± 1.1 µg/mlNABreastNone
7134
353234572022
L(N-Me-L)LPL
Z-15CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerSyntheticA-549Lung CancerMTT assayIC50 = 4.92 ± 0.84 µg/mlNALungNone
7135
353234572022
LPLPL
Z-25CyclicLNoneCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 4.68 ± 1.22 µg/mlNABreastNone
7132
353234572022
L(N-Me-L)LPL
Z-15CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 17.81 ± 0.6 µg/mlNABreastNone
7133
353234572022
L(N-Me-L)LPL
Z-15CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 11.56 ± 0.65 µg/mlNACervixNone
7130
353234572022
L(N-Me-L)LPL
Z-15CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 5.85 ± 1.28 µg/mlNABreastNone
7131
353234572022
L(N-Me-L)LPL
Z-15CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerSyntheticHepG-2Liver CancerMTT assayIC50 = 7.57 ± 0.17 µg/mlNALiverNone
7128
353234572022
(N-Me-L)L(N-Me-L)LL
Galaxamide5CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerGalaxaura filamentosaMDA-MB-231Breast CancerMTT assayIC50 = 8.73 ± 0.29 µg/mlNABreastNone
7129
353234572022
(N-Me-L)L(N-Me-L)LL
Galaxamide5CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerGalaxaura filamentosaA-549Lung CancerMTT assayIC50 = 6.99 ± 0.63 µg/mlNALungNone
7126
353234572022
(N-Me-L)L(N-Me-L)LL
Galaxamide5CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerGalaxaura filamentosaMCF-7Breast CancerMTT assayIC50 = 11.33 ± 2.95 µg/mlNABreastNone
7127
353234572022
(N-Me-L)L(N-Me-L)LL
Galaxamide5CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerGalaxaura filamentosaHeLaCervical CancerMTT assayIC50 = 8.53 ± 0.73 µg/mlNACervixNone
7125
353234572022
(N-Me-L)L(N-Me-L)LL
Galaxamide5CyclicLN-Me-L = N-methyl-LysineCyclizedCyclizedAnticancerGalaxaura filamentosaHepG-2Liver CancerMTT assayIC50 = 5.20 ± 0.52 µg/mlNALiverNone
7123
357408842022
FLPLiiGALSSLLPKiF
Temporin-PKE-3i17LinearMixNoneAmidationFreeAntimicrobialSyntheticHCT-116Colorectal CancerMTT assayIC50 = 72.06 μM24-hColonNone
7124
357408842022
FLPLiiGALSSLLPKiF
Temporin-PKE-3i17LinearMixNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 71.18 μM24-hLungNone
7122
357408842022
FLPLiiGALSSLLPKiF
Temporin-PKE-3i17LinearMixNoneAmidationFreeAntimicrobialSyntheticH-838Lung CancerMTT assayIC50 = 193.4 μM24-hLungNone
7121
357408842022
FLPLiiGALSSLLPKiF
Temporin-PKE-3i17LinearMixNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 167 μM24-hProstateNone
7120
357408842022
FLPLiiGALSSLLPKiF
Temporin-PKE-3i17LinearMixNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 120.6 μM24-hBrainNone
7119
357408842022
FLPLIIGALSSLLPKiF
Temporin-PKE-i17LinearMixNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 2.94 μM24-hLungNone
7117
357408842022
FLPLIIGALSSLLPKiF
Temporin-PKE-i17LinearMixNoneAmidationFreeAntimicrobialSyntheticH-838Lung CancerMTT assayIC50 = 5.28 μM24-hLungNone
7118
357408842022
FLPLIIGALSSLLPKiF
Temporin-PKE-i17LinearMixNoneAmidationFreeAntimicrobialSyntheticHCT-116Colorectal CancerMTT assayIC50 = 3.07 μM24-hColonNone
7116
357408842022
FLPLIIGALSSLLPKiF
Temporin-PKE-i17LinearMixNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 3.35 μM24-hProstateNone
7115
357408842022
FLPLIIGALSSLLPKiF
Temporin-PKE-i17LinearMixNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 4.46 μM24-hBrainNone
7114
357408842022
FLPKIIGKLSSKLPKIF
Temporin-PKE-4K17LinearLNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 27.76 μM24-hLungNone
7113
357408842022
FLPKIIGKLSSKLPKIF
Temporin-PKE-4K17LinearLNoneAmidationFreeAntimicrobialSyntheticHCT-116Colorectal CancerMTT assayIC50 = 99.36 μM24-hColonNone
7111
357408842022
FLPKIIGKLSSKLPKIF
Temporin-PKE-4K17LinearLNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 49.50 μM24-hProstateNone
7112
357408842022
FLPKIIGKLSSKLPKIF
Temporin-PKE-4K17LinearLNoneAmidationFreeAntimicrobialSyntheticH-838Lung CancerMTT assayIC50 = 35.28 μM24-hLungNone
7110
357408842022
FLPKIIGKLSSKLPKIF
Temporin-PKE-4K17LinearLNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 85.52 μM24-hBrainNone
7109
357408842022
FLPKIIGKLSSLLPKIF
Temporin-PKE-3K17LinearLNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 3.29 μM24-hLungNone
7108
357408842022
FLPKIIGKLSSLLPKIF
Temporin-PKE-3K17LinearLNoneAmidationFreeAntimicrobialSyntheticHCT-116Colorectal CancerMTT assayIC50 = 0.38 μM24-hColonNone
7106
357408842022
FLPKIIGKLSSLLPKIF
Temporin-PKE-3K17LinearLNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 3.01 μM24-hProstateNone
7107
357408842022
FLPKIIGKLSSLLPKIF
Temporin-PKE-3K17LinearLNoneAmidationFreeAntimicrobialSyntheticH-838Lung CancerMTT assayIC50 = 0.51 μM24-hLungNone
7105
357408842022
FLPKIIGKLSSLLPKIF
Temporin-PKE-3K17LinearLNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 2.83 μM24-hBrainNone
7103
357408842022
FLPLIIGALSSKLPKIF
Temporin-PKE-K1217LinearLNoneAmidationFreeAntimicrobialSyntheticHCT-116Colorectal CancerMTT assayIC50 = 22.09 μM24-hColonNone
7104
357408842022
FLPLIIGALSSKLPKIF
Temporin-PKE-K1217LinearLNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 24.03 μM24-hLungNone
7102
357408842022
FLPLIIGALSSKLPKIF
Temporin-PKE-K1217LinearLNoneAmidationFreeAntimicrobialSyntheticH-838Lung CancerMTT assayIC50 = 22.67 μM24-hLungNone
7101
357408842022
FLPLIIGALSSKLPKIF
Temporin-PKE-K1217LinearLNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 27.32 μM24-hProstateNone
7100
357408842022
FLPLIIGALSSKLPKIF
Temporin-PKE-K1217LinearLNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 25.75 μM24-hBrainNone
7099
357408842022
FLPLIIGKLSSLLPKIF
Temporin-PKE-2K17LinearLNoneAmidationFreeAntimicrobialSyntheticH-157Lung CancerMTT assayIC50 = 2.78 μM24-hLungNone
7098
357408842022
FLPLIIGKLSSLLPKIF
Temporin-PKE-2K17LinearLNoneAmidationFreeAntimicrobialSyntheticHCT-116Colorectal CancerMTT assayIC50 = 2.84 μM24-hColonNone
7097
357408842022
FLPLIIGKLSSLLPKIF
Temporin-PKE-2K17LinearLNoneAmidationFreeAntimicrobialSyntheticH-838Lung CancerMTT assayIC50 = 3.07 μM24-hLungNone
7096
357408842022
FLPLIIGKLSSLLPKIF
Temporin-PKE-2K17LinearLNoneAmidationFreeAntimicrobialSyntheticPC-3Prostate CancerMTT assayIC50 = 2.64 μM24-hProstateNone
7095
357408842022
FLPLIIGKLSSLLPKIF
Temporin-PKE-2K17LinearLNoneAmidationFreeAntimicrobialSyntheticU251-MGBrain TumorMTT assayIC50 = 2.49 μM24-hBrainNone
7094
357408842022
FLPLIIGALSSLLPKIF
Temporin-PKE17LinearLNoneAmidationFreeAntimicrobialskin secretion of Pelophylax kl. esculentusH-157Lung CancerMTT assayIC50 = 17.40 μM24-hLungNone
7093
357408842022
FLPLIIGALSSLLPKIF
Temporin-PKE17LinearLNoneAmidationFreeAntimicrobialskin secretion of Pelophylax kl. esculentusHCT-116Colorectal CancerMTT assayIC50 = 21.31 μM24-hColonNone
7092
357408842022
FLPLIIGALSSLLPKIF
Temporin-PKE17LinearLNoneAmidationFreeAntimicrobialskin secretion of Pelophylax kl. esculentusH-838Lung CancerMTT assayIC50 = 16.38 μM24-hLungNone
7091
357408842022
FLPLIIGALSSLLPKIF
Temporin-PKE17LinearLNoneAmidationFreeAntimicrobialskin secretion of Pelophylax kl. esculentusPC-3Prostate CancerMTT assayIC50 = 7.29 μM24-hProstateNone
7089
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMNT-1Skin CancerResazurin dye assayIC50 = 57.03 ± 6.09 µM48-hSkinUS_10550155_B2
7090
357408842022
FLPLIIGALSSLLPKIF
Temporin-PKE17LinearLNoneAmidationFreeAntimicrobialskin secretion of Pelophylax kl. esculentusU251-MGBrain TumorMTT assayIC50 = 23.24 μM24-hBrainNone
7088
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaPC-3Prostate CancerResazurin dye assayIC50 = 57.99 ± 5.04 µM48-hProstateUS_10550155_B2
7086
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-2780Ovarian CancerResazurin dye assayIC50 = 33.92 ± 5.90 µM48-hOvaryUS_10550155_B2
7087
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMiaPaCa.2Pancreatic CancerResazurin dye assayIC50 = 57.45 ± 6.03 µM48-hPancreasUS_10550155_B2
7084
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMCF-7Breast CancerResazurin dye assayIC50 = 35.71 ± 8.50 µM48-hBreastUS_10550155_B2
7085
357408952022
FLSGIVGMLaKLF-jeff-FLSGIVGMLaKLF
Jeff-[G10a]2-SHa26LinearMixJeffamine linkerAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-549Lung CancerResazurin dye assayIC50 = 70.71 ± 5.39 µM48-hLungUS_10550155_B2
7082
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaPC-3Prostate CancerResazurin dye assayIC50 = 1.84 ± 0.17 µM48-hProstateUS_10550155_B2
7083
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMNT-1Skin CancerResazurin dye assayIC50 = 2.24 ± 0.05 µM48-hSkinUS_10550155_B2
7080
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-2780Ovarian CancerResazurin dye assayIC50 = 2.31 ± 0.08 µM48-hOvaryUS_10550155_B2
7081
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMiaPaCa.2Pancreatic CancerResazurin dye assayIC50 = 6.94 ± 0.27 µM48-hPancreasUS_10550155_B2
7079
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-549Lung CancerResazurin dye assayIC50 = 3.74 ± 3.46 µM48-hLungUS_10550155_B2
7077
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMCF-7Breast CancerResazurin dye assayIC50 = 3.77 ± 0.12 µM48-hBreastUS_10550155_B2
7078
357408952022
FLSGIVGMLaKLFFLSGIVGMLaKLFFLSGIVGMLaKLFKK
