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Detailed description page of AntiTbPdb

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antitb_1745 details
Primary information
IDantitb_1745
Peptide NameFKAB-1Ge
SequenceG-Tic-Oic-K-Tic-Oic-G-Tic-Oic-K-Tic-KKKK
N-terminal ModificationAcetylation
C-terminal ModificationAmidation
Chemical ModificationTic = tetrahydroisoquinolinecarboxylic acid, Oic = Octahydroindolecarboxylic acid
Linear/ CyclicLinear
Length15
ChiralityL
NatureHydrophobic
SourceSynthetic
OriginNA
SpeciesMycobacterium ranae
StrainMycobacterium ranae
Inhibition ConcentartionMIC = 3 μM
In vitro/In vivoBoth
Cell LineRBC
Inhibition ConcentartionNA
Cytotoxicity26.7 % hemolysis at 100 μM and 9.2 % at 25 μM
In vivo ModelMice
Lethal DoseNo observed toxicity at 1, 5 and 25 mg/kg
Immune ResponseNA
Mechanism of ActionNA
TargetNA
Combination TherapyNone
Other ActivitiesAnti-bacterial (Salmonella typhimurium, Staphylococcus aureus, Bacillus subtillis)
Pubmed IDUS 2012/0197004
Year of Publication2012
3-D StructureNA