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Details of CPPsite entry with Sequence RQIKIWFQNRRMKWAK
Primary information
PEPTIDE SEQUENCERQIKIWFQNRRMKWAK
CPPsite ID 1129,
PEPTIDE NAMEAla57 substitution mutant of pAntp (43-58)
CHIRALITYL
LINEAR/CYCLICLinear
SOURCEProtein derived
CATEGORYProbably Amphipathic
SUB CELLULAR LOCALIZATIONProbably Cytosol and nucleus, nucleoi
N-TERMINAL MODIFICATIONBiotinylation (Labeled with Biotinyl-beta-Alanine)
C-TERMINAL MODIFICATIONAmidation
UPTAKE EFFICIENCYLow (20% relative to (pAntp) (43-58))
PROPOSED UPTAKE MECHANISMNon-endocytic pathway
INVITRO/INVIVOIn vitro
CELL LINEHaCat/ A549 cells
CARGOBiotin
PMID10784032
PATENTUS 7153931
Tertiary Structure
(Technique)
1129 (PEPstrMOD),