[G10a]3-SHa41LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaHepG-2Liver CancerResazurin dye assayIC50 = 5.49 ± 0.37 µM48-hLiverUS_10550155_B2
7076
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMNT-1Skin CancerResazurin dye assayIC50 = 4.72 ± 0.36 µM48-hSkinUS_10550155_B2
7075
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaPC-3Prostate CancerResazurin dye assayIC50 = 6.31 ± 0.66 µM48-hProstateUS_10550155_B2
7074
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMiaPaCa.2Pancreatic CancerResazurin dye assayIC50 = 8.71 ± 0.35 µM48-hPancreasUS_10550155_B2
7073
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-2780Ovarian CancerResazurin dye assayIC50 = 4.42 ± 0.06 µM48-hOvaryUS_10550155_B2
7072
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-549Lung CancerResazurin dye assayIC50 = 3.79 ± 1.61 µM48-hLungUS_10550155_B2
7071
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaHepG-2Liver CancerResazurin dye assayIC50 = 14.31 ± 1.37 µM48-hLiverUS_10550155_B2
7070
357408952022
FLSGIVGMLaKLFKFLKaLMFLSGIVG
[G10a]2-SHa27LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMCF-7Breast CancerResazurin dye assayIC50 = 5.69 ± 1.46 µM48-hBreastUS_10550155_B2
7069
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMNT-1Skin CancerResazurin dye assayIC50 = 15.25 ± 0.80 µM48-hSkinUS_10550155_B2
7068
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaPC-3Prostate CancerResazurin dye assayIC50 = 13.04 ± 1.99 µM48-hProstateUS_10550155_B2
7067
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMiaPaCa.2Pancreatic CancerResazurin dye assayIC50 = 22.36 ± 6.07 µM48-hPancreasUS_10550155_B2
7066
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-2780Ovarian CancerResazurin dye assayIC50 = 14.75 ± 7.35 µM48-hOvaryUS_10550155_B2
7065
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaA-549Lung CancerResazurin dye assayIC50 = 14.52 ± 1.44 µM48-hLungUS_10550155_B2
7064
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaHepG-2Liver CancerResazurin dye assayIC50 = 31.63 ± 1.56 µM48-hLiverUS_10550155_B2
7063
357408952022
FLSGIVGMLaKLF
[G10a]-SHa13LinearMixNoneAmidationFreeAntimicrobial and AnticancerAnalog of temporin SHaMCF-7Breast CancerResazurin dye assayIC50 = 15.05 ± 8.51 µM48-hBreastUS_10550155_B2
7061
356315152022
KKKKFFFFFFKKKK
K4F6K414LinearLNoneFreeFreeAntimicrobialSyntheticA-549Lung CancerAnnexinV-FITC/PI double staining assayapoptotic cells (early and late) increased from 9.59 ± 1.00% to 43.03 ± 2.13%12-hLungNone
7060
356315152022
KKKKFFFFFFFFKKKK
K4F8K416LinearLNoneFreeFreeAntimicrobialSyntheticA-549Lung CancerCCK-8 assayIC50 = 571.87 ± 66.23 μg/mL48-hLungNone
7059
356315152022
KKKKFFFFFFKKKK
K4F6K414LinearLNoneFreeFreeAntimicrobialSyntheticA-549Lung CancerCCK-8 assayIC50 = 62.64 ± 9.55 μg/mL48-hLungNone
7057
356315152022
KKFFFFFFKK
K2F6K210LinearLNoneFreeFreeAntimicrobialSyntheticA-549Lung CancerCCK-8 assayIC50 = 1146.23 ± 346.83 μg/mL48-hLungNone
7058
356315152022
KKKFFFFFFKKK
K3F6K312LinearLNoneFreeFreeAntimicrobialSyntheticA-549Lung CancerCCK-8 assayIC50 = 123.10 ± 35.19 μg/mL48-hLungNone
7056
363641562022
PTECQVGTTCKVES
PS1414LinearLNoneFreeFreeAnticancer and Anti-inflammatoryAphanomyces invadansHep-2Larynx CancerLDH leakage assay45.56 ± 2% LDH release at 20 µM24-hLarynxNone
7055
363641552022
PTECQVGTTCKVES
PS1414LinearLNoneFreeFreeAnticancer and Anti-inflammatoryAphanomyces invadansHep-2Larynx CancerMTT assayIC50 = 21 µM24-hLarynxNone
7054
352469612022
GllellelllkaaGw
d-EEK15LinearMixNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 4.78 ± 0.02 µM72-hBoneNone
7053
352469612022
GllellelllkaaGw
d-EEK15LinearMixNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 0.29 ± 0.01 µM72-hBreastNone
7052
352469612022
GllellelllkaaGw
d-EEK15LinearMixNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 0.29 ± 0.01 µM72-hBreastNone
7051
352469612022
GlldllelllkaaGw
d-DEK15LinearMixNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 5.84 ± 0.04 µM72-hBoneNone
7050
352469612022
GlldllelllkaaGw
d-DEK15LinearMixNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 0.36 ± 0 µM72-hBreastNone
7049
352469612022
GlldllelllkaaGw
d-DEK15LinearMixNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 0.44 ± 0.10 µM72-hBreastNone
7048
352469612022
GlldllhlllkaaGw
d-DHK15LinearMixNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 1.24 ± 0.03 µM72-hBoneNone
7046
352469612022
GlldllhlllkaaGw
d-DHK15LinearMixNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 0.32 ± 0.07 µM72-hBreastNone
7047
352469612022
GlldllhlllkaaGw
d-DHK15LinearMixNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 0.23 ± 0.04 µM72-hBreastNone
7045
352469612022
GLLKLLKLLLKAAGW
KKK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 9.65 ± 1.20 µM72-hBoneNone
7044
352469612022
GLLKLLKLLLKAAGW
KKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.35 ± 0.40 µM72-hBreastNone
7042
352469612022
GLLHLLKLLLKAAGW
HKK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 12.23 ± 0.11 µM72-hBoneNone
7043
352469612022
GLLKLLKLLLKAAGW
KKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.57 ± 0.24 µM72-hBreastNone
7041
352469612022
GLLHLLKLLLKAAGW
HKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.60 ± 0.42 µM72-hBreastNone
7039
352469612022
GLLELLKLLLKAAGW
EKK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 12.20 ± 1.84 µM72-hBoneNone
7040
352469612022
GLLHLLKLLLKAAGW
HKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.40 ± 0.71 µM72-hBreastNone
7038
352469612022
GLLELLKLLLKAAGW
EKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.19 ± 0.40 µM72-hBreastNone
7037
352469612022
GLLELLKLLLKAAGW
EKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.72 ± 0.21 µM72-hBreastNone
7035
352469612022
GLLDLLKLLLKAAGW
DKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.20 ± 0.14 µM72-hBreastNone
7036
352469612022
GLLDLLKLLLKAAGW
DKK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 10.40 ± 1.70 µM72-hBoneNone
7034
352469612022
GLLDLLKLLLKAAGW
DKK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.95 ± 0.35 µM72-hBreastNone
7033
352469612022
GLLKLLHLLLKAAGW
KHK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 12.88 ± 1.24 µM72-hBoneNone
7031
352469612022
GLLKLLHLLLKAAGW
KHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.59 ± 0.92 µM72-hBreastNone
7032
352469612022
GLLKLLHLLLKAAGW
KHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.40 ± 0.14 µM72-hBreastNone
7030
352469612022
GLLHLLHLLLKAAGW
HHK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 12.65 ± 1.91 µM72-hBoneNone
7028
352469612022
GLLHLLHLLLKAAGW
HHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.15 ± 0.07 µM72-hBreastNone
7029
352469612022
GLLHLLHLLLKAAGW
HHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.75 ± 0.21 µM72-hBreastNone
7027
352469612022
GLLELLHLLLKAAGW
EHK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 25.00 ± 0 µM72-hBoneNone
7025
352469612022
GLLELLHLLLKAAGW
EHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.35 ± 0.35 µM72-hBreastNone
7026
352469612022
GLLELLHLLLKAAGW
EHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 0.71 ± 0.13 µM72-hBreastNone
7024
352469612022
GLLDLLHLLLKAAGW
DHK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 20.45 ± 2.05 µM72-hBoneNone
7022
352469612022
GLLDLLHLLLKAAGW
DHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.75 ±0.49 µM72-hBreastNone
7023
352469612022
GLLDLLHLLLKAAGW
DHK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.02 ± 0.12 µM72-hBreastNone
7021
352469612022
GLLKLLELLLKAAGW
KEK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 8.15 ± 0.49 µM72-hBoneNone
7019
352469612022
GLLKLLELLLKAAGW
KEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.60 ± 0.14 µM72-hBreastNone
7020
352469612022
GLLKLLELLLKAAGW
KEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.35 ± 0.07 µM72-hBreastNone
7018
352469612022
GLLHLLELLLKAAGW
HEK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 143.20 ± 80.33 µM72-hBoneNone
7017
352469612022
GLLHLLELLLKAAGW
HEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 3.45 ± 2.19 µM72-hBreastNone
7016
352469612022
GLLHLLELLLKAAGW
HEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.35 ± 1.06 µM72-hBreastNone
7015
352469612022
GLLELLELLLKAAGW
EEK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 32.88 ± 4.07 µM72-hBoneNone
7014
352469612022
GLLELLELLLKAAGW
EEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.08 ± 0.18 µM72-hBreastNone
7013
352469612022
GLLELLELLLKAAGW
EEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.10 ± 0.14 µM72-hBreastNone
7012
352469612022
GLLDLLELLLKAAGW
DEK15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 19.88 ± 2.65 µM72-hBoneNone
7011
352469612022
GLLDLLELLLKAAGW
DEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 0.70 ± 0.07 µM72-hBreastNone
7010
352469612022
GLLDLLELLLKAAGW
DEK15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.14 ± 0.52 µM72-hBreastNone
7009
352469612022
GLLKLLKLLLHAAGW
KKH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 13.30 ± 0.99 µM72-hBoneNone
7008
352469612022
GLLKLLKLLLHAAGW
KKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.20 ± 0.42 µM72-hBreastNone
7007
