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Browse result page of B3Pdb
The total number entries retrieved from this search are
318
, scroll left/right for detailed information.
B3pdbID
PEPTIDE NAME
PEPTIDE SEQUENCE (1-letter)
PEPTIDE SEQUENCE (3-letter)
N-TERMINAL MODIFICATION
C-TERMINAL MODIFICATION
CHEMICAL MODIFICATION
PEPTIDE LENGTH
PEPTIDE CONFORMATION
PEPTIDE NATURE
SOURCE/ORIGIN OF PEPTIDE
SMILES
CELL LINE
In vitro
CONCENTRATION
In vitro
METHOD
In vitro
RESULT
ANIMAL MODEL
In vivo
CONCENTRATION
In vivo
MODE OF DELIVERY
In vivo
METHOD
In vivo
RESULT
ACTION
TRANSPORT TYPE
SUBCELLULAR LOCALISATION
COMBINATION
PHYSICAL CONDITION
RESPONSE
RESULT
LABEL
PMID
b3pdb_0093
BVDO2
DmtNmeAFS-NH15
H-Dmt-Nme-D-Ala-Phe-Ser-NH2
Methylation
Amidation
NA
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
80% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0094
BVDO2
DmtNmeAFS-NH16
H-Dmt-Nme-D-Ala-Phe-Ser-NH2
Methylation
Amidation
NA
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0095
BVDO3
Dmt-N-Me-D-AAbaG-NH2
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
10% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0096
BVDO3
Dmt-N-Me-D-AAbaG-NH3
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
40% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0097
BVDO3
Dmt-N-Me-D-AAbaG-NH4
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
70% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0098
BVDO3
Dmt-N-Me-D-AAbaG-NH5
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
70% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0099
BVDO3
Dmt-N-Me-D-AAbaG-NH6
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
50% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0100
BVDO3
Dmt-N-Me-D-AAbaG-NH7
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
10% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0101
BVDO3
Dmt-N-Me-D-AAbaG-NH8
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
50% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0102
BVDO3
Dmt-N-Me-D-AAbaG-NH9
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
70% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0103
BVDO3
Dmt-N-Me-D-AAbaG-NH10
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
90% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0104
BVDO3
Dmt-N-Me-D-AAbaG-NH11
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
90% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0105
BVDO3
Dmt-N-Me-D-AAbaG-NH12
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0106
BVDO3
Dmt-N-Me-D-AAbaG-NH13
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
40% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0107
BVDO3
Dmt-N-Me-D-AAbaG-NH14
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
40% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0108
BVDO3
Dmt-N-Me-D-AAbaG-NH15
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
90% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0109
BVDO3
Dmt-N-Me-D-AAbaG-NH16
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
90% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0110
BVDO3
Dmt-N-Me-D-AAbaG-NH17
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.25mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0111
BVDO3
Dmt-N-Me-D-AAbaG-NH18
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.25mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0112
BVDO3
Dmt-N-Me-D-AAbaG-NH19
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.25mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0113
BVDO3
Dmt-N-Me-D-AAbaG-NH20
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.25mg/Kg
Intravenous
Hot water tail flick test
40% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0114
BVDO3
Dmt-N-Me-D-AAbaG-NH21
Dmt-N-Me-D-Ala-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at alanine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.25mg/Kg
Intravenous
Hot water tail flick test
50% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0115
BVDO3
H-Dmt-D-RAbaG-NH2
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0116
BVDO3
H-Dmt-D-RAbaG-NH3
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0117
BVDO3
H-Dmt-D-RAbaG-NH4
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0118
BVDO3
H-Dmt-D-RAbaG-NH5
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0119
BVDO3
H-Dmt-D-RAbaG-NH6
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
4 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0120
BVDO3
H-Dmt-D-RAbaG-NH7
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0121
BVDO3
H-Dmt-D-RAbaG-NH8
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
60% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0122
BVDO3
H-Dmt-D-RAbaG-NH9
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
90% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0123
BVDO3
H-Dmt-D-RAbaG-NH10
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0124
BVDO3
H-Dmt-D-RAbaG-NH11
