Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0003118
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1CDK5/p25----59.83±0.5510 µM---
2CK1a1----100.18±3.1210 µM---
3CK2a----77.02±1.0810 µM---
4EGFR----32.67±0.6810 µM---
5ERK1----109.58±1.3210 µM---
6GSK-3b----18.57±0.0710 µM---
7IGF1R----96.24±3.8810 µM---
8JNK1----93.28±0.7910 µM---
9MAPKAPK2----78.23±0.9010 µM---
10TYRO3/SKY----96.72±1.4310 µM---