352469612022
GLLKLLKLLLHAAGW
KKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.40 ± 0.85 µM72-hBreastNone
7006
352469612022
GLLHLLKLLLHAAGW
HKH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 18.88 ± 1.24 µM72-hBoneNone
7005
352469612022
GLLHLLKLLLHAAGW
HKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 3.10 ± 0.57 µM72-hBreastNone
7004
352469612022
GLLHLLKLLLHAAGW
HKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.45 ± 0.21 µM72-hBreastNone
7003
352469612022
GLLELLKLLLHAAGW
EKH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 23.83 ± 0.81 µM72-hBoneNone
7002
352469612022
GLLELLKLLLHAAGW
EKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.18 ± 0.31 µM72-hBreastNone
7001
352469612022
GLLELLKLLLHAAGW
EKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.75 ± 0.07 µM72-hBreastNone
7000
352469612022
GLLDLLKLLLHAAGW
DKH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 21.13 ± 3.01 µM72-hBoneNone
6999
352469612022
GLLDLLKLLLHAAGW
DKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.80 ± 0.28 µM72-hBreastNone
6998
352469612022
GLLDLLKLLLHAAGW
DKH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.45 ± 0.07 µM72-hBreastNone
6997
352469612022
GLLKLLHLLLHAAGW
KHH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 39.75 ± 5.30 µM72-hBoneNone
6996
352469612022
GLLKLLHLLLHAAGW
KHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 4.45 ± 0.49 µM72-hBreastNone
6995
352469612022
GLLKLLHLLLHAAGW
KHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 5.20 ± 0.71 µM72-hBreastNone
6994
352469612022
GLLHLLHLLLHAAGW
HHH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 185 ± 7 µM72-hBoneNone
6993
352469612022
GLLHLLHLLLHAAGW
HHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 9.50 ± 0.99 µM72-hBreastNone
6991
352469612022
GLLELLHLLLHAAGW
EHH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 117 ± 7 µM72-hBoneNone
6992
352469612022
GLLHLLHLLLHAAGW
HHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 21.10 ± 6.93 µM72-hBreastNone
6990
352469612022
GLLELLHLLLHAAGW
EHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 16.05 ± 3.18 µM72-hBreastNone
6989
352469612022
GLLELLHLLLHAAGW
EHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 25.35 ± 2.76 µM72-hBreastNone
6987
352469612022
GLLDLLHLLLHAAGW
DHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 11.90 ± 0.14 µM72-hBreastNone
6988
352469612022
GLLDLLHLLLHAAGW
DHH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 55.85 ± 18.88 µM72-hBoneNone
6986
352469612022
GLLDLLHLLLHAAGW
DHH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 21.45 ± 2.47 µM72-hBreastNone
6985
352469612022
GLLKLLELLLHAAGW
KEH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 49.25 ± 5.30 µM72-hBoneNone
6984
352469612022
GLLKLLELLLHAAGW
KEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.35 ± 0.07 µM72-hBreastNone
6983
352469612022
GLLKLLELLLHAAGW
KEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.30 ± 0.42 µM72-hBreastNone
6982
352469612022
GLLHLLELLLHAAGW
HEH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 106 ± 14 µM72-hBoneNone
6981
352469612022
GLLHLLELLLHAAGW
HEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 10.95 ± 1.06 µM72-hBreastNone
6979
352469612022
GLLELLELLLHAAGW
EEH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 19.60 ± 3.96 µM72-hBoneNone
6980
352469612022
GLLHLLELLLHAAGW
HEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 28.60 ± 10.75 µM72-hBreastNone
6977
352469612022
GLLELLELLLHAAGW
EEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.30 ± 0.14 µM72-hBreastNone
6978
352469612022
GLLELLELLLHAAGW
EEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 3.60 ± 0.85 µM72-hBreastNone
6976
352469612022
GLLDLLELLLHAAGW
DEH15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 36.48 ± 3.92 µM72-hBoneNone
6975
352469612022
GLLDLLELLLHAAGW
DEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 3.60 ± 0.42 µM72-hBreastNone
6974
352469612022
GLLDLLELLLHAAGW
DEH15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 5.35 ± 1.91 µM72-hBreastNone
6973
352469612022
GLLKLLKLLLEAAGW
KKE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 12.75 ± 1.20 µM72-hBoneNone
6972
352469612022
GLLKLLKLLLEAAGW
KKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.70 ± 0 µM72-hBreastNone
6971
352469612022
GLLKLLKLLLEAAGW
KKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.05 ± 0.64 µM72-hBreastNone
6970
352469612022
GLLHLLKLLLEAAGW
HKE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 15.95 ± 0.78 µM72-hBoneNone
6969
352469612022
GLLHLLKLLLEAAGW
HKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.90 ± 0.42 µM72-hBreastNone
6968
352469612022
GLLHLLKLLLEAAGW
HKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.70 ± 0.28 µM72-hBreastNone
6967
352469612022
GLLELLKLLLEAAGW
EKE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 8.00 ± 0.71 µM72-hBoneNone
6966
352469612022
GLLELLKLLLEAAGW
EKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.30 ± 0.14 µM72-hBreastNone
6965
352469612022
GLLELLKLLLEAAGW
EKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 1.80 ± 0.28 µM72-hBreastNone
6964
352469612022
GLLDLLKLLLEAAGW
DKE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 9.93 ± 0.25 µM72-hBoneNone
6963
352469612022
GLLDLLKLLLEAAGW
DKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 1.57 ± 0.33 µM72-hBreastNone
6962
352469612022
GLLDLLKLLLEAAGW
DKE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 2.10 ± 0 µM72-hBreastNone
6961
352469612022
GLLKLLHLLLEAAGW
KHE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 53 ± 2.83 µM72-hBoneNone
6960
352469612022
GLLKLLHLLLEAAGW
KHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.92 ± 0.17 µM72-hBreastNone
6959
352469612022
GLLKLLHLLLEAAGW
KHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.70 ± 0.14 µM72-hBreastNone
6958
352469612022
GLLHLLHLLLEAAGW
HHE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 53.25 ± 5.30 µM72-hBoneNone
6957
352469612022
GLLHLLHLLLEAAGW
HHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 10.75 ± 0.78 µM72-hBreastNone
6956
352469612022
GLLHLLHLLLEAAGW
HHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 16.70 ± 2.26 µM72-hBreastNone
6955
352469612022
GLLELLHLLLEAAGW
EHE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 18.25 ± 1.06 µM72-hBoneNone
6954
352469612022
GLLELLHLLLEAAGW
EHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.55 ± 0.07 µM72-hBreastNone
6953
352469612022
GLLELLHLLLEAAGW
EHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.90 ± 0.28 µM72-hBreastNone
6952
352469612022
GLLDLLHLLLEAAGW
DHE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 17.25 ± 1.06 µM72-hBoneNone
6951
352469612022
GLLDLLHLLLEAAGW
DHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.80 ± 0.14 µM72-hBreastNone
6950
352469612022
GLLDLLHLLLEAAGW
DHE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.75 ± 0.92 µM72-hBreastNone
6949
352469612022
GLLKLLELLLEAAGW
KEE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 49.38 ± 13.26 µM72-hBoneNone
6948
352469612022
GLLKLLELLLEAAGW
KEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 2.05 ± 0.21 µM72-hBreastNone
6947
352469612022
GLLKLLELLLEAAGW
KEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 3.75 ± 0.78 µM72-hBreastNone
6946
352469612022
GLLHLLELLLEAAGW
HEE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 47.50 ± 11 µM72-hBoneNone
6945
352469612022
GLLHLLELLLEAAGW
HEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 4.95 ± 0.49 µM72-hBreastNone
6944
352469612022
GLLHLLELLLEAAGW
HEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 6.50 ± 0.71 µM72-hBreastNone
6943
352469612022
GLLELLELLLEAAGW
EEE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 78.75 ± 5.30 µM72-hBoneNone
6942
352469612022
GLLELLELLLEAAGW
EEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 10.55 ± 3.46 µM72-hBreastNone
6941
352469612022
GLLELLELLLEAAGW
EEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 6.25 ± 1.77 µM72-hBreastNone
6940
352469612022
GLLDLLELLLEAAGW
DEE15LinearLNoneAmidationFreeAnticancerSyntheticU-2 OSBone CancerMTT assayIC50 = 61.00 ± 1.41 µM72-hBoneNone
6939
352469612022
GLLDLLELLLEAAGW
DEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLER-shEcadBreast CancerMTT assayIC50 = 6.05 ± 2.76 µM72-hBreastNone
6938
352469612022
GLLDLLELLLEAAGW
DEE15LinearLNoneAmidationFreeAnticancerSyntheticHMLERBreast CancerMTT assayIC50 = 5.55 ± 0.35 µM72-hBreastNone
6937
363550262022
TFKHG
LJP-125LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.72 ± 0.05 mM48-hLiverNone
6935
363550262022
TFKHG
LJP-125LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 0.41 ± 0.04 mM48-hLiverNone
6936
363550262022
TFKHG
LJP-125LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 0.60 ± 0.08 mM48-hLiverNone
6934
363550262022
YEHSHG
LJP-116LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.70 ± 0.07 mM48-hLiverNone
6933
363550262022
YEHSHG
LJP-116LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 0.61 ± 0.07 mM48-hLiverNone
6931
363550262022
HASWEH
LJP-106LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 3.53 ± 0.34 mM48-hLiverNone
