A database of hormones and their receptors
Receptor

Search Result - 1

HMRbase accession number21207
Swiss-prot Accession numberQ9TT90 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismCanis familiaris (Dog)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Laurasiatheria; Carnivora; Caniformia; Canidae;Canis.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-522 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length907 Amino acids
Molecular weight98727
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 11768233
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Gene ID403588      
PDB IDN/A
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Search Result - 2

HMRbase accession number21208
Swiss-prot Accession numberQ8MIK0 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismCrocuta crocuta (Spotted hyena)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Laurasiatheria; Carnivora; Feliformia; Hyaenidae;Crocuta.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length912 Amino acids
Molecular weight99958
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 12242031
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Gene IDN/A
PDB IDN/A
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Search Result - 3

HMRbase accession number21209
Swiss-prot Accession numberO97776 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismEulemur fulvus collaris (Collared brown lemur)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Strepsirrhini;Lemuriformes; Lemuridae; Eulemur.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-499 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length884 Amino acids
Molecular weight95611
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 9732460
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Gene IDN/A
PDB IDN/A
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Search Result - 4

HMRbase accession number21210
Swiss-prot Accession numberP10275 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismHomo sapiens (Human)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Hominidae; Homo.
Subcellular locationNucleus
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Sumoylated on Lys-386 (major) and Lys-520. Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-534 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression.
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3.
Protein Length919 Amino acids
Molecular weight98989
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 3216866
2  PubMed abstract 2594783
3  PubMed abstract 2342476
4  PubMed abstract 3174628
5  PubMed abstract 2911578
6  PubMed abstract 2293020
7  PubMed abstract 15489334
8  PubMed abstract 2917688
9  PubMed abstract 3353726
10  PubMed abstract 3377788
11  PubMed abstract 2546571
12  PubMed abstract 3353727
13  PubMed abstract 1775137
14  PubMed abstract 1561105
15  PubMed abstract 9096391
16  PubMed abstract 10332029
17  PubMed abstract 10075738
18  PubMed abstract 10383460
19  PubMed abstract 10400640
20  PubMed abstract 10625666
21  PubMed abstract 10930412
22  PubMed abstract 11121022
23  PubMed abstract 12361945
24  PubMed abstract 12415108
25  PubMed abstract 14609956
26  PubMed abstract 14664718
27  PubMed abstract 12612053
28  PubMed abstract 16027218
29  PubMed abstract 16051670
30  PubMed abstract 17045208
31  PubMed abstract 17550981
32  PubMed abstract 10840043
33  PubMed abstract 11906285
34  PubMed abstract 15525515
35  PubMed abstract 15563469
36  PubMed abstract 16129672
37  PubMed abstract 16641486
38  PubMed abstract 18007036
39  PubMed abstract 17311914
40  PubMed abstract 17591767
41  PubMed abstract 17711855
42  PubMed abstract 17911242
43  PubMed abstract 1458719
44  PubMed abstract 8339746
45  PubMed abstract 8240973
46  PubMed abstract 7937057
47  PubMed abstract 7626493
48  PubMed abstract 9016528
49  PubMed abstract 2260966
50  PubMed abstract 2082179
51  PubMed abstract 1856263
52  PubMed abstract 1999491
53  PubMed abstract 2010552
54  PubMed abstract 2062380
55  PubMed abstract 1609793
56  PubMed abstract 1424203
57  PubMed abstract 1426313
58  PubMed abstract 1487249
59  PubMed abstract 1307250
60  PubMed abstract 1569163
61  PubMed abstract 1464650
