Details of CPPsite entry with Sequence KRPTMRFRYTWNPMK |
| Primary information | |
|---|---|
| PEPTIDE SEQUENCE | KRPTMRFRYTWNPMK |
| CPPsite ID | 2735, |
| PEPTIDE NAME | 44 |
| CHIRALITY | L |
| LINEAR/CYCLIC | Linear |
| SOURCE | Synthetic |
| UPTAKE EFFICIENCY | primary myelogenous leukaemic cells (AML) showed uptake of CPP44, but not of TAT or CPP2 at comparable concentrations, showed poor penetration into normal fibroblasts |
| INVITRO/INVIVO | In vitro and in vivo |
| CELL LINE | Many Human neoplastic cells including HeLa, Lovo, A549, MCF-7,MKN45,HepG2, LNCap, KPK,U2OS, RC-15,RD-ES,H28,K562,U251,NHDF |
| In VIVO MODEL | NOD-SCID mice model of xenograft human tumour cells |
| CARGO | Fluorophore (FITC) |
| PMID | 22805558 |
| PATENT | Unknown |
| Tertiary Structure (Technique) | 2735 (PEPstrMOD), |