Browse result page of ImmunoSPdb

The total number entries retrieved from this search are 5
IDNameSequenceLengthChiralityN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicNatureSourceTargetMechanism of ActionIn vivo/ In vitroCell LineIC-50In vivo ModelAssay TypeLethal DoseCombination TherapyPubmed IDYear of Publication
1392SEQ ID19RSCIDTIPKSQCTAFQCKHSXKYRLSFCRKTCGTC35LNoneNoneX = norleucine (nL)LinearNaturalShk toxin of S.helianthusT Lymphocytes Kv1.3 channelsBy blocking the potassium channel, Kv1.3 of T lymphocytesBothPeripheral blood human lymhocytes1 nMCD18-nullPL/J miceEnzyme-linked immunosorbent assay (ELISA), HPLCNACharybdotoxin (ChTX)US 60776802000
1394SEQ ID21RSCIDTIPKSRCTAFQCKHSMXYRLSFCRKTCGTC35LNoneNoneX = norleucine (nL)LinearNaturalShk toxin of S.helianthusT Lymphocytes Kv1.3 channelsBy blocking the potassium channel, Kv1.3 of T lymphocytesBothPeripheral blood human lymhocytes1 nMCD18-nullPL/J miceEnzyme-linked immunosorbent assay (ELISA), HPLCNACharybdotoxin (ChTX)US 60776802000
1463SEQ ID35R-nL-nL-nL-R-nL-nL-nLGY10LAcetylationAmidationnL = norleucineLinearProtein Derived(HLA-B) α1-domainNAInhibited T-cell proliferation, various inflammatory cytokines production.BothRAW264.7 macrophages cellsNACBA miceEnzyme-linked immunosorbent assay (ELISA)NALPSUS 6696545 B12004
1493SEQ ID1r-nL-nL-nL-r-nL-nL-nLgy10DNoneNonenL = norleucineLinearProtein Derived(HLA-B) α1-domainGut Associated Lymphoid Tissue (GALT)Increased CD4+ and CD8+ T-cellsIn vivoNoneNARhesus macaquesNANANAUS 7094413 B22006
1520SEQ ID13r-nL-nL-nL-r-nL-nL-nLGy10MixAcetylationAmidationnL = norleucineLinearSyntheticNANAInhibited T-cell proliferation, various inflammatory cytokines production.In vivoNone2.5-10micromolar against binding to peptides to HSC95C57BL6/J, Balb/c and CBA/J miceEnzyme-linked immunosorbent assay (ELISA)NALPSUS 7267822 B22007