NPACT- Naturally occuring Plant based Anticancerous Compound-Activity-Target DataBase

Compound: Cucurbitacin I

TargetsGene NameGene IDCancerCell LinesIC50ED50EC50GI50RemarkReferences
JAK2Janus kinase 23717Breast CarcinomaMDA-MB-4350.18±0.07 µM---Cucurbitacin I treatment suppressed P-JAK2.15735720
JAK2Janus kinase 23717Lung adenocarcinomaA5490.25±0.09 µM---Cucurbitacin I treatment suppressed P-JAK2.15735720
JAK2Janus kinase 23717Breast CarcinomaMDA-MB-4680.40±0.26 µM---Cucurbitacin I treatment suppressed P-JAK2.15735720
STAT3signal transducer and activator of transcription 3 (acute-phase response factor)6774Lung adenocarcinomaA5490.8±0.7 µM---Cucurbitacin I treatment suppressed P-STAT3.15735720
STAT3signal transducer and activator of transcription 3 (acute-phase response factor)6774Breast CarcinomaMDA-MB-4354.6±1.9 µM---Cucurbitacin I treatment suppressed P-STAT3.15735720
STAT3signal transducer and activator of transcription 3 (acute-phase response factor)6774Breast CarcinomaMDA-MB-4687.5±1.5 µM---Cucurbitacin I treatment suppressed P-STAT3.15735720

 






Copyright © 2012. Subhash M. Agagrwal. All Rights Reserved.