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Browse result page of AntiTbPdb

The total number entries retrieved from this search are 202
IDNameSequenceN-Terminal ModificationC-Terminal ModificationChemical ModificationLinear/CyclicLengthChiralityNatureSourceOriginSpeciesStrainInhibition ConcentrationIn vitro/ In vivoCell LineIntracellular InhibitionCytotoxicityAnimal ModelEffective Dose in model organismImmune ResponceMechanism of ActionTargetCombination TherapyOther ActivitiesYear of PublicationPubmed ID/ Patent No.
antitb_1390LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /ml (after 6 hours)in vitroJ774.A1 macrophage cell lines34% bacteria is cleared NANA NANANANANANA201121790937
antitb_1391LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg/mlin vitroJ774.A1 macrophage cell lines41% bacteria is clearedNANA NANANANANANA201121790937
antitb_1392LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTES FreeFreeNoneLinear38LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg /ml (after 6 hours incubation)in vitroJ774.A1 macrophage cell lines67% bacteria is cleared NANA NANANANANANA201121790937
antitb_1393GEK-31RKSKEKIGKEFKRIVQR IKDFLRNLVPRTES FreeFreeNoneLinear33LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155NAin vitroJ774.A1 macrophage cell linesNANANA NANANANANANA201121790937
antitb_1394LL-18KEFKRIVQRIKDFLRNLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155NAin vitroJ774.A1 macrophage cell linesNANANA NANANANANANA201121790937
antitb_1395LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /mlin vitroJ774.A1 macrophage cell lines67% bacteria is cleared NANA NANANANANANA201121790937
antitb_1396LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /ml (after 6 hours)in vitroJ774.A1 macrophage cell lines89% bacteria is cleared NANA NANANANANANA201121790937
antitb_1397LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg/mlin vitroJ774.A1 macrophage cell lines81% bacteria is cleared NANA NANANANANANA201121790937
antitb_1398LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg /ml (after 6 hours incubation)in vitroJ774.A1 macrophage cell lines98% bacteria is cleared NANA NANANANANANA201121790937
antitb_1401LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 1μg /mlin vitroJ774.A1 macrophage cell lines51% bacteria is cleared NANA NANANANANANA201121790937
antitb_1402LLKKK-18KEFKRIVKRIKKFLRKLV FreeFreeNoneLinear19LCationicNaturalMurine macrophagesMycobacteria smegmatisM. smegmatis mc2 155MIC = 25μg/mlin vitroJ774.A1 macrophage cell lines80% bacteria is clearedNANA NANANANANANA201121790937
antitb_1485Dihydromycoplanecin A (DHMP A)not availableNANANABranched cyclic0DCationicNaturalDerived from ActinoplanesawajinensisMycobacteria smegmatisMycobacteria smegmatis ATCC 607MIC = 12.5 μg/mLin vitroNANANANA NANANANADHMP A + INHNA201525681127
antitb_1506SP508AR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 31.25 μg/mlin vitroNANANANA NANASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1507SP508BR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue Cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1508SP22AR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 7.8 μg/mlin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1509SP22BR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 31.25 μg/mlin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1510SP508AR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to15 mm at 31.25 mg/Lin vitroNANANANA NANASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1511SP508BR-(zDhb)-PVLALVAAVAATSAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue Cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to 18 mm at 62.5 mg/Lin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1512SP22AR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acidLinear18LCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to 12 mm 7.8 mg/Lin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1513SP22BR-(zDhb)-PVVAAVVAVAASAAYR =3-hydroxyldodecanoylFreeDhb= Dihydrobutyric acid, o-C=o linkage between 12 and 16 amino acid residue cyclic18DCationicNaturalDerived from Pseudomonas syringaeMycobacterium smegmatisMycobacterium smegmatis ATCC14468Reduction in zone to 14 mm at 31.25 mg/Lin vitroNANANANA NASpecific interaction with membraneNANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1520PR-39RRRPRPPYLPRPRPPPFFPPRLPPRIPPGFPPRFPPRFPFreeFreeNoneLinear39LCationicNaturalDerived from pig porcineMycobacterium smegmatis Mycobacterium smegmatis susceptible strain50 mg/Lin vitroNANANANA NANANANAAntibacterial against E.coli, S.aureus, bacillus, pseudomonas201525681127
