Details of CPPsite entry with Sequence RXRRBRRXRYQFLIRXRBRXRB |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | RXRRBRRXRYQFLIRXRBRXRB |
| CPPsite ID | 2315, |
| PEPTIDE NAME | Pip6a |
| CHIRALITY | Modified |
| LINEAR/CYCLIC | Linear |
| SOURCE | Synthetic |
| SUB CELLULAR LOCALIZATION | Vesicles |
| N-TERMINAL MODIFICATION | Acetylation |
| C-TERMINAL MODIFICATION | Free |
| CHEMICAL MODIFICATION | B, Beta-Alanine and X, 6-aminohexanoic acid (Ahx) |
| UPTAKE EFFICIENCY | Dose dependent uptake |
| PROPOSED UPTAKE MECHANISM | Energy and caveolae-mediated endocytosis |
| INVITRO/INVIVO | In vitro and in vivo |
| CELL LINE | Murine H2k mdx myoblasts and C2C12 cells |
| In VIVO MODEL | 1- to 2-day-old newborn wild-type C57BL/6 J mice |
| CARGO | Nucleic acid [phosphorodiamidate morpholino oligomers (PMO)] |
| PMID | 24366877 |
| PATENT | Unknown |
| Tertiary Structure (Technique) | Not Predicted), |