Epidermal Growth Factor Receptor Inhibitor Database
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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0002633 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | MAP | - | >25000nM | - | - | - | - | - | - | - | ||||
| 2 | PKA | - | >50000nM | - | - | - | - | - | - | - | ||||
| 3 | PKC | - | >50000nM | - | - | - | - | - | - | - | ||||
| 4 | CDK1/CycB1 | - | 130nM | - | - | - | - | - | - | - | ||||
| 5 | CDK2/CycE | - | 2110nM | - | - | - | - | - | - | - | ||||
| 6 | CDK4/Cyc | - | 6150nM | - | - | - | - | - | - | - | ||||