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KKLALALAKKWLALAKKLALALAKK details
Primary information
ID antitb_1408,
Name25154927
N-Terminal modificationD-LAK120-A
C-Terminal ModificationKKLALALAKKWLALAKKLALALAKK
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature25
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium tuberculosis
In Vitro/ In vivoMycobacterium tuberculosis MDR strain
Cell LineMIC = 25 μM
Inhibition Concentrationin vitro
Sequence2014
CytotoxicityNA
In vivo ModelNA
Lethal DoseNA
Immune ResponceNA
Mechanism of ActionNA
TargetNA
Combination TherapyNA
Other activitiesNA
PMIDNA
Year of PublicationNA
Tertiary Structure
(Technique)
Not Predicted),
Primary information
ID antitb_1413,
Name25154927
N-Terminal modificationD-LAK120-A
C-Terminal ModificationKKLALALAKKWLALAKKLALALAKK
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature25
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium tuberculosis
In Vitro/ In vivoMycobacterium tuberculosis XDR strain
Cell LineMIC = 100 μM
Inhibition Concentrationin vitro
Sequence2014
CytotoxicityNA
In vivo ModelNA
Lethal DoseNA
Immune ResponceNA
Mechanism of ActionNA
TargetNA
Combination TherapyNA
Other activitiesNA
PMIDNA
Year of PublicationNA
Tertiary Structure
(Technique)
Not Predicted),
Primary information
ID antitb_1419,
Name25154927
N-Terminal modificationD-LAK120-A
C-Terminal ModificationKKLALALAKKWLALAKKLALALAKK
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature25
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium tuberculosis
In Vitro/ In vivoMycobacterium tuberculosis XDR strain
Inhibition Concentrationin vitro
Sequence2014
CytotoxicityTHP-1 cell line
In vivo ModelEC50 = 31.9 ± 9.5 μM
Lethal DoseCytotoxic at > 25 μM
Immune ResponceNA
Mechanism of ActionNA
TargetNA
Combination TherapyNA
Other activitiesNA
PMIDNA
Year of PublicationNA
Tertiary Structure
(Technique)
Not Predicted),
Primary information
ID antitb_1425,
Name25154927
N-Terminal modificationD-LAK120-A
C-Terminal ModificationKKLALALAKKWLALAKKLALALAKK
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature25
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium tuberculosis
In Vitro/ In vivoMycobacterium tuberculosis MDR strain GB2
Inhibition ConcentrationEx vivo
Sequence2014
CytotoxicityTHP-1 cell line
In vivo ModelNA
Lethal DoseCytotoxic at12.5 μM
Immune ResponceNA
Mechanism of ActionNA
TargetNA
Combination TherapyNA
Other activitiesNA
PMIDNA
Year of PublicationNA
Tertiary Structure
(Technique)
Not Predicted),
Primary information
ID antitb_1429,
Name25154927
N-Terminal modificationD-LAK120-A
C-Terminal ModificationKKLALALAKKWLALAKKLALALAKK
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature25
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium tuberculosis
In Vitro/ In vivoMycobacterium tuberculosis XDR strain WYC-11
Inhibition ConcentrationEx vivo
Sequence2014
CytotoxicityTHP-1 cell line
In vivo ModelNA
Lethal DoseCytotoxic at12.5 μM
Immune ResponceNA
Mechanism of ActionNA
TargetNA
Combination TherapyNA
Other activitiesNA
PMIDNA
Year of PublicationNA
Tertiary Structure
(Technique)
Not Predicted),