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Browse result page of AntiTbPdb

The total number entries retrieved from this search are 738
IDNameSequenceN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicLengthChiralityNatureSourceOriginSpeciesStrainInhibition ConcentrationIn vitro/ In vivoCell LineIntracellular InhibitionCytotoxicityAnimal ModelEffective Dose in model organismImmune ResponceMechanism of ActionTargetCombination TherapyOther ActivitiesYear of PublicationPubmed ID/ Patent No.
antitb_1875GranF2VCRTGRSRWRDVCRNFMRRYQSRFreeFreeNoneLinear23LCationicProtein DerivedPeptide derived from Granulysin proteinMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1876Dhvar4KRLFKKLLFSLRKYFreeFreeNoneLinear14LCationicProtein DerivedHuman salivary Histatin derivativeMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1877Crot(1–9,38–42)YKQCHKKGGKKGSGFreeFreeNoneLinear14LCationicNaturalCrotamine, a toxin of Crotalus durissus terrificusMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1878CM15KWKLFKKIGAVLKVLFreeFreeNoneLinear15LCationicSyntheticFrom Cecropin A and Melittin sequencesMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at 18.9 ± 1.71 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1879MelittinGIGAVLKVLTTGLPALISWIKRKRQQFreeFreeNoneLinear26LCationicNaturalVenom of Apis melliferaMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at 0.339 ± 0.0854 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1880OT20TKPKGTKPKGTKPKGTKPKGFreeFreeNoneLinear20LCationicSyntheticTetramer derivative of tuftsin sequenceMycobacterium tuberculosisMycobacterium tuberculosis H37Rv (ATCC 27294)MIC >300 μMIn vitroRBCNA50% hemolysis at >300 μMNA NANANANANAAntibacterial (Streptococcus pneumoniae)201728314993
antitb_1881Polydim-I AVAGEKLWLLPHLLKMLLTPTPFreeFreeNoneLinear22LAmphipathicNaturalIsolated from the venom of the Neotropical wasp Polybia dimorpha Mycobacterium abscessusMycobacterium abscessus subsp. massiliense isolates GO 01, GO 06, GO 07, GO 08, GO 13, and GO 18, CRM0020 (Mycobacterium abscessus subsp. massiliense), and ATCC19977 (Mycobacterium abscessus subsp. abscessus)MIC = 60.8 μg/mL BothPeritoneal macrophages, J774 macrophages cells, human red blood cells Treatment of infected macrophages with 7.6 μg/mL of Polydim-I decreased approximately 50% of the bacterial load Non-cytotoxic, 10% cytotoxicity on J774 cells at concentrations above 121.6 μg/mL (10%) and concentrations up to 121.6 μg/mL presented less than 2.5% of hemolytic activity6 to 8 weeks old BALB/c and IFN-γKO (Knockout) female mice 2 mg/kg/mLW shows 90% reduction in bacterial loadNACell wall disruption Cell wallNoneNA201626930596
antitb_1893Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC50 = 15.8 ± 4.5 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1894Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC90 = 34.6 ± 22.4 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1895Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC50 = 11.0 ± 4.1 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1896Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC90 = 65.8 ± 19.13 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1897Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC50 = 15.2± 2.9 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1898Human lactoferricin 1-11GRRRRSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC90 = 37.9 ± 15.9 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1899Human lactoferricin 1-11GKKKKSVQWCAFreeFreeNoneLinear11LCationicNaturalDerived from human lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1900Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC50 = 14.2 ± 1.5 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1901Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2447 smTIC90 = 18.9 ± 4.0 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1902Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC50 = 8.0 ± 1.5 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1903Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smTIC90 = 22.8 ± 9.1 