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
1 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0125
BVDO3
H-Dmt-D-RAbaG-NH12
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
10% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0126
BVDO3
H-Dmt-D-RAbaG-NH13
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
40% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0127
BVDO3
H-Dmt-D-RAbaG-NH14
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
60% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0128
BVDO3
H-Dmt-D-RAbaG-NH15
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
70% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0129
BVDO3
H-Dmt-D-RAbaG-NH16
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.5 mg/Kg
Intravenous
Hot water tail flick test
100% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0130
BVDO3
H-Dmt-D-RAbaG-NH17
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.1mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 5 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0131
BVDO3
H-Dmt-D-RAbaG-NH18
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.1mg/Kg
Intravenous
Hot water tail flick test
30% maximum possible effect after 15 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0132
BVDO3
H-Dmt-D-RAbaG-NH19
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.1mg/Kg
Intravenous
Hot water tail flick test
50% maximum possible effect after 30 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0133
BVDO3
H-Dmt-D-RAbaG-NH20
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.1mg/Kg
Intravenous
Hot water tail flick test
50% maximum possible effect after 60 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0134
BVDO3
H-Dmt-D-RAbaG-NH21
H-Dmt-D-Arg-Aba-Gly-NH2
Methylation
Amidation
Addition of amiNAbenzoic acid at arginine
4
Tetrapeptide
Cationic
NA
NA
NA
NA
NA
NA
C57BL6 mice
0.1mg/Kg
Intravenous
Hot water tail flick test
50% maximum possible effect after 120 minutes
Cross BBB and shows morphine like action with analgesic effects
NA
NA
NA
NA
NA
NA
NA
22289619
b3pdb_0136
G23
HLNILSTLWKYR
HisLeuAsnIleLeuSerThrLeuTrpLysTyrArg
NA
NA
NA
12
Linear
NA
Phage display of prion proteins
NA
NA
NA
NA
NA
BALB/c mice
NA
Intravenous
Radioimaging
0.052 + 0.019 of fluoroscent measured in btain tissue after 4 hours
NA
Transcytosis as well as BBB penetration
NA
NA
NA
NA
NA
NA
22536790
b3pdb_0137
G23
HLNILSTLWKYR
HisLeuAsnIleLeuSerThrLeuTrpLysTyrArg
NA
NA
NA
12
Linear
NA
Phage display of prion proteins
NA
NA
NA
NA
NA
BALB/c mice
NA
Intravenous
Radioimaging
0.047 + 0.031 of fluoroscent measured in btain tissue after 24 hours
NA
Transcytosis as well as BBB penetration
NA
NA
NA
NA
NA
NA
22536790
b3pdb_0138
Scr-G23
KISHLLNYRTWL
LysIleSerHisLeuLeuAsnTyrArgThrTrpLeu
NA
NA
NA
12
Linear
NA
Phage display of prion proteins
NA
NA
NA
NA
NA
BALB/c mice
NA
Intravenous
Radioimaging
0.013 + 0.006 of fluoroscent measured in btain tissue after 4 hours
NA
Transcytosis as well as BBB penetration
NA
NA
NA
NA
NA
NA
22536790
b3pdb_0139
Scr-G23
KISHLLNYRTWL
LysIleSerHisLeuLeuAsnTyrArgThrTrpLeu
NA
NA
NA
12
Linear
NA
Phage display of prion proteins
NA
NA
NA
NA
NA
BALB/c mice
NA
Intravenous
Radioimaging
0.008 + 0.002 of fluoroscent measured in btain tissue after 24 hours
NA
Transcytosis as well as BBB penetration
NA
NA
NA
NA
NA
NA
22536790
b3pdb_0151
MPEG-PCL-Tat
NA
NA
Addition of MPEG and ploygalactolactone
NA
Addition of MPEG and PCL
NA
Linear
NA
Chemically synthesized
NA
NA
NA
NA
NA
Adult Sprague-Dawley rats
100 microliter
Intravenous
Fluoroscent screening by FITC labbled peptide maass in brain tissue
0.5% fluoroscence observed in brain tissue
NA
NA
NA
NA
NA
NA
NA
NA
23992922
b3pdb_0175
Angiopep-2
TFFYGGSRGKRNNFKTEEY
ThrPhePheTyrGlyGlySerArgGlyLysArgAsnAsnPheLysThrGluGluTyr
NA
NA
Conjugated with Tratuzumab
19
Linear
NA
NA
NA
NA
NA
NA
NA
Male Crl:Cd-1 nude mice
10mg/Kg
Intravenous
Fluoroscent screening by FITC labbled peptide maass in brain tissue
Significant fluoroscdnt observed in brain tissue
NA
NA
NA
NA
Breast cancer metastasis
NA
NA
NA
25492620
b3pdb_0176
Angiopep-2
TFFYGGSRGKRNNFKTEEY
ThrPhePheTyrGlyGlySerArgGlyLysArgAsnAsnPheLysThrGluGluTyr
NA
NA
Conjugated with Tratuzumab
19
Linear
NA
NA
NA
NA
NA
NA
NA
Male mice xenograft for BT 474 cell line intracerebrally
6 ml/kg
Intravenous
In situ brain perfusion assay
10 time increase of Mab as compared to control in brain tissue
NA
NA
NA
NA
Breast cancer metastasis
NA
NA
NA
25492620
b3pdb_0232
NA
RGD
ArgGlyAsp
NA
NA
NA
3
Linear
Cationic
Chemically synthesized
NA
NA
NA
NA
NA
BALB/c mice xenograft for U87MG glioma cells
5mg/Kg
Intravenous
Fluoroscent measurement
Significant amount of drugsa delivered in brain tissue
Peptide can deliver drugs into brain tissue
NA
NA
Doxorubicin+paclitaxel in 5mg/Kg combination
Brain glioma therapy
NA
NA
NA
27143884
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IIITD/CB
Raghava's Group
IMTECH
CellPPDMOD