62  PubMed abstract 1430233
63  PubMed abstract 1562539
64  PubMed abstract 1316540
65  PubMed abstract 1480178
66  PubMed abstract 1303262
67  PubMed abstract 1631125
68  PubMed abstract 8213813
69  PubMed abstract 8224266
70  PubMed abstract 8103398
71  PubMed abstract 8281139
72  PubMed abstract 8281140
73  PubMed abstract 8325932
74  PubMed abstract 8325950
75  PubMed abstract 8097257
76  PubMed abstract 8096390
77  PubMed abstract 8274409
78  PubMed abstract 8446106
79  PubMed abstract 8413310
80  PubMed abstract 8145761
81  PubMed abstract 7511268
82  PubMed abstract 8292051
83  PubMed abstract 8187068
84  PubMed abstract 7910529
85  PubMed abstract 7909256
86  PubMed abstract 8205256
87  PubMed abstract 8033918
88  PubMed abstract 8162033
89  PubMed abstract 7981687
90  PubMed abstract 7981689
91  PubMed abstract 8126121
92  PubMed abstract 7962294
93  PubMed abstract 8040309
94  PubMed abstract 7929841
95  PubMed abstract 7993455
96  PubMed abstract 7970939
97  PubMed abstract 8830623
98  PubMed abstract 7712463
99  PubMed abstract 7641413
100  PubMed abstract 7671849
101  PubMed abstract 7633398
102  PubMed abstract 7537149
103  PubMed abstract 7581399
104  PubMed abstract 7591265
105  PubMed abstract 7673412
106  PubMed abstract 8530589
107  PubMed abstract 7649358
108  PubMed abstract 7723794
109  PubMed abstract 8723113
110  PubMed abstract 9816170
111  PubMed abstract 9039340
112  PubMed abstract 9001799
113  PubMed abstract 8824883
114  PubMed abstract 8550758
115  PubMed abstract 8626869
116  PubMed abstract 8768864
117  PubMed abstract 8823308
118  PubMed abstract 8918984
119  PubMed abstract 8683794
120  PubMed abstract 8647313
121  PubMed abstract 8809734
122  PubMed abstract 8628719
123  PubMed abstract 8827083
124  PubMed abstract 9106550
125  PubMed abstract 9000575
126  PubMed abstract 9196614
127  PubMed abstract 9160185
128  PubMed abstract 9007482
129  PubMed abstract 8990010
130  PubMed abstract 9438000
131  PubMed abstract 9184448
132  PubMed abstract 9255042
133  PubMed abstract 9329414
134  PubMed abstract 9252933
135  PubMed abstract 9328206
136  PubMed abstract 9302173
137  PubMed abstract 9544375
138  PubMed abstract 9698822
139  PubMed abstract 9788719
140  PubMed abstract 9610419
141  PubMed abstract 9856504
142  PubMed abstract 9554754
143  PubMed abstract 9554755
144  PubMed abstract 9543136
145  PubMed abstract 9768671
146  PubMed abstract 9851768
147  PubMed abstract 9627582
148  PubMed abstract 9607727
149  PubMed abstract 10470409
150  PubMed abstract 10363963
151  PubMed abstract 10502786
152  PubMed abstract 10571951
153  PubMed abstract 10221692
154  PubMed abstract 10404311
155  PubMed abstract 10022458
156  PubMed abstract 10629558
157  PubMed abstract 10569618
158  PubMed abstract 10543676
159  PubMed abstract 10221770
160  PubMed abstract 10598582
161  PubMed abstract 10590024
162  PubMed abstract 10458483
163  PubMed abstract 10092153
164  PubMed abstract 10706109
165  PubMed abstract 10690872
166  PubMed abstract 11587068
167  PubMed abstract 11231320
168  PubMed abstract 11744994
169  PubMed abstract 15902657
170  PubMed abstract 16595706
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Gene ID367      
PDB ID1E3G   1GS4   1T5Z   1T63   1T65   1XJ7   1XOW   1XQ3   1Z95   2AM9   2AMA   2AMB   2AO6   2AX6   2AX7   2AX8   2AX9   2AXA   2HVC   2OZ7   2PIO   2PIP   2PIQ   2PIR   2PIT   2PIU   2PIV   2PIW   2PIX   2PKL   2PNU   2Q7I   2Q7J   2Q7K   2Q7L   2Z4J   3B5R   3B65   3B66   3B67   3B68      
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Search Result - 5

HMRbase accession number21211
Swiss-prot Accession numberO97952 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismMacaca fascicularis (Crab eating macaque) (Cynomolgus monkey)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Cercopithecidae; Cercopithecinae; Macaca.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-510 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length895 Amino acids
Molecular weight96495
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 9732460
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Gene IDN/A
PDB IDN/A
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Search Result - 6