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1904Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC50 = 12.4± 0.3 μMIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1905Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium avium 2-151 smDIC90 = 21.5± 4.0 μMIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1906Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14DCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1907Bovine lactoferricin 17-30FKCRRWQWRMKKLGFreeFreeNoneLinear14DCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1908Bovine lactoferricin 17-30 all KFKCKKWQWKMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1909Bovine lactoferricin 17-30 all KFKCKKWQWKMKKLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1910Bovine lactoferricin 17-30 all RFRCRRWQWRMRRLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 50% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1911Bovine lactoferricin 17-30 all RFRCRRWQWRMRRLGFreeFreeNoneLinear14LCationicNaturalDerived from bovine lactoferricin proteinMycobacterium aviumMycobacterium aviumMycobacterium avium 2447 smTIn vitroNATratment with this concentration inhibit 90% bacterial growthNANA NANANALipid bilayerNANA201424709266
antitb_1912NoneILSLRWRWKWWKKFreeFreeNoneLinear13LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatisMIC = 8 μMIn vitroJ774.16 mouse macrophages and A549 human lung epithelial cellsNANo cytotoxicity against J774.16 mouse macrophages and A549 human lung epithelial cellsNA NANANALipid bilayerNAAntibacterial against Streptococcus pyogenes, Streptococcus agalactiae, Streptococcus pneumoniae ATCC 49619, Klebsiella pneumoniae, Pseudomonas aeruginosa ATCC27853, Bacillus subtilis BGSC 1A1. 201626902758
antitb_1913NoneILSLRWRWKWWKKFreeFreeNoneLinear13LCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis mc2 6020MIC = 32 μMIn vitroJ774.16 mouse macrophages and A549 human lung epithelial cellsNANo cytotoxicity against J774.16 mouse macrophages and A549 human lung epithelial cellsNA NANANALipid bilayerNAAntibacterial against Streptococcus pyogenes, Streptococcus agalactiae, Streptococcus pneumoniae ATCC 49619, Klebsiella pneumoniae, Pseudomonas aeruginosa ATCC 27853, Bacillus subtilis BGSC 1A1. 201626902758
antitb_1914NoneILSLRWRWKWWKKFreeFreeNoneLinear13LCationicSyntheticNAMycobacterium bovis Mycobacterium bovis BCG pasteur strainMIC = 32 μMIn vitroJ774.16 mouse macrophages and A549 human lung epithelial cellsNANo cytotoxicity against J774.16 mouse macrophages and A549 human lung epithelial cellsNA NANANALipid bilayerNAAntibacterial against Streptococcus pyogenes, Streptococcus agalactiae, Streptococcus pneumoniae ATCC 49619, Klebsiella pneumoniae, Pseudomonas aeruginosa ATCC 27853, Bacillus subtilis BGSC 1A1. 201626902758
antitb_1915Laterosporulin 10ACVNQCPDAIDRFIVKDKGCHGVEKKYYKQVYVACMNGQHLYCRTEWGGPCQLFreeFreeDisulphide bond between residues 2-43, 6-35 and 20-51 Cyclic53DCationicNaturalDerived from Brevibacillus species SKDU10Mycobacterium smegmatisMycobacterium smegmatis MC2 155MIC = 45 μMIn vitro and ex vivoRAW 264.7 murine macrophageNANo cytotoxicity upto 40 μM/ml concentrationNA NANANACell wall pore formation0.00625 μM of rifampicin with 0.25 μM of peptide, a fourfold reduction in MIC of rifampicin against H37 RVAntibacterial against Staphylococcus aureus MTCC 1430, Bacillus subtilis MTCC 121, Pseudomonas aeruginosa MTCC 1934, Vibrio cholerae MTCC 3904, Escherichia coli MTCC 1610201627267959
antitb_1949YD-1APKGVQGPNGFreeAmidationNoneLinear10LNANaturalDerived from Bacillus amyloliquefaciens CBSYD1Mycobacterium smegmatisMycobacterium smegmatis ATCC 9341MIC = 8 μg/mlIn vitroNANANANA NANANACell wall pore formationNAAntibacterial against gram negative such as Alcaligenes faecalis ATCC 1004, Salmonella Typhimurium KCTC 1925 etc and gram positive bacteria such as Enterococcus faecalis ATCC 29212, Micrococcus luteus ATCC 9341, Staphylococcus aureus KCTC 1928201728050849
antitb_1950NDBP-5IFSAIAGLLSNLLFreeFreeNoneLinear13LCationicNaturalDerived from scorpion hadrurus gertschiMycobacterium abscessus Mycobacterium abscessus subsp. Massiliene GO01MIC = 100 μMIn vitroHuman erythrocyteNANo cytotoxicityBALB/c mice 2mg/kgIFN-y productionNANANANA201728275372
