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FWGALAKGALKLIGSLFSSFSKKD details |
Primary information | |
---|---|
ID | antitb_1187, |
Name | 25019413 |
N-Terminal modification | Pin2 [G] |
C-Terminal Modification | FWGALAKGALKLIGSLFSSFSKKD |
Chemical Modification | Free |
Linear/Cyclic | Free |
Length | None |
Chirality | Linear |
Nature | 24 |
Source | L |
Origin | Cationic |
Species | Synthetic |
Strain | Amino acid substitution at one postion of Pin2 (P at 14 by G) |
Inhibition Concentration | Mycobacterium tuberculosis |
In Vitro/ In vivo | Mycobacterium tuberculosis H37Rv |
Cell Line | MIC = 48.1 μg/ml or 18.7 μM |
Inhibition Concentration | In vitro |
Sequence | 2014 |
Cytotoxicity | RBC |
In vivo Model | NA |
Lethal Dose | Hemolysis ( IC-50 = 1.4 [0.4–4.3] ) |
Immune Responce | None |
Mechanism of Action | NA |
Target | NA |
Combination Therapy | Cell wall disruption |
Other activities | Cell wall |
PMID | None |
Year of Publication | Anti-bacterial (E. coli, S. aureus) |
Tertiary Structure (Technique) | Not Predicted), |
Primary information | |
---|---|
ID | antitb_1188, |
Name | 25019413 |
N-Terminal modification | Pin2 [G] |
C-Terminal Modification | FWGALAKGALKLIGSLFSSFSKKD |
Chemical Modification | Free |
Linear/Cyclic | Free |
Length | None |
Chirality | Linear |
Nature | 24 |
Source | L |
Origin | Cationic |
Species | Synthetic |
Strain | Amino acid substitution at one postion of Pin2 (P at 14 by G) |
Inhibition Concentration | Mycobacterium tuberculosis |
In Vitro/ In vivo | Mycobacterium tuberculosis muti-drug resistant strain (MDR) clinical isolate |
Cell Line | MIC = 48.1 μg/ml or 18.7 μM |
Inhibition Concentration | In vitro |
Sequence | 2014 |
Cytotoxicity | RBC |
In vivo Model | NA |
Lethal Dose | Hemolysis ( IC-50 = 1.4 [0.4–4.3] ) |
Immune Responce | None |
Mechanism of Action | NA |
Target | NA |
Combination Therapy | Cell wall disruption |
Other activities | Cell wall |
PMID | None |
Year of Publication | Anti-bacterial (E. coli, S. aureus) |
Tertiary Structure (Technique) | Not Predicted), |