HMRbase accession number21212
Swiss-prot Accession numberQ6QT55 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismMacaca mulatta (Rhesus macaque)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Cercopithecidae; Cercopithecinae; Macaca.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-510 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length895 Amino acids
Molecular weight96537
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 10208992
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Gene ID574293      
PDB IDN/A
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Search Result - 7

HMRbase accession number21213
Swiss-prot Accession numberP19091 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismMus musculus (Mouse)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Glires; Rodentia; Sciurognathi;Muroidea; Muridae; Murinae; Mus.
Subcellular locationNucleus
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-514 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3.
Protein Length899 Amino acids
Molecular weight98194
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 2403358
2  PubMed abstract 2178222
3  PubMed abstract 1883336
4  PubMed abstract 1681426
5  PubMed abstract 12058073
6  PubMed abstract 15199138
7  PubMed abstract 15882980
8  PubMed abstract 15988012
9  PubMed abstract 17911242
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Gene ID11835      
PDB ID2QPY      
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Search Result - 8

HMRbase accession number21214
Swiss-prot Accession numberO97775 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismPan troglodytes (Chimpanzee)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Hominidae; Pan.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-526 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length911 Amino acids
Molecular weight98403
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 9732460
2  PubMed abstract 15328534
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Gene ID449595      
PDB ID1T73   1T74   1T76   1T79   1T7F   1T7M   1T7R   1T7T      
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Search Result - 9

HMRbase accession number21215
Swiss-prot Accession numberO97960 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismPapio hamadryas (Hamadryas baboon)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Cercopithecidae; Cercopithecinae; Papio.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-510 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length895 Amino acids
Molecular weight96479
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 9732460
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Gene IDN/A
PDB IDN/A
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Search Result - 10

HMRbase accession number21216
Swiss-prot Accession numberQ9GKL7 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismSus scrofa (Pig)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Laurasiatheria; Cetartiodactyla; Suina; Suidae;Sus.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-511 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length896 Amino acids
Molecular weight97166
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 11086548
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Gene ID397582      
PDB IDN/A
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Search Result - 11

HMRbase accession number21217
Swiss-prot Accession numberP49699 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4; Fragment;
Source organismOryctolagus cuniculus (Rabbit)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Glires; Lagomorpha; Leporidae;Oryctolagus.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-324 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length709 Amino acids
Molecular weight77392
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 7559153
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PDB IDN/A
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Search Result - 12

HMRbase accession number21218
Swiss-prot Accession numberQ7T1K4 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;bfAR;
Source organismRana catesbeiana (Bull frog)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Amphibia; Batrachia; Anura; Neobatrachia; Ranoidea; Ranidae; Rana;Aquarana.
Subcellular locationNucleus (By similarity)
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityDetected in somatic Leydig and Sertoli cells in testis with high level expression. Also detected at lower expression levels in forebrain and heart.
Post translational modificationN/A
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins (By similarity).
Protein Length777 Amino acids
Molecular weight86436
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 13129498
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PDB IDN/A
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Search Result - 13

HMRbase accession number21219
Swiss-prot Accession numberP15207 (Sequence in FASTA format)
DescriptionRecName: Androgen receptor;Alternative Name: Dihydrotestosterone receptor;Alternative Name: Nuclear receptor subfamily 3 group C member 4;
Source organismRattus norvegicus (Rat)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Glires; Rodentia; Sciurognathi;Muroidea; Muridae; Murinae; Rattus.
Subcellular locationNucleus
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. NR3 subfamily. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityHighest levels in the seminal vesicle, ventral prostate and coagulating gland with lower levels in the kidney and levator ani muscle.
Post translational modification Phosphorylated in prostate cancer cells in response to several growth factors including EGF. Phosphorylation is induced by c-Src kinase (CSK). Tyr-517 is one of the major phosphorylation sites and an increase in phosphorylation and Src kinase activity is associated with prostate cancer progression (By similarity).
Function Steroid hormone receptors are ligand-activated transcription factors that regulate eukaryotic gene expression and affect cellular proliferation and differentiation in target tissues. Transcription factor activity is modulated by bound coactivator and corepressor proteins. Transcription activation is down-regulated by NR0B2. Activated, but not phosphorylated, by HIPK3 (By similarity).
Protein Length902 Amino acids
Molecular weight98218
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 3216867
2  PubMed abstract 3174628
3  PubMed abstract 2341409
4  PubMed abstract 9725910
5  PubMed abstract 12350225
6  PubMed abstract 11320241
7  PubMed abstract 15037741
8  PubMed abstract 15603938
9  PubMed abstract 17181141
10  PubMed abstract 17008401
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Gene ID24208      
PDB ID1I37   1I38   1R4I   1XNN   2IHQ   2NW4      
Drugpediawiki
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Search Result - 14

