Detailed description page of ImmunoSPdb

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1062 details
Primary information
ID1062
Peptide NameCharybdotoxin (ChTX)
SequenceEFTNVSCTTSKECWSVCQRLHNTSRGKCMNKKCRCYS
Length37
ChiralityL
N-terminal ModificationNone
C-terminal ModificationNone
Chemical ModificationNone
Linear/ CyclicLinear
NatureNatural
Source of OriginVenom of the scorpion Leiurusquin questriatus var. hebraeus
TargetK+ channels
Mechanism of ActionPotent selective block of apamin-insensitive Ca2+- activated K+ channels
In vitro/In vivoIn vitro
Cell LineGH3 pitutary cells and aortic smooth muscle
Inhibition ConcentartionNA
In vivo ModelNA
AssayNA
Lethal DoseNA
Combination TherapyNA
Pubmed ID2453055
Year of Publication1988
3-D Structure View in Jmol or Download Structure