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Details of RareLED ID Assay_1049
Primary information
GENETPP1
NUMBER OF ASSAY17
ASSAY IDs214629 214628 282917 214627 214626 214630 329747 329748 52104 52099 49450 49447 47574 329749 52105 52100 48563
Assay Name1. Inhibition potency against Cholecystokinin-8-Inactivating Peptidase (Serine Peptidase).,2. Inhibition potency against Cholecystokinin-8-Inactivating Peptidase (Serine Peptidase).,3. Inhibition of TPPII in rat cerebral membrane,4. Inhibitory activity against tripeptidyl peptidase II purified from rat liver,5. Inhibition of Tripeptidyl-peptidase II purified from a rat liver post-lysosomal fraction.,6. Inhibition of Tripeptidyl-peptidase II purified from a rat liver post-lysosomal fraction.,7. Inhibition of human tripeptidyl peptidase2 from erythrocytes,8. Agonist activity at mu opioid receptor in mouse model,9. Compound was tested for the inhibitory activity against chitin synthetase,10. Compound was tested for the inhibitory activity against chitin synthetase in the mixed membrane preparation from Candida albicans,11. Concentration at which 50% of the Candida albicans cells were not viable,12. Compound was tested for the inhibitory activity against Candida albicans cell growth,13. Millimolar concentration at which some morphological effects in Candida albicans cells (about 5% of cells) was determined,14. Agonist activity at mouse delta opioid receptor in mouse model,15. Inhibition constant (KI) for the mmf chitin synthetase assay performed at constant inhibitor and varying substrate concentrations,16. Compound was tested for the inhibitory activity against chitin synthetase in the permeabilised cell assay,17. Millimolar concentration of the lowest concentration that clearly inhibited the cell growth of Candida albicans was determined
ACTIVITYSubstance BioActivity: 16 Active, 1 Activity <= 1 µM, 59 Tested Substance BioActivity: 1 Tested Substance BioActivity: 32 Active, 15 Activity <= 1 µM, 36 Tested Substance BioActivity: 5 Active, 5 Activity <= 1 µM, 8 Tested Substance BioActivity: 12 Active, 8 Activity <= 1 µM, 15 Tested Substance BioActivity: 13 Active, 11 Activity <= 1 µM, 21 Tested Substance BioActivity: 1 Active, 1 Activity <= 1 µM, 1 Tested Substance BioActivity: 2 Active, 1 Activity <= 1 nM, 2 Activity <= 1 µM, 2 Tested Substance BioActivity: 2 Active, 3 Tested Substance BioActivity: 3 Active, 8 Tested Substance BioActivity: 5 Tested Substance BioActivity: 3 Tested Substance BioActivity: 2 Active, 8 Tested Substance BioActivity: 2 Active, 1 Activity <= 1 nM, 2 Activity <= 1 µM, 2 Tested Substance BioActivity: 1 Active, 1 Activity <= 1 µM, 5 Tested Substance BioActivity: 1 Active, 1 Activity <= 1 µM, 8 Tested Substance BioActivity: 8 Tested