Details of CPPsite entry with Sequence VKRGLKLRHVRPRVTRMDV |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | VKRGLKLRHVRPRVTRMDV |
| CPPsite ID | 1212, |
| PEPTIDE NAME | DPV1047 |
| CHIRALITY | L |
| LINEAR/CYCLIC | Linear |
| SOURCE | Protein derived |
| CATEGORY | Unknown |
| SUB CELLULAR LOCALIZATION | Nucleus |
| N-TERMINAL MODIFICATION | Cys addition |
| C-TERMINAL MODIFICATION | Free |
| UPTAKE EFFICIENCY | Lower than other DPVs and tat (48-60) |
| PROPOSED UPTAKE MECHANISM | Energy-dependent caveolar endocytic independent mechanism |
| INVITRO/INVIVO | In vitro |
| CELL LINE | HeLa, HCT116, HL-60, K562, Molt4, NIH-3T3 and primary hepatocyte cultures |
| CARGO | Protein (PO and IgG) |
| PMID | 15859953 |
| PATENT | Unknown |
| Tertiary Structure (Technique) | 1212 (PEPstrMOD), |