Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0002357
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1VEGFR1-160100 ± 28900nM-------
2PDGFR beta-40300 ± 5100nM-------
3VEGFR-2/Flk-1-56300 ± 7100nM-------