Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0004339
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1Lck%ACTIVITY RELATIVE TO 100%DMSO---110 µM---
2YES1%ACTIVITY RELATIVE TO 100%DMSO---410 µM---
3EPH-B3%ACTIVITY RELATIVE TO 100%DMSO---510 µM---
4RIPK2%ACTIVITY RELATIVE TO 100%DMSO---1010 µM---
5MINK1%ACTIVITY RELATIVE TO 100%DMSO---1210 µM---
6Src%ACTIVITY RELATIVE TO 100%DMSO---1310 µM---
7PKD1%ACTIVITY RELATIVE TO 100%DMSO---1410 µM---
8MNK2%ACTIVITY RELATIVE TO 100%DMSO---2110 µM---
9MELK%ACTIVITY RELATIVE TO 100%DMSO---2510 µM---
10EPH-A2%ACTIVITY RELATIVE TO 100%DMSO---2610 µM---
11PHK%ACTIVITY RELATIVE TO 100%DMSO---2610 µM---
12CHK2%ACTIVITY RELATIVE TO 100%DMSO---2710 µM---
13CAMK1%ACTIVITY RELATIVE TO 100%DMSO---3010 µM---
14GCK%ACTIVITY RELATIVE TO 100%DMSO---3010 µM---
15p38a%ACTIVITY RELATIVE TO 100%DMSO---3010 µM---
16FGF-R1%ACTIVITY RELATIVE TO 100%DMSO---3110 µM---
17DYRK3%ACTIVITY RELATIVE TO 100%DMSO---3210 µM---
18AuroraB%ACTIVITY RELATIVE TO 100%DMSO---3310 µM---
19BRSK2%ACTIVITY RELATIVE TO 100%DMSO---3610 µM---
20BTK%ACTIVITY RELATIVE TO 100%DMSO---3610 µM---
21PRK2%ACTIVITY RELATIVE TO 100%DMSO---3610 µM---
22VEGFR%ACTIVITY RELATIVE TO 100%DMSO---3610 µM---
23NUAK1%ACTIVITY RELATIVE TO 100%DMSO---3710 µM---
24CK1%ACTIVITY RELATIVE TO 100%DMSO---4410 µM---
25MKK1%ACTIVITY RELATIVE TO 100%DMSO---4510 µM---
26BRSK1%ACTIVITY RELATIVE TO 100%DMSO---4610 µM---
27PIM1%ACTIVITY RELATIVE TO 100%DMSO---4610 µM---
28SmMLCK%ACTIVITY RELATIVE TO 100%DMSO---4810 µM---
29JNK1%ACTIVITY RELATIVE TO 100%DMSO---4910 µM---
30JNK2%ACTIVITY RELATIVE TO 100%DMSO---5010 µM---
31DYRK2%ACTIVITY RELATIVE TO 100%DMSO---5210 µM---
32SYK%ACTIVITY RELATIVE TO 100%DMSO---5710 µM---
33PKBb%ACTIVITY RELATIVE TO 100%DMSO---6110 µM---
34IKKB%ACTIVITY RELATIVE TO 100%DMSO---6210 µM---
35JNK3%ACTIVITY RELATIVE TO 100%DMSO---6210 µM---
36p38b%ACTIVITY RELATIVE TO 100%DMSO---6310 µM---
37MetNK1%ACTIVITY RELATIVE TO 100%DMSO---6410 µM---
38PIM3%ACTIVITY RELATIVE TO 100%DMSO---6610 µM---
39PAK5%ACTIVITY RELATIVE TO 100%DMSO---6810 µM---
40IRAK4%ACTIVITY RELATIVE TO 100%DMSO---7010 µM---
41IGF-1R%ACTIVITY RELATIVE TO 100%DMSO---7110 µM---
42MAPKAP-K3%ACTIVITY RELATIVE TO 100%DMSO---7210 µM---
43CSK%ACTIVITY RELATIVE TO 100%DMSO---7310 µM---
44CAMKKb%ACTIVITY RELATIVE TO 100%DMSO---7410 µM---
45RSK2%ACTIVITY RELATIVE TO 100%DMSO---7410 µM---
46MARK4%ACTIVITY RELATIVE TO 100%DMSO---7510 µM---
