Browse result page of B3Pdb

The total number entries retrieved from this search are 318, scroll left/right for detailed information.
B3pdbIDPEPTIDE NAMEPEPTIDE SEQUENCE (1-letter)PEPTIDE SEQUENCE (3-letter)N-TERMINAL MODIFICATIONC-TERMINAL MODIFICATION CHEMICAL MODIFICATIONPEPTIDE LENGTHPEPTIDE CONFORMATIONPEPTIDE NATURESOURCE/ORIGIN OF PEPTIDESMILESCELL LINEIn vitro CONCENTRATIONIn vitro METHODIn vitro RESULTANIMAL MODELIn vivo CONCENTRATIONIn vivo MODE OF DELIVERYIn vivo METHODIn vivo RESULTACTIONTRANSPORT TYPESUBCELLULAR LOCALISATIONCOMBINATIONPHYSICAL CONDITIONRESPONSERESULTLABELPMID
b3pdb_0983pVECLLIILRRRIRKQAHAHSK-NH2Leu-Leu-Ile-Ile-Leu-Arg-Arg-Arg-Ile-Arg-Lys-Gln-Ala-His-Ala-His-Ser-Lys-NH2NANANA18LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00602 mL/(g x min) Direct iodination 26465925
b3pdb_0984pVECLLIILRRRIRKQAHAHSK-NH2Leu-Leu-Ile-Ile-Leu-Arg-Arg-Arg-Ile-Arg-Lys-Gln-Ala-His-Ala-His-Ser-Lys-NH2NANANA18LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.02313 ml/g Direct iodination 26465925
b3pdb_0988Transportan 10AGYLLGKINLKALAALAKKIL-NH2Ala-Gly-Tyr-Leu-Leu-Gly-Lys-Ile-Asn-Leu-Lys-Ala-Leu-Ala-Ala-Leu-Ala-Lys-Lys-Ile-Leu-NH2NANANA21LinearNAsynthetic,viralNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00005 mL/(g x min) Direct iodination 26465925
b3pdb_0989Transportan 10AGYLLGKINLKALAALAKKIL-NH2Ala-Gly-Tyr-Leu-Leu-Gly-Lys-Ile-Asn-Leu-Lys-Ala-Leu-Ala-Ala-Leu-Ala-Lys-Lys-Ile-Leu-NH2NANANA21LinearNAsynthetic,viralNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.00988 ml/g Direct iodination 26465925
b3pdb_0993TP10-2AGYLLGKINLKPLAALAKKIL-NH2Ala-Gly-Tyr-Leu-Leu-Gly-Lys-Ile-Asn-Leu-Lys-Pro-Leu-Ala-Ala-Leu-Ala-Lys-Lys-Ile-Leu-NH2NANANA21LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.000359 mL/(g x min) Direct iodination 26465925
b3pdb_0994TP10-2AGYLLGKINLKPLAALAKKIL-NH2Ala-Gly-Tyr-Leu-Leu-Gly-Lys-Ile-Asn-Leu-Lys-Pro-Leu-Ala-Ala-Leu-Ala-Lys-Lys-Ile-Leu-NH2NANANA21LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.01007 ml/g Direct iodination 26465925
b3pdb_0998D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00113 mL/(g x min) Direct iodination 3440215
b3pdb_0999D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.0226 ml/g Direct iodination 3440215
b3pdb_1000D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.0025 mL/(g x min) Direct iodination 3440215
b3pdb_1001D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.0177 ml/g Direct iodination 3440215
b3pdb_1002D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00292 mL/(g x min) Direct iodination 3440215
b3pdb_1003D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.0199 ml/g Direct iodination 3440215
b3pdb_1004D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.0025 mL/(g x min) Direct iodination 3440215
b3pdb_1005D-[Ala1]-peptide T-aaSTTTNYT-NH2(D)Ala-Ser-Thr-Thr-Thr-Asn-Tyr-Thr-NH2NANANA8LinearNAChemically synthesizedC[C@H]([C@@H](C(=O)N)NC(=O)[C@H](CC1=CC=C(C=C1)O)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@@H](C)N)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.0227 ml/g Direct iodination 3440215
b3pdb_1009NT1, Neurotensin8-13(NαMe)RK-(3,4-dehydro)PWtLL(NαMe)Arg-Lys-(3,4-dehydro)Pro-Trp-tLeu-LeuNANANA6LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA saturable NA NA NA Unidirectional influx rate constant 0.000512 mL/(g x min) H3/C14 8574648