6932
363550262022
YEHSHG
LJP-116LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 0.49 ± 0.05 mM48-hLiverNone
6930
363550262022
HASWEH
LJP-106LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 2.69 ± 0.22 mM48-hLiverNone
6928
363550262022
FEHSG
LJP-95LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.51 ± 0.07 mM48-hLiverNone
6929
363550262022
HASWEH
LJP-106LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 3.52 ± 0.35 mM48-hLiverNone
6927
363550262022
FEHSG
LJP-95LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 0.69 ± 0.08 mM48-hLiverNone
6925
363550262022
FSHTYV
LJP-86LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.76 ± 0.08 mM48-hLiverNone
6926
363550262022
FEHSG
LJP-95LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 0.53 ± 0.05 mM48-hLiverNone
6924
363550262022
FSHTYV
LJP-86LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 0.63 ± 0.05 mM48-hLiverNone
6923
363550262022
FSHTYV
LJP-86LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 0.44 ± 0.04 mM48-hLiverNone
6921
363550262022
HAGYSWA
LJP-77LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 1.66 ± 0.11 mM48-hLiverNone
6922
363550262022
HAGYSWA
LJP-77LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 1.44 ± 0.12 mM48-hLiverNone
6920
363550262022
HAGYSWA
LJP-77LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 2.53 ± 0.24 mM48-hLiverNone
6918
363550262022
FSTHGG
LJP-56LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 1.49 ± 0.13 mM48-hLiverNone
6919
363550262022
FKEHGY
LJP-66LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 3.06 ± 0.31 mM48-hLiverNone
6917
363550262022
FSTHGG
LJP-56LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 2.78 ± 0.26 mM48-hLiverNone
6915
363550262022
EGHGF
LJP-45LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.68 ± 0.07 mM48-hLiverNone
6916
363550262022
FSTHGG
LJP-56LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 2.44 ± 0.22 mM48-hLiverNone
6914
363550262022
EGHGF
LJP-45LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 0.65 ± 0.07 mM48-hLiverNone
6912
363550262022
FSHRGH
LJP-36LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 1.70 ± 0.15 mM48-hLiverNone
6913
363550262022
EGHGF
LJP-45LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 0.62 ± 0.07 mM48-hLiverNone
6911
363550262022
FSHRGH
LJP-36LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 1.42 ± 0.12 mM48-hLiverNone
6909
363550262022
LWEHSH
LJP-26LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 1.71 ± 0.13 mM48-hLiverNone
6910
363550262022
LWEHSH
LJP-26LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.62 ± 0.05 mM48-hLiverNone
6908
363550262022
LWEHSH
LJP-26LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 2.25 ± 0.22 mM48-hLiverNone
6906
363550262022
EGFHL
LJP-15LinearLNoneFreeFreeAnticancerLaminaria japonicaHepG-2Liver CancerMTT assayIC50 = 0.45 ± 0.05 mM48-hLiverNone
6907
363550262022
EGFHL
LJP-15LinearLNoneFreeFreeAnticancerLaminaria japonicaH-22Liver CancerMTT assayIC50 = 0.36 ± 0.03 mM48-hLiverNone
6905
363550262022
EGFHL
LJP-15LinearLNoneFreeFreeAnticancerLaminaria japonicaHuh-7Liver CancerMTT assayIC50 = 0.48 ± 0.05 mM48-hLiverNone
6904
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisB16-F10Skin CancerMTS assayIC50 = 6.65 ± 0.33 μM48-hSkinNone
6903
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisSMMC-7721Liver CancerMTS assayIC50 = 6.87 ± 0.51 μM48-hLiverNone
6902
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisA-549Lung CancerMTS assayIC50 = 5.81 ± 0.23 μM48-hLungNone
6901
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisSW-480Blood CancerMTS assayIC50 = 10.37 ± 0.40 μM48-hBloodNone
6900
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisMDA-MB-231Breast CancerMTS assayIC50 = 5.44 ± 0.33 μM48-hBreastNone
6898
343617282021
Structure given in figure
GA - 8Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HCT-116Colon CancerMTT assayIC50 = 60.70 ± 0.6 µg/mL24-hColonNone
6899
339167892021
FFPLIAGLAARFLPKIFCSITKRC
Brevinin-1RL124Cyclic(C18-C24)LNoneFreeFreeAntimicrobialRana limnocharisHCT-116Colon CancerMTS assayIC50 = 5.87 ± 0.15 μM48-hColonNone
6896
343617282021
Structure given in figure
GA - 7Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HepG-2Liver CancerMTT assayIC50 = 3.30 ± 0.1 µg/mL24-hLiverNone
6897
343617282021
Structure given in figure
GA - 8Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)MCF-7Breast CancerMTT assayIC50 = 6.90 ± 1.1 µg/mL24-hBreastNone
6894
343617282021
Structure given in figure
GA - 7Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)MCF-7Breast CancerMTT assayIC50 = 3.70 ± 0.2 µg/mL24-hBreastNone
6895
343617282021
Structure given in figure
GA - 7Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HCT-116Colon CancerMTT assayIC50 = 3.0 ± 1.1 µg/mL24-hColonNone
6892
343617282021
Structure given in figure
GA - 5Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)MCF-7Breast CancerMTT assayIC50 = 5.0 ± 0.3 µg/mL24-hBreastNone
6893
343617282021
Structure given in figure
GA - 5Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HCT-116Colon CancerMTT assayIC50 = 5.2 ± 0.8 µg/mL24-hColonNone
6891
343617282021
Structure given in figure
GA - 4Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HCT-116Colon CancerMTT assayIC50 = 73.0 ± 1.4 µg/mL24-hColonNone
6889
343617282021
Structure given in figure
GA - 3Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HCT-116Colon CancerMTT assayIC50 = 7.40 ± 0.4 µg/mL24-hColonNone
6890
343617282021
Structure given in figure
GA - 4Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)MCF-7Breast CancerMTT assayIC50 = 6.10 ± 0.4 µg/mL24-hBreastNone
6887
343617282021
Structure given in figure
GA - 2Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)HCT-116Colon CancerMTT assayIC50 = 70.30 ± 0.9 µg/mL24-hColonNone
6888
343617282021
Structure given in figure
GA - 3Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)MCF-7Breast CancerMTT assayIC50 = 5.1 ± 0.7 µg/mL24-hBreastNone
6886
343617282021
Structure given in figure
GA - 2Not AvailableLinearLNoneFree18beta-glycyrrhetinic-acidAntimicrobial and AnticancerSynthetic (glycyrrhetinic acid (GA)-based peptides)MCF-7Breast CancerMTT assayIC50 = 7.70 ± 1.3 µg/mL24-hBreastNone
6885
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisHeLaCervical CancerMTT assayIC50 = 1.97 µM24-hCervixNone
6884
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisHeLaCervical CancerMTT assayIC50 = 18.1 µM24-hCervixNone
6883
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisA-549Lung CancerMTT assayIC50 = 2.99 µM24-hLungNone
6882
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisA-549Lung CancerMTT assayIC50 = 21.6 µM24-hLungNone
6881
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 5.25 µM24-hBreastNone
6880
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 17.5 µM24-hBreastNone
6879
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLCu2+ boundFreeFreeAnticancerMorone chrysops x Morone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 5.52 µM24-hNot AvailableNone
6878
341353702021
FIHHIFRGIVHAGRSIGRFLTG
Piscidin 322LinearLNoneFreeFreeAnticancerMorone chrysops x Morone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 26.01 µM24-hNot AvailableNone
6877
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisHeLaCervical CancerMTT assayIC50 = 2.17 µM24-hCervixNone
6876
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisHeLaCervical CancerMTT assayIC50 = 2.22 µM24-hCervixNone
6875
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisA-549Lung CancerMTT assayIC50 = 2.15 µM24-hLungNone
6874
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisA-549Lung CancerMTT assayIC50 = 4.2 µM24-hLungNone
6873
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 3.92 µM24-hBreastNone
6872
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisMDA-MB-231Breast CancerMTT assayIC50 = 5.83 µM24-hBreastNone
6871
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLCu2+ boundFreeFreeAnticancerMorone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 5.31 µM24-hNot AvailableNone
6870
341353702021
FFHHIFRGIVHVGKTIHRLVTG
Piscidin 1, Moronecidin22LinearLNoneFreeFreeAnticancerMorone saxatilisHT-1080FibrosarcomaMTT assayIC50 = 5.58 µM24-hNot AvailableNone
6863
336030332021
RYGFTEVAGNFQQHNFGRG
L. squarrosulus purifed fraction19LinearLNoneFreeFreeAnticancerLentinus squarrosulus (Mont.)H-460Lung CancerMTT assayGraph Figure 224-hLungNone
6862
347897532021
GFLDIIKDTGKEFAVKILNNLKCKLAGGCPP
Palustrin - Ca31LinearLNoneFreeFreeHost Defence PeptideLithobates catesbeianusSGC-7901Gastric CancerNot AvailableIC50 = 0.951 μg/mlNot AvailableStomachNone
6861
336770232021
GKLRLIKKLWVKKWKKKGWKA
Pep21LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 2 µM24-hBreastNone
6860
336770232021
GKLRLIKKLWVKKWKKKGWKA
Pep21LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticA-549Lung CancerMTT assayIC50 = 4 µM24-hLungNone
6859
345314302021
KKRKKKAFALKFVVDLI
PCC-117LinearLNoneAmidationFreeAntimicrobialPoecilocoris lewisiG361Skin CancerMTS assayIC50 = 57.8 µM48-hSkinNone
6858
345314302021