antitb_1607TP-5RKDVYFreeAmidationNoneLinear4LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = > 1000mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1608RR-6RRRRRRFreeAmidationNoneLinear5LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = 125 mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1609RR-11RKDVYRRRRRRFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = 125 mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1610RY-11RRRRRRRKDVYFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-susceptible MIC = 125 mg/Lin vitro RAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1611TP-5RKDVYFreeAmidationNoneLinear4LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceNAin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1612RR-6RRRRRRFreeAmidationNoneLinear5LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1613RR-11RKDVYRRRRRRFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1614RY-11RRRRRRRKDVYFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNANANA201424411680
antitb_1615RY-11RRRRRRRKDVYFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis RIF-ResistanceMIC = 125 mg/Lin vitroRAW 264.7 mouse macrophageNAHC50= > 2000 mg/L on Human RBCNA NAStimulate TNF-α production Disrupt the mycobacterial membraneNARR-11 Peptide(31.25 mg/L) + Rifampicin (1.95mg/L)NA201424411680
antitb_1616LKLLKKLLKKFreeAmidationNoneLinear8LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 125 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1617PPPLLKKLLKKPFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 250 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1618CCCLLKKLLKKCFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 250 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1619IIILLKKLLKKIFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1620MMMLLKKLLKKMFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1621WWWLLKKLLKKWFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNANANA201526380930
antitb_1622LKLLKKLLKKFreeAmidationNoneLinear8LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 62.5 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1623PPPLLKKLLKKPFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 125 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1624CCCLLKKLLKKCFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 250 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1625IIILLKKLLKKIFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 15.6 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1626MMMLLKKLLKKMFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 15.6 μg/mlin vitroRAW 264.7 mouse macrophageNAHC50= >500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1627WWWLLKKLLKKWFreeAmidationNoneLinear10LCationicSyntheticNAMycobacterium smegmatisMycobacterium smegmatis ATCC14468MIC = 0.98 μg/mlin vitroRAW 264.7 mouse macrophageNA>500 μg/mlNA NANABacterial membrane pore formationNAPeptide + Rifampicin (0.98 μg/ml)NA201526380930
antitb_1628LL-37LLGDFFRKSKEKIGKEFKRIVQRIKDFLRNLVPRTESFreeFreeNoneLinear37LCationicSyntheticNAMycobacterium smegmatisMycobacteria smegmatis mc2 155MIC = 2400 μg/mlin vitro J774 macrophage cell linesNAIC50= 11226 μg/mlNA NAStimulation of TNF-α productioninhibit bacterial Atpase activityNANANA201526218806
antitb_1629LLAPRKSAKKIGKRAKRFreeFreeNoneLinear13LCationicNaturalNAMycobacterium smegmatisMycobacteria smegmatis mc2 155MIC = 600 μg/mlin vitro J774 macrophage cell linesNAIC50= 11226 μg/mlNA NAStimulation of TNF-α productioninhibit bacterial Atpase activityNANANA201526218806
antitb_1654Trichoderins Anot availableNANANANA0NANANaturalTrichoderma speciesMycobacteria smegmatisMycobacteria smegmatis (aerobic)IC90= 0.1 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201020483615
antitb_1657Trichoderins Anot availableNANANANA0NANANaturalTrichoderma speciesMycobacteria smegmatisMycobacteria smegmatis (hypoxic)IC90= 0.1 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201020483615
antitb_1660Trichoderins Anot availableNANANANA0NANANaturalTrichoderma speciesMycobacteria smegmatisMycobacteria smegmatis (aerobic)IC90= 0.02 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201020483615
antitb_1663Trichoderins Anot availableNANANANA0NANANaturalTrichoderma speciesMycobacteria smegmatisMycobacteria smegmatis (hypoxic)IC90= 0.02 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201020483615
antitb_1666Trichoderins Anot availableNANANANA0NANANaturalTrichoderma speciesMycobacteria smegmatisMycobacteria smegmatis (aerobic)IC90= 0.12 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201020483615
antitb_1669Trichoderins Anot availableNANANANA0NANANaturalTrichoderma speciesMycobacteria smegmatisMycobacteria smegmatis (hypoxic)IC90= 0.12 μg/mlin vitroHuman THP-1 cell linesNANANA NANAMicrobial membrane disruptionNANANA201020483615