Details of CPPsite entry with Sequence RQIKIWFPNRRMKWKK |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | RQIKIWFPNRRMKWKK |
| CPPsite ID | 1093, 1132, |
| PEPTIDE NAME | pAntpHD (Pro50), Penetratin (pAntp) (43-58) |
| CHIRALITY | L, L |
| LINEAR/CYCLIC | Linear, Linear |
| SOURCE | Protein derived, Protein derived |
| CATEGORY | Unknown, Amphipathic |
| SUB CELLULAR LOCALIZATION | Cytoplasm, Cytosol and nucleus, nucleoi |
| N-TERMINAL MODIFICATION | Biotinylation, Conjugation with fluorescein |
| C-TERMINAL MODIFICATION | Amidation, Amidation |
| CHEMICAL MODIFICATION | NA, NA |
| UPTAKE EFFICIENCY | High, comparbale to (pAntp) (43-58), Unknown |
| PROPOSED UPTAKE MECHANISM | Non-receptor mdiated endocytic pathway, Non-endocytic pathway |
| INVITRO/INVIVO | In vitro, In vitro |
| CELL LINE | Cortical striatal cells, HaCat/ A549 cells |
| In VIVO MODEL | NA, NA |
| CARGO | Biotin, Fluorophore (fluorescein) |
| PMID | 8663410, 10784032 |
| PATENT | Unknown, Unknown |
| Tertiary Structure (Technique) | 1093 (PEPstrMOD), 1132 (PEPstrMOD), |