KKRKKKAFALKFVVDLI
PCC-117LinearLNoneAmidationFreeAntimicrobialPoecilocoris lewisiSK-Mel-28Skin CancerMTS assayIC50 = 50.8 µM48-hSkinNone
6856
339813632021
GBKRLVQRLKDBLRNLV
17BIPHE217LinearLNoneFreeFreeAntimicrobialDerivative of LL-37NCI-H-1975Lung CancerMTT assayIC50 = 71.42 µmol/L24-hLungNone
6857
336909772021
zffygwyggmekllrggrgerppr
NMTP-524LinearDZ = C10H7CH2C(O), M, 4-(Trifluoromethyl)-D-phenylalanineFreeFreeAnticancerNot AvailableSK-HEP-1Liver CancerMTT assayIC50 = 53.84 ± 4.35 µM48-hLiverNone
6853
335677892021
KnLAKnLAK
Si157LinearLnL = nor-LeuAmidationCaffeic acid (Caf)Antimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 140.3 ± 7.12 µM72-hBreastNone
6854
335677892021
KnLAKnLAK
Si157LinearLnL = nor-LeuAmidationCaffeic acid (Caf)Antimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 346.3 ± 7.91 µM72-hBreastNone
6855
339813632021
GBKRLVQRLKDBLRNLV
17BIPHE217LinearLNoneFreeFreeAntimicrobialDerivative of LL-37A-549Lung CancerMTT assayIC50 = 34.33 µmol24-hLungNone
6851
335677892021
KnLAKnLAK
Si147LinearLnL = nor-LeuAmidation1,8-naphthalimide-GlyAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 593.3 ± 60.3 µM72-hBreastNone
6852
335677892021
KnLAKnLAK
Si147LinearLnL = nor-LeuAmidation1,8-naphthalimide-GlyAntimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 1049 ± 49.77 µM72-hBreastNone
6849
335677892021
KL(Beta-A)KL(Beta-A)K
Si117LinearLβ-AlaAmidationCaffeic acid (Caf)Antimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 1087 ± 70.71 µM72-hBreastNone
6850
335677892021
KnLAKnLAK
Si137LinearLnL = nor-LeuAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 1704 ± 112 µM72-hBreastNone
6847
335677892021
KL(Beta-A)KL(Beta-A)K
Si27LinearLβ-AlaAmidation1,8-naphthalimide-GlyAntimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 840 ± 21.18 µM72-hBreastNone
6848
335677892021
KL(Beta-A)KLAK
Si117LinearLβ-AlaAmidationCaffeic acid (Caf)Antimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 228.8 ± 7.18 µM72-hBreastNone
6846
335677892021
KL(Beta-A)KL(Beta-A)K
Si27LinearLβ-AlaAmidation1,8-naphthalimide-GlyAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 662.9 ± 20.02 µM72-hBreastNone
6844
335677892021
KLAKLAK
Si87LinearLNoneAmidationCaffeic acid (Caf)Antimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 514.3 ± 26.82 µM72-hBreastNone
6845
335677892021
KL(Beta-A)KL(Beta-A)AK
Si38LinearLβ-AlaAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 176.3 ± 4.66 µM72-hBreastNone
6842
335677892021
KLAKLAK
Si77LinearLNoneAmidation1,8-naphthalimide-GlyAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 1195 ± 131.5 µM72-hBreastNone
6843
335677892021
KLAKLAK
Si87LinearLNoneAmidationCaffeic acid (Caf)Antimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 128.6 ± 8.03 µM72-hBreastNone
6841
335677892021
(KLAKLAK)2
Si114LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 746.5 ± 7.6 µM72-hBreastNone
6840
335677892021
(KLAKLAK)2
Si114LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 124.1 ± 8.12 µM72-hBreastNone
6839
334285072021
LHHLLHLLHHLLHL
L8H614LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 16.4 µM24-hCervixNone
6838
334285072021
LHLLLHLLHHLLHL
L9H5-114LinearLNoneAmidationFreeAnticancerSyntheticHeLaCervical CancerMTT assayIC50 = 5.4 µM24-hCervixNone
6837
None2021
FPLPCAYKGTYC
SKACP00312LinearLNoneFreeFreeAnticancerSyntheticMDA-MB-453Breast CancerMTT assayIC50 = 156 ± 0.5 µM24-hBreastNone
6836
None2021
FPLPCAYKGTYC
SKACP00312LinearLNoneFreeFreeAnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 212 ± 0.5 µM24-hBreastNone
6835
None2021
FPLPCAYKGTYC
SKACP00312LinearLNoneFreeFreeAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 193 ± 0.5 µM24-hBreastNone
6834
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticHT-29Colon CancerMTT assayNot AvailableNot AvailableColonNone
6833
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticRKOColon CancerMTT assay25% cell viability at at 20 μM24-hColonNone
6832
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticHCT-15Colon CancerMTT assayNot AvailableNot AvailableColonNone
6831
323811042021
YGRKKRRQRRRKDHRISTFKNWPFLEGCACTPERM
Sur-X35LinearLNoneFreeTAT PeptideAnticancerSyntheticHCT-116Colon CancerMTT assay20% cell viability at at 20 μM24-hColonNone
6830
344401852021
SFIPRAKSTWLNNIKLL
HMP-S717LinearLNoneFreeFreeAnticancerHuman MilkSup-B15Blood CancerTrypan blue assayIC50 = 90 ± 14 µM24-hBloodNone
6828
344401852021
SFIPRAKSTWLNNIKLL
HMP-S717LinearLNoneFreeFreeAnticancerHuman MilkRS4;11Blood CancerTrypan blue assayIC50 = 184 ± 23 µM24-hBloodNone
6829
344401852021
SFIPRAKSTWLNNIKLL
HMP-S717LinearLNoneFreeFreeAnticancerHuman MilkRajiLymphoma CancerTrypan blue assayIC50 = 89 ± 24 µM24-hBloodNone
6827
344401852021
SFIPRAKSTWLNNIKLL
HMP-S717LinearLNoneFreeFreeAnticancerHuman MilkJurkatBlood CancerTrypan blue assayIC50 = 186 ± 37 µM24-hBloodNone
6826
334428812021
FLGALWNVAKRVF
[Arg]11-VmCT113LinearLNoneAmidationFreeAnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 25.8 ± 5.2 μmol/L24-hBreastNone
6825
334428812021
FLGALWRVAKSVF
[Arg]7-VmCT113LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 18.0 ± 2.7 μmol/L24-hBreastNone
6824
334428812021
FLRALWNVAKSVF
[Arg]3-VmCT113LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 20.6 ± 3.1 μmol/L24-hBreastNone
6823
334428812021
FLGALWNVAKSVF
VmCT113LinearLNoneAmidationFreeAntimicrobial and AnticancerVaejovis mexicanus smithiMCF-7Breast CancerMTT assayIC50 = 8.3 ± 1.4 μmol/L24-hBreastNone
6821
349417052021
ASIGALIQKAIALIKAKAA
LVTX-9-C1819LinearLNoneAmidationCH3-(CH2)16-COAnticancerSyntheticHepG-2Liver CancerCCK-8 assayIC50 = 7.0 ± 1.0 µM24-hLiverNone
6822
349417052021
ASIGALIQKAIALIKAKAA
LVTX-9-C1819LinearLNoneAmidationCH3-(CH2)16-COAnticancerSyntheticHeLaCervical CancerCCK-8 assayIC50 = 4.7 ± 1.4 µM24-hCervixNone
6819
349417052021
ASIGALIQKAIALIKAKAA
LVTX-9-C1819LinearLNoneAmidationCH3-(CH2)16-COAnticancerSyntheticA-549Lung CancerCCK-8 assayIC50 = 6.2 ± 1.4 µM24-hLungNone
6820
349417052021
ASIGALIQKAIALIKAKAA
LVTX-9-C1819LinearLNoneAmidationCH3-(CH2)16-COAnticancerSynthetic4T1Breast CancerCCK-8 assayIC50 = 7.6 ± 1.3 µM24-hBreastNone
6818
349417052021
ASIGALIQKAIALIKAKAA
LVTX-919LinearLNoneAmidationFreeAnticancerLycosa vittataA-549Lung CancerCCK-8 assayIC50 = 51.7 ± 4.3 µM24-hLungNone
6817
332448882021
IFGTILGFLKGL
Protonectin-F12LinearLNoneAmidationFreeAntimicrobialProtonoectinHCT-116Colon CancerResazurin dye assayCC50 = 9.8 ± 1.2 µM24-hColonNone
6816
332448882021
IFGTILGFLKGL
Protonectin-F12LinearLNoneAmidationFreeAntimicrobialProtonoectinMM96LSkin CancerResazurin dye assayCC50 = 16.0 ± 1.2 µM24-hSkinNone
6815
332448882021
ILGTILGLLKGL
Protonectin12LinearLNoneAmidationFreeAntimicrobialParachartergus fraternusHCT-116Colon CancerResazurin dye assayCC50 = 8.0 ± 0.5 µM24-hColonNone
6814
332448882021
ILGTILGLLKGL
Protonectin12LinearLNoneAmidationFreeAntimicrobialParachartergus fraternusMM96LSkin CancerResazurin dye assayCC50 = 14.8 ± 0.9 µM24-hSkinNone
6813
343093732021
FPWWWPFLRDVFTKGYGFGLGRKKRRQRRRPQ
Pal-pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinMCF-7Breast CancerMTT assayIC50 = 11.85 μM24-hBreastNone
6812
343093732021
FPWWWPFLRDVFTKGYGFGLGRKKRRQRRRPQ
Pal-pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-549Lung CancerMTT assayIC50 = 31.17 μM24-hLungNone
6811
343093732021
FPWWWPFLRDVFTKGYGFGLGRKKRRQRRRPQ
Pal-pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acid; pFL - a hydrophobic peptide fragment (FPWWWPFL) rich in tryptophan (W)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50 = 5.5 ± 1.1 μM24-hSkinNone
6810
343093732021
FPWWWPFL-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
pFL-N-Ter-TAT32LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATpFL = hydrophobic peptide fragment (FPWWWPFL)AnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50 = 11.1 ± 0.1 μM24-hSkinNone
6809
343093732021
Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
Pal-N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acidAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinMCF-7Breast CancerMTT assayIC50 = 27.26 μM24-hBreastNone
6808
343093732021
Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
Pal-N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acidAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-549Lung CancerMTT assayIC50 = 44.98 μM24-hLungNone
6807
343093732021
Pal-RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
Pal-N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATPalmitic acidAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50 = 36.67(Supplementary material)/15.2 ± 0.7 μM(Published paper)24-hSkinNone
6806
343093732021
RDVFTKGYGFGL
N-Ter12LinearLNoneFreeFreeAnticancerAnalogue of N-terminal fragment of the VDAC1 proteinA-375Skin CancerMTT assayIC50(A-375)> 50.0 μM24-hSkinNone
6803
341179172021
FKKLKKLFSKLWNWK
HPRP-A115LinearLNoneAmidationAcetylationAnticancerN-terminal region of Helicobacter pylori ribosomal protein L1HT-29Colon CancerMTT assayIC50 ~ 0.5 µg/mL24-hColonNone
6802
341179172021
FKKLKKLFSKLWNWK
