Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0004326
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1Abl1-<0.5 nM-------
2B-Raf V600E2.1nM-------
3C-Raf-2.5nM-------
4DDR2-7nM-------
5EPHA2-11nM-------
6KDR-6.2nM-------
7LCK-170nM-------
8MEK-1400nM-------
9p38R-42nM-------
10PDGFR-47nM-------
11RET-0.8nM-------
12B-Rafwt4.2nM-------