47PIM2%ACTIVITY RELATIVE TO 100%DMSO---7510 µM---
48SRPK1%ACTIVITY RELATIVE TO 100%DMSO---7510 µM---
49p38d%ACTIVITY RELATIVE TO 100%DMSO---7610 µM---
50MARK2%ACTIVITY RELATIVE TO 100%DMSO---7710 µM---
51PDK1%ACTIVITY RELATIVE TO 100%DMSO---7810 µM---
52IRR%ACTIVITY RELATIVE TO 100%DMSO---7910 µM---
53MLK1%ACTIVITY RELATIVE TO 100%DMSO---7910 µM---
54PAK2%ACTIVITY RELATIVE TO 100%DMSO---7910 µM---
55PAK4%ACTIVITY RELATIVE TO 100%DMSO---7910 µM---
56MST4%ACTIVITY RELATIVE TO 100%DMSO---8010 µM---
57MST2%ACTIVITY RELATIVE TO 100%DMSO---8110 µM---
58PKCa%ACTIVITY RELATIVE TO 100%DMSO---8210 µM---
59SGK1%ACTIVITY RELATIVE TO 100%DMSO---8210 µM---
60CHK1%ACTIVITY RELATIVE TO 100%DMSO---8310 µM---
61ERK1%ACTIVITY RELATIVE TO 100%DMSO---8310 µM---
62PAK6%ACTIVITY RELATIVE TO 100%DMSO---8310 µM---
63AMPK%ACTIVITY RELATIVE TO 100%DMSO---8410 µM---
64MLK3%ACTIVITY RELATIVE TO 100%DMSO---8410 µM---
65PRAK%ACTIVITY RELATIVE TO 100%DMSO---8410 µM---
66TBK1%ACTIVITY RELATIVE TO 100%DMSO---8410 µM---
67DYRK1A%ACTIVITY RELATIVE TO 100%DMSO---8510 µM---
68ERK8%ACTIVITY RELATIVE TO 100%DMSO---8510 µM---
69IR-HIS%ACTIVITY RELATIVE TO 100%DMSO---8510 µM---
70NEK6%ACTIVITY RELATIVE TO 100%DMSO---8510 µM---
71TTK%ACTIVITY RELATIVE TO 100%DMSO---8510 µM---
72MAPKAP-K2%ACTIVITY RELATIVE TO 100%DMSO---8610 µM---
73PKA%ACTIVITY RELATIVE TO 100%DMSO---8610 µM---
74PKCz%ACTIVITY RELATIVE TO 100%DMSO---8610 µM---
75S6K1%ACTIVITY RELATIVE TO 100%DMSO---8710 µM---
76AuroraA%ACTIVITY RELATIVE TO 100%DMSO---8810 µM---
77CDK2-CycA%ACTIVITY RELATIVE TO 100%DMSO---8810 µM---
78ERK2%ACTIVITY RELATIVE TO 100%DMSO---8810 µM---
79ROCK2%ACTIVITY RELATIVE TO 100%DMSO---8810 µM---
80GSK3b%ACTIVITY RELATIVE TO 100%DMSO---8910 µM---
81RSK1%ACTIVITY RELATIVE TO 100%DMSO---8910 µM---
82CK2%ACTIVITY RELATIVE TO 100%DMSO---9010 µM---
83IKKe%ACTIVITY RELATIVE TO 100%DMSO---9210 µM---
84LKB1%ACTIVITY RELATIVE TO 100%DMSO---9410 µM---
85MARK3%ACTIVITY RELATIVE TO 100%DMSO---9410 µM---
86p38g%ACTIVITY RELATIVE TO 100%DMSO---9410 µM---
87NEK2a%ACTIVITY RELATIVE TO 100%DMSO---9510 µM---
88HIPK3%ACTIVITY RELATIVE TO 100%DMSO---9610 µM---
89MSK1%ACTIVITY RELATIVE TO 100%DMSO---9610 µM---
90EF2K%ACTIVITY RELATIVE TO 100%DMSO---9910 µM---
91PKBa%ACTIVITY RELATIVE TO 100%DMSO---10010 µM---
92HIPK1%ACTIVITY RELATIVE TO 100%DMSO---10310 µM---
93HIPK2%ACTIVITY RELATIVE TO 100%DMSO---10410 µM---
94PLK1%ACTIVITY RELATIVE TO 100%DMSO---10910 µM---