HPRP-A115LinearLNoneAmidationAcetylationAnticancerN-terminal region of Helicobacter pylori ribosomal protein L1CT-26Colorectal CancerMTT assayIC50 between 0.5 and 1 µg/mL24-hColonNone
6801
348487292021
TGIATSGLATFTLHTGSLAPAT
AtMP222LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MDA-MB-231Breast CancerMTT assayIC50 = 6.97 ± 0.24 μg/ml48-hBreastNone
6800
348487292021
TGIATSGLATFTLHTGSLAPAT
AtMP222LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MCF-7Breast CancerMTT assayIC50 = 5.89 ± 0.14 μg/ml48-hBreastNone
6799
348487292021
THPPTTTTTTTTTTTTTAAPATTT
AtMP124LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MDA-MB-231Breast CancerMTT assayIC50 = 9.35 ± 0.25 μg/ml48-hBreastNone
6798
348487292021
THPPTTTTTTTTTTTTTAAPATTT
AtMP124LinearLNoneFreeFreeAntimicrobial and AnticancerAnabastestudineus skin mucus fraction 2MCF-7Breast CancerMTT assayIC50 = 8.25 ± 0.14 μg/ml48-hBreastNone
6797
335172642021
ICIFCCGCCHRSKCGMCCKT
Hepcidin20LinearLNoneFreeFreeAntimicrobial and AnticancerHomo sapiensU-266Lymphoma CancerMTT assayNANABloodNone
6796
347969032021
FLGWLFKVASK
A4W-GGN511LinearLNoneAmidationFreeAnticancerGaegurin 5SW-620Colorectal CancerSulforhodamine B assayEC50 = 22.07 ± 1.63 µM48-hColonNone
6795
347969032021
FLGWLFKVASK
A4W-GGN511LinearLNoneAmidationFreeAnticancerGaegurin 5SW-480Colorectal CancerSulforhodamine B assayEC50 = 98.63 ± 1.17 µM48-hColonNone
6793
347969032021
TYFNAVKPPITA
Loop2-PS2Aa12LinearLNoneAmidationFreeAnticancerParasporin-2Aa1SW-620Colorectal CancerSulforhodamine B assayEC50 = 15.95 ± 0.69 µM48-hColonNone
6794
347969032021
FKPQSGGGKCF
Loop1-HCoV-229E11LinearLNoneAmidationFreeAnticancerAlphacoronavirus (HCoV-229E)SW-480Colorectal CancerSulforhodamine B assayEC50 = 125.0 ± 1.32 µM48-hColonNone
6792
347969032021
TYFNAVKPPITA
Loop2-PS2Aa12LinearLNoneAmidationFreeAnticancerParasporin-2Aa1SW-480Colorectal CancerSulforhodamine B assayEC50 = 92.99 ± 0.98 µM48-hColonNone
6791
347969032021
NNETYFNAVKP
Loop1-PS2Aa11LinearLNoneAmidationFreeAnticancerParasporin-2Aa1SW-620Colorectal CancerSulforhodamine B assayEC50 = 106.2 ± 1.67 µM48-hColonNone
6790
347969032021
NNETYFNAVKP
Loop1-PS2Aa11LinearLNoneAmidationFreeAnticancerParasporin-2Aa1SW-480Colorectal CancerSulforhodamine B assayEC50 = 23.76 ± 1.25 µM48-hColonNone
6789
347969032021
PARDVLNTTSG
P264-G27411LinearLNoneAmidationFreeAnticancerParasporin-2Aa1SW-620Colorectal CancerSulforhodamine B assayEC50 = 11.28 ± 0.52 µM48-hColonNone
6788
347969032021
PARDVLNTTSG
P264-G27411LinearLNoneAmidationFreeAnticancerParasporin-2Aa1SW-480Colorectal CancerSulforhodamine B assayEC50 = 90.98 ± 0.75 µM48-hColonNone
6787
332451892021
KWCFRVCYRGICYIRRCR
Tachyplesin17LinearLNoneAmidationFreeAntibacterialHorseshoe crabH-460Lung CancerMTT assayIC50 = 25 µg/ml24-hLungNone
6786
332451892021
KWCFRVCYRGICYIRRCR
Tachyplesin17LinearLNoneAmidationFreeAntibacterialHorseshoe crabA-549Lung CancerMTT assayIC50 = 35 µg/ml24-hLungNone
6785
335626812021
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusAska-SSSynovial SarcomaMTS assayIC50 = 32.41 μg/mLNAMuscleNone
6784
335626812021
FIHHIIGGLFSAGKAIHRLIRRRRR
TP425LinearLNoneFreeFreeAntimicrobialOreochromis niloticusSW982Synovial SarcomaMTS assayIC50 = 29.20 μg/mLNAMuscleNone
6783
344493222021
PMPVSQECFETLRGHERILSILRHQNLLKELQDLALQGAKERAHQQ
rhCGA-N4646LinearLNoneFreeFreeAntimicrobialFound in neurons and endocrine cells in HumansHCT-116Colon CancerMTT assayIC50 = 1.997 µg/ml24-hColonNone
6782
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaLoVoColon CancerMTT assayIC50 = 128 µM24-hColonNone
6781
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaHeLaCervical CancerMTT assayIC50 > 128 µM24-hCervixNone
6780
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaMCF-7Breast CancerMTT assayIC50 > 128 µM24-hBreastNone
6779
340732032021
GLFLDTLKGAAKDVAGKLEGLKCKITGCKLP
Ranatuerin-231LinearLNoneFreeFreeAnticancerRana catesbeianaA-549Lung CancerMTT assayIC50 > 128 µM24-hLungNone
6778
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticMDA-MB-435 DOX-RBreast CancerMTS assayIC50 = 3.4 µM24-hBreastNone
6777
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticMDA-MB-435 WTBreast CancerMTS assayIC50 = 3.5 µM24-hBreastNone
6776
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticCT-26Colorectal CancerMTS assayIC50 = 2.2 µM24-hColonNone
6775
344614562021
gigavlkvlttglpaliswikrkrqqc
D-melittin27LinearDNoneFreeFreeAnticancerSyntheticA-549Lung CancerMTS assayIC50 = 4.5 µM24-hLungNone
6774
334629442021
FSHTYV
GP-36LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideColo-320Colon CancerMTT assayIC50 = 149 ± 15.2 µM48-hColonNone
6772
334629442021
FSHTYV
GP-36LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideCT-26Colorectal CancerMTT assayIC50 = 133 ± 12.5 µM48-hColonNone
6773
334629442021
FSHTYV
GP-36LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideCaCo-2Colon CancerMTT assayIC50 = 162 ± 17.1 µM48-hColonNone
6770
334629442021
EGFHL
GP-25LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideCaCo-2Colon CancerMTT assayIC50 = 154 ± 15.8 µM48-hColonNone
6771
334629442021
EGFHL
GP-25LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideColo-320Colon CancerMTT assayIC50 = 142 ± 14.9 µM48-hColonNone
6768
334629442021
FKEHGY
GP-16LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideColo-320Colon CancerMTT assayIC50 = 111 ± 12.0 µM48-hColonNone
6769
334629442021
EGFHL
GP-25LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideCT-26Colorectal CancerMTT assayIC50 = 114 ± 12.1 µM48-hColonNone
6767
334629442021
FKEHGY
GP-16LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideCaCo-2Colon CancerMTT assayIC50 = 104 ± 11.3 µM48-hColonNone
6766
334629442021
FKEHGY
GP-16LinearLNoneAmidationFreeAnticancerGinseng Leaf PeptideCT-26Colorectal CancerMTT assayIC50 = 86.4 ± 9.46 µM48-hColonNone
6765
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiLoVoColon CancerMTT assayIC50 = 35.05 µM24-hColonNone
6764
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiHeLaCervical CancerMTT assayIC50 = 23.26 µM24-hCervixNone
6763
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiMCF-7Breast CancerMTT assayIC50 = 37.84 µM24-hBreastNone
6762
340732032021
GLFDVVKGVLKGAGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYb33LinearLNoneFreeFreeAnticancerRana dybowskiiA-549Lung CancerMTT assayIC50 = 24.01 µM24-hLungNone
6761
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiLoVoColon CancerMTT assayIC50 = 55.22 µM24-hColonNone
6760
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiHeLaCervical CancerMTT assayIC50 = 52.83 µM24-hCervixNone
6759
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiMCF-7Breast CancerMTT assayIC50 = 41.21 µM24-hBreastNone
6758
340732032021
GVLGAVKDLLIGAGKSAAQSVLKTLSCKLSNDC
Odorranain-C133LinearLNoneFreeFreeAnticancerOdorrana grahamiA-549Lung CancerMTT assayIC50 = 27.31 µM24-hLungNone
6757
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisLoVoColon CancerMTT assayIC50 = 59.78 µM24-hColonNone
6755
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisMCF-7Breast CancerMTT assayIC50 = 45.25 µM24-hBreastNone
6756
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisHeLaCervical CancerMTT assayIC50 = 37.23 µM24-hCervixNone
6754
340732032021
GILSSIKGVAKGVAKNVAAQLLDTLKCKITGC
Ranatuerin-2Lb32LinearLNoneFreeFreeAnticancerRana luteiventrisA-549Lung CancerMTT assayIC50 = 15.32 µM24-hLungNone
6753
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiLoVoColon CancerMTT assayIC50 = 8.05 µg/ml24-hColonNone
6752
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiHeLaCervical CancerMTT assayIC50 = 19.69 µg/ml24-hCervixNone
6751
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiMCF-7Breast CancerMTT assayIC50 = 25.74 µg/ml24-hBreastNone
6750
340732032021
GIFDVVKGVLKGVGKNVAGSLLEQLKCKLSGGC
Brevinin-2DYd33LinearLNoneFreeFreeAnticancerRana dybowskiiA-549Lung CancerMTT assayIC50 = 2.975 µg/ml24-hLungNone
6749
339196392021
RMMRIFWVIKLAR
Pugnin B13LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax)PC-3Prostate CancerMTT assay90% Cytotoxicity at 100 µM24-hProstateNone
6748
339196392021
RMMRIFWVIKLAR
Pugnin B13LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax)MCF-7Breast CancerMTT assay5% Cytotoxicity at 100 µM24-hBreastNone
6747
339196392021
RLMRIFRILKLAR
Pugnin A13LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax)PC-3Prostate CancerMTT assay74% Cytotoxicity at 100 µM24-hProstateNone
6745
349352532021
WHLV
LCP-34CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaCaCo-2Colon CancerMTT assayIC50 = 68.2 ± 7.11 μM48-hColonNone
6746
339196392021
RLMRIFRILKLAR
Pugnin A13LinearLNoneFreeFreeAntibacterial and AnticancerSynthetic; Using Skin Transcriptome of Treefrog ( Boana pugnax)MCF-7Breast CancerMTT assay12% Cytotoxicity at 100 µM24-hBreastNone
6743
349352532021
WHLV
LCP-34CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaMKN-45Gastric CancerMTT assayIC50 = 86.9 ± 9.11 μM48-hStomachNone
6744
349352532021
WHLV
LCP-34CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaHepG-2Gastric CancerMTT assayIC50 = 85.2 ± 9.27 μM48-hStomachNone
6740
349352532021
WAHT