HMRbase accession number21901
Swiss-prot Accession numberO93244 (Sequence in FASTA format)
DescriptionAndrogen receptor alpha
Source organismOncorhynchus mykiss (Rainbow trout) (Salmo gairdneri)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei;Protacanthopterygii; Salmoniformes; Salmonidae; Salmoninae;Oncorhynchus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length854 Amino acids
Molecular weight96237
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 10026186
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Gene ID100135788      
PDB IDN/A
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Search Result - 15

HMRbase accession number21902
Swiss-prot Accession numberO93245 (Sequence in FASTA format)
DescriptionAndrogen receptor beta
Source organismOncorhynchus mykiss (Rainbow trout) (Salmo gairdneri)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei;Protacanthopterygii; Salmoniformes; Salmonidae; Salmoninae;Oncorhynchus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length853 Amino acids
Molecular weight95777
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 10026186
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Gene ID100135789      
PDB IDN/A
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Search Result - 16

HMRbase accession number21904
Swiss-prot Accession numberO93497 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismPagrus major (Red sea bream) (Chrysophrys major)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Perciformes; Percoidei;Sparidae; Pagrus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length769 Amino acids
Molecular weight86082
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 10395960
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PDB IDN/A
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Search Result - 17

HMRbase accession number21925
Swiss-prot Accession numberP70048 (Sequence in FASTA format)
DescriptionAndrogen receptor alpha isoform
Source organismXenopus laevis (African clawed frog)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Amphibia; Batrachia; Anura; Mesobatrachia; Pipoidea; Pipidae;Xenopodinae; Xenopus; Xenopus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length790 Amino acids
Molecular weight86974
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 7690145
2  PubMed abstract 7601302
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Gene ID399456      
PDB IDN/A
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Search Result - 18

HMRbase accession number21941
Swiss-prot Accession numberQ13771 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismHomo sapiens (Human)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Hominidae; Homo.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length730 Amino acids
Molecular weight79150
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 2342476
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PDB IDN/A
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Search Result - 19

HMRbase accession number22053
Swiss-prot Accession numberQ60I32 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismGambusia affinis (Western mosquitofish)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Atherinomorpha;Cyprinodontiformes; Poeciliidae; Gambusia.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length755 Amino acids
Molecular weight84333
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 15388345
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Search Result - 20

HMRbase accession number22076
Swiss-prot Accession numberQ66VR6 (Sequence in FASTA format)
DescriptionNuclear androgen receptor
Source organismMicropogonias undulatus (Atlantic croaker)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Perciformes; Percoidei;Sciaenidae; Micropogonias.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length757 Amino acids
Molecular weight85377
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
HormoneN/A
Gene IDN/A
PDB IDN/A
Drugpediawiki
Comments!Hormone for this Receptor are either unknown or have not yet been curated


Search Result - 21

HMRbase accession number22241
Swiss-prot Accession numberQ76LM5 (Sequence in FASTA format)
DescriptionAndrogen receptor alpha
Source organismOryzias latipes (Medaka fish) (Japanese ricefish)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Atherinomorpha;Beloniformes; Adrianichthyidae; Oryziinae; Oryzias.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length744 Amino acids
Molecular weight82424
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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Gene ID100049233      
PDB IDN/A
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Search Result - 22

HMRbase accession number22318
Swiss-prot Accession numberQ800S7 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismAcanthopagrus schlegeli (Black porgy)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Perciformes; Percoidei;Sparidae; Acanthopagrus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length771 Amino acids
Molecular weight86155
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 12672663
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Search Result - 23

