ID Reference Source Clone name Sequence Motif Target-tumor Target-cell Receptors-biomarker Phage/Library In vitro/Ex-vivo In vivo Homing/targeting Payloads patent
1160Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.LSDCLSDGKRKCNAHuman melanomaLymphatic vesselPodoplanin, Prox-1,LYVE-1 and VEGFR-10T7 phage/CX7C peptide libraryC8161 human melanoma, MDA-MB-435 human breast cancerMice bearing C8161 cells human cancer xenograftsHomingRadioactive indium, proapoptotic peptideUS 2007/0219134A1
1161Zhang L et al. Cancer Res. 2006 Jun 1;66(11):5696-706.NACLDGGRPKCNAHuman melanomaLymphatic vesselPodoplanin,Prox-1,LYVE-1 and VEGFR-10T7 phage/CX7C peptide libraryC8161 human melanoma, MDA-MB-435 human breast cancerMice bearing C8161 cells human cancer xenograftsHomingFluoresceineNA
1226Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAPRPGAPLAGSWPGTSPRPMelanoma, Pancreatic, Brain cancerAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryHuman tumor tissues of islet cells of pancreas, glioblastoma of brain.5-week-old C57BL/6 male bearing B16BL6 melanoma cellsHomingRadionuclide PRP-Lip -Andramycin drugEP1122262A4
1227Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAADGAPRPGAPLAPRPMelanomaAngiogenic endothelial cellVEGFNANA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHomingNANA
1228Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NADRWRPALPVVLFPLHWRPMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHomingNAUS 6,753,310 B1
1229Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAASSSYPLIHWRPWARNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHomingNAUS 6,753,310 B1
1230Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NADRWRPALPWRPMelanomaAngiogenic endothelial cellVEGFNANA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHomingNANA
1231Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAIHWRPWARWRPMelanomaAngiogenic endothelial cellVEGF-CNANA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHomingNANA
1232Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAAAEWLDAFFVRHVDRNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHoming (Phage display clone)NAUS 6,753,310 B1
1233Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAGDVWLFLTSTSHFARNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHoming (Phage display clone)NAUS 6,753,310 B1
1234Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAGCSVSSVGALCTHVNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHoming (Phage display clone)NANA
1235Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAAPCCSHLDASPFQRPNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHoming (Phage display clone)NAUS 6,753,310 B1
1236Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NAAQSNFVTWGYNVAVNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHoming (Phage display clone)NANA
1237Oku N et al. Oncogene. 2002 Apr 18;21(17):2662-9.NARASDVGSDVVPRYPFNAMelanomaAngiogenic endothelial cellVEGFM13 phage/15 mer peptide libraryNA5-week-old C57BL/6 male bearing B16BL6 melanoma cells derived tumorHoming (Phage display clone)NAUS 6,753,310 B1
1262Chen Y et al. Cancer Res. 2001 Mar 15;61(6):2434-8.NACRGDCGGKWCFRVCYRGICYRRCRRGDProstate cancer, MelanomaTumor cell and Endothelial cellIntegrinsNAThe TSU human prostate cancer cells, B16 melanoma, nontumorigenic cell lines Cos-7, and NIH-3T3CAMs of 10-day-old chicken embryos, C57BL/6 mice bearing B16 melanoma HomingAntimicrobial peptideNA
1293Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NATAASGVRSMHNAMelanomaTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NG2 knockout mice, NG2 expressing wild mice.HomingNAUS 6,528,481 B1
1294Burg MA et al. Cancer Res. 1999 Jun 15;59(12):2869-74.NALTLRWVGLMSNAMelanomaTumor cell and angiogenic tumor vasculatureProteoglycanPhage/linear 10 mer peptide libraryNG2 fragments (transfected human embryonic kidney 293 cells )NG2 knockout mice, NG2 expressing wild mice.HomingNAUS 6,528,481 B1
1311Arap W et al. Science. 1998 Jan 16;279(5349):377-80.NACVLNGRMECNGRMouse melanomaEndothelial cellIntegrinM13 Phage/CX3CX3CX3C peptide libraryNAMice bearing MDA-MB-435derived tumors, SLK cell derived human Kaposi's sarcoma xenograftsHomingNAUS2009/0257951 A1
1316Iida J et al. J Biol Chem. 1998 Mar 6;273(10):5955-62.SG1KKEKDIMKKTINAMelanomaNAAlpha- 4 beta -1NAHuman melanoma cells (A375SM)NATargetingOVANA
1317Yun Z et al. Cancer Res. 1996 Jul 1;56(13):3103-11.NAGRGDSPKNAMelanomaNAAlpha- 4 beta -1NAMurine RAW117NATargetingFITCNA
1325Samanta S et al. Biomaterials. 2010 Mar;31(7):1787-97.NACRGDGWCRGDMelanomaTumor vesselIntegrins Alpha- 5 beta -1NANAMice bearing the aggressive B16F10 tumorHomingNANA
1326Samanta S et al. Biomaterials. 2010 Mar;31(7):1787-97.RGDGWK-lipopeptideRGDGWKRGDMelanomaTumor vesselIntegrins Alpha -5 beta- 1NANAMice bearing the aggressive B16F10 tumorHomingAnticancer-p-53 geneNA