LCP-24CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaHepG-2Gastric CancerMTT assayIC50 = 96.9 ± 9.91 μM48-hStomachNone
6741
349352532021
WAHT
LCP-24CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaCaCo-2Colon CancerMTT assayIC50 = 100 ± 11.6 μM48-hColonNone
6742
349352532021
WHLV
LCP-34CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaSGC-7901Gastric CancerMTT assayIC50 = 101 ± 10.6 μM48-hStomachNone
6738
349352532021
WAHT
LCP-24CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaSGC-7901Gastric CancerMTT assayIC50 = 116 ± 12.4 μM48-hStomachNone
6739
349352532021
WAHT
LCP-24CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaMKN-45Gastric CancerMTT assayIC50 = 107 ± 11.8 μM48-hStomachNone
6735
349352532021
FHVL
LCP-14CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaMKN-45Gastric CancerMTT assayIC50 = 128 ± 13.5 μM48-hStomachNone
6736
349352532021
FHVL
LCP-14CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaHepG-2Gastric CancerMTT assayIC50 = 123 ± 12.9 μM48-hStomachNone
6737
349352532021
FHVL
LCP-14CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaCaCo-2Colon CancerMTT assayIC50 = 131 ± 13.4 μM48-hColonNone
6733
337571452021
RALGWSCL
P28LinearLNoneFreeFreeAnticancerZingiber officinaleRajiLymphoma CancerMTT assayIC50 = 700 μg/mL24-hBloodNone
6734
349352532021
FHVL
LCP-14CyclicLNoneCyclizedCyclizedAnticancerLaminaria japonicaSGC-7901Gastric CancerMTT assayIC50 = 111 ± 10.6 μM48-hStomachNone
6732
337571452021
RALGWSCL
P28LinearLNoneFreeFreeAnticancerZingiber officinaleMOLT-4Luekemia CancerMTT assayIC50 = 700 μg/mL24-hBloodNone
6730
343093732021
RDVFTKGYGFGL-GRK(Dansylglycine)KRRQRRRPQ
N-Ter-TAT24LinearLDansylglycine = fluorescent amino acid residue located in the side chain of lysineTATFreeAnticancerSyntheticA-375Skin CancerMTT assayIC50 > 50.0 μM24-hSkinNone
6731
337571452021
RALGWSCL
P28LinearLNoneFreeFreeAnticancerZingiber officinaleNB-4Luekemia CancerMTT assayIC50 = 600 μg/mL24-hBloodNone
6729
343943842021
SLSLSVAR
MIPP8LinearLNoneFreeFreeAnticancerMorchella importunaHeLaCervical CancerMTT assayInhibitory rate = 59.36 ± 3.67% at 400 μg/mL24-hCervixNone
6728
335822212021
ALWKDLLKNVGIAAGKAALNKVTDMVNQ
Dermaseptin-TO28LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tomopternaPC-3Prostate CancerMTT assayGraph Figure-724-hProstateNone
6727
335822212021
ALWKDLLKNVGIAAGKAALNKVTDMVNQ
Dermaseptin-TO28LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tomopternaH-157Lung CancerMTT assayGraph Figure-724-hLungNone
6726
335822212021
ALWKDLLKNVGIAAGKAALNKVTDMVNQ
Dermaseptin-TO28LinearLNoneAmidationFreeAntimicrobialPhyllomedusa tomopternaU251-MGBrain TumorMTT assayGraph Figure-724-hBrainNone
6725
345727192021
IWLTALKFLGKNLGKLAKQQLAKL
LyeTxI-b24LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMDA-MB-231Breast CancerMTT assayIC50 = 5.77 ± 0.83 µM48-hBreastNone
6724
345727192021
IWLTALKFLGKNLGKLAKQQLAKL
LyeTxI-b24LinearLNoneAmidationFreeAntimicrobial and AnticancerSyntheticMCF-7Breast CancerMTT assayIC50 = 7.34 ± 3.09 µM48-hBreastNone
6723
345727192021
IWLTALKFLGKNLGKLAKQQLAKL
LyeTxI-b24LinearLNoneAmidationFreeAntimicrobial and AnticancerSynthetic4T1Breast CancerMTT assayIC50 = 6.5 ± 5.30 µM48-hBreastNone
6722
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkMDA-MB-231Breast CancerAnnexin V-FITC assay~80% cell death at 200 µg/ml48-hBreastNone
6721
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkMCF-7Breast CancerAnnexin V-FITC assay~50% cell death at 300 µg/ml48-hBreastNone
6720
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkSK-BR-3Breast CancerAnnexin V-FITC assay~80% cell death at 100 µg/ml48-hBreastNone
6719
342361342021
FKCRRWQWRMKKLGAPSITCVRRAF
Bovine Lactoferricin (LfcinB)25LinearLNoneFreeFreeAntimicrobialBovine MilkMDA-MB-468Breast CancerAnnexin V-FITC assay~60% cell death at 300 µg/ml48-hBreastNone
6718
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSHCT-116Colon CancerMTT assayIC50 = 3.721 µM24-hColonNone
6717
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSMCF-7Breast CancerMTT assayIC50 = 3.17 µM24-hBreastNone
6716
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSU251-MGBrain TumorMTT assayIC50 = 3.492 µM24-hBrainNone
6715
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSPC-3Prostate CancerMTT assayIC50 = 2.629 µM24-hProstateNone
6714
345646152021
FlPLIASLAGNVVPKIFCKITKRC
B1OS-D-L24LinearMixNoneFreeFreeAntimicrobialB-1OSH-838Lung CancerMTT assayIC50 = 2.553 µM24-hLungNone
6713
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSHCT-116Colon CancerMTT assayIC50 = 11.03 µM24-hColonNone
6712
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSMCF-7Breast CancerMTT assayIC50 = 8.883 µM24-hBreastNone
6711
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSU251-MGBrain TumorMTT assayIC50 = 8.629 µM24-hBrainNone
6710
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSPC-3Prostate CancerMTT assayIC50 = 5.473 µM24-hProstateNone
6709
345646152021
FLPLIASLAGNVVPKIFCKITKRC
B1OS-L24LinearLNoneFreeFreeAntimicrobialB-1OSH-838Lung CancerMTT assayIC50 = 3.976 µM24-hLungNone
6708
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriHCT-116Colon CancerMTT assayIC50 = 33.69 µM24-hColonNone
6707
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriMCF-7Breast CancerMTT assayIC50 = 112 µM24-hBreastNone
6706
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriU251-MGBrain TumorMTT assayIC50 = 233.0 µM24-hBrainNone
6705
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriPC-3Prostate CancerMTT assayIC50 = 95.94 µM24-hProstateNone
6704
345646152021
FPLIASLAGNVVPKIFCKITKRC
B1OS23LinearLNoneFreeFreeAntimicrobialOdorrana schmackeriH-838Lung CancerMTT assayIC50 = 36.84 µM24-hLungNone
6703
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HHCT-116Colon CancerMTT assayIC50 = 3.583 µM24-hColonNone
6702
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HH-157Lung CancerMTT assayIC50 = 2.811 µM24-hLungNone
6701
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HMDA-MB-435SBreast CancerMTT assayIC50 = 2.243 µM24-hBreastNone
6700
328126942021
FALGAVTKVLYKLFCLITRKC
Brevinin-1HY21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HPC-3Prostate CancerMTT assayIC50 = 5.425 µM24-hProstateNone
6699
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HHCT-116Colon CancerMTT assayIC50 = 342.8 µM24-hColonNone
6698
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HH-157Lung CancerMTT assayIC50 = 278.9 µM24-hLungNone
6697
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HMDA-MB-435SBreast CancerMTT assayIC50 = 214.7 µM24-hBreastNone
6696
328126942021
FALGAVTCLIRTKCKVLPKLF
Brevinin-1Ha21LinearLNoneFreeFreeAntimicrobialAnalogue of Brevinin-1HPC-3Prostate CancerMTT assayIC50 = 186.9 µM24-hProstateNone
6695
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisHCT-116Colon CancerMTT assayIC50 = 2.599 µM24-hColonNone
6694
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisH-157Lung CancerMTT assayIC50 = 3.37 µM24-hLungNone
6693
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisMDA-MB-435SBreast CancerMTT assayIC50 = 3.47 µM24-hBreastNone
6692
328126942021
FALGAVTKVLPKLFCLITRKC
Brevinin-1H21LinearLNoneFreeFreeAntimicrobialAmolops hainanensisPC-3Prostate CancerMTT assayIC50 = 5.87 µM24-hProstateNone
6691
334896812021
ADLPGLK
Chickpea7LinearLNoneFreeFreeAnticancerCicer arietinum L.MCF-7Breast CancerSulforhodamine B assayIC50 = 110.3 ± 2.97µMNABreastNone
6690
334896812021
ADLPGLK
Chickpea7LinearLNoneFreeFreeAnticancerCicer arietinum L.MDA-MB-231Breast CancerSulforhodamine B assayIC50 = 107.2 ± 1.62µMNABreastNone
6688
334896812021
ADLPGLK
Chickpea7LinearLNoneFreeFreeAnticancerCicer arietinum L.A-549Lung CancerSulforhodamine B assayIC50 = 126.4 ± 1.98 µMNALungNone
6689
334896812021
ADLPGLK
Chickpea7LinearLNoneFreeFreeAnticancerCicer arietinum L.HepG-2Liver CancerSulforhodamine B assayIC50 = 113.7 ± 0.99 µMNALiverNone
6687
334896812021
ADLPGLK
Chickpea7LinearLNoneFreeFreeAnticancerCicer arietinum L.IshikawaEndometrial CancerSulforhodamine B assayIC50 = 101.5 ± 1.83 µMNAEndometriumNone
6686
334896812021
ADLPGLK
Chickpea7LinearLNoneFreeFreeAnticancerCicer arietinum L.PA-1Ovarian CancerSulforhodamine B assayIC50 = 133.4 ± 0.70µMNAOvaryNone
6685
335958762021
VKLRSLLCS
VS-99LinearLNoneFreeFreeAnticancerAllium sativumK-562Blood CancerMTT assayIC50 = 1.57 mM48-hBloodNone
6684
335958762021
VKLRSLLCS
VS-99LinearLNoneFreeFreeAnticancerAllium sativumMOLT-4Blood CancerMTT assayIC50 = 0.84 mM48-hBloodNone
6681
348679622021
FLPLLISALTSLFPKLGK
SSTP118LinearLNoneFreeFreeHost Defense PeptideIndosylvirana aurantiacaHSC-4Tongue Squamous Cell CarcinomaMTT assayIC50 = 10.22 μM48-hTongueNone
6680
348679622021
FLPLLISALTSLFPKLGK
SSTP118LinearLNoneFreeFreeHost Defense PeptideIndosylvirana aurantiacaMDA-MB-231Breast CancerMTT assayIC50 = 4.5 μM48-hBreastNone
6679
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 1499 μM24-hBrainNone
6678
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 427.3 μM24-hLungNone
6677
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 180.8 μM24-hLungNone
6676
349437412021
WLWKKIKNVAKAAGKAAKGAL
t-DPH1-6KW21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 118.4 μM24-hProstateNone