HMRbase accession number22321
Swiss-prot Accession numberQ801Z1 (Sequence in FASTA format)
DescriptionAndrogen receptor beta 1
Source organismGasterosteus aculeatus (Three-spined stickleback)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Gasterosteiformes;Gasterosteidae; Gasterosteus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length682 Amino acids
Molecular weight76625
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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PDB IDN/A
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Search Result - 24

HMRbase accession number22322
Swiss-prot Accession numberQ801Z2 (Sequence in FASTA format)
DescriptionAndrogen receptor beta 2; Fragment
Source organismGasterosteus aculeatus (Three-spined stickleback)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Gasterosteiformes;Gasterosteidae; Gasterosteus.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length735 Amino acids
Molecular weight82153
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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PDB IDN/A
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Search Result - 25

HMRbase accession number22494
Swiss-prot Accession numberQ8QFV2 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismCarassius auratus (Goldfish)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Ostariophysi; Cypriniformes;Cyprinidae; Carassius.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length839 Amino acids
Molecular weight93171
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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PDB IDN/A
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Search Result - 26

HMRbase accession number22495
Swiss-prot Accession numberQ8QFV7 (Sequence in FASTA format)
DescriptionAndrogen receptor beta
Source organismHaplochromis burtoni (Burton's mouthbrooder)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Perciformes; Labroidei;Cichlidae; African cichlids; Pseudocrenilabrinae; Haplochromini;Haplochromis.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length763 Amino acids
Molecular weight84869
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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PDB IDN/A
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Search Result - 27

HMRbase accession number22533
Swiss-prot Accession numberQ8UWB7 (Sequence in FASTA format)
DescriptionAndrogen receptor beta
Source organismOreochromis niloticus (Nile tilapia) (Tilapia nilotica)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Euteleostei; Neoteleostei;Acanthomorpha; Acanthopterygii; Percomorpha; Perciformes; Labroidei;Cichlidae; African cichlids; Pseudocrenilabrinae; Tilapiini;Oreochromis.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length763 Amino acids
Molecular weight85024
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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PDB IDN/A
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Search Result - 28

HMRbase accession number22791
Swiss-prot Accession numberQ9I8F5 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismPimephales promelas
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Ostariophysi; Cypriniformes;Cyprinidae; Pimephales.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length839 Amino acids
Molecular weight92818
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 15597887
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PDB IDN/A
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Search Result - 29

HMRbase accession number22853
Swiss-prot Accession numberQ9PWG5 (Sequence in FASTA format)
DescriptionAndrogen receptor-beta
Source organismAnguilla japonica (Japanese eel)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Anguilliformes; Anguillidae;Anguilla.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length797 Amino acids
Molecular weight89925
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 10464240
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Search Result - 30

HMRbase accession number22906
Swiss-prot Accession numberQ9UN21 (Sequence in FASTA format)
DescriptionAndrogen receptor
Source organismHomo sapiens (Human)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Mammalia; Eutheria; Euarchontoglires; Primates; Haplorrhini;Catarrhini; Hominidae; Homo.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length906 Amino acids
Molecular weight97885
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References----
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Gene IDN/A
PDB IDN/A
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Search Result - 31

HMRbase accession number22948
Swiss-prot Accession numberQ9YGV9 (Sequence in FASTA format)
DescriptionAndrogen receptor alpha
Source organismAnguilla japonica (Japanese eel)
Taxonomical ClassificationEukaryota; Metazoa; Chordata; Craniata; Vertebrata; Euteleostomi;Actinopterygii; Neopterygii; Teleostei; Anguilliformes; Anguillidae;Anguilla.
Subcellular locationN/A
Developmental StageN/A
Similarity Belongs to the nuclear hormone receptor family. Contains 1 nuclear receptor DNA-binding domain.
Tissue SpecificityN/A
Post translational modification N/A
Function N/A
Protein Length848 Amino acids
Molecular weight94693
Domain NameAndrogen_recep  Hormone_recep  zf-C4  
References1  PubMed abstract 9918846
HormoneDetail in HMRbase   
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Detail in HMRbase   
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Gene IDN/A
PDB IDN/A
Drugpediawiki
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