| Primary information |
|---|
| ID | 12276 |
| Uniprot ID | P0DL36 |
| Description | Mu-scoloptoxin(03)-Ssm2a (Mu-SLPTX(03)-Ssm2a) (Mu-scoloptoxin-Ssm6a) (Mu-SLPTX-Ssm6a) |
| Organism | Scolopendra subspinipes |
| Txonomy | Eukaryota; Opisthokonta; Metazoa; Eumetazoa; Bilateria; Protostomia; Ecdysozoa; Panarthropoda; Arthropoda; Mandibulata; Myriapoda; Chilopoda (centipedes); Pleurostigmophora; Epimorpha; Scolopendromorpha; Scolopendridae; Scolopendra; Scolopendra subspinipes (Vietnamese centipede) |
| Subcellular Location | Secreted |
| Developmental Stage | NA |
| Similarity | Belongs to the scoloptoxin-03 family. |
| Tissue Specificity | Expressed by the venom gland. |
| Post Translational Modification | NA |
| Function | Gating-modifier toxin that inhibits voltage-gated sodium channel with a preference for hNav1.7/SCN9A (IC(50)=25.4 nM) over hNav1.1/SCN1A (IC(50)=4.1 uM); hNav1.2/SCN2A (IC(50)=813 nM); and hNav1.6/SCN8A (IC(50)=15.2 uM) |
| Length | 112 |
| Molecular Weight | 12 |
| Name | NA |
| Sequence | NA |
| Sequence map | NA |
| PDB ID | 2MUN; 2MZ4; |
| Drugpedia | NA |
| Receptor | NA |
| Domain | Is exclusively composed of 4 tightly packed alpha |
| Pharmaceutical Use | NA
|