Epidermal Growth Factor Receptor Inhibitor Database
|
|
|
|
|
|
|
|
|
|
|
| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0002634 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | CDK4/Cyc | - | 1000000nM | - | - | - | - | - | - | - | ||||
| 2 | PKC | - | 1000000nM | - | - | - | - | - | - | - | ||||
| 3 | PKA | - | 2000000nM | - | - | - | - | - | - | - | ||||
| 4 | MAP | - | 30000nM | - | - | - | - | - | - | - | ||||
| 5 | CDK1/CycB1 | - | 7000nM | - | - | - | - | - | - | - | ||||
| 6 | CDK2/CycE | - | 7000nM | - | - | - | - | - | - | - | ||||