Epidermal Growth Factor Receptor Inhibitor Database


Activity against kinases
Molecule Id: EGIN0002045
S.No. Kinase Mutant IC50 Ki Kd Enz. inhib. (%) Inhib. Conc. Cellular IC50 Cell line Growth Factor
1VEGFR1->200000nM-------
2PDGFR beta->500000nM-------
3VEGFR2-132100 ± 16700nM-------