6675
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 593.7 μM24-hBrainNone
6674
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 88.28 μM24-hLungNone
6673
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 186.1 μM24-hLungNone
6672
349437412021
GLWKKIKNVAKAAGKAAKGAL
t-DPH1-6K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 55.65 μM24-hProstateNone
6671
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 2.679 μM24-hBrainNone
6670
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 1.546 μM24-hLungNone
6669
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 1.796 μM24-hLungNone
6668
349437412021
GLWKKIKNVAKAAGKAALGAL
t-DPH1-5K21LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 2.605 μM24-hProstateNone
6667
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1U251-MGBrain TumorMTT assayIC50 = 32.18 μM24-hBrainNone
6666
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-157Lung CancerMTT assayIC50 = 6.143 μM24-hLungNone
6665
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1H-838Lung CancerMTT assayIC50 = 10.11 μM24-hLungNone
6664
349437412021
GLWKKIKNVAAAAGKAALGAL
t-DPH1-K421LinearLNoneAmidationFreeAntimicrobialAnalogue of t-DPH1PC-3Prostate CancerMTT assayIC50 = 18.99 μM24-hProstateNone
6663
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisU251-MGBrain TumorMTT assayIC50 = 34.25 μM24-hBrainNone
6662
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisH-157Lung CancerMTT assayIC50 = 10.20 μM24-hLungNone
6661
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisH-838Lung CancerMTT assayIC50 = 23.51 μM24-hLungNone
6660
349437412021
GLWSKIKNVAAAAGKAALGAL
t-DPH121LinearLNoneAmidationFreeAntimicrobialPhyllomedusa hypochondrialisPC-3Prostate CancerMTT assayIC50 = 14.67 μM24-hProstateNone
6659
None2021
ILGKIWKGIVSDF
DN413LinearLNoneFreeFreeAntimicrobialSyntheticHepG-2Liver CancerMTT assay191.67 ± 12.02 μM24-hLiverNone
6658
None2021
ILGKIVKKLVSDF
DN113LinearLNoneFreeFreeAntimicrobialSyntheticHepG-2Liver CancerMTT assay152.17 ± 7.73 μM24-hLiverNone
7781
None2023
KRWHWWRRHWVVW
MAD113LinearLNoneAmidationFreeAntimicrobialSyntheticOVCAR-3Ovarian CancerMTT assayIC50 = 14.2 μM48-hOvaryUS11571454 B2
7782
None2023
KRWHWWRRHWVVW
MAD113LinearLNoneAmidationFreeAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 36.2 μM48-hLungUS11571454 B2
7783
None2023
KRWHWWRRHWVVW
MAD113LinearLNoneAmidationFreeAntimicrobialSyntheticNCI/ADR-RESOvarian CancerMTT assayIC50 = 85.6 μM48-hOvaryUS11571454 B2
7784
None2023
LWKRWVGVWRKWL
DAP113LinearLNoneAmidationFreeAntimicrobialSyntheticA-549Lung CancerMTT assayIC50 = 11.9 μM48-hLungUS11571454 B2
7785
None2023
LWKRWVGVWRKWL
DAP113LinearLNoneAmidationFreeAntimicrobialSyntheticOVCAR-3Ovarian CancerMTT assayIC50 = 8.6 μM48-hOvaryUS11571454 B2
7786
None2023
LWKRWVGVWRKWL
DAP113LinearLNoneAmidationFreeAntimicrobialSyntheticNCI/ADR-RESOvarian CancerMTT assayIC50 = 14.0 μM48-hLungUS11571454 B2
7787
None2023
LWKRWVGVWRKWL
DAP113LinearLNoneAmidationFreeAntimicrobialSyntheticT-24Bladder CancerMTT assayIC50 = 15.3 μM48-hBladderUS11571454 B2
7788
None2023
WKWLKKWIK
AMP19LinearLNoneAmidationFreeAntimicrobialSyntheticOVCAR-3Ovarian CancerMTT assayIC50 = 51.1 μM48-hOvaryUS11571454 B2
7789
None2023
KRWWKWWRR
AMP29LinearLNoneAmidationFreeAntimicrobialSyntheticOVCAR-3Ovarian CancerMTT assayIC50 = 53.5 μM48-hOvaryUS11571454 B2
7808
None2022
YKSIEFC
P1C7LinearLNoneAcetylationFreeAnticancerSyntheticBXPC-3Pancreatic CancerCell Proliferation assay~40% reduction in cell growth at 20 μM72-hPancreasUS011214593B2
7809
None2022
YKSIEFC
P1A7LinearLNoneFreeFreeAnticancerSyntheticBXPC-4Pancreatic CancerCell Proliferation assay~50% reduction in cell growth at 20 μM72-hPancreasUS011214593B2
7810
None2022
YKSVEFC
P1B7LinearLNoneAcetylationFreeAnticancerSyntheticBXPC-5Pancreatic CancerCell Proliferation assay~50% reduction in cell growth at 20 μM72-hPancreasUS011214593B2
7816
None2022
LTSVVFILICCFHLENIFVLLKKRTLRKNDRKKR
Sample Peptide 1 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 48% at 25 μM48-hKidneyUS011339203B2
7817
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 0.4% at 25 μM48-hKidneyUS011339203B2
7818
None2022
WFLREGSMFVALSASVFSLLAIKKRTLRKNDRKKR
Sample Peptide 3 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 45.8% at 25 μM48-hKidneyUS011339203B2
7819
None2022
FLLISACWVISLILGGLPIMGWKKRTLRKNDRKKR
Sample Peptide 4 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 85.6% at 25 μM48-hKidneyUS011339203B2
7820
None2022
LYHKHYILECTTVFTLLLLSIVILYCRIKKRTLRKNDRKKR
Sample Peptide 5 from US011339203B241LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 77.6% at 25 μM48-hKidneyUS011339203B2
7821
None2022
VIIVLSVFIACWAPLFILLLLKKRTLRKNDRKKR
Sample Peptide 6 from US011339203B234LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 59.7% at 25 μM48-hKidneyUS011339203B2
7822
None2022
LFRAEYFLVLAVLNSGTNPIIKKRTLRKNDRKKR
Sample Peptide 7 from US011339203B234LinearLNoneAmidationFreeAnticancerSyntheticCAKI-2Renal CancerCCK-8 assayCell Viability = 66.3% at 25 μM48-hKidneyUS011339203B2
7823
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticPC-3Prostate CancerCCK-8 assayCell Viability = 2.5% at 25 μM48-hKidneyUS011339203B2
7824
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticA-2058Skin CancerCCK-8 assayCell Viability = 0.2% at 25 μM48-hSkinUS011339203B2
7825
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 assayCell Viability = 0.6% at 25 μM48-hLungUS011339203B2
7826
None2022
FIGNLALSDLLAGVAYTANLLLKKRTLRKNDRKKR
Sample Peptide 2 from US011339203B235LinearLNoneAmidationFreeAnticancerSyntheticA-549Lung CancerCCK-8 assayCell Viability = 1.4% at 25 μM48-hLungUS011339203B2
7827
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 / WST-8Cell Viability = 6.8% at 25 μM48-hLungEP3604345B1;US11352408B2
7828
None2023
MQIPQAPWPVVWAVLQLGWRRKKRRQRRR
Sample Peptide 2 from EP3604345B129LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 / WST-8Cell Viability = 3.6% at 25 μM48-hLungEP3604345B1
7829
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticNCI-H2444Lung CancerCCK-8 / WST-8Cell Viability = 87.7% at 25 μM48-hLungEP3604345B1
7830
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 11.8% at 25 μM48-hLungEP3604345B1
7831
None2023
MQIPQAPWPVVWAVLQLGWRRKKRRQRRR
Sample Peptide 2 from EP3604345B129LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 4.9% at 25 μM48-hLungEP3604345B1
7832
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 120.6% at 25 μM48-hLungEP3604345B1
7833
None2023
PWWWPPVVVQQQMILLIGAARKKRTLRKNDRKKR
Sample Peptide 4 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 102.6% at 25 μM48-hLungEP3604345B1
7834
None2023
KKRTLRKNDRKKR
Sample Peptide 5 from EP3604345B113LinearLNoneAmidationFreeAnticancerSyntheticHCC-827Lung CancerCCK-8 / WST-8Cell Viability = 106.5% at 25 μM48-hLungEP3604345B1
7835
None2023
MQIPQAPWPVVWAVLQLGWRRKKRRQRRR
Sample Peptide 2 from EP3604345B129LinearLNoneAmidationFreeAnticancerSyntheticA-549Lung CancerCCK-8 / WST-8Cell Viability = 9.1% at 25 μM48-hLungEP3604345B1
7836
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticNCI-H446Lung CancerCCK-8 / WST-8Cell Viability = 0.5% at 25 μM48-hLungEP3604345B1
7837
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticNCI-H446Lung CancerCCK-8 / WST-8Cell Viability = 56.7% at 25 μM48-hLungEP3604345B1
7838
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticA-2058Skin CancerCCK-8 / WST-8Cell Viability = 6.7% at 25 μM48-hSkinEP3604345B1
7839
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticA-2058Skin CancerCCK-8 / WST-8Cell Viability = 87.5% at 25 μM48-hSkinEP3604345B1
7840
None2023
MQIPQAPWPVVWAVLQLGWRKKRTLRKNDRKKR
Sample Peptide 1 from EP3604345B133LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerCCK-8 / WST-8Cell Viability = 62.3% at 25 μM48-hBreastEP3604345B1
7841
None2023
MRIFAVFIFMTYWHLLNAKKRTLRKNDRKKR
Sample Peptide 3 from EP3604345B131LinearLNoneAmidationFreeAnticancerSyntheticMDA-MB-231Breast CancerCCK-8 / WST-8Cell Viability = 81.7% at 25 μM48-hBreastEP3604345B1
7842
378746702023
Not Available
LUNA18Not AvailableCyclicLNoneFreeAlkylationAnticancer and AntitumorSyntheticNCI-H2122NSCLCCellTiter-Glo Cell Viability assayIC50 = 1.4 ± 0.3 nmol/LNot availableLungNone
7843
378746702023
Not Available
LUNA18Not AvailableCyclicLNoneFreeAlkylationAnticancer and AntitumorSyntheticMiaPaCa.2Pancreatic CancerCellTiter-Glo Cell Viability assayIC50 = 1.4 ± 0.2 nmol/LNot availablePancreasNone
7844
378746702023
Not Available
LUNA18Not AvailableCyclicLNoneFreeAlkylationAnticancer and AntitumorSyntheticNCI-H441NSCLCCellTiter-Glo Cell Viability assayIC50 = 2.9 ± 0.7 nmol/LNot availableLungNone
7845
378746702023
Not Available
LUNA18Not AvailableCyclicLNoneFreeAlkylationAnticancer and AntitumorSyntheticLS 180Colon CancerCellTiter-Glo Cell Viability assayIC50 = 2.7 ± 0.4 nmol/LNot availableColonNone
7846
378746702023
Not Available
LUNA18Not AvailableCyclicLNoneFreeAlkylationAnticancer and AntitumorSyntheticGSUStomach CancerCellTiter-Glo Cell Viability assayIC50 = 0.17 ± 0.02 nmol/LNot availableStomachNone