Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0002343
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1PDGFR beta->500000nM-------
2VEGFR2-17400 ± 1500nM-------
3DHFR human-42100nM-------