Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0003200
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1IGF->>10000nM-------
2JAK2->50000nM-------
3JAK3->50000nM-------
4JNK->50000nM-------
5LCK-1400 ± 100nM-------
6Insulin R-33000 ± 5000nM-------
7PDGFr-76 ± 13nM-------