antitb_1951NDBP-5IFSAIAGLLSNLLFreeFreeNoneLinear13LCationicNaturalDerived from scorpion hadrurus gertschiMycobacterium abscessusMycobacterium abscessus subsp. Massiliene GO06MIC = 100 μMIn vitroHuman erythrocyteNANo cytotoxicityBALB/c mice 2mg/kgIFN-y productionNANANANA201728275372
antitb_1952NDBP-5IFSAIAGLLSNLLFreeFreeNoneLinear13LCationicNaturalDerived from scorpion hadrurus gertschiMycobacterium abscessusMycobacterium abscessus subsp. Massiliene GO08MIC = 100 μMIn vitroHuman erythrocyteNANo cytotoxicityBALB/c mice 2mg/kgIFN-y productionNANANANA201728275372
antitb_1953Wollamide- BWAlVNxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC > 80 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1954Wollamide- BALlVNxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC > 80 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1955Wollamide- BWLlVAxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC > 20 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1956Wollamide- BWLlANxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC > 80 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1957Wollamide- BWLaVNxFreeFreeThird residue is D-alanine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC > 80 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1958Wollamide- BWLlINxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 1.1 μMIn vitroHepG2 cell lineNACytoxic above > 50 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1959Wollamide- BWLlMNxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC > 80 μMIn vitroNANANANA NANANAcell wall pore formationNANA201728423019
antitb_1960Wollamide- BWLlVxxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC =2.5 μMIn vitroHepG2 cell lineNACytoxic above > 50 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1961Wollamide- BWLlISxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC =15 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1962Wollamide- BWLlIXxFreeFreeThird residue is D-leucine, fifth residue is tertiary butyl serine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 40 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1963Wollamide- BWLlIIxFreeFreeThird residue is D-leucine and x= ornithineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 3.1 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1964Wollamide- BWLlINrFreeFreeThird residue is D-leucine and r= D- arginineCyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 0.6 μMIn vitroNANANANA NANANAcell wall pore formationNANA201728423019
antitb_1965Wollamide- BxLlVNxFreeFreeFirst residue is D- phenyalanine, Third is D-leucine and sixth is D-ornithine Cyclic6DCationicSyntheticNAMycobacterium tuberculosisMycobacterium tuberculosis H37RvMIC = 40 μMIn vitroHepG2 cell lineNACytoxic above > 100 μMNA NANANAcell wall pore formationNANA201728423019
antitb_1966HIDFS1GFGCPFNARRCHRHCRSIRRRAGYCAGRLRLTCTCVRFreeFreeNoneLinear37LCationicNaturalDerived from Haemaphysalis longicornisMycobacterium bovisMycobacterium bovisMIC50 = 0.2 μMIn vitroA549, 293 T, K562 and THP1 cellsNANo cytotoxicity at 20 μMNA NANANANANAAntiibacterial against Bacillus pumilus, Micrococcus luteus, Pseudomonas aeruginosa, Escherichia coli201728446822
antitb_1967HIDFS2GFGCPLNQGACHRHCRSIRRRGGYCSGIIKQTCYFreeFreeNoneLinear34LCationicNaturalDerived from Haemaphysalis longicornisMycobacterium bovisMycobacterium bovisMIC50 = 0.5μMIn vitroA549, 293 T, K562 and THP1 cellsNANo cytotoxicity at 20 μMNA NANANANANAAntiibacterial against Bacillus pumilus, Micrococcus luteus, Pseudomonas aeruginosa, Escherichia coli201728446822
antitb_1968HIDFS1GFGCPFNARRCHRHCRSIRRRAGYCAGRLRLTCTCVRFreeFreeNoneLinear37LCationicNaturalDerived from Haemaphysalis longicornisMycobacterium bovisMycobacterium bovisMIC50 = 0.5 μMIn vitroA549, 293 T, K562 and THP1 cellsNANo cytotoxicity at 20 μMNA NANANANANAAntiibacterial against Bacillus pumilus, Micrococcus luteus, Pseudomonas aeruginosa, Escherichia coli201728446822