Epidermal Growth Factor Receptor Inhibitor Database
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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0001093 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | EphB4 | - | 1.4 ± 0.2 nM | - | - | - | - | - | - | - | ||||
| 2 | Flt4 | - | 8.7 ± 0.6 nM | - | - | - | - | - | - | - | ||||
| 3 | IGF1R | - | >10000 nM | - | - | - | - | - | - | - | ||||
| 4 | InsR | - | >26000 nM | - | - | - | - | - | - | - | ||||
| 5 | KDR | - | 1.5 ± 0.2 nM | - | - | - | - | - | - | - | ||||