Details of CPPsite entry with Sequence GRKKRRQRRRPWQ |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | GRKKRRQRRRPWQ |
| CPPsite ID | 1137, 1138, |
| PEPTIDE NAME | TatP59W, TatP59W |
| CHIRALITY | L, L |
| LINEAR/CYCLIC | Linear, Linear |
| SOURCE | Protein derived, Protein derived |
| CATEGORY | Cationic, Cationic |
| SUB CELLULAR LOCALIZATION | Cytoplasm and nucleus, Cytoplasm and nucleus |
| N-TERMINAL MODIFICATION | Conjugation with fluorescein, Conjugation with fluorescein |
| C-TERMINAL MODIFICATION | Amidation, Amidation |
| CHEMICAL MODIFICATION | NA, NA |
| UPTAKE EFFICIENCY | Comparable to that of (pAntp) (43-58), Comparable to that of (pAntp) (43-58) |
| PROPOSED UPTAKE MECHANISM | Endocytic pathway, Non-endocytic pathway |
| INVITRO/INVIVO | In vitro, In vitro |
| CELL LINE | PC-12 cells, V79 cells |
| In VIVO MODEL | NA, NA |
| CARGO | Fluorophore (fluorescein), Fluorophore (fluorescein) |
| PMID | 12849987, 12849987 |
| PATENT | Unknown, Unknown |
| Tertiary Structure (Technique) | 1137 (PEPstrMOD), 1138 (PEPstrMOD), |