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Activity against kinases | ||||||||||||||
Molecule Id: EGIN0001289 | ||||||||||||||
S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
1 | VEGF-R2 | - | - | - | - | 30 | 100 µM | - | - | - | ||||
2 | Aurora-A | - | - | - | - | 73 | 100 µM | - | - | - | ||||
3 | CDK1 | - | - | - | - | <10 | 100 µM | - | - | - |