b3pdb_1010NT1, Neurotensin8-13(NαMe)RK-(3,4-dehydro)PWtLL(NαMe)Arg-Lys-(3,4-dehydro)Pro-Trp-tLeu-LeuNANANA6LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA saturable NA NA NA Initial disrobution volume 0.0151 ml/g H3/C14 8574648
b3pdb_1011NT1, Neurotensin8-13(NαMe)RK-(3,4-dehydro)PWtLL(NαMe)Arg-Lys-(3,4-dehydro)Pro-Trp-tLeu-LeuNANANA6LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA saturable NA NA NA % injected dose 0.087 %/g H3/C14 8574648
b3pdb_1037MIF-1PLG-NH2Pro-Leu-Gly-NH2NANANA3LinearNANACC(C)CC(C(=O)NCC(=O)N)NC(=O)C1CCCN1NANANANANANAIntravenous NANA NA partially saturable NA NA NA Unidirectional influx rate constant 0.0237 mL/(g x min) H3/C14 7912427
b3pdb_1038MIF-1PLG-NH2Pro-Leu-Gly-NH2NANANA3LinearNANACC(C)CC(C(=O)NCC(=O)N)NC(=O)C1CCCN1NANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume -0.0173 ml/g H3/C14 7912427
b3pdb_1043β-Amyloid1-28DAEFRHDSGYQVHHQKLVFFAEDVGSNKAsp-Ala-Glu-Phe-Arg-His-Asp-Ser-Gly-Tyr-Gln-Val-His-His-Gln-Lys-Leu-Val-Phe-Phe-Ala-Glu-Asp-Val-Gly-Ser-Asn-LysNANANA28LinearNANAN[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(CC1=CN=C-N1)C(=O)N[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(CO)C(=O)NCC(=O)N[C@@]([H])(Cc1ccc(O)cc1)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(CC1=CN=C-N1)C(=O)N[C@@]([H])(CC1=CN=C-N1)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(CCCCN)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(C(C)C)C(=O)NCC(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(CC(=O)N)C(=O)N[C@@]([H])(CCCCN)C(=O)ONANANANANANAIntravenous NANA NA non saturable NA NA NA Unidirectional influx rate constant 0.000386 mL/(g x min) Direct iodination 1786560
b3pdb_1044β-Amyloid1-28DAEFRHDSGYQVHHQKLVFFAEDVGSNKAsp-Ala-Glu-Phe-Arg-His-Asp-Ser-Gly-Tyr-Gln-Val-His-His-Gln-Lys-Leu-Val-Phe-Phe-Ala-Glu-Asp-Val-Gly-Ser-Asn-LysNANANA28LinearNANAN[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(CC1=CN=C-N1)C(=O)N[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(CO)C(=O)NCC(=O)N[C@@]([H])(Cc1ccc(O)cc1)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(CC1=CN=C-N1)C(=O)N[C@@]([H])(CC1=CN=C-N1)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(CCCCN)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(C(C)C)C(=O)NCC(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(CC(=O)N)C(=O)N[C@@]([H])(CCCCN)C(=O)ONANANANANANAIntravenous NANA NA non saturable NA NA NA Initial disrobution volume 0.0159 ml/g Direct iodination 1786560
b3pdb_1046β-Amyloid1-40DAEFRHDSGYEVHHQKLVFFAEDVGSNKGAIIGLMVGGVVAsp-Ala-Glu-Phe-Arg-His-Asp-Ser-Gly-Tyr-Glu-Val-His-His-Gln-Lys-Leu-Val-Phe-Phe-Ala-Glu-Asp-Val-Gly-Ser-Asn-Lys-Gly-Ala-Ile-Ile-Gly-Leu-Met-Val-Gly-Gly-Val-ValNANANA40LinearNAhumanCC[C@H](C)[C@@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](C(C)C)C(=O)NCC(=O)NCC(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)O)NC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](CC3=CNC=N3)NC(=O)[C@H](CC4=CNC=N4)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC5=CC=C(C=C5)O)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC6=CNC=N6)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC7=CC=CC=C7)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NNANANANANANAIntravenous NANA NA Permeability NA NA NA RadioactiInitial disrobution volumety ratio 7 (cpm brain/mg)/(cpm blood/µl) direct iodination 26971931