1362Wu J et al. J Biosci. 2009 Jun;34(2):213-20.Clone AAHLPIVRASLPSLIIPP/LPI/IL/PMelanomaNAADAM15, ADAMs (A Disintegrin and Metalloproteinases)M13 phage/12-mer peptide libraryHuman melanoma A375-M cellsNATargetingNANA
1363Wu J et al. J Biosci. 2009 Jun;34(2):213-20.Clone DTPMNHHSQHAERNAMelanomaNANAM13 phage/12-mer peptide libraryHuman melanoma A375-M cellsNATargetingNANA
1364Wu J et al. J Biosci. 2009 Jun;34(2):213-20.Clone BGNIIPDRPMHPTNAMelanomaNANAM13 phage/12-mer peptide libraryHuman melanoma A375-M cellsNATargetingNANA
1365Wu J et al. J Biosci. 2009 Jun;34(2):213-20.Clone CFPSSLIIPPLPNNAMelanomaNANAM13 phage/12-mer peptide libraryHuman melanoma A375-M cellsNATargetingNANA
1483Pasqualini R et al. Nat Biotechnol. 1997 Jun;15(6):542-6.NACDCRGDCFCNAMalignant melanomas and breast carcinomaNAAlpha -5 beta-1 integrinPhage /RGD-4CLibraryMDA-MB-435 breast cancer cells, murine B16B15b melanoma,C8161 human melanomaFemale 2-month old BALB/ C miceHomingNANA
1586NAClone 4CLSGSLSCNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1587NA Clone 18WGTGLCNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1588NAClone 107GICKDDWCQNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1589NAClone 108TSCDPSLCENAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1590NAClone 109KGCGTRQCWNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1591NAClone 110YRCREVLCQNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1592NAClone 111CWGTGLCNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1593NAClone 112WSCADRTCMNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1594NAClone 113AGCRLKSCANAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1595NAClone 114SRCKTGLCQNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1596NAClone 115PICEVSRCWNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1597NAClone 116WTCRASWCSNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1598NAClone 117GRCLLMQCRNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1599NAClone 118TECDMSRCMNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1600NA Clone 119ARCRVDPCVNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1601NA Clone120CIEGVLGGCNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1602NA Clone 121CSVANSCNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1603NAClone 122CSSTMRCNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1604NAClone 123SIDSTTFNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1605NAClone 124GPSRVGGNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1606NAClone125WWSGLEANAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1607NAClone126LGTDVRQNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1608NAClone 127LVGVRLLNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1609NAClone 128GRPGDJWNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1610NAClone 129TVWNPVGNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1611NAClone 130GLLLVVPNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1612NAClone131FAATSAENAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1613NAClone 132WCCRQFNNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1614NAClone 133VGFGKALNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1615NAClone 134DSSLRLPNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1616NAClone 135KLWCAMSNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1617NAClone 136SLVSFLGNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1618NAClone 137GSFAFLVNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1619NAClone 138IASVRWANAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1620NAClone 139TWGHLRANAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1621NAClone 140QYREGLVNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1622NAClone 141QSADRSVNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1623NAClone 142YMFWTSRNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1624NAClone 143LVRRWYLNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1625NAClone 144TARGSSRNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1626NAClone 145TTREKNLNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1627NAClone 146PKWLLFSNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1628NAClone 147LRTNVVHNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1629NAClone 148AVMGLAANAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1630NAClone 149VRNSLRNNAMouse melanoma tumorNANAM13 phage /CX5 C , CX 6C ) or CX7C peptide libraryNAMice bearing B16B15b MelanomaHoming (Phage display clone)NAUS 6,180,084 B1
1684NAClone 7IELLQARNAMelanomaNAE-selectinT7 phage /(CX7C) peptide libraryHL-60 Cell lineMice bearing B16 cellsHomingBiotinUS 7,470,658 B2
1750Dai W et al. Nanomedicine. 2012 Jan 31.NAPHSCNKNAMelanomaNAIntegrinsNAB16F10 cells overexpressing integrinMale C57BL/6 mice HomingLiposomes loaded doxorubicinNA
1755Matsuo AL et al . Mol Cancer Res 2011 Nov;9(11):NACVNHPAFACNAMelanomaNA NA T7 phage / CX7C peptide libraryNASyngeneic miceHoming Antiangiogenic peptide (HTMYYHHYQHHL)NA