Epidermal Growth Factor Receptor Inhibitor Database
Activity against kinases |
Molecule Id: EGIN0003428 |
S.No. |
Kinase |
Mutant |
IC50 |
Ki |
Kd |
Enz. inhib. (%) |
Inhib. Conc. |
Cellular IC50 |
Cell line |
Growth Factor |
1 | AKT | - | >5000 nM | - | - | - | - | - | - | - |
2 | CaMKII | - | >50000 nM | - | - | - | - | - | - | - |
3 | CDK2 | - | >10000 nM | - | - | - | - | - | - | - |
4 | c-kit | - | 370nM | - | - | - | - | - | - | - |
5 | FGFR1 | - | >5000 nM | - | - | - | - | - | - | - |
6 | Flk-1 | - | 40nM | - | - | - | - | - | - | - |
7 | GSK-3 | - | >5000 nM | - | - | - | - | - | - | - |
8 | IGF1R | - | >25000 nM | - | - | - | - | - | - | - |
9 | IKK | - | >10000 nM | - | - | - | - | - | - | - |
10 | Itk | - | >50000 nM | - | - | - | - | - | - | - |
11 | JAK3 | - | >50000 nM | - | - | - | - | - | - | - |
12 | Lck | - | >50000 nM | - | - | - | - | - | - | - |
13 | MAPKAPK2 | - | >50000 nM | - | - | - | - | - | - | - |
14 | MEK | - | >5000 nM | - | - | - | - | - | - | - |
15 | p38 | - | >5000 nM | - | - | - | - | - | - | - |
16 | PDGFR beta | - | 200nM | - | - | - | - | - | - | - |
17 | PKC alpha | - | >40000 nM | - | - | - | - | - | - | - |
18 | PKC beta | - | >40000 nM | - | - | - | - | - | - | - |
19 | PKC tau | - | >40000 nM | - | - | - | - | - | - | - |
20 | PKC zeta | - | >40000 nM | - | - | - | - | - | - | - |
21 | Src | - | >10000 nM | - | - | - | - | - | - | - |
22 | SRPK1 | - | >10000 nM | - | - | - | - | - | - | - |
23 | Syk | - | >50000 nM | - | - | - | - | - | - | - |
24 | VEGFR1 | - | 400nM | - | - | - | - | - | - | - |
25 | VEGFR2 | - | 23nM | - | - | - | - | - | - | - |