b3pdb_1087Insulin detemir, LevA-chain: Gly-Ile-Val-Glu-Gln-Cys-Cys-Thr-Ser-Ile-Cys-Ser-Leu-Tyr-Gln-Leu-Glu-Asn-Tyr-Cys-Asn B-chain:Phe-Val-Asn-Gln-His-Leu-Cys-Gly-Ser-His-Leu-Val-Glu-Ala-Leu-Tyr-Leu-Val-Cys-Gly-Glu-Arg-Gly-Phe-Phe-Tyr-Thr-Pro-Lys-myristic acidA-chain:GIVEQCCTSICSLYQLENYCN B-chain: FVNQHLCGSHLVEALYLVCGERGFFYTPK-myristic acidNANACysA6-CysA11; CysA7-CysB7; CysA20-CysB1950LinearNAChemically synthesizedCCCCCCCCCCCCCC(=O)NCCCC[C@@H](C(=O)O)NC(=O)[C@@H]1CCCN1C(=O)[C@H]([C@@H](C)O)NC(=O)[C@H](CC2=CC=C(C=C2)O)NC(=O)[C@H](CC3=CC=CC=C3)NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)CNC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@@H]5CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]6CSSC[C@@H](C(=O)N[C@@H](CSSC[C@@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N5)C(C)C)CC(C)C)CC7=CC=C(C=C7)O)CC(C)C)C)CCC(=O)O)C(C)C)CC(C)C)CC8=CN=CN8)CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC9=CN=CN9)NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC1=CC=CC=C1)N)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N6)[C@@H](C)CC)CO)[C@@H](C)O)NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C(C)C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)CN)CO)CC(C)C)CC1=CC=C(C=C1)O)CCC(=O)N)CC(C)C)CCC(=O)O)CC(=O)N)CC1=CC=C(C=C1)O)C(=O)N[C@@H](CC(=O)N)C(=O)ONANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0 mL/(g x min) Direct iodination 20868713
b3pdb_1109PhrANTH2SKDYNSer-Lys-Asp-Tyr-AsnNANANA5LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00018 mL/(g x min) Direct iodination 26536593
b3pdb_1110PhrANTH2SKDYNSer-Lys-Asp-Tyr-AsnNANANA5LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.00659 ml/g Direct iodination 26536593
b3pdb_1114BIP-2GLWEDLLYNINRYAHYITGly-Leu-Trp-Glu-Asp-Leu-Leu-Tyr-Asn-Ile-Asn-Arg-Tyr-Ala-His-Tyr-Ile-ThrNANANA18LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00035 mL/(g x min) Direct iodination 26536593
b3pdb_1115BIP-2GLWEDLLYNINRYAHYITGly-Leu-Trp-Glu-Asp-Leu-Leu-Tyr-Asn-Ile-Asn-Arg-Tyr-Ala-His-Tyr-Ile-ThrNANANA18LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.01267 ml/g Direct iodination 26536593
b3pdb_1119PhrCACET1SYPGWSWSer-Tyr-Pro-Gly-Trp-Ser-TrpNANANA7LinearNAbacterialNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00133 mL/(g x min) Direct iodination 26536593
b3pdb_1120PhrCACET1SYPGWSWSer-Tyr-Pro-Gly-Trp-Ser-TrpNANANA7LinearNAbacterialNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.03553 ml/g Direct iodination 26536593
b3pdb_1124Neuromedin UYKVNEYQGPVAPSGGFFLFRPRNTyr-Lys-Val-Asn-Glu-Tyr-Gln-Gly-Pro-Val-Ala-Pro-Ser-Gly-Gly-Phe-Phe-Leu-Phe-Arg-Pro-Arg-AsnNANANA25LinearNAbacterialNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00131 mL/(g x min) Direct iodination 27040796
b3pdb_1128NeurotensinELYENLPRRPYILpGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-LeuNANANA13LinearNAbacterialNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.03383 ml/g Direct iodination 27040796
b3pdb_1129NeurotensinELYENLPRRPYILpGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-LeuNANANA13LinearNAbacterialNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00075 mL/(g x min) Direct iodination 27040796
b3pdb_1130NeurotensinELYENLPRRPYILpGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-LeuNANANA13LinearNAbacterialNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.01125 ml/g Direct iodination 27040796
b3pdb_1134Neuromedin NKIPYILLys-Ile-Pro-Tyr-Ile-LeuNANANA6LinearNAhumanNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant,initial 0.02299 ml/(g x min) Direct iodination 27040796
b3pdb_1137Neuromedin BGNLWATGHFMGly-Asn-Leu-Trp-Ala-Thr-Gly-His-Phe-Met-NH2NANANA10LinearNAhumanNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.00012 mL/(g x min) Direct iodination 27040796
b3pdb_1138Neuromedin BGNLWATGHFMGly-Asn-Leu-Trp-Ala-Thr-Gly-His-Phe-Met-NH2NANANA10LinearNAhumanNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.00799 ml/g Direct iodination 27040796
b3pdb_1153BeauvericinNANANANANA6LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.01115 mL/(g x min) Direct iodination 27349679
b3pdb_1154BeauvericinNANANANANA6LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.02191 ml/g Direct iodination 27349679
b3pdb_1156PepH1VQQLTKRFSLValGlnGlnLeuThrLysArgPheSerLeuNANANA10LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA % injected dose 0.02 %/g 99mTc(CO)3+ 28263555
b3pdb_1159PepH3AGILKRWAlaGlyIleLeuLysArgTrpNANANA7LinearNAviralNANANANANANANAIntravenous NANA NA Permeability NA NA NA % injected dose 0.03 %/g 99mTc(CO)3+ 28263555
b3pdb_1177L57TWPKHFDKHTFYSILKLGKHThr-Trp-Pro-Lys-His-Phe-Asp-Lys-His-Thr-Phe-Tyr-Ser-Ile-Leu-Lys-Leu-Gly-Lys-HisNANANA20LinearNAHemoglobinNANANANANANANAIntravenous NANA NA Permeability NA NA NA % injected dose 0.042 %/g Direct iodination 29090274
b3pdb_1178D3D3RPRTRLHTHRNRRPRTRLHTHRNRArg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAHemoglobinNANANANANANANAIntravenous NANA NA Permeability NA NA NA Brain to plasma ratio 0.6 H3/C14 27086111
b3pdb_1179RD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Brain to plasma ratio 0.6 H3/C14 27086111
b3pdb_1180RD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Peak response 0.3 µL/(g x min) H3/C14 27086111
b3pdb_1181RD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.0003 ml/(g x min) H3/C14 27086111
b3pdb_1182RD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.0512 ml/g H3/C14 27086111
b3pdb_1183cRD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Peak response 2 µL/(g x min) H3/C14 29225107
b3pdb_1184cRD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.002 ml/(g x min) H3/C14 29225107
b3pdb_1185cRD2D3PTLHTHNRRRRRRPRTRLHTHRNRPro-Thr-Leu-His-Thr-His-Asn-Arg-Arg-Arg-Arg-Arg-Arg-Pro-Arg-Thr-Arg-Leu-His-Thr-His-Arg-Asn-ArgNANANA24LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Initial disrobution volume 0.1955 ml/g H3/C14 29225107
b3pdb_1186AH-DSGSWLRDVWDWICTVLTDFKTWLQSKLSer-Gly-Ser-Trp-Leu-Arg-Asp-Val-Trp-Asp-Trp-Ile-Cys-Thr-Val-Leu-Thr-Asp-Phe-Lys-Thr-Trp-Leu-Gln-Ser-Lys-LeuNANANA27LinearNAChemically synthesizedNANANANANANANAIntravenous NANA NA Permeability NA NA NA Unidirectional influx rate constant 0.0003853 mL/(g x min) NA 30349030