|
|
|
|
|
|
|
|
|
|
Activity against kinases | ||||||||||||||
Molecule Id: EGIN0002357 | ||||||||||||||
S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
1 | VEGFR1 | - | 160100 ± 28900nM | - | - | - | - | - | - | - | ||||
2 | PDGFR beta | - | 40300 ± 5100nM | - | - | - | - | - | - | - | ||||
3 | VEGFR-2/Flk-1 | - | 56300 ± 7100nM | - | - | - | - | - | - | - |