Epidermal Growth Factor Receptor Inhibitor Database
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| Activity against kinases | ||||||||||||||
| Molecule Id: EGIN0000597 | ||||||||||||||
| S.No. | Kinase | Mutant | IC50 | Ki | Kd | Enz. inhib. (%) | Inhib. Conc. | Cellular IC50 | Cell line | Growth Factor | ||||
| 1 | FGFR1 | - | >50000nM | - | - | - | - | - | - | - | ||||
| 2 | PDGFR beta | - | >50000nM | - | - | - | - | - | - | - | ||||
| 3 | VEGFR2 | - | - | - | - | 0.8 | 20 µM | - | - | - | ||||
| 4 | FGFR1 | - | - | - | - | 10.5 | 20 µM | - | - | - | ||||
| 5 | PDGFR beta | - | - | - | - | 12.7 | 20 